Sfoglia per Autore
A Multidisciplinary Approach for the Identification of Novel HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: S-DABOCs and DAVPs
2008-01-01 Radi, Marco; Chiara, Falciani; Lorenzo, Contemori; Elena, Petricci; Giovanni, Maga; Alberta, Samuele; Samantha, Zanoli; Montserrat, Terrazas; Marinunzia, Castria; Andrea, Togninelli; Esté, J. o. s. é. . A.; Imma Clotet, Codina; Mercedes Armand, Ugón; Maurizio, Botta
Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents
2008-01-01 Radi, Marco; Emmanuele, Crespan; Giorgia, Botta; Federico, Falchi; Giovanni, Maga; Fabrizio, Manetti; Valentina, Corradi; Manuela, Mancini; Maria Alessandra, Santucci; Silvia, Schenone; Maurizio, Botta
The fight against AIDS: new avenues for inhibiting reverse transcriptase (RT), an old target
2008-01-01 Maurizio, Botta; Lucilla, Angeli; Radi, Marco; Giovanni, Maga
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis
2008-01-01 Daniele, Castagnolo; Alessandro De, Logu; Radi, Marco; Beatrice, Bechi; Fabrizio, Manetti; Matteo, Magnani; Sibilla, Supino; Rita, Meleddu; Lorenza, Chisu; Maurizio, Botta
A one-pot, two-step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs)
2008-01-01 Radi, Marco; Sara, Saletti; Maurizio, Botta
4-Amino-Substituted Pyrazolo[3,4-d]Pyrimidines: Synthesis and Biological Properties
2009-01-01 Silvia, Schenone; Olga, Bruno; Radi, Marco; Maurizio, Botta
Recent highlights in the synthesis of highly functionalized pyrimidines
2009-01-01 Radi, Marco; Silvia, Schenone; Maurizio, Botta
Discovery of Chiral Cyclopropyl Dihydro-Alkylthio-Benzyl-Oxopyrimidine (S-DABO) Derivatives as Potent HIV-1 Reverse Transcriptase Inhibitors with High Activity Against Clinically Relevant Mutants
2009-01-01 Radi, Marco; Giovanni, Maga; Maddalena, Alongi; Lucilla, Angeli; Alberta, Samuele; Samantha, Zanoli; Luca, Bellucci; Andrea, Tafi; Gianni, Casaluce; Gianluca, Giorgi; Mercedes Armand, Ugon; Emmanuel, Gonzalez; José A., Esté; Mireille, Baltzinger; Guillaume, Bec; Philippe, Dumas; Eric, Ennifar; Maurizio, Botta
Crystal structure of HIV-1 reverse transcriptase bound to a nucleotide-competitive reverse transcriptase inhibitor and the use thereof
2009-01-01 Radi, Marco; Maurizio, Botta; Lucilla, Angeli; Giovanni, Maga; Eric, Ennifar; Philippe, Dumas; Philippe, Wolff; Guillaume, Bec; Severine, Freisz
Compounds with DDX3 inhibitory activity and uses thereof
2009-01-01 Radi, Marco; Maurizio, Botta; Federico, Falchi; Giovanni, Maga; Fausto, Baldanti; Stefania, Paolucci
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones
2009-01-01 Daniele, Castagnolo; Fabrizio, Manetti; Radi, Marco; Beatrice, Bechi; Mafalda, Pagano; Alessandro De, Logu; Rita, Meleddu; Manuela, Saddi; Maurizio, Botta
Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis
2009-01-01 Daniele, Castagnolo; Radi, Marco; Filippo, Dessì; Fabrizio, Manetti; Manuela, Saddi; Rita, Meleddu; Alessandro De, Logu; Maurizio, Botta
Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles
2009-01-01 Radi, Marco; Vincenzo, Bernardo; Beatrice, Bechi; Daniele, Castagnolo; Mafalda, Pagano; Maurizio, Botta
A Convergent Approach for the Synthesis of Ara-Neplanocin a Analogues Under Subzero Microwave Assisted Conditions
2009-01-01 Radi, Marco; Jagadeeshwar R., Rao; Ashok K., Jha; Chu, Chung K.
