IRIS
INCERTI, Matteo
 Distribuzione geografica
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Continente #
NA - Nord America 6.095
AS - Asia 5.283
EU - Europa 4.358
SA - Sud America 755
AF - Africa 345
Continente sconosciuto - Info sul continente non disponibili 183
OC - Oceania 2
Totale 17.021
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Nazione #
US - Stati Uniti d'America 5.923
SG - Singapore 1.763
CN - Cina 1.520
IT - Italia 1.015
VN - Vietnam 921
IE - Irlanda 643
FI - Finlandia 609
BR - Brasile 597
SE - Svezia 589
DE - Germania 425
HK - Hong Kong 396
UA - Ucraina 310
ZA - Sudafrica 240
FR - Francia 197
BD - Bangladesh 165
NL - Olanda 141
TR - Turchia 117
GB - Regno Unito 115
CA - Canada 102
IN - India 94
AR - Argentina 77
RU - Federazione Russa 76
AT - Austria 51
JP - Giappone 43
MX - Messico 40
BE - Belgio 39
CI - Costa d'Avorio 39
ID - Indonesia 34
IQ - Iraq 34
PH - Filippine 32
KR - Corea 31
ES - Italia 26
CZ - Repubblica Ceca 22
EC - Ecuador 22
TH - Thailandia 22
GR - Grecia 21
VE - Venezuela 20
MA - Marocco 17
PK - Pakistan 16
HU - Ungheria 15
EG - Egitto 14
LT - Lituania 14
PL - Polonia 14
SA - Arabia Saudita 12
UZ - Uzbekistan 11
CO - Colombia 10
JO - Giordania 10
KE - Kenya 10
TN - Tunisia 10
CL - Cile 9
AL - Albania 6
IL - Israele 6
JM - Giamaica 6
LB - Libano 6
PY - Paraguay 6
BO - Bolivia 5
ET - Etiopia 5
IR - Iran 5
NP - Nepal 5
PE - Perù 5
SN - Senegal 5
TW - Taiwan 5
AE - Emirati Arabi Uniti 4
AZ - Azerbaigian 4
CH - Svizzera 4
HN - Honduras 4
KZ - Kazakistan 4
OM - Oman 4
RO - Romania 4
SV - El Salvador 4
UY - Uruguay 4
CR - Costa Rica 3
DK - Danimarca 3
KG - Kirghizistan 3
MY - Malesia 3
NI - Nicaragua 3
NO - Norvegia 3
PA - Panama 3
AM - Armenia 2
AU - Australia 2
BG - Bulgaria 2
BH - Bahrain 2
HR - Croazia 2
KH - Cambogia 2
LK - Sri Lanka 2
NG - Nigeria 2
RS - Serbia 2
SI - Slovenia 2
SY - Repubblica araba siriana 2
AD - Andorra 1
BB - Barbados 1
BY - Bielorussia 1
CY - Cipro 1
DO - Repubblica Dominicana 1
DZ - Algeria 1
EE - Estonia 1
GD - Grenada 1
GT - Guatemala 1
KY - Cayman, isole 1
LU - Lussemburgo 1
Totale 16.828
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Città #
Singapore 880
Dublin 643
Ashburn 630
Chandler 551
San Jose 514
Beijing 442
Santa Clara 416
Hong Kong 360
Jacksonville 350
Parma 322
Dallas 292
Ho Chi Minh City 266
Ann Arbor 251
Johannesburg 228
Hanoi 217
Council Bluffs 208
Boardman 199
Dearborn 185
Nanjing 155
Los Angeles 142
New York 136
Shanghai 113
Lauterbourg 111
Princeton 108
Izmir 89
Munich 87
Wilmington 83
San Mateo 79
Hefei 70
Bremen 66
São Paulo 61
Toronto 61
Helsinki 55
Chicago 50
Shenyang 50
Vienna 49
Buffalo 48
Kunming 44
Rome 43
Milan 42
Abidjan 39
Grafing 39
Haiphong 37
Moscow 37
Bologna 36
Hebei 36
Jinan 36
Nanchang 36
Da Nang 35
Guangzhou 34
Tokyo 34
Columbus 33
Brussels 32
Des Moines 29
Tianjin 29
Frankfurt am Main 27
Houston 27
Turku 26
Modena 25
Seattle 25
Rio de Janeiro 22
Woodbridge 22
Jiaxing 21
Pune 20
The Dalles 20
Changsha 19
Jakarta 18
London 18
Montreal 17
Orem 17
Atlanta 16
Chennai 16
Denver 16
Mexico City 16
Seoul 16
Belo Horizonte 15
Brasília 15
Poplar 15
San Francisco 15
Brooklyn 14
Can Tho 14
Fremont 14
Phoenix 14
Biên Hòa 13
Brescia 13
Hangzhou 13
Ninh Bình 13
Nuremberg 13
Athens 12
Brno 12
Hải Dương 12
Norwalk 12
Zhengzhou 12
Ankara 11
Boston 11
Bắc Ninh 11
Curitiba 11
Baghdad 10
Bangkok 10
Düsseldorf 10
Totale 9.937
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Nome #
A New ABCB1 Inhibitor Enhances the Anticancer Effect of Doxorubicin in Both In Vitro and In Vivo Models of NSCLC 299
Hydroxyphenyl thiosemicarbazones as inhibitors of mushroom tyrosinase and antibrowning agents. 274
