IRIS
BORDI, Fabrizio
 Distribuzione geografica
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Continente #
EU - Europa 1.772
NA - Nord America 1.713
AS - Asia 688
SA - Sud America 3
OC - Oceania 2
AF - Africa 1
Continente sconosciuto - Info sul continente non disponibili 1
Totale 4.180
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Nazione #
US - Stati Uniti d'America 1.677
CN - Cina 566
FI - Finlandia 538
SE - Svezia 360
IE - Irlanda 328
UA - Ucraina 208
DE - Germania 182
TR - Turchia 90
IT - Italia 80
CA - Canada 35
GB - Regno Unito 33
BE - Belgio 27
IN - India 16
SG - Singapore 10
AT - Austria 4
IR - Iran 4
CL - Cile 3
ES - Italia 3
AU - Australia 2
CZ - Repubblica Ceca 2
KR - Corea 2
NL - Olanda 2
EE - Estonia 1
EG - Egitto 1
EU - Europa 1
FR - Francia 1
HR - Croazia 1
PA - Panama 1
RO - Romania 1
RU - Federazione Russa 1
Totale 4.180
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Città #
Chandler 337
Dublin 328
Jacksonville 284
Ann Arbor 159
Dearborn 129
Beijing 116
Nanjing 103
Ashburn 91
Izmir 90
Princeton 63
New York 58
San Mateo 56
Parma 43
Wilmington 37
Shanghai 36
Shenyang 35
Toronto 33
Bremen 32
Nanchang 32
Hefei 29
Helsinki 29
Kunming 29
Brussels 27
Hebei 27
Jinan 25
Des Moines 22
Grafing 22
Boardman 17
Tianjin 16
Changsha 12
Guangzhou 11
Woodbridge 9
Los Angeles 8
Zhengzhou 8
Augusta 7
Jiaxing 7
Norwalk 7
Pune 7
Seattle 7
Taiyuan 7
Fuzhou 6
Haikou 6
Mordano 6
Düsseldorf 5
Auburn Hills 4
Hangzhou 4
Ningbo 4
Chengdu 3
Dallas 3
Fremont 3
Houston 3
Lanzhou 3
Madrid 3
Reggio Nell'emilia 3
Taizhou 3
Vienna 3
Xian 3
Baotou 2
Belluno 2
Borås 2
Chongqing 2
Collebeato 2
Milan 2
Monmouth Junction 2
Prague 2
Sabz 2
Wuhan 2
Ardabil 1
Bari 1
Berlin 1
Birmingham 1
Brisbane 1
Cairo 1
Canberra 1
Changchun 1
Charlotte 1
Dundee 1
Edinburgh 1
Fairfield 1
Fiorano Modenese 1
Fornovo Di Taro 1
Huizen 1
Jinhua 1
Las Vegas 1
Leawood 1
Lissone 1
London 1
Madison 1
Mountain View 1
Mumbai 1
New Delhi 1
Niles 1
Panama City 1
Prata Di Pordenone 1
Puxian 1
Quzhou 1
Redmond 1
Stevenage 1
Tallinn 1
Tappahannock 1
Totale 2.513
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Nome #
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain. 104
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides. 98
Azionifarmacologiche di composti alchilaminoalchilfenilbenzisotiazolici sul trattogastrointestinale 98
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors 95
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays 92
Synthesis and 3D-QSAR Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group 90
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion 85
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity 84
Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups 83
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists 80
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line 80
A New Potent and Selective Histamine H3-Receptor Antagonist, 4(5)-{2-[4(5)-cyclohexylimidazol-2-ylthio]ethyl}imidazole 79
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano 78
Plasma concentration and brain penetration of the H3-receptor antagonist Thioperamide in rats 75
4-(1,2-benzisothiazol-3-)alkanoic and phenylalkanoic acids: synthesis and anti-inflammatory, analgesic and antipyretic activities 75
Action of histamine and ofdifferent synthetic P^ receptor stimulants on the isolated gastric fundus of theguinea pig 74
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity 74
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. 73
HPLC detection ofthioperamide from biological samples and its determination in rat blood and brainafter systemic administration 72
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists 72
Functional Studies of New Imidazole H3-Antagonists on Guinea-Pig Isolated Preparations 71
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. 71
Effects of antimuscarinic agents, H2-blockers and omeprazole on rat chronic gastric ulcer after long-a and short-term administration 69
Dual mechanisms of action of the 5-benzylidene-hydantoin UPR1024 on lung cancer cell lines 68
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine 67
Structure-Property Relationships on Histamine H3-Antagonists: Binding of Phenyl-substituted Alkylthioimidazole Derivatives to Rat Plasma Proteins 66
Heteroarylaminoethyl and heteroarylthioethylimidazoles. Synthesis and H3-receptor affinity 66
4-(3-Oxo-1,2-benzisothiazolin-2-yl)alkanoic, phenyl and phenoxyalkanoic acids: synthesis and anti-inflammatory, analgesic, and antipyretic properties 66
