IRIS
BORDI, Fabrizio
 Distribuzione geografica
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Continente #
NA - Nord America 3.102
AS - Asia 2.727
EU - Europa 2.275
SA - Sud America 356
AF - Africa 149
OC - Oceania 5
Continente sconosciuto - Info sul continente non disponibili 1
Totale 8.615
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Nazione #
US - Stati Uniti d'America 3.013
SG - Singapore 976
CN - Cina 883
FI - Finlandia 581
VN - Vietnam 393
SE - Svezia 367
IE - Irlanda 328
DE - Germania 290
BR - Brasile 272
UA - Ucraina 215
HK - Hong Kong 183
IT - Italia 146
TR - Turchia 100
ZA - Sudafrica 94
NL - Olanda 80
GB - Regno Unito 79
FR - Francia 75
CA - Canada 62
IN - India 37
CI - Costa d'Avorio 33
BE - Belgio 29
AR - Argentina 28
BD - Bangladesh 23
RU - Federazione Russa 22
EC - Ecuador 15
JP - Giappone 15
MX - Messico 15
PL - Polonia 15
ES - Italia 14
IQ - Iraq 14
PH - Filippine 12
PK - Pakistan 11
TH - Thailandia 11
KR - Corea 9
CZ - Repubblica Ceca 8
ID - Indonesia 8
UZ - Uzbekistan 8
VE - Venezuela 8
BO - Bolivia 6
CO - Colombia 6
MA - Marocco 6
CL - Cile 5
JO - Giordania 5
LT - Lituania 5
PE - Perù 5
PY - Paraguay 5
UY - Uruguay 5
AT - Austria 4
AU - Australia 4
AZ - Azerbaigian 4
BY - Bielorussia 4
DZ - Algeria 4
IR - Iran 4
OM - Oman 4
SA - Arabia Saudita 4
EG - Egitto 3
HR - Croazia 3
KZ - Kazakistan 3
LB - Libano 3
NP - Nepal 3
TW - Taiwan 3
AE - Emirati Arabi Uniti 2
DO - Repubblica Dominicana 2
EE - Estonia 2
ET - Etiopia 2
GE - Georgia 2
HN - Honduras 2
IL - Israele 2
LY - Libia 2
MD - Moldavia 2
NI - Nicaragua 2
PA - Panama 2
TN - Tunisia 2
TT - Trinidad e Tobago 2
AL - Albania 1
AM - Armenia 1
AO - Angola 1
BB - Barbados 1
BW - Botswana 1
CH - Svizzera 1
EU - Europa 1
GA - Gabon 1
GY - Guiana 1
JM - Giamaica 1
LV - Lettonia 1
MN - Mongolia 1
MY - Malesia 1
RO - Romania 1
RS - Serbia 1
SK - Slovacchia (Repubblica Slovacca) 1
SY - Repubblica araba siriana 1
TJ - Tagikistan 1
TV - Tuvalu 1
Totale 8.615
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Città #
Singapore 477
Ashburn 366
Chandler 337
Dublin 328
Jacksonville 284
San Jose 234
Beijing 210
Santa Clara 189
Hong Kong 178
Ann Arbor 159
Dearborn 129
Dallas 127
Ho Chi Minh City 118
Nanjing 105
Boardman 96
Izmir 90
Johannesburg 88
New York 86
Hanoi 78
Los Angeles 68
Munich 68
Princeton 63
Shanghai 63
San Mateo 56
Lauterbourg 54
Toronto 44
Parma 43
Helsinki 41
Wilmington 38
Shenyang 36
Abidjan 33
Hefei 33
Bremen 32
Nanchang 32
Turku 31
Brussels 29
Kunming 29
Hebei 27
Jinan 26
Haiphong 25
Des Moines 22
Grafing 22
São Paulo 22
Frankfurt am Main 21
Buffalo 20
Columbus 20
Da Nang 18
Tianjin 18
London 17
Guangzhou 16
Changsha 13
Moscow 13
Tokyo 13
Brooklyn 11
The Dalles 11
Warsaw 11
Atlanta 9
Woodbridge 9
Zhengzhou 9
Can Tho 8
Phoenix 8
Seattle 8
Augusta 7
Council Bluffs 7
Denver 7
Jiaxing 7
Milan 7
Montreal 7
Norwalk 7
Pune 7
Rio de Janeiro 7
Stockholm 7
Taiyuan 7
Wuhan 7
Bexley 6
Biên Hòa 6
Falkenstein 6
Fuzhou 6
Haikou 6
Lahore 6
Mordano 6
Redondo Beach 6
San Francisco 6
Tashkent 6
Tân Tiến 6
Amman 5
Amsterdam 5
Baghdad 5
Belo Horizonte 5
Chengdu 5
Curitiba 5
Düsseldorf 5
Genoa 5
Guayaquil 5
Manchester 5
Montevideo 5
Mumbai 5
Orem 5
Poplar 5
Quito 5
Totale 5.094
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Nome #
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides. 209
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity 205
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain. 204
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors 192
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line 191
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists 190
Azionifarmacologiche di composti alchilaminoalchilfenilbenzisotiazolici sul trattogastrointestinale 189
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion 176
4-(1,2-benzisothiazol-3-)alkanoic and phenylalkanoic acids: synthesis and anti-inflammatory, analgesic and antipyretic activities 173
