BORDI, Fabrizio
 Distribuzione geografica
Continente #
NA - Nord America 2.018
EU - Europa 1.819
AS - Asia 965
AF - Africa 35
SA - Sud America 24
OC - Oceania 2
Continente sconosciuto - Info sul continente non disponibili 1
Totale 4.864
Nazione #
US - Stati Uniti d'America 1.981
CN - Cina 610
FI - Finlandia 543
SE - Svezia 361
IE - Irlanda 328
SG - Singapore 234
UA - Ucraina 208
DE - Germania 199
TR - Turchia 90
IT - Italia 89
CA - Canada 36
GB - Regno Unito 35
CI - Costa d'Avorio 33
BE - Belgio 29
BR - Brasile 16
IN - India 16
CZ - Repubblica Ceca 7
AT - Austria 4
IR - Iran 4
CL - Cile 3
EC - Ecuador 3
ES - Italia 3
FR - Francia 3
AU - Australia 2
EE - Estonia 2
KR - Corea 2
NL - Olanda 2
AE - Emirati Arabi Uniti 1
AM - Armenia 1
AZ - Azerbaigian 1
BY - Bielorussia 1
DZ - Algeria 1
EG - Egitto 1
EU - Europa 1
HR - Croazia 1
IL - Israele 1
JO - Giordania 1
LT - Lituania 1
MD - Moldavia 1
PA - Panama 1
RO - Romania 1
RU - Federazione Russa 1
SA - Arabia Saudita 1
TH - Thailandia 1
TJ - Tagikistan 1
UY - Uruguay 1
UZ - Uzbekistan 1
VE - Venezuela 1
Totale 4.864
Città #
Chandler 337
Dublin 328
Jacksonville 284
Santa Clara 176
Singapore 175
Ann Arbor 159
Dearborn 129
Beijing 118
Nanjing 103
Ashburn 92
Izmir 90
Boardman 82
Princeton 63
Shanghai 60
New York 58
San Mateo 56
Parma 43
Wilmington 37
Shenyang 35
Helsinki 34
Toronto 34
Abidjan 33
Bremen 32
Nanchang 32
Brussels 29
Hefei 29
Kunming 29
Hebei 27
Jinan 25
Los Angeles 23
Des Moines 22
Grafing 22
Tianjin 16
Changsha 12
Guangzhou 11
Munich 9
Woodbridge 9
Zhengzhou 8
Augusta 7
Jiaxing 7
Norwalk 7
Pune 7
Seattle 7
Taiyuan 7
Fuzhou 6
Haikou 6
Milan 6
Mordano 6
Dallas 5
Düsseldorf 5
Auburn Hills 4
Brno 4
Hangzhou 4
Ningbo 4
Chengdu 3
Fremont 3
Houston 3
Lanzhou 3
Leipzig 3
Madrid 3
Magdeburg 3
Prague 3
Reggio Nell'emilia 3
Taizhou 3
Vienna 3
Wuhan 3
Xian 3
Baotou 2
Belluno 2
Borås 2
Chongqing 2
Clifton 2
Collebeato 2
Frankfurt am Main 2
London 2
Marseille 2
Monmouth Junction 2
Quito 2
Sabz 2
São Paulo 2
Tallinn 2
Amman 1
Ardabil 1
Baku 1
Baoding 1
Bari 1
Bauru 1
Berlin 1
Birmingham 1
Boa Vista 1
Bragança Paulista 1
Brisbane 1
Cairo 1
Campinas 1
Campo Grande 1
Canberra 1
Changchun 1
Charlotte 1
Chisinau 1
Dubai 1
Totale 3.039
Nome #
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides. 146
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain. 117
Azionifarmacologiche di composti alchilaminoalchilfenilbenzisotiazolici sul trattogastrointestinale 111
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors 108
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays 100
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity 99
Synthesis and 3D-QSAR Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group 96
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion 96
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line 95
4-(1,2-benzisothiazol-3-)alkanoic and phenylalkanoic acids: synthesis and anti-inflammatory, analgesic and antipyretic activities 94
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists 93
A New Potent and Selective Histamine H3-Receptor Antagonist, 4(5)-{2-[4(5)-cyclohexylimidazol-2-ylthio]ethyl}imidazole 91
Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups 90
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano 88
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine 86
HPLC detection ofthioperamide from biological samples and its determination in rat blood and brainafter systemic administration 85
Plasma concentration and brain penetration of the H3-receptor antagonist Thioperamide in rats 84
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. 83
Action of histamine and ofdifferent synthetic P^ receptor stimulants on the isolated gastric fundus of theguinea pig 83
Effects of antimuscarinic agents, H2-blockers and omeprazole on rat chronic gastric ulcer after long-a and short-term administration 80
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity 80
Functional Studies of New Imidazole H3-Antagonists on Guinea-Pig Isolated Preparations 79
4-(3-Oxo-1,2-benzisothiazolin-2-yl)alkanoic, phenyl and phenoxyalkanoic acids: synthesis and anti-inflammatory, analgesic, and antipyretic properties 79
Dual mechanisms of action of the 5-benzylidene-hydantoin UPR1024 on lung cancer cell lines 79
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. 79
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists 78
A possible physiological role ofhistamine H^-receptors in rat mesenteric circulation 77
