Advances in the set-up of a fluorescence- anisotropy assay for the search of novel inhibitors of the tead-4 complexes
2019-01-01 Romito, Filippo; Tagliazucchi, Lorenzo; Pozzi, Cecilia; Mangani, Stefano; Lopresti, Ludovica; Ponterini, Glauco; Paola Costi, Maria
Development of a sensitive biochemical tool to assess the expression levels of recombinant ectopic proteins in in vitro engineered cellular systems
2022-01-01 Moschella, Mg; Marverti, G; Cassanelli, Valentina; Venuti, Federica; Tagliazucchi, L; Costi, Mp; D’Arca., D
MS Proteomics And Biochemical Characterization Of Thymidylate Synthase Dimer Destabilizer E7 To Halt Colorectal Carcinoma
2024-01-01 Tagliazucchi, Lorenzo; Di Persio, Sara; Gaetana Moschella, Maria; Malpezzi, Giulia; Aiello, Daniele; Saporito, Giulia; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro; Marverti, Gaetano; Venturelli, Alberto; D’Arca, Domenico; Paola Costi, Maria
One Health Approach in Drug Discovery for Leishmaniasis by Targeting Calpain cys-protease
2024-01-01 Aiello, Daniele; Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mazzorana, Marco; Pozzi, Cecilia; Brancale, Andrea; Costi Maria, Paola
Investigating the mechanism of action of the antiparasitic agent H80 through imaging techniques
2023-01-01 Malpezzi, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Venturelli, Alberto; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Ponterini, Glauco; Paola Costi, Maria
Integrating MS proteomics in the Medicinal Chemistry pipeline as powerful tool to overcome drug resistance issues in colorectal cancer
2024-01-01 Tagliazucchi, Lorenzo; Piazzi, Manuela; D'Arca, Domenico; Marverti, Gaetano; Moschella Maria, Gaetana; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro; Costi, M Paola
Lead-optimization process and characterization of the dissociative effect applied to new dimer disrupters of human Thymidylate Synthase
2022-01-01 Aiello, Daniele; Ascione, Cristian; Tagliazucchi, Lorenzo; Malpezzi, Giulia; Cassanelli, Valentina; Ponterini, Glauco; D’Arca, Domenico; Marverti, Gaetano; Gaetana Moschella, Maria; Falchi, Federico; Venturelli, Alberto; Paola Costi, Maria
Development of a novel class of YAP:TEAD interface-3 molecular disruptors to treat colorectal carcinoma
2023-01-01 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Aiello, Daniele; Zappaterra, Dana; Elisi, Gian Marco; Venturelli, Alberto; Gaetana Moschella, Maria; D’Arca, Domenico; Marverti, Gaetano; Lopresti, Ludovica; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Ponterini, Glauco; Paola Costi, Maria
Coupling a microwave-assisted process with HPLC-ELSD for the extraction, purification and analysis of bioactive policosanols from beeswax
2021-01-01 Venturelli, Alberto; Brighenti, Virginia; Tagliazucchi, Lorenzo; Paola Costi, Maria; Pellati, Federica
Precision medicine through proteomics studies in drug resistant colorectal cancer
2024-01-01 Paola Costi, Maria; Piazzi, Manuela; Tagliazucchi, Lorenzo; Marverti, Gaetano; D’Arca, Domenico; Gaetana Moschella, Maria; Losi, Lorena; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro
LC-MS serum proteomics reveals a panel of proteins prognostic of positive responsiveness to bevacizumab therapy in late-stages ovarian cancer patients
2022-01-01 Tagliazucchi, Lorenzo; Gaetana Moschella, Maria; D'Addese, Gianluca; Califano, Daniela; Arenare, Laura; Mezzanzanico, Delia; Chinello, Clizia; Magni, Fulvio; Villani, Marco; Losi, Lorena; Marverti, Gaetano; D’Arca, Domenico; Chiodini, Paolo; Pignata, Sandro; Paola Costi, Maria
Applying optical tweezers technology to reveal Thymidylate Synthase interactions with its consensus mRNA
2023-01-01 Malpezzi, Giulia; Viader, Xvaier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Gaetana Moschella, Maria; Paola Costi, Maria; D’Arca, Domenico; Cecconi, Ciro
LC-MS/MS Helps Characterizing THP-1 Cells Proteome After Infection with Drug Resistant Leishmania Strains
2022-01-01 Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; García-Hernández, Raquel; Genovese, Filippo; Pinetti, Diego; Gamarro, Francisco; Paola Costi, Maria
Promoting A Sustainable Medicinal Chemistry Approach With The Cost Action CA21111 - One Health Drugs Against Parasitic Vector Borne Diseases In Europe And Beyond
