Applying optical tweezers technology to reveal Thymidylate Synthase interactions with its consensus mRNA
2023-01-01 Malpezzi, Giulia; Viader, Xvaier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Gaetana Moschella, Maria; Paola Costi, Maria; D’Arca, Domenico; Cecconi, Ciro
LC-MS/MS Helps Characterizing THP-1 Cells Proteome After Infection with Drug Resistant Leishmania Strains
2022-01-01 Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; García-Hernández, Raquel; Genovese, Filippo; Pinetti, Diego; Gamarro, Francisco; Paola Costi, Maria
Promoting A Sustainable Medicinal Chemistry Approach With The Cost Action CA21111 - One Health Drugs Against Parasitic Vector Borne Diseases In Europe And Beyond
2024-01-01 Aiello, Daniele; Cordeiro-da-Silva, Anabela; Tagliazucchi, Lorenzo; Saporito, Giulia; Malpezzi, Giulia; Action Ca2111 Members, Cost; Paola Costi, Maria
Development of guanidino-containing benzimidazoles as novel folate enzymes inhibitors for the treatment of Human African Trypanosomiasis
2021-01-01 Rizzo, Marco; Francesconi, Valeria; Cichero, Elena; Schenone, Silvia; Tagliazucchi, Lorenzo; Cordeiro Da Silva, Anabela; Paola Costi, Maria; Tonelli, Michele
Lead optimization of human thymidylate synthase dimer disrupters: from computational studies to evaluation of their biological profiles
2023-01-01 Daniele, Aiello; Giulia, Malpezzi; Tagliazucchi, Lorenzo; Maria Gaetana, Moschella; Saporito, Giulia; Venturelli, Alberto; Ponterini, Gluaco; D’Arca, Domenico; Marverti, Gaetano; Falchi, Federico; Paola Costi, Maria
Targeting of the Cysteines Surface domain of the Transcriptional Enhancer Associate Domain (TEAD) for anticancer drug discovery
2021-01-01 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mangani, Stefano; Lopresti, Ludovica; Pozzi, Cecilia; Ponterini, Glauco; Venturelli, Alberto; Paola Costi, Maria
Structural insight into YAP-TEAD4 protein-protein interactions as target for cancer treatment
2021-01-01 Lopresti, Ludovica; Pozzi, Cecilia; Tagliazucchi, L; D’Arca, D; Marverti, G; Costi, Mp; Mangani, Stefano
Expression, purification, and characterization of Transcriptional Enhancer Associated Domain (hTEAD4), a promising target for anticancer agents
2022-01-01 Tagliazucchi, L; Rossi, Marianna; Pozzi, Cecilia; Lopresti, Ludovica; Aiello, D; Venturelli, A; Ponterini, G; Costi, Mp
Optimization of chemical-biological tools for characterizing the activity of dissociative inhibitor of human thymidylate synthase
2024-01-01 Saporito, Giulia; Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Venturelli, Alberto; Falchi, Federico; Ponterini, Glauco; Costi, Maria Paola
Development of a fluorescent anisotropy displacement assay for the optimization of YAP:TEAD molecular disrupters with anticancer activity
2024-01-01 Malpezzi, Giulia; Elisi, Gianmarco; Scalvini, Laura; Tagliazucchi, Lorenzo; Aiello, Daniele; Guerrini, Remo; D’Arca, Domenico; Marverti, Gaetano; Pozzi, Cecilia; Venturelli, Alberto; Ponterini, Glauco; Mor, Marco; Paola Costi, Maria
Leveraging proteomic, bioinformatic and ecotoxicology models to select new targets overcoming L. Infantum drug resistent
2024-01-01 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Brooks, Brain V.; Thorè, Eli S. J.; Bertram, Michael G.; Gammarro, Francisco; Paola Costi, Maria
Discovery of guanidino-containing benzimidazoles as novel antifolates for Trypanosomiasis
2022-01-01 Francesconi, Valeria; Rizzo, Marco; Tagliazucchi, Lorenzo; Pozzi, Cecilia; Cordeiro-da-Silva, Anabela; Venuti, Federica; Konchie, Claude; Paola Costi, Maria; Michele, Tonelli
