IRIS
RIVARA, Mirko
 Distribuzione geografica
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Continente #
NA - Nord America 1.524
EU - Europa 1.507
AS - Asia 726
SA - Sud America 71
AF - Africa 28
Continente sconosciuto - Info sul continente non disponibili 1
OC - Oceania 1
Totale 3.858
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Nazione #
US - Stati Uniti d'America 1.486
CN - Cina 416
FI - Finlandia 291
IT - Italia 271
SE - Svezia 240
SG - Singapore 240
IE - Irlanda 230
UA - Ucraina 137
DE - Germania 128
NL - Olanda 66
BR - Brasile 60
GB - Regno Unito 50
CA - Canada 34
RU - Federazione Russa 34
TR - Turchia 34
CI - Costa d'Avorio 25
IN - India 17
CZ - Repubblica Ceca 16
BE - Belgio 14
FR - Francia 8
PT - Portogallo 6
AT - Austria 5
CL - Cile 5
LT - Lituania 4
EC - Ecuador 3
ES - Italia 3
HK - Hong Kong 3
IQ - Iraq 3
AR - Argentina 2
AZ - Azerbaigian 2
BD - Bangladesh 2
ID - Indonesia 2
MA - Marocco 2
MX - Messico 2
AL - Albania 1
AM - Armenia 1
AU - Australia 1
BH - Bahrain 1
CY - Cipro 1
EG - Egitto 1
EU - Europa 1
JO - Giordania 1
LI - Liechtenstein 1
NI - Nicaragua 1
NP - Nepal 1
PA - Panama 1
PH - Filippine 1
PS - Palestinian Territory 1
RO - Romania 1
RS - Serbia 1
VE - Venezuela 1
Totale 3.858
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Città #
Dublin 230
Chandler 226
Jacksonville 154
Singapore 149
Santa Clara 134
Ashburn 118
Beijing 99
Ann Arbor 97
Parma 79
Boardman 70
Dearborn 67
Nanjing 62
Shanghai 49
Princeton 45
Milan 42
Helsinki 34
New York 33
Wilmington 32
Izmir 31
San Mateo 29
Chicago 27
Abidjan 25
Toronto 23
Moscow 22
Munich 22
Los Angeles 18
Shenyang 18
Turku 18
Nanchang 17
Guangzhou 16
Kunming 16
Hefei 15
Jinan 15
London 15
Bremen 14
Brussels 14
Des Moines 14
Hebei 14
Seattle 14
The Dalles 13
Council Bluffs 12
Jiaxing 11
Brno 10
Woodbridge 10
Nuremberg 8
Bengaluru 7
Changsha 7
Frankfurt am Main 7
Dallas 6
Ottawa 6
Piacenza 6
Reggio Emilia 6
Tianjin 6
Auburn Hills 5
Bologna 5
Brooklyn 5
Chengdu 5
Falls Church 5
Modena 5
Norwalk 5
Vienna 5
Abbiategrasso 4
Brescia 4
Chennai 4
Düsseldorf 4
Roncadelle 4
Belo Horizonte 3
Buccinasco 3
Castelo Branco 3
Columbus 3
Falkenstein 3
Fremont 3
Grafing 3
Gualtieri 3
Haikou 3
Hangzhou 3
Ningbo 3
Novi di Modena 3
Pavia 3
Reggio Nell'emilia 3
St Andrews 3
Taiyuan 3
Taizhou 3
Trezzano Sul Naviglio 3
Vobarno 3
Wuhan 3
Zhengzhou 3
Amsterdam 2
Baku 2
Baotou 2
Brasília 2
Castelcovati 2
Cereda 2
Cesena 2
Charlotte 2
Chongqing 2
Contagem 2
Ferrara 2
Florence 2
Fuzhou 2
Totale 2.381
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Nome #
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays 112
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line 112
QSAR study of 2-aminobenzimidazole derivatives as H3 antagonists 110
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists 108
3D proteome-wide scale screening and activity evaluation of a new ALKBH5 inhibitor in U87 glioblastoma cell line 108
Cognition enhancing effect in rats of a selected histamine H3 receptor antagonist with good brain penetration 105
Gene-Delivery Ability of New Hydrogenated and Partially Fluorinated Gemini bispyridinium Surfactants with Six Methylene Spacers 98
Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design 95
Novel Sodium Channel Antagonists in the Treatment of Neuropathic Pain 94
COMPOSITIONS AND METHODS FOR BLOCKING SODIUM CHANNELS 93
Development of a GPCR model for SAR interpretation of classical and new H3 antagonists 93
Antioxidant and cytoprotective activity of indole derivatives related to melatonin 92
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine 91