2024-01-01 Aiello, Daniele; Cordeiro-da-Silva, Anabela; Tagliazucchi, Lorenzo; Saporito, Giulia; Malpezzi, Giulia; Action Ca2111 Members, Cost; Paola Costi, Maria
Development of guanidino-containing benzimidazoles as novel folate enzymes inhibitors for the treatment of Human African Trypanosomiasis
2021-01-01 Rizzo, Marco; Francesconi, Valeria; Cichero, Elena; Schenone, Silvia; Tagliazucchi, Lorenzo; Cordeiro Da Silva, Anabela; Paola Costi, Maria; Tonelli, Michele
Lead optimization of human thymidylate synthase dimer disrupters: from computational studies to evaluation of their biological profiles
2023-01-01 Daniele, Aiello; Giulia, Malpezzi; Tagliazucchi, Lorenzo; Maria Gaetana, Moschella; Saporito, Giulia; Venturelli, Alberto; Ponterini, Gluaco; D’Arca, Domenico; Marverti, Gaetano; Falchi, Federico; Paola Costi, Maria
Targeting of the Cysteines Surface domain of the Transcriptional Enhancer Associate Domain (TEAD) for anticancer drug discovery
2021-01-01 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mangani, Stefano; Lopresti, Ludovica; Pozzi, Cecilia; Ponterini, Glauco; Venturelli, Alberto; Paola Costi, Maria
Structural insight into YAP-TEAD4 protein-protein interactions as target for cancer treatment
2021-01-01 Lopresti, Ludovica; Pozzi, Cecilia; Tagliazucchi, L; D’Arca, D; Marverti, G; Costi, Mp; Mangani, Stefano
Expression, purification, and characterization of Transcriptional Enhancer Associated Domain (hTEAD4), a promising target for anticancer agents
2022-01-01 Tagliazucchi, L; Rossi, Marianna; Pozzi, Cecilia; Lopresti, Ludovica; Aiello, D; Venturelli, A; Ponterini, G; Costi, Mp
Optimization of chemical-biological tools for characterizing the activity of dissociative inhibitor of human thymidylate synthase
2024-01-01 Saporito, Giulia; Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Venturelli, Alberto; Falchi, Federico; Ponterini, Glauco; Costi, Maria Paola
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Advances in the set-up of a fluorescence- anisotropy assay for the search of novel inhibitors of the tead-4 complexes | 1-gen-2019 | Romito, Filippo; Tagliazucchi, Lorenzo; Pozzi, Cecilia; Mangani, Stefano; Lopresti, Ludovica; Ponterini, Glauco; Paola Costi, Maria | |
| Development of a sensitive biochemical tool to assess the expression levels of recombinant ectopic proteins in in vitro engineered cellular systems | 1-gen-2022 | Moschella, Mg; Marverti, G; Cassanelli, Valentina; Venuti, Federica; Tagliazucchi, L; Costi, Mp; D’Arca., D | |
| MS Proteomics And Biochemical Characterization Of Thymidylate Synthase Dimer Destabilizer E7 To Halt Colorectal Carcinoma | 1-gen-2024 | Tagliazucchi, Lorenzo; Di Persio, Sara; Gaetana Moschella, Maria; Malpezzi, Giulia; Aiello, Daniele; Saporito, Giulia; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro; Marverti, Gaetano; Venturelli, Alberto; D’Arca, Domenico; Paola Costi, Maria | |
| One Health Approach in Drug Discovery for Leishmaniasis by Targeting Calpain cys-protease | 1-gen-2024 | Aiello, Daniele; Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mazzorana, Marco; Pozzi, Cecilia; Brancale, Andrea; Costi Maria, Paola | |
| Investigating the mechanism of action of the antiparasitic agent H80 through imaging techniques | 1-gen-2023 | Malpezzi, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Venturelli, Alberto; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Ponterini, Glauco; Paola Costi, Maria | |
| Integrating MS proteomics in the Medicinal Chemistry pipeline as powerful tool to overcome drug resistance issues in colorectal cancer | 1-gen-2024 | Tagliazucchi, Lorenzo; Piazzi, Manuela; D'Arca, Domenico; Marverti, Gaetano; Moschella Maria, Gaetana; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro; Costi, M Paola | |
| Lead-optimization process and characterization of the dissociative effect applied to new dimer disrupters of human Thymidylate Synthase | 1-gen-2022 | Aiello, Daniele; Ascione, Cristian; Tagliazucchi, Lorenzo; Malpezzi, Giulia; Cassanelli, Valentina; Ponterini, Glauco; D’Arca, Domenico; Marverti, Gaetano; Gaetana Moschella, Maria; Falchi, Federico; Venturelli, Alberto; Paola Costi, Maria | |