Hz-agonistiimidazolici: importanza della 2-amino sostituzione per 1'attivita farmacologica 77
Heteroarylaminoethyl and heteroarylthioethylimidazoles. Synthesis and H3-receptor affinity 76
H3-antagonists: synthesis and activity of 2-amino-5-thiazolyl derivatives 76
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. 76
Structural researcheson H^-agonists: the structures of the dipicrates of 2-(2-amino-4-imidazolyl)ethylamine, its 5-methyl derivative and N^f-dimeihyl-2-(2-am'mo-l,3-thiazol-5-yl)ethylamine 75
Irreversible EGFR inhibitor compounds with antiproliferative activity 74
Biological studies on 1,2-benzisothiazole derivatives. V. Antimicrobial properties of N-alkanoic, N-arylalkanoic and N-aryloxyalkanoic derivatives of 1,2-benzisothiazolin-3-one: QSAR study and genotoxicity evaluation 74
Sviluppo e caratterizzazione farmacologica di un nuovo potente e selettivo H3-bloccante istaminico non-tioureico 73
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors 73
Structure-Property Relationships on Histamine H3-Antagonists: Binding of Phenyl-substituted Alkylthioimidazole Derivatives to Rat Plasma Proteins 72
Ligands for the histamine H3-receptor: new potent antagonists of the 2-thioimidazole type 70
Pharmacological activities of two new histamine analogs 70
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series 70
Histamine H3-antagonists: the basicity of the polar group in quantitative structure-activity and structure-property relationship 70
In vitro characterization of potency, affinity and selectivity of H3-antagonists: from thioperamide to thioperamide unrelated derivatives 69
H3-receptor antagonists: Synthesis and structure relationships of para- and meta-substituted 4(5)-phenyl-2-((2-(4(5)-imidazolyl)ethyl)thio)imidazoles 68
Are histamine receptors involved in the stimulant activities of thiazolylethylamines supposed as cyclic models of dimaprit? 67
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma. 67
A possible physiological role of histamine H2-receptors in rat mesenteric circulation 65
Pharmacological profile of original potent H3 receptor antagonists 64
Auxin-like activity of 1,2-benzisothiazole derivatives 64
Action of histamine and of different synthetic H2 receptor stimulants on the isolated gastric fundus of the guinea pig 64
Influence of urea-equivalent groups in position 5 of 2-amino, 2-(1-aminoethylidenamino) and 2-guanidino thiazole derivatives on H3-receptor antagonist activity in gastric fistula cat 63
Studio di sostanze analoghe alDimaprit sulla secrezione gastrica "in vitro" 62
Pharmacological characterization of H3 receptor antagonists with imidazole, thioimidazole and thioimidazoline polar groups in the side chain 62
Pharmacological profile of new thioperamide derivatives at histamine peripheral H1-, H2, H3-receptors in guinea-pig 61
Rat protein binding and cerebral phospholipid affinity of the H3-receptor antagonist thioperamide 61
Antipyretic activity of new compounds "4-(3-OXO-1,2-BENZISOTHIAZOLIN-2-YL) PHENYLALKANOIC acids, their esters, amides and 1,1-dioxide derivatives 61
null 61
Synthesis and binding assays of H3-receptor ligands. 57
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. 57
QSAR study on H3-receptor affinity of benzothiazole derivatives of thioperamide 56
Melatonin Receptor Ligands: Synthesis of New Melatonin Derivatives and Comprehensive Comparative Molecular Field Analysis (CoMFA) Study. 49
Antipyreticactivity of new compounds 4-(3-oxo-l,2-benzisothiazolin-2-yl)puenyialkanoicacids, their esters, amides and 1,1 dioxide derivatives 44
null 37
Influence of urea-equivalent groups in position 5 of 2-amino, 2-(1-aminoethylidenamino) and 2-guanidino thiazole derivatives on H2-receptor antagonist activity in gastric fistula cat. 36
Pharmacological activities of two new histamine analogs 36
THIAZOLYLALKYLAMINES - SYNTHESIS OF ANALOGS OF IMIDAZOLYLETHYLAMINES AND THEIR INFLUENCE ON GASTRIC-SECRETION 35
Are histamine receptors involved in the stimulant activities ofthiazolylethylamines supposed as cyclic models of dimaprit? 18
Totale 4.886
Categoria #
all - tutte 18.183
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 18.183


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020414 0 0 0 0 0 0 117 18 122 44 48 65
2020/2021440 8 65 30 9 60 2 59 5 101 8 91 2
2021/2022344 7 3 3 30 17 33 45 49 19 24 21 93
2022/20231.308 156 143 89 86 121 162 18 74 411 10 30 8
2023/2024410 22 45 3 10 31 137 39 17 14 19 27 46
2024/2025599 51 78 89 93 105 183 0 0 0 0 0 0
Totale 4.886