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Mostrati risultati da 21 a 40 di 97
Titolo Data di pubblicazione Autore(i) File
Discovery and SAR of 1,3,4-thiadiazole derivatives as potent Abl tyrosine kinase inhibitors and cytodifferentiating agents 1-gen-2008 Radi, Marco; Emmanuele, Crespan; Giorgia, Botta; Federico, Falchi; Giovanni, Maga; Fabrizio, Manetti; Valentina, Corradi; Manuela, Mancini; Maria Alessandra, Santucci; Silvia, Schenone; Maurizio, Botta
A one-pot, two-step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs) 1-gen-2008 Radi, Marco; Sara, Saletti; Maurizio, Botta
Synthesis of an Original Oxygenated Taxuspine X Analogue: a Versatile “Non-Natural” Natural Product with Remarkable P-gp Modulating Activity 1-gen-2008 Avramova, S. t. a. n. i. s. l. a. v. a.  . I.; Elena, Galletti; Renzulli, M. i. c. h. e. l. a.  . L.; Gianluca, Giorgi; Gianpietro, Sgaragli; Daniela, Alderighi; Chiara, Ghiron; Federico, Corelli; Radi, Marco; Maurizio, Botta
Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis 1-gen-2008 Daniele, Castagnolo; Alessandro De, Logu; Radi, Marco; Beatrice, Bechi; Fabrizio, Manetti; Matteo, Magnani; Sibilla, Supino; Rita, Meleddu; Lorenza, Chisu; Maurizio, Botta
A Multidisciplinary Approach for the Identification of Novel HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: S-DABOCs and DAVPs 1-gen-2008 Radi, Marco; Chiara, Falciani; Lorenzo, Contemori; Elena, Petricci; Giovanni, Maga; Alberta, Samuele; Samantha, Zanoli; Montserrat, Terrazas; Marinunzia, Castria; Andrea, Togninelli; Esté, J. o. s. é.  . A.; Imma Clotet, Codina; Mercedes Armand, Ugón; Maurizio, Botta
4-Amino-Substituted Pyrazolo[3,4-d]Pyrimidines: Synthesis and Biological Properties 1-gen-2009 Silvia, Schenone; Olga, Bruno; Radi, Marco; Maurizio, Botta
Crystal structure of HIV-1 reverse transcriptase bound to a nucleotide-competitive reverse transcriptase inhibitor and the use thereof 1-gen-2009 Radi, Marco; Maurizio, Botta; Lucilla, Angeli; Giovanni, Maga; Eric, Ennifar; Philippe, Dumas; Philippe, Wolff; Guillaume, Bec; Severine, Freisz
Compounds with DDX3 inhibitory activity and uses thereof 1-gen-2009 Radi, Marco; Maurizio, Botta; Federico, Falchi; Giovanni, Maga; Fausto, Baldanti; Stefania, Paolucci
A Convergent Approach for the Synthesis of Ara-Neplanocin a Analogues Under Subzero Microwave Assisted Conditions 1-gen-2009 Radi, Marco; Jagadeeshwar R., Rao; Ashok K., Jha; Chu, Chung K.
Synthesis and biological evaluation of new enantiomerically pure azole derivatives as inhibitors of Mycobacterium tuberculosis 1-gen-2009 Daniele, Castagnolo; Radi, Marco; Filippo, Dessì; Fabrizio, Manetti; Manuela, Saddi; Rita, Meleddu; Alessandro De, Logu; Maurizio, Botta
Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones 1-gen-2009 Daniele, Castagnolo; Fabrizio, Manetti; Radi, Marco; Beatrice, Bechi; Mafalda, Pagano; Alessandro De, Logu; Rita, Meleddu; Manuela, Saddi; Maurizio, Botta
Discovery of Chiral Cyclopropyl Dihydro-Alkylthio-Benzyl-Oxopyrimidine (S-DABO) Derivatives as Potent HIV-1 Reverse Transcriptase Inhibitors with High Activity Against Clinically Relevant Mutants 1-gen-2009 Radi, Marco; Giovanni, Maga; Maddalena, Alongi; Lucilla, Angeli; Alberta, Samuele; Samantha, Zanoli; Luca, Bellucci; Andrea, Tafi; Gianni, Casaluce; Gianluca, Giorgi; Mercedes Armand, Ugon; Emmanuel, Gonzalez; José A., Esté; Mireille, Baltzinger; Guillaume, Bec; Philippe, Dumas; Eric, Ennifar; Maurizio, Botta
Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles 1-gen-2009 Radi, Marco; Vincenzo, Bernardo; Beatrice, Bechi; Daniele, Castagnolo; Mafalda, Pagano; Maurizio, Botta
C6-Unsubstituted Pyrazolo[3,4-d]pyrimidines Are Dual Src/Abl Inhibitors Effective against Imatinib Mesylate Resistant Chronic Myeloid Leukemia Cell Lines 1-gen-2009 Maria Alessandra, Santucci; Valentina, Corradi; Manuela, Mancini; Fabrizio, Manetti; Radi, Marco; Silvia, Schenone; Maurizio, Botta
Recent highlights in the synthesis of highly functionalized pyrimidines 1-gen-2009 Radi, Marco; Silvia, Schenone; Maurizio, Botta
Design and Synthesis of Thiadiazoles and Thiazoles Targeting the Bcr-Abl T315I Mutant: from Docking False Positives to ATP-Noncompetitive Inhibitors 1-gen-2010 Radi, Marco; Emmanuele, Crespan; Federico, Falchi; Vincenzo, Bernardo; Samantha, Zanoli; Fabrizio, Manetti; Silvia, Schenone; Giovanni, Maga; Maurizio, Botta
Molecular Characterization of c-Abl/c-Src Kinase Inhibitors Targeted against Murine Tumour Progenitor Cells that Express Stem Cell Markers 1-gen-2010 Thomas, Kruewel; Silvia, Schenone; Radi, Marco; Giovanni, Maga; Astrid, Rohrbeck; Maurizio, Botta; Juergen, Borlak
Dual Src and Abl inhibitors target wild type Abl and the AblT315I Imatinib-resistant mutant with different mechanisms 1-gen-2010 Emmanuele, Crespan; Radi, Marco; Samantha, Zanoli; Silvia, Schenone; Maurizio, Botta; Giovanni, Maga
HIV-1 RT Inhibitors with a Novel Mechanism of Action: NNRTIs that Compete with the Nucleotide Substrate 1-gen-2010 Giovanni, Maga; Radi, Marco; Marie Aline, Gerard; Maurizio, Botta; Eric, Ennifar
Crystal Structure of HIV-1 Reverse Transcriptase Bound to a Non-Nucleoside Inhibitor with a Novel Mechanism of Action 1-gen-2010 Séverine, Freisz; Guillaume, Bec; Radi, Marco; Philippe, Wolff; Emmanuele, Crespan; Lucilla, Angeli; Philippe, Dumas; Giovanni, Maga; Maurizio, Botta; Eric, Ennifar
Mostrati risultati da 21 a 40 di 97
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