LC-MS/MS proteomics for the rapid and selective screening of drug resistances in Leishmania infantum clinical isolates
2023-01-01 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Perea Martinez, Ana; Ignacio Manzano, José; Garcia-Hernandez, Raquel; Pinetti, Diego; Genovese, Filippo; Paola Costi, Maria
Exploiting the Optical Tweezer technology to reveal thymidylate synthase interactions with its consensus mRNA
2023-01-01 Malpezzi, Giulia; Viander, Xavier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, Maria; Paola Costi, Maria; D’Arca, Domenico; Cecconi, Ciro
Exploiting Forster Resonance Energy Transfer (FRET) in the characterization of YAP:TEAD complex disruption
2022-01-01 Tagliazucchi, Lorenzo; Rossi, Marianna; Malpezzi, Giulia; Zappaterra, Dana; Aiello, Daniele; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Venturelli, Alberto; Ponterini, Glauco; Paola Costi, Maria
Drug discovery of pyrazolo-piperidinone inhibitors targeting YAP:TEAD interaction and development of a fluorescence anisotropy assay for high-throughput screening
2025-01-01 Malpezzi, Giulia; Scalvini, Laura; Tagliazucchi, Lorenzo; Chiaravalle, Annalisa; Aiello, Daniele; Saporito, Giulia; Illuminati, Davide; Pacifico, Salvatore; Guerrini, Remo; Pozzi, Cecilia; Venturelli, Alberto; Ponterini, Glauco; Mor Sheraz Gul, Marco; Paola Costi, Maria
Preclinical investigation of H80 compared to miltefosine: imaging and proteomics for sustainable drug development
2024-01-01 Malpezzi, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Venturelli, Alberto; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Ponterini, Glauco; Paola Costi, Maria
Targeting the dimer-monomer equilibrium of thymidylate synthase, to accelerate protein degradation and cancer cell growth inhibition
2022-01-01 Costi Maria, Paola; Venturelli, A; Ponterini, G; Pozzi, C; Wade, Rebecca; Giovannetti, E; Rimessi, A; Tagliazucchi, L; Moschella, M; Marverti, G; D’Arca, D
A dual-Omics approach to identify the modulated proteins/genes in THP-1 cells infected with different drug resistant L. infantum clinical isolates
2023-01-01 Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; García-Hernández, Raquel; Genovese, Filippo; Pinetti, Diego; Gamarro, Francisco; Paola Costi, Maria
UHPLC-MS/MS screening of the hTEAD surface for the identification of novel allosteric inhibitors with anticancer activity
2021-01-01 Tagliazucchi, Lorenzo; Malpezzi, Giulia; Pozzi, Cecilia; Lopresti, Ludovica; Mangani, Stefano; Abdel Latif, Andrea; Ponterini, Glauco; Venturelli, Alberto; Paola Costi, Maria
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Applying optical tweezers technology to reveal Thymidylate Synthase interactions with its consensus mRNA | 1-gen-2023 | Malpezzi, Giulia; Viader, Xvaier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Gaetana Moschella, Maria; Paola Costi, Maria; D’Arca, Domenico; Cecconi, Ciro | |
| LC-MS/MS Helps Characterizing THP-1 Cells Proteome After Infection with Drug Resistant Leishmania Strains | 1-gen-2022 | Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; García-Hernández, Raquel; Genovese, Filippo; Pinetti, Diego; Gamarro, Francisco; Paola Costi, Maria | |
| Promoting A Sustainable Medicinal Chemistry Approach With The Cost Action CA21111 - One Health Drugs Against Parasitic Vector Borne Diseases In Europe And Beyond | 1-gen-2024 | Aiello, Daniele; Cordeiro-da-Silva, Anabela; Tagliazucchi, Lorenzo; Saporito, Giulia; Malpezzi, Giulia; Action Ca2111 Members, Cost; Paola Costi, Maria | |