A potentiometric and spectrofluorimetric approach to unravel inhibitory effects of semi- and thiosemicarbazones on mushroom tyrosinase activity 249
Inhibition of Eph/ephrin interaction with the small molecule UniPR500 improves glucose tolerance in healthy and insulin-resistant mice 244
Pharmacological evaluation of new bioavailable small molecules targeting Eph/ephrin interaction 228
Effetto di derivati dell'urea sulla radicazione avventizia in vitro di microtalee micropropagate di corbezzolo 227
Development of an orally bioavailable small molecule targeting Eph-ephrin system: in vitro and in vivo anticancer activity. 223
Complete 1H and 13C NMR spectral assignment of benzo[d]isothiazole derivatives and of an isoindole isoster 222
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. 221
Probucol treatment is associated with an ABCA1-independent mechanism of cholesterol efflux to lipid poor apolipoproteins from foam cell macrophages 221
Effect of Cl-Substitution on Rooting- or Cytokinin-like Activity of Diphenylurea Derivatives 220
Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3α-carbamoyloxy derivative with antiangiogenetic properties 220
Metabolic Soft Spot and Pharmacokinetics: Functionalization of C-3 Position of an Eph–Ephrin Antagonist Featuring a Bile Acid Core as an Effective Strategy to Obtain Oral Bioavailability in Mice 215
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties 207
Combining ligand- and structure-based approaches for the discovery of new inhibitors of the EPHA2-ephrin-A1 interaction 204
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses 202
A new efficient route to 7-aryl-6-fluoro-8-nitroquinolones as potent antibacterial agents 201
UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations. 199
Adventitious rooting adjuvant activity of 1,3-di(benzo[d]oxazol-5-yl) urea and 1,3-di(benzo[d]oxazol-6-yl)urea: new insights and perspectives 196
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists 189
Discovery and development of small molecules targeting Eph-ephrin system in glioblastoma: an academic history 179
4-Chloro-N-(4-chlorophenylsulfonyl)-N-(3-oxo-2,3-dihydro-1,2-benzisothiazol-2-yl)benzenesulfonamide 178
Lithocholic acid is an Eph-ephrin ligand interfering with Eph-kinase activation 178
inibitori eph-ephrin biodisponibili oralmente 177
A one-pot PPh3-promoted synthesis of new functionalized heterocycles derived from 2-aminobenzo[d]isothiazol-3-one 177
Structure–Activity Relationships and Mechanism of Action of Eph–ephrin Antagonists: Interaction of Cholanic Acid with the EphA2 Receptor 177
270 Discovery, development and optimization of low molecular weight EPH–ephrin protein–protein inhibitors 175
Probing the effects of MR120 in preclinical chronic colitis: A first-in-class anti-IBD agent targeting the CCL20/CCR6 axis 174
2-Benzo[d]isothiazolylimino-5-arylidene-4-thiazolidinones: Synthesis and antimicrobial activity 172
Dual-Acting Drugs: an in vitro Study of Nonimidazole Histamine H(3) Receptor Antagonists Combining Anticholinesterase Activity 168
4-Methyl-N-(3-oxo-2,3-dihydro-1,2-benzisothiazol-2-yl)benzenesulfonamide 168
2-Heteroarylimino-5-benzylidene-4-thiazolidinones analogues of 2-thiazolylimino-5-benzylidene-4-thiazolidinones with antimicrobial activity: synthesis and structure-activity relationship. 166
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis 165
A ONE-POT ENTRY TO A NOVEL 3-H-BENZO[D]PYRAZOLO[1,5-B]ISOTHIAZOLE RING SYSTEM. 164
Multiple approaches for the discovery and development of small molecules targeting Eph-ephrin protein-protein interaction 162
Eph/ephrin targeting with a small molecule improves glucose tolerance in healthy and insulin-resistant mice 160