Drug repurposing approaches to fight Dengue virus infection and related diseases 91
COMPOSITIONS AND METHODS FOR BLOCKING SODIUM CHANNELS 91
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. 90
Chiral NMR discrimination of the diastereoisomeric salts of the H(3)-antagonist 2-[3-(1H-imidazol-4-ylmethyl)piperidin-1-yl]-1H-benzimidazole. 88
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists 88
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity. 87
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. 86
Advances in Design and Development of Sodium Channel Blockers. 84
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. 84
Chemico-Physical Properties of Some 1,1′-Bis-alkyl-2,2′-hexane-1,6-diyl-bispyridinium Chlorides Hydrogenated and Partially Fluorinated for Gene Delivery 81
2,4(5)-Diarylimidazoles: Synthesis and Biological Evaluation of a New Class of Sodium Channel Blockers against hNav1.2 81
Anticonvulsant Activity of 2,4(5)-Diarylimidazoles in Mice and Rat Models 78
Inhibition of NaV1.6 sodium channel currents by a novel series of 1,4-disubstituted-triazole derivatives obtained via copper-catalyzed click chemistry 78
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series 77
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors 77
NMR Analysis of a Series of Imidazobenzoxazines 74
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity 74
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships 73
Anticonvulsant Activity of 2,4(1H)-Diarylimidazoles in Mice and Rats Acute Seizure Models 73
COMPOSITIONS AND METHODS FOR BLOCKING SODIUM CHANNELS 73
Biological evaluation of imidazobenzoxazines, imidazobenzoxazin-5-ones and imidazobenzoxazin-5-thiones as sodium channel blockers 72
Sodium Channel Blocking Activity and In-vivo Testing of New Phenyl-imidazole Derivatives. 70
NEW ALKBH2 AND ALKBH5 INHIBITORS FOR TREATING GLIOBLASTOMA 68
A Practical Synthesis of 2,4(5)-Diarylimidazoles from Simple Building Blocks 65
Sodium channel blockers: a patent review (2010 - 2014) 64
Recent Advances in the Medicinal Chemistry of Sodium Channel Blockers and their Therapeutic Potential 63
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. 62
Sodium Channel Blockers as Therapeutic Target for Treating Epilepsy: Recent Updates 62
MV1035 Overcomes Temozolomide Resistance in Patient-Derived Glioblastoma Stem Cell Lines 60
In vivo Screening of Diarylimidazoles as Anticonvulsant Agents 59
Sodium channel blockers for neuropathic pain. 57
Microwave Assisted Efficient Synthesis of Imidazole-based Privileged Structure 54
New ALKBH2 and ALKBH5 inhibitors for treating glioblastoma 53
NaV1.1 and NaV1.6 selective compounds reduce the behavior phenotype and epileptiform activity in a novel zebrafish model for Dravet syndrome 53
Potential in-vitro antiviral activity of MV1035 on SARS-CoV-2 wild type viruses 51
Subtype-selective small molecule inhibitors reveal a fundamental role for Nav1.7 in nociceptor electrogenesis, axonal conduction and presynaptic release 39
IMIDAZOBENZOXAZIN-5-THIONE (MV1035) TO OVERCOME THE BLOOD-BRAIN BARRIER AND TARGET CNS DISEASES 35
Totale 3.926
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Categoria #
all - tutte 16.928
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 16.928
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/202054 0 0 0 0 0 0 0 0 0 0 11 43
2020/2021304 11 39 24 16 31 9 47 10 55 16 42 4
2021/2022229 3 2 5 18 14 7 29 26 21 17 17 70
2022/2023929 106 108 68 57 71 118 17 44 275 12 36 17
2023/2024411 22 32 11 14 43 84 38 29 19 21 35 63
2024/20251.000 64 78 99 90 72 137 41 77 101 114 127 0
Totale 3.926