C6-Unsubstituted Pyrazolo[3,4-d]pyrimidines Are Dual Src/Abl Inhibitors Effective against Imatinib Mesylate Resistant Chronic Myeloid Leukemia Cell Lines
2009-01-01 Maria Alessandra, Santucci; Valentina, Corradi; Manuela, Mancini; Fabrizio, Manetti; Radi, Marco; Silvia, Schenone; Maurizio, Botta
Crystal Structure of HIV-1 Reverse Transcriptase Bound to a Non-Nucleoside Inhibitor with a Novel Mechanism of Action
2010-01-01 Séverine, Freisz; Guillaume, Bec; Radi, Marco; Philippe, Wolff; Emmanuele, Crespan; Lucilla, Angeli; Philippe, Dumas; Giovanni, Maga; Maurizio, Botta; Eric, Ennifar
Dual Src and Abl inhibitors target wild type Abl and the AblT315I Imatinib-resistant mutant with different mechanisms
2010-01-01 Emmanuele, Crespan; Radi, Marco; Samantha, Zanoli; Silvia, Schenone; Maurizio, Botta; Giovanni, Maga
Arylation of 2-Furyl 4-Fluorophenyl Ketone: An Extension of Heck Chemistry towards Novel Integrase Inhibitors
2010-01-01 Luigi, Franchi; Marta, Rinaldi; Giulia, Vignaroli; Anna, Innitzer; Radi, Marco; Maurizio, Botta
Molecular Characterization of c-Abl/c-Src Kinase Inhibitors Targeted against Murine Tumour Progenitor Cells that Express Stem Cell Markers
2010-01-01 Thomas, Kruewel; Silvia, Schenone; Radi, Marco; Giovanni, Maga; Astrid, Rohrbeck; Maurizio, Botta; Juergen, Borlak
Practical One-Pot Two-Step Protocol for the Microwave-Assisted Synthesis of Highly Functionalized Rhodanine Derivatives
2010-01-01 Radi, Marco; Lorenzo, Botta; Gianni, Casaluce; Martina, Bernardini; Maurizio, Botta
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
A Multidisciplinary Approach for the Identification of Novel HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: S-DABOCs and DAVPs | 1-gen-2008 | Radi, Marco; Chiara, Falciani; Lorenzo, Contemori; Elena, Petricci; Giovanni, Maga; Alberta, Samuele; Samantha, Zanoli; Montserrat, Terrazas; Marinunzia, Castria; Andrea, Togninelli; Esté, J. o. s. é. . A.; Imma Clotet, Codina; Mercedes Armand, Ugón; Maurizio, Botta | |
Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents | 1-gen-2008 | Radi, Marco; Emmanuele, Crespan; Giorgia, Botta; Federico, Falchi; Giovanni, Maga; Fabrizio, Manetti; Valentina, Corradi; Manuela, Mancini; Maria Alessandra, Santucci; Silvia, Schenone; Maurizio, Botta | |
The fight against AIDS: new avenues for inhibiting reverse transcriptase (RT), an old target | 1-gen-2008 | Maurizio, Botta; Lucilla, Angeli; Radi, Marco; Giovanni, Maga | |
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis | 1-gen-2008 | Daniele, Castagnolo; Alessandro De, Logu; Radi, Marco; Beatrice, Bechi; Fabrizio, Manetti; Matteo, Magnani; Sibilla, Supino; Rita, Meleddu; Lorenza, Chisu; Maurizio, Botta | |
A one-pot, two-step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs) | 1-gen-2008 | Radi, Marco; Sara, Saletti; Maurizio, Botta | |
4-Amino-Substituted Pyrazolo[3,4-d]Pyrimidines: Synthesis and Biological Properties | 1-gen-2009 | Silvia, Schenone; Olga, Bruno; Radi, Marco; Maurizio, Botta | |
Recent highlights in the synthesis of highly functionalized pyrimidines | 1-gen-2009 | Radi, Marco; Silvia, Schenone; Maurizio, Botta | |