Biochemical characterization of EphA2 antagonists with improved physico-chemical properties by cell-based assays and surface plasmon resonance analysis 159
Amidinobenzisothiazole derivatives with antidegenerative activity on cartilage 156
2-Benzisothiazolylimino-5-benzylidene-4-thiazolidinones as protective agents against cartilage destruction 155
New ALKBH2 and ALKBH5 inhibitors for treating glioblastoma 154
2-Benzisothiazolylimino-5-benzylidene-4-thiazolidinones as protective agents against cartilage destruction. 153
Δ5-Cholenoyl-amino acids as selective and orally available antagonists of the Eph-ephrin system 153
Structure activity relationship of new EphA2 ligands 152
Evaluation of the anti-tumor activity of small molecules targeting eph/ephrins in apcmin j mice 152
Aminoderivatives of benzothiazole/benzisothiazole heterocycles as intermediates in the synthesis of novel therapeutic agents 151
Design and structure-activity relationships of amino acid derivatives of lithocholic acid as novel EphA2 receptor antagonists. 151
Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return 151
New MDR1 inhibitors for overcoming multidrug resistance 150
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction. 150
Comparative Analysis of Virtual Screening Approaches in the Search for Novel EphA2 Receptor Antagonists 148
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity 147
Synthesis and NMR spectral assignments of novel 1,4-benzothiazepine-5-one derivatives 146
2-BENZO[d]ISOTHIAZOLYLIMINO-5-ARYLIDENE-4-THIAZOLIDINONES: SYNTHESIS AND ANTIMICROBIAL ACTIVITY 145
Target-hopping: a useful approach to identify novel Eph receptor antagonists 141
Effects of a dietary intervention with Mediterranean vs lacto-ovo vegetarian diets on HDL function: results from the CARDIVEG study 140
Metadynamics for perspective drug design: Computationally driven synthesis of new protein-protein interaction inhibitors targeting the EphA2 receptor 139
Computer-Aided Design of Novel Antagonists of the EphA2 Receptor 138
A one-pot PPh3-promoted synthesis of new functionalized heterocycles derived from 2-aminobenzo[d]isothiazol-3-one 137
Target Hopping as a Useful Tool for the Identification of Novel EphA2 Protein–Protein Antagonists 137
4-thiazolidinone derivatives as MMP inhibitors in tissue damage: Synthesis, biological evaluation and docking studies 137
Diheteroarylurea derivatives as adventitious rooting adjuvants in mung bean shoots and M26 apple rootstock. 136
Structure-activity relationships of N-phenyl-N’-benzothiazol-6-ylurea synthetic derivatives: cytokinin-like activity and adventitious rooting enhancement 136
Lomitapide modifies high-density lipoprotein function in homozygous familial hypercholesterolaemia 132
Lithocholic acid competitively inhibitis EphA2-ephrinA1 binding: pharmacological and structural considerations. 128
Are we using the right pharmacological tools to target EphA4? 128
QSAR analysis of 4-thiazolidinone derivatives with antimicrobial activity. 127
Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor. 127
Weakly cytokinin-active diphenylurea derivatives influence adventitious rooting in M26 Malus pumila microcuttings 126
Synthesis and antiproliferative activity of novel benzo[d]isothiazole compounds bearing a 2,4-dinitrophenyl group. 126
Lithocholic acid competitively inhibits EphA2-ephrinA1 binding: pharmacological and structural considerations. 126
Attività antiproliferativa di N-(1,2-benzisothiaziol-3-il)benzaamidine su cellule di carcinoma colon-rettale umano 126
Lithocholic Acid Is an Eph-ephrin Ligand Interfering with Eph-kinase Activation. 125
Synthesis and antimicrobial properties of 2-(benzylidene -amino)-benzo[d]isothiazol-3-ones 124
Benzisothiazolylimino-5-benzylidene-4-thiazolidinones as potential biologically active agents 123
Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties 121
Synthesis and antimicrobial properties of benzothiazole benzenesulfonamides 121
Anti-HIV evaluation of benzo[d]isothiazole hydrazones. 121
Synthesis and biological evaluation of tetracyclic fluoroquinolones as antibacterial and anticancer agents 119
Synthesis and pharmacological properties of benzisothiazole/benzimidazole derivatives with acidic groups 118
Benzisothiazolyliminothiazolidin-4-ones with chondroprotective properties: searching for potent and selective inhibitors of MMP-13. 116
Design synthesis and antibacterial activity studies of new thiadiazoloquinolone compounds 115
Antidegenerative activity of heteroarylimino-4-thiazolidinones on human chondrocyte cultures stimulated by IL-1ß 115
Synthesis of benzisoxazole and benzisothiazole derivatives with potential antitumor activity 115
On the Use of 2,5-Dimethyl-Pyrrol-1-yl-Benzoic Acid Derivatives as EPH-Ephrin Antagonists. 114
Investigation of the reaction between 3-benzisothiazolones, an isoindole isoster and activated acetylenes: synthesis of novel heterocyclic backbones for building bioactive molecules 114
Heterocycles [h]-fused to 4-oxoquinoline-3-carboxylic acid. Part XI: Synthesis and antibacterial activity of 4-fluoro-6-oxoimidazo[4,5-h]quinoline-7-carboxylic acids 113
A Microwave‐Assisted One‐Pot Three‐Step Metal‐Free [4+2] Annulation for the Sustainable Synthesis of Highly Substituted 1,2,4‐Triazines 113
Synthesis and biological evaluation of benzo[d]isothiazole, benzothiazole and thiazole Schiff bases 112
Synthesis and biological evaluation of tetracyclic thienopyridones as antibacterial and antitumor agents 111
Thiazolyl and isothiazolyl azomethine derivatives with antiinflammatory and antioxidant activities. Synthesis, biological evaluation and structure activity relationships study 110
Lipophilicity estimation of new benzisothiazolone derivatives with anti HIV-1 activity for a rational study of structure-activity relationship 110
Multi-target-directed ligands: new histamine H3 receptor antagonists with anticholinesterase activity 110
Stereospecific effects of benzo(d)isothiazolyloxypropanolamine derivatives at beta-adrenoceptors: synthesis, chiral resolution, and biological activity in vitro 106
PHARMACOLOGICAL, ATP-BINDING CASSETTE TRANSPORTER A1 (ABCA1)-DEPENDENT MEMBRANE FREE CHOLESTEROL POOL REDUCTION LEADS TO ATHEROPROTECTIVE MODULATION OF MACROPHAGE FUNCTIONS 106
Phenyl thiosemicarbazide cyclization leads to the versatile 1,3,4-thiadiazole scaffold: Structural analysis of its copper(I) complex 104
Synthesis and effect of new N-(1,2-benzo[d]isothiazol-3-yl) benzamidines on IL-1- induced alteration in cartilage metabolism 103
Synthesis and evaluation as antimicrobial agents of novel heteroaryl sulfonamides 102
Synthesis of novel 5-arylidene-thiazol-4-ones 2-heteroarylamino substituted as potential antimicrobials 102
Synthesis and Antiproliferative Activity of Benzo[d]isothiazole Hydrazones. 99
Synthesis and biological activity of hydrazones of benzo[d]isothiazole hydrazides 99
Totale 15.422
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Categoria #
all - tutte 56.940
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 56.940
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022650 0 15 20 70 24 55 70 87 37 55 25 192
2022/20232.326 245 261 126 169 217 240 44 145 763 20 62 34
2023/2024858 56 64 40 23 60 191 95 65 20 36 68 140
2024/20252.731 92 166 189 150 305 298 138 127 295 235 241 495
2025/20266.360 545 576 683 629 836 342 642 254 966 427 259 201
2026/2027472 167 305 0 0 0 0 0 0 0 0 0 0
Totale 17.021