A possible physiological role ofhistamine H^-receptors in rat mesenteric circulation 66
Hz-agonistiimidazolici: importanza della 2-amino sostituzione per 1'attivita farmacologica 66
Sviluppo e caratterizzazione farmacologica di un nuovo potente e selettivo H3-bloccante istaminico non-tioureico 65
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors 65
Structural researcheson H^-agonists: the structures of the dipicrates of 2-(2-amino-4-imidazolyl)ethylamine, its 5-methyl derivative and N^f-dimeihyl-2-(2-am'mo-l,3-thiazol-5-yl)ethylamine 64
Irreversible EGFR inhibitor compounds with antiproliferative activity 64
H3-antagonists: synthesis and activity of 2-amino-5-thiazolyl derivatives 63
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. 63
Ligands for the histamine H3-receptor: new potent antagonists of the 2-thioimidazole type 62
Pharmacological activities of two new histamine analogs 62
Biological studies on 1,2-benzisothiazole derivatives. V. Antimicrobial properties of N-alkanoic, N-arylalkanoic and N-aryloxyalkanoic derivatives of 1,2-benzisothiazolin-3-one: QSAR study and genotoxicity evaluation 62
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series 61
In vitro characterization of potency, affinity and selectivity of H3-antagonists: from thioperamide to thioperamide unrelated derivatives 61
null 61
H3-receptor antagonists: Synthesis and structure relationships of para- and meta-substituted 4(5)-phenyl-2-((2-(4(5)-imidazolyl)ethyl)thio)imidazoles 60
Studio di sostanze analoghe alDimaprit sulla secrezione gastrica "in vitro" 58
Histamine H3-antagonists: the basicity of the polar group in quantitative structure-activity and structure-property relationship 58
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma. 58
Pharmacological profile of original potent H3 receptor antagonists 57
Are histamine receptors involved in the stimulant activities of thiazolylethylamines supposed as cyclic models of dimaprit? 57
Pharmacological profile of new thioperamide derivatives at histamine peripheral H1-, H2, H3-receptors in guinea-pig 54
Rat protein binding and cerebral phospholipid affinity of the H3-receptor antagonist thioperamide 53
Influence of urea-equivalent groups in position 5 of 2-amino, 2-(1-aminoethylidenamino) and 2-guanidino thiazole derivatives on H3-receptor antagonist activity in gastric fistula cat 53
Auxin-like activity of 1,2-benzisothiazole derivatives 52
A possible physiological role of histamine H2-receptors in rat mesenteric circulation 51
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. 51
Pharmacological characterization of H3 receptor antagonists with imidazole, thioimidazole and thioimidazoline polar groups in the side chain 51
Synthesis and binding assays of H3-receptor ligands. 50
Antipyretic activity of new compounds "4-(3-OXO-1,2-BENZISOTHIAZOLIN-2-YL) PHENYLALKANOIC acids, their esters, amides and 1,1-dioxide derivatives 49
Action of histamine and of different synthetic H2 receptor stimulants on the isolated gastric fundus of the guinea pig 46
QSAR study on H3-receptor affinity of benzothiazole derivatives of thioperamide 45
Melatonin Receptor Ligands: Synthesis of New Melatonin Derivatives and Comprehensive Comparative Molecular Field Analysis (CoMFA) Study. 44
null 37
Antipyreticactivity of new compounds 4-(3-oxo-l,2-benzisothiazolin-2-yl)puenyialkanoicacids, their esters, amides and 1,1 dioxide derivatives 33
Influence of urea-equivalent groups in position 5 of 2-amino, 2-(1-aminoethylidenamino) and 2-guanidino thiazole derivatives on H2-receptor antagonist activity in gastric fistula cat. 31
Pharmacological activities of two new histamine analogs 30
THIAZOLYLALKYLAMINES - SYNTHESIS OF ANALOGS OF IMIDAZOLYLETHYLAMINES AND THEIR INFLUENCE ON GASTRIC-SECRETION 27
Are histamine receptors involved in the stimulant activities ofthiazolylethylamines supposed as cyclic models of dimaprit? 7
Totale 4.202
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Categoria #
all - tutte 12.961
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 12.961
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2018/2019124 0 0 0 0 0 0 0 0 0 3 120 1
2019/2020953 134 158 64 12 76 95 117 18 122 44 48 65
2020/2021440 8 65 30 9 60 2 59 5 101 8 91 2
2021/2022344 7 3 3 30 17 33 45 49 19 24 21 93
2022/20231.308 156 143 89 86 121 162 18 74 411 10 30 8
2023/2024325 22 45 3 10 31 137 39 17 14 7 0 0
Totale 4.202