Action of histamine and ofdifferent synthetic P^ receptor stimulants on the isolated gastric fundus of theguinea pig 172
4-(3-Oxo-1,2-benzisothiazolin-2-yl)alkanoic, phenyl and phenoxyalkanoic acids: synthesis and anti-inflammatory, analgesic, and antipyretic properties 171
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays 169
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists 163
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. 162
A New Potent and Selective Histamine H3-Receptor Antagonist, 4(5)-{2-[4(5)-cyclohexylimidazol-2-ylthio]ethyl}imidazole 162
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine 157
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano 156
Synthesis and 3D-QSAR Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group 148
H3-antagonists: synthesis and activity of 2-amino-5-thiazolyl derivatives 148
Effects of antimuscarinic agents, H2-blockers and omeprazole on rat chronic gastric ulcer after long-a and short-term administration 148
Biological studies on 1,2-benzisothiazole derivatives. V. Antimicrobial properties of N-alkanoic, N-arylalkanoic and N-aryloxyalkanoic derivatives of 1,2-benzisothiazolin-3-one: QSAR study and genotoxicity evaluation 148
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. 146
Functional Studies of New Imidazole H3-Antagonists on Guinea-Pig Isolated Preparations 143
Structural researcheson H^-agonists: the structures of the dipicrates of 2-(2-amino-4-imidazolyl)ethylamine, its 5-methyl derivative and N^f-dimeihyl-2-(2-am'mo-l,3-thiazol-5-yl)ethylamine 143
Are histamine receptors involved in the stimulant activities of thiazolylethylamines supposed as cyclic models of dimaprit? 143
Dual mechanisms of action of the 5-benzylidene-hydantoin UPR1024 on lung cancer cell lines 142
A possible physiological role ofhistamine H^-receptors in rat mesenteric circulation 139
Hz-agonistiimidazolici: importanza della 2-amino sostituzione per 1'attivita farmacologica 137
A possible physiological role of histamine H2-receptors in rat mesenteric circulation 136
HPLC detection ofthioperamide from biological samples and its determination in rat blood and brainafter systemic administration 135
Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups 135
Heteroarylaminoethyl and heteroarylthioethylimidazoles. Synthesis and H3-receptor affinity 133
Irreversible EGFR inhibitor compounds with antiproliferative activity 129
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity 129
Histamine H3-antagonists: the basicity of the polar group in quantitative structure-activity and structure-property relationship 129
Action of histamine and of different synthetic H2 receptor stimulants on the isolated gastric fundus of the guinea pig 129
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. 127
Antipyretic activity of new compounds "4-(3-OXO-1,2-BENZISOTHIAZOLIN-2-YL) PHENYLALKANOIC acids, their esters, amides and 1,1-dioxide derivatives 123
Auxin-like activity of 1,2-benzisothiazole derivatives 119
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series 119
In vitro characterization of potency, affinity and selectivity of H3-antagonists: from thioperamide to thioperamide unrelated derivatives 119
Plasma concentration and brain penetration of the H3-receptor antagonist Thioperamide in rats 115
Pharmacological activities of two new histamine analogs 114
H3-receptor antagonists: Synthesis and structure relationships of para- and meta-substituted 4(5)-phenyl-2-((2-(4(5)-imidazolyl)ethyl)thio)imidazoles 113
Influence of urea-equivalent groups in position 5 of 2-amino, 2-(1-aminoethylidenamino) and 2-guanidino thiazole derivatives on H3-receptor antagonist activity in gastric fistula cat 112
QSAR study on H3-receptor affinity of benzothiazole derivatives of thioperamide 112
Sