IRIS
RIVARA, Mirko
 Distribuzione geografica
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Continente #
NA - Nord America 1.472
EU - Europa 1.466
AS - Asia 712
SA - Sud America 60
AF - Africa 27
Continente sconosciuto - Info sul continente non disponibili 1
OC - Oceania 1
Totale 3.739
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Nazione #
US - Stati Uniti d'America 1.438
CN - Cina 416
FI - Finlandia 273
IT - Italia 266
SE - Svezia 240
SG - Singapore 238
IE - Irlanda 230
UA - Ucraina 136
DE - Germania 122
NL - Olanda 65
BR - Brasile 51
GB - Regno Unito 44
RU - Federazione Russa 34
TR - Turchia 34
CA - Canada 32
CI - Costa d'Avorio 25
CZ - Repubblica Ceca 15
BE - Belgio 14
FR - Francia 8
IN - India 6
PT - Portogallo 6
AT - Austria 5
LT - Lituania 4
CL - Cile 3
EC - Ecuador 3
HK - Hong Kong 3
IQ - Iraq 3
AR - Argentina 2
AZ - Azerbaigian 2
ID - Indonesia 2
AL - Albania 1
AM - Armenia 1
AU - Australia 1
BD - Bangladesh 1
BH - Bahrain 1
CY - Cipro 1
EG - Egitto 1
EU - Europa 1
JO - Giordania 1
LI - Liechtenstein 1
MA - Marocco 1
NI - Nicaragua 1
NP - Nepal 1
PA - Panama 1
PH - Filippine 1
PS - Palestinian Territory 1
RO - Romania 1
RS - Serbia 1
VE - Venezuela 1
Totale 3.739
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Città #
Dublin 230
Chandler 226
Jacksonville 154
Singapore 147
Santa Clara 133
Ashburn 114
Beijing 99
Ann Arbor 97
Parma 77
Boardman 70
Dearborn 67
Nanjing 62
Shanghai 49
Princeton 45
Milan 42
Helsinki 34
New York 32
Wilmington 32
Izmir 31
San Mateo 29
Chicago 27
Abidjan 25
Toronto 23
Moscow 22
Shenyang 18
Nanchang 17
Guangzhou 16
Kunming 16
Munich 16
Hefei 15
Jinan 15
Los Angeles 15
Bremen 14
Brussels 14
Des Moines 14
Hebei 14
Seattle 14
Council Bluffs 12
Jiaxing 11
London 11
Brno 10
Woodbridge 10
Nuremberg 8
Changsha 7
Frankfurt am Main 7
Ottawa 6
Piacenza 6
Reggio Emilia 6
Tianjin 6
Auburn Hills 5
Bologna 5
Chengdu 5
Dallas 5
Falls Church 5
Modena 5
Norwalk 5
The Dalles 5
Vienna 5
Abbiategrasso 4
Brescia 4
Düsseldorf 4
Roncadelle 4
Belo Horizonte 3
Buccinasco 3
Castelo Branco 3
Falkenstein 3
Fremont 3
Grafing 3
Gualtieri 3
Haikou 3
Hangzhou 3
Ningbo 3
Novi di Modena 3
Pavia 3
Reggio Nell'emilia 3
St Andrews 3
Taiyuan 3
Taizhou 3
Trezzano Sul Naviglio 3
Vobarno 3
Wuhan 3
Zhengzhou 3
Amsterdam 2
Baku 2
Baotou 2
Castelcovati 2
Cereda 2
Cesena 2
Chongqing 2
Contagem 2
Florence 2
Fuzhou 2
Grezzago 2
Hertford 2
Istanbul 2
Jakarta 2
Lanzhou 2
Miami 2
Montepulciano 2
Mãe do Rio 2
Totale 2.322
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Nome #
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays 111
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line 109
QSAR study of 2-aminobenzimidazole derivatives as H3 antagonists 108
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists 106
3D proteome-wide scale screening and activity evaluation of a new ALKBH5 inhibitor in U87 glioblastoma cell line 105
Cognition enhancing effect in rats of a selected histamine H3 receptor antagonist with good brain penetration 101
Gene-Delivery Ability of New Hydrogenated and Partially Fluorinated Gemini bispyridinium Surfactants with Six Methylene Spacers 97
Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design 91
COMPOSITIONS AND METHODS FOR BLOCKING SODIUM CHANNELS 91
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine 90
Drug repurposing approaches to fight Dengue virus infection and related diseases 90
Antioxidant and cytoprotective activity of indole derivatives related to melatonin 90
Development of a GPCR model for SAR interpretation of classical and new H3 antagonists 90
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. 89
Novel Sodium Channel Antagonists in the Treatment of Neuropathic Pain 89
COMPOSITIONS AND METHODS FOR BLOCKING SODIUM CHANNELS 89
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity. 86
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists 86
Chiral NMR discrimination of the diastereoisomeric salts of the H(3)-antagonist 2-[3-(1H-imidazol-4-ylmethyl)piperidin-1-yl]-1H-benzimidazole. 85
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. 84
2,4(5)-Diarylimidazoles: Synthesis and Biological Evaluation of a New Class of Sodium Channel Blockers against hNav1.2 80
Advances in Design and Development of Sodium Channel Blockers. 80
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. 80
Chemico-Physical Properties of Some 1,1′-Bis-alkyl-2,2′-hexane-1,6-diyl-bispyridinium Chlorides Hydrogenated and Partially Fluorinated for Gene Delivery 76
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series 75
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors 75
Inhibition of NaV1.6 sodium channel currents by a novel series of 1,4-disubstituted-triazole derivatives obtained via copper-catalyzed click chemistry 75
Anticonvulsant Activity of 2,4(5)-Diarylimidazoles in Mice and Rat Models 74
NMR Analysis of a Series of Imidazobenzoxazines 73
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity 73
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships 72
COMPOSITIONS AND METHODS FOR BLOCKING SODIUM CHANNELS 72
Anticonvulsant Activity of 2,4(1H)-Diarylimidazoles in Mice and Rats Acute Seizure Models 70
Biological evaluation of imidazobenzoxazines, imidazobenzoxazin-5-ones and imidazobenzoxazin-5-thiones as sodium channel blockers 69
Sodium Channel Blocking Activity and In-vivo Testing of New Phenyl-imidazole Derivatives. 68
A Practical Synthesis of 2,4(5)-Diarylimidazoles from Simple Building Blocks 63
Sodium channel blockers: a patent review (2010 - 2014) 63
Recent Advances in the Medicinal Chemistry of Sodium Channel Blockers and their Therapeutic Potential 61
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. 61
Sodium Channel Blockers as Therapeutic Target for Treating Epilepsy: Recent Updates 60
NEW ALKBH2 AND ALKBH5 INHIBITORS FOR TREATING GLIOBLASTOMA 59
In vivo Screening of Diarylimidazoles as Anticonvulsant Agents 58
MV1035 Overcomes Temozolomide Resistance in Patient-Derived Glioblastoma Stem Cell Lines 58
Sodium channel blockers for neuropathic pain. 56
Microwave Assisted Efficient Synthesis of Imidazole-based Privileged Structure 53
NaV1.1 and NaV1.6 selective compounds reduce the behavior phenotype and epileptiform activity in a novel zebrafish model for Dravet syndrome 52
Potential in-vitro antiviral activity of MV1035 on SARS-CoV-2 wild type viruses 49
New ALKBH2 and ALKBH5 inhibitors for treating glioblastoma 47
Subtype-selective small molecule inhibitors reveal a fundamental role for Nav1.7 in nociceptor electrogenesis, axonal conduction and presynaptic release 37
IMIDAZOBENZOXAZIN-5-THIONE (MV1035) TO OVERCOME THE BLOOD-BRAIN BARRIER AND TARGET CNS DISEASES 31
Totale 3.807
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Categoria #
all - tutte 16.583
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 16.583
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/202054 0 0 0 0 0 0 0 0 0 0 11 43
2020/2021304 11 39 24 16 31 9 47 10 55 16 42 4
2021/2022229 3 2 5 18 14 7 29 26 21 17 17 70
2022/2023929 106 108 68 57 71 118 17 44 275 12 36 17
2023/2024411 22 32 11 14 43 84 38 29 19 21 35 63
2024/2025881 64 78 99 90 72 137 41 77 101 114 8 0
Totale 3.807