IRIS
PIERONI, Marco
 Distribuzione geografica
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Continente #
NA - Nord America 1.290
EU - Europa 1.094
AS - Asia 492
AF - Africa 4
SA - Sud America 2
Totale 2.882
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Nazione #
US - Stati Uniti d'America 1.278
CN - Cina 345
IE - Irlanda 292
IT - Italia 254
SE - Svezia 222
FI - Finlandia 109
TR - Turchia 93
DE - Germania 73
AT - Austria 43
GB - Regno Unito 18
BE - Belgio 17
FR - Francia 17
IN - India 16
NL - Olanda 15
SG - Singapore 14
KR - Corea 11
CZ - Repubblica Ceca 9
CA - Canada 8
LU - Lussemburgo 6
ES - Italia 5
PK - Pakistan 4
PA - Panama 3
VN - Vietnam 3
CH - Svizzera 2
EG - Egitto 2
GH - Ghana 2
HK - Hong Kong 2
SI - Slovenia 2
BG - Bulgaria 1
BR - Brasile 1
CL - Cile 1
CY - Cipro 1
HR - Croazia 1
IR - Iran 1
JP - Giappone 1
LT - Lituania 1
ME - Montenegro 1
MX - Messico 1
NO - Norvegia 1
NP - Nepal 1
PL - Polonia 1
PT - Portogallo 1
RU - Federazione Russa 1
SK - Slovacchia (Repubblica Slovacca) 1
UA - Ucraina 1
Totale 2.882
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Città #
Chandler 339
Dublin 290
Ann Arbor 146
Ashburn 91
Parma 79
Dearborn 72
Izmir 72
Nanjing 61
Princeton 57
Beijing 56
Wilmington 43
Helsinki 42
Shanghai 42
Bremen 40
Vienna 35
Kocaeli 21
New York 19
San Mateo 18
Hefei 17
Nanchang 17
Falls Church 16
Hebei 16
Shenyang 16
Brussels 14
Changsha 14
Guangzhou 14
Jinan 13
Milan 13
Seattle 13
Jiaxing 12
Norwalk 12
Los Angeles 11
Houston 9
Boardman 8
Bologna 8
Des Moines 8
Fremont 8
Sassari 6
Woodbridge 6
Birmingham 5
Fairfield 5
Luxembourg 5
Modena 5
New Brunswick 5
Ningbo 5
Chongqing 4
Dordrecht 4
Haikou 4
Kunming 4
London 4
Pune 4
San Giuliano Milanese 4
Washington 4
Zhengzhou 4
Ahmedabad 3
Amstelveen 3
Edinburgh 3
Florence 3
Gonzaga 3
Grafing 3
Lucca 3
Ottawa 3
Panama City 3
Rockville 3
Rome 3
Sissa 3
Ancona 2
Angers 2
Antwerpen 2
Basel 2
Brno 2
Cairo 2
Carpi 2
Chengdu 2
Chiniot 2
Daejeon 2
Dong Ket 2
Evanston 2
Figline Valdarno 2
Formigine 2
Gwanak-gu 2
Hangzhou 2
Hong Kong 2
Lanzhou 2
Lattes 2
Ljubljana 2
Maddaloni 2
Madrid 2
Mira Loma 2
Montechiarugolo 2
Mumbai 2
Prato 2
Riverside 2
Segrate 2
Soriano nel Cimino 2
Taiyuan 2
Taizhou 2
Tianjin 2
Trecasali 2
Trezzano Sul Naviglio 2
Totale 1.944
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Nome #
Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants 136
Nuovi composti antimicrobici 131
Investigational Studies on a Hit Compound Cyclopropane-Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin Adjuvant 96
Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets 84
Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases 83
Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms 81
Rational Design, Synthesis and Preliminary Structure-Activity Relationships of α-Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella Typhimurium O-Acetylserine Sulfhydrylase 77
Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design 76
Inhibitors of the sulfur assimilation pathway in bacterial pathogens as enhancers of antibiotic therapy 70
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor 69
Antituberculosis agents: Beyond medicinal chemistry rules 68
Aspergillus fumigatus tryptophan metabolic route differently affects host immunity 66
Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections 65
A competitive o‐acetylserine sulfhydrylase inhibitor modulates the formation of cysteine synthase complex 64
Cyclopropane derivatives as potential human serine racemase inhibitors: unveiling novel insights into a difficult target 64
Blocking cysteine biosynthesis in Salmonella typhimurium: the moonlighting enzyme CysK as a potential antibiotic target 62
Modulation of bacterial metabolism by the microenvironment controls MAIT cell stimulation 62
Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR 56
Design, Synthesis and Investigation onthe Structure–Activity Relationships of N-Substituted 2-Aminothiazole Derivatives as Antitubercular Agents 55
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents 55
Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases 54
Substituted N-Phenyl-5-(2-(phenylamino)thiazol-4-yl)isoxazole-3-carboxamides Are Valuable Antitubercular Candidates that Evade Innate Efflux Machinery 52
Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting Mycobacterium tuberculosis energetics 51
Sodium Hyaluronate Microparticles for Pulmonary Delivery of Anti-mycobacterial Drugs 49
Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A 49
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design 49
Exploring the chemical space around N-(5-nitrothiazol-2-yl)-1,2,3-thiadiazole-4-carboxamide, a hit compound with serine acetyltransferase (SAT) inhibitory properties 48