| Development of a novel class of YAP:TEAD interface-3 molecular disruptors to treat colorectal carcinoma | 1-gen-2023 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Aiello, Daniele; Zappaterra, Dana; Elisi, Gian Marco; Venturelli, Alberto; Gaetana Moschella, Maria; D’Arca, Domenico; Marverti, Gaetano; Lopresti, Ludovica; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Ponterini, Glauco; Paola Costi, Maria | |
| Coupling a microwave-assisted process with HPLC-ELSD for the extraction, purification and analysis of bioactive policosanols from beeswax | 1-gen-2021 | Venturelli, Alberto; Brighenti, Virginia; Tagliazucchi, Lorenzo; Paola Costi, Maria; Pellati, Federica | |
| Precision medicine through proteomics studies in drug resistant colorectal cancer | 1-gen-2024 | Paola Costi, Maria; Piazzi, Manuela; Tagliazucchi, Lorenzo; Marverti, Gaetano; D’Arca, Domenico; Gaetana Moschella, Maria; Losi, Lorena; Bedeschi, Martina; Tesei, Anna; Passardi, Alessandro | |
| LC-MS serum proteomics reveals a panel of proteins prognostic of positive responsiveness to bevacizumab therapy in late-stages ovarian cancer patients | 1-gen-2022 | Tagliazucchi, Lorenzo; Gaetana Moschella, Maria; D'Addese, Gianluca; Califano, Daniela; Arenare, Laura; Mezzanzanico, Delia; Chinello, Clizia; Magni, Fulvio; Villani, Marco; Losi, Lorena; Marverti, Gaetano; D’Arca, Domenico; Chiodini, Paolo; Pignata, Sandro; Paola Costi, Maria | |
| Applying optical tweezers technology to reveal Thymidylate Synthase interactions with its consensus mRNA | 1-gen-2023 | Malpezzi, Giulia; Viader, Xvaier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Gaetana Moschella, Maria; Paola Costi, Maria; D’Arca, Domenico; Cecconi, Ciro | |
| LC-MS/MS Helps Characterizing THP-1 Cells Proteome After Infection with Drug Resistant Leishmania Strains | 1-gen-2022 | Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; García-Hernández, Raquel; Genovese, Filippo; Pinetti, Diego; Gamarro, Francisco; Paola Costi, Maria | |
| Promoting A Sustainable Medicinal Chemistry Approach With The Cost Action CA21111 - One Health Drugs Against Parasitic Vector Borne Diseases In Europe And Beyond | 1-gen-2024 | Aiello, Daniele; Cordeiro-da-Silva, Anabela; Tagliazucchi, Lorenzo; Saporito, Giulia; Malpezzi, Giulia; Action Ca2111 Members, Cost; Paola Costi, Maria | |
| Development of guanidino-containing benzimidazoles as novel folate enzymes inhibitors for the treatment of Human African Trypanosomiasis | 1-gen-2021 | Rizzo, Marco; Francesconi, Valeria; Cichero, Elena; Schenone, Silvia; Tagliazucchi, Lorenzo; Cordeiro Da Silva, Anabela; Paola Costi, Maria; Tonelli, Michele | |
| Lead optimization of human thymidylate synthase dimer disrupters: from computational studies to evaluation of their biological profiles | 1-gen-2023 | Daniele, Aiello; Giulia, Malpezzi; Tagliazucchi, Lorenzo; Maria Gaetana, Moschella; Saporito, Giulia; Venturelli, Alberto; Ponterini, Gluaco; D’Arca, Domenico; Marverti, Gaetano; Falchi, Federico; Paola Costi, Maria | |
| Targeting of the Cysteines Surface domain of the Transcriptional Enhancer Associate Domain (TEAD) for anticancer drug discovery | 1-gen-2021 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mangani, Stefano; Lopresti, Ludovica; Pozzi, Cecilia; Ponterini, Glauco; Venturelli, Alberto; Paola Costi, Maria | |
| Structural insight into YAP-TEAD4 protein-protein interactions as target for cancer treatment | 1-gen-2021 | Lopresti, Ludovica; Pozzi, Cecilia; Tagliazucchi, L; D’Arca, D; Marverti, G; Costi, Mp; Mangani, Stefano | |
| Expression, purification, and characterization of Transcriptional Enhancer Associated Domain (hTEAD4), a promising target for anticancer agents | 1-gen-2022 | Tagliazucchi, L; Rossi, Marianna; Pozzi, Cecilia; Lopresti, Ludovica; Aiello, D; Venturelli, A; Ponterini, G; Costi, Mp | |
| Optimization of chemical-biological tools for characterizing the activity of dissociative inhibitor of human thymidylate synthase | 1-gen-2024 | Saporito, Giulia; Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Venturelli, Alberto; Falchi, Federico; Ponterini, Glauco; Costi, Maria Paola |
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