Discovery of Chiral Cyclopropyl Dihydro-Alkylthio-Benzyl-Oxopyrimidine (S-DABO) Derivatives as Potent HIV-1 Reverse Transcriptase Inhibitors with High Activity Against Clinically Relevant Mutants | 1-gen-2009 | Radi, Marco; Giovanni, Maga; Maddalena, Alongi; Lucilla, Angeli; Alberta, Samuele; Samantha, Zanoli; Luca, Bellucci; Andrea, Tafi; Gianni, Casaluce; Gianluca, Giorgi; Mercedes Armand, Ugon; Emmanuel, Gonzalez; José A., Esté; Mireille, Baltzinger; Guillaume, Bec; Philippe, Dumas; Eric, Ennifar; Maurizio, Botta | |
Crystal structure of HIV-1 reverse transcriptase bound to a nucleotide-competitive reverse transcriptase inhibitor and the use thereof | 1-gen-2009 | Radi, Marco; Maurizio, Botta; Lucilla, Angeli; Giovanni, Maga; Eric, Ennifar; Philippe, Dumas; Philippe, Wolff; Guillaume, Bec; Severine, Freisz | |
Compounds with DDX3 inhibitory activity and uses thereof | 1-gen-2009 | Radi, Marco; Maurizio, Botta; Federico, Falchi; Giovanni, Maga; Fausto, Baldanti; Stefania, Paolucci | |
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones | 1-gen-2009 | Daniele, Castagnolo; Fabrizio, Manetti; Radi, Marco; Beatrice, Bechi; Mafalda, Pagano; Alessandro De, Logu; Rita, Meleddu; Manuela, Saddi; Maurizio, Botta | |
Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis | 1-gen-2009 | Daniele, Castagnolo; Radi, Marco; Filippo, Dessì; Fabrizio, Manetti; Manuela, Saddi; Rita, Meleddu; Alessandro De, Logu; Maurizio, Botta | |
Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles | 1-gen-2009 | Radi, Marco; Vincenzo, Bernardo; Beatrice, Bechi; Daniele, Castagnolo; Mafalda, Pagano; Maurizio, Botta | |
A Convergent Approach for the Synthesis of Ara-Neplanocin a Analogues Under Subzero Microwave Assisted Conditions | 1-gen-2009 | Radi, Marco; Jagadeeshwar R., Rao; Ashok K., Jha; Chu, Chung K. | |
C6-Unsubstituted Pyrazolo[3,4-d]pyrimidines Are Dual Src/Abl Inhibitors Effective against Imatinib Mesylate Resistant Chronic Myeloid Leukemia Cell Lines | 1-gen-2009 | Maria Alessandra, Santucci; Valentina, Corradi; Manuela, Mancini; Fabrizio, Manetti; Radi, Marco; Silvia, Schenone; Maurizio, Botta | |
Crystal Structure of HIV-1 Reverse Transcriptase Bound to a Non-Nucleoside Inhibitor with a Novel Mechanism of Action | 1-gen-2010 | Séverine, Freisz; Guillaume, Bec; Radi, Marco; Philippe, Wolff; Emmanuele, Crespan; Lucilla, Angeli; Philippe, Dumas; Giovanni, Maga; Maurizio, Botta; Eric, Ennifar | |
Dual Src and Abl inhibitors target wild type Abl and the AblT315I Imatinib-resistant mutant with different mechanisms | 1-gen-2010 | Emmanuele, Crespan; Radi, Marco; Samantha, Zanoli; Silvia, Schenone; Maurizio, Botta; Giovanni, Maga | |
Arylation of 2-Furyl 4-Fluorophenyl Ketone: An Extension of Heck Chemistry towards Novel Integrase Inhibitors | 1-gen-2010 | Luigi, Franchi; Marta, Rinaldi; Giulia, Vignaroli; Anna, Innitzer; Radi, Marco; Maurizio, Botta | |
Molecular Characterization of c-Abl/c-Src Kinase Inhibitors Targeted against Murine Tumour Progenitor Cells that Express Stem Cell Markers | 1-gen-2010 | Thomas, Kruewel; Silvia, Schenone; Radi, Marco; Giovanni, Maga; Astrid, Rohrbeck; Maurizio, Botta; Juergen, Borlak | |
Practical One-Pot Two-Step Protocol for the Microwave-Assisted Synthesis of Highly Functionalized Rhodanine Derivatives | 1-gen-2010 | Radi, Marco; Lorenzo, Botta; Gianni, Casaluce; Martina, Bernardini; Maurizio, Botta |
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