In vitro digestion of zingiber officinale extract and evaluation of stability as a first step to determine its bioaccesibility 48
Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: Implications for Primary Hyperoxaluria type 1 48
Crystal structure of Aspergillus fumigatus AroH, an aromatic amino acid aminotransferase 47
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin 43
Preliminary structure - Activity relationships and biological evaluation of novel antitubercular indolecarboxamide derivatives against drug-susceptible and drug-resistant Mycobacterium tuberculosis strains 42
Derivatives of 3-isoxazolecarboxylic acid esters - a potent and selective compound class against replicating and nonreplicating Mycobacterium tuberculosis 41
Challenging the drug-likeness dogma for new drug discovery in Tuberculosis 41
Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria 40
Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches 40
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis 40
Biochemical characterization of Aspergillus fumigatus AroH, a putative aromatic amino acid aminotransferase 39
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry 39
Nitric oxide-releasing cyclodextrins as biodegradable antibacterial scaffolds: a patent evaluation of US2019343869(A1) 38
Synthesis of 7-desmethyl analogs of (+)- and (-)-huperzine A 37
Modulation of bacterial metabolism by the microenvironment controls MAIT cell stimulation article 37
From 6-aminoquinolone antibacterials to 6-amino-7- thiopyranopyridinylquinolone ethyl esters as inhibitors of staphylococcus aureus multidrug efflux pumps 35
Towards the sustainable discovery and development of new antibiotics 35
Rational Design and Synthesis of Thioridazine Analogues as Enhancers of the Antituberculosis Therapy 35
Identification of Human Alanine-Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1 34
Structural analogs of huperzine A improve survival in guinea pigs exposed to soman 33
An Experimental Model for the Rapid Screening of Compounds with Potential Use Against Mycobacteria 32
Indoleamides are active against drug-resistant mycobacterium tuberculosis 27
NOC chemistry for tuberculosis - Further investigations on the structure-activity relationships of antitubercular isoxazole-3-carboxylic acid ester derivatives 27
Synthesis and Structure-Activity Relationships of Lansine Analogues as Antileishmanial Agents 26
Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains 26
Pyrido[1,2-a]benzimidazole-Based Agents Active Against Tuberculosis (TB), Multidrug-Resistant (MDR) TB and Extensively Drug-Resistant (XDR) TB 24
Spectinamides: A challenge, a proof, and a suggestion 24
Searching for innovative quinolone-like scaffolds: Synthesis and biological evaluation of 2,1-benzothiazine 2,2-dioxide derivatives 23
From serendipity to rational antituberculosis drug discovery of mefloquine-isoxazole carboxylic acid esters 23
Mutation of Rv2887, a marR-Like gene, confers mycobacterium tuberculosis resistance to an imidazopyridine-based agent 22
Novel N-benzoyl-2-hydroxybenzamide disrupts unique parasite secretory pathway 22
Synthesis, biological evaluation, and structure-activity relationships of N -benzoyl-2-hydroxybenzamides as agents active against P. falciparum (K1 strain), trypanosomes, and leishmania 20
Rational design of 5-phenyl-3-isoxazolecarboxylic acid ethyl esters as growth inhibitors of Mycobacterium tuberculosis. A potent and selective series for further drug development 19
Synthesis, biological evaluation, and structure-activity relationships for 5-[(E)-2-arylethenyl]-3-isoxazolecarboxylic acid alkyl ester derivatives as valuable antitubercular chemotypes 18
Expanding the knowledge around antitubercular 5-(2-aminothiazol-4-yl)isoxazole-3-carboxamides: Hit–to–lead optimization and release of a novel antitubercular chemotype via scaffold derivatization 17
In pursuit of natural product leads: Synthesis and biological evaluation of 2-[3-hydroxy-2-[(3-hydroxypyridine-2-carbonyl)amino]phenyl]benzoxazole-4- carboxylic acid (A-33853) and its analogues: Discovery of N-(2-benzoxazol-2- ylphenyl)benzamides as novel antileishmanial chemotypes 17
Totale 3.031
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Categoria #
all - tutte 12.640
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 12.640
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/201990 0 0 0 0 0 0 0 0 0 0 85 5
2019/2020436 99 56 3 7 42 74 47 8 27 49 17 7
2020/2021201 3 5 8 10 6 12 8 24 46 41 17 21
2021/2022379 15 28 25 25 10 38 20 26 35 22 21 114
2022/20231.261 118 138 79 100 146 149 7 65 374 15 41 29
2023/2024379 24 40 17 28 49 72 48 44 26 28 3 0
Totale 3.031