| Development of guanidino-containing benzimidazoles as novel folate enzymes inhibitors for the treatment of Human African Trypanosomiasis | 1-gen-2021 | Rizzo, Marco; Francesconi, Valeria; Cichero, Elena; Schenone, Silvia; Tagliazucchi, Lorenzo; Cordeiro Da Silva, Anabela; Paola Costi, Maria; Tonelli, Michele | |
| Lead optimization of human thymidylate synthase dimer disrupters: from computational studies to evaluation of their biological profiles | 1-gen-2023 | Daniele, Aiello; Giulia, Malpezzi; Tagliazucchi, Lorenzo; Maria Gaetana, Moschella; Saporito, Giulia; Venturelli, Alberto; Ponterini, Gluaco; D’Arca, Domenico; Marverti, Gaetano; Falchi, Federico; Paola Costi, Maria | |
| Targeting of the Cysteines Surface domain of the Transcriptional Enhancer Associate Domain (TEAD) for anticancer drug discovery | 1-gen-2021 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Mangani, Stefano; Lopresti, Ludovica; Pozzi, Cecilia; Ponterini, Glauco; Venturelli, Alberto; Paola Costi, Maria | |
| Structural insight into YAP-TEAD4 protein-protein interactions as target for cancer treatment | 1-gen-2021 | Lopresti, Ludovica; Pozzi, Cecilia; Tagliazucchi, L; D’Arca, D; Marverti, G; Costi, Mp; Mangani, Stefano | |
| Expression, purification, and characterization of Transcriptional Enhancer Associated Domain (hTEAD4), a promising target for anticancer agents | 1-gen-2022 | Tagliazucchi, L; Rossi, Marianna; Pozzi, Cecilia; Lopresti, Ludovica; Aiello, D; Venturelli, A; Ponterini, G; Costi, Mp | |
| Optimization of chemical-biological tools for characterizing the activity of dissociative inhibitor of human thymidylate synthase | 1-gen-2024 | Saporito, Giulia; Aiello, Daniele; Malpezzi, Giulia; Tagliazucchi, Lorenzo; Venturelli, Alberto; Falchi, Federico; Ponterini, Glauco; Costi, Maria Paola | |
| Development of a fluorescent anisotropy displacement assay for the optimization of YAP:TEAD molecular disrupters with anticancer activity | 1-gen-2024 | Malpezzi, Giulia; Elisi, Gianmarco; Scalvini, Laura; Tagliazucchi, Lorenzo; Aiello, Daniele; Guerrini, Remo; D’Arca, Domenico; Marverti, Gaetano; Pozzi, Cecilia; Venturelli, Alberto; Ponterini, Glauco; Mor, Marco; Paola Costi, Maria | |
| Leveraging proteomic, bioinformatic and ecotoxicology models to select new targets overcoming L. Infantum drug resistent | 1-gen-2024 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Brooks, Brain V.; Thorè, Eli S. J.; Bertram, Michael G.; Gammarro, Francisco; Paola Costi, Maria | |
| Discovery of guanidino-containing benzimidazoles as novel antifolates for Trypanosomiasis | 1-gen-2022 | Francesconi, Valeria; Rizzo, Marco; Tagliazucchi, Lorenzo; Pozzi, Cecilia; Cordeiro-da-Silva, Anabela; Venuti, Federica; Konchie, Claude; Paola Costi, Maria; Michele, Tonelli | |
| LC-MS/MS proteomics for the rapid and selective screening of drug resistances in Leishmania infantum clinical isolates | 1-gen-2023 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Perea Martinez, Ana; Ignacio Manzano, José; Garcia-Hernandez, Raquel; Pinetti, Diego; Genovese, Filippo; Paola Costi, Maria | |
| Exploiting the Optical Tweezer technology to reveal thymidylate synthase interactions with its consensus mRNA | 1-gen-2023 | Malpezzi, Giulia; Viander, Xavier; Zaltron, Annamaria; Neri, Benedetta; Di Felice, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Moschella, Maria; Paola Costi, Maria; D’Arca, Domenico; Cecconi, Ciro | |
| Exploiting Forster Resonance Energy Transfer (FRET) in the characterization of YAP:TEAD complex disruption | 1-gen-2022 | Tagliazucchi, Lorenzo; Rossi, Marianna; Malpezzi, Giulia; Zappaterra, Dana; Aiello, Daniele; Pozzi, Cecilia; Pacifico, Salvatore; Guerrini, Remo; Venturelli, Alberto; Ponterini, Glauco; Paola Costi, Maria | |
| Drug discovery of pyrazolo-piperidinone inhibitors targeting YAP:TEAD interaction and development of a fluorescence anisotropy assay for high-throughput screening | 1-gen-2025 | Malpezzi, Giulia; Scalvini, Laura; Tagliazucchi, Lorenzo; Chiaravalle, Annalisa; Aiello, Daniele; Saporito, Giulia; Illuminati, Davide; Pacifico, Salvatore; Guerrini, Remo; Pozzi, Cecilia; Venturelli, Alberto; Ponterini, Glauco; Mor Sheraz Gul, Marco; Paola Costi, Maria | |
| Preclinical investigation of H80 compared to miltefosine: imaging and proteomics for sustainable drug development | 1-gen-2024 | Malpezzi, Giulia; Tagliazucchi, Lorenzo; Aiello, Daniele; Venturelli, Alberto; Cordeiro-da-Silva, Anabela; Santarem, Nuno; Ponterini, Glauco; Paola Costi, Maria | |
| Targeting the dimer-monomer equilibrium of thymidylate synthase, to accelerate protein degradation and cancer cell growth inhibition | 1-gen-2022 | Costi Maria, Paola; Venturelli, A; Ponterini, G; Pozzi, C; Wade, Rebecca; Giovannetti, E; Rimessi, A; Tagliazucchi, L; Moschella, M; Marverti, G; D’Arca, D | |
| A dual-Omics approach to identify the modulated proteins/genes in THP-1 cells infected with different drug resistant L. infantum clinical isolates | 1-gen-2023 | Tagliazucchi, Lorenzo; Perea-Martinez, Ana; Fiorini, Greta; Ignacio Manzano, José; García-Hernández, Raquel; Genovese, Filippo; Pinetti, Diego; Gamarro, Francisco; Paola Costi, Maria | |
| UHPLC-MS/MS screening of the hTEAD surface for the identification of novel allosteric inhibitors with anticancer activity | 1-gen-2021 | Tagliazucchi, Lorenzo; Malpezzi, Giulia; Pozzi, Cecilia; Lopresti, Ludovica; Mangani, Stefano; Abdel Latif, Andrea; Ponterini, Glauco; Venturelli, Alberto; Paola Costi, Maria |
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Scopri
Tipologia
- 4 Contributo in atti di convegno ...3357
Data di pubblicazione
- In corso di stampa1
- 2020 - 2026534
- 2010 - 20191567
- 2000 - 2009667
- 1990 - 1999394
- 1980 - 1989192
- 1977 - 19792
Editore
- -63
- Società Italiana di Igiene, Medic...23
- EGU20
- European Society of Clinical Micr...20
- Società Chimica Italiana19
- .18
- Società Geologica Italiana17
- Società Italiana di Microbiologia16
- IEEE15
- s.n15
Rivista
- GIORNALE ITALIANO DI PSICOPATOLOGIA28
- ACTA BIO-MEDICA DE L'ATENEO PARMENSE21
- GIORNALE ITALIANO DI ORTOPEDIA E ...14
- ITALIAN JOURNAL OF ANIMAL SCIENCE13
- SCIENZA E TECNICA LATTIERO-CASEARIA13
- BLOOD11
- JOURNAL OF CARDIAC FAILURE11
- SURGICAL ENDOSCOPY10
- HAEMATOLOGICA9
- EUROPEAN HEART JOURNAL8
Serie
- ANNUAL MEETING OF THE EUROPEAN AS...9
- BOOK OF ABSTRACTS OF THE ENTRENOV...1
- International Conference on Quali...1
- MAPPE PARASSITOLOGICHE1
- MATERIALS SCIENCE FORUM1
Keyword
- phosphate glasses12
- Raman Spectroscopy10
- dog7
- erbium5
- micro-Raman spectroscopy5
- Aspergillus flavus4
- immigrazione4
- media education4
- ab-initio vibrational calculations3
- BIOHYDROGEN3
Lingua
- eng1860
- ita596
- fre4
- ger3
- spa3
- afr1
- lit1
- nah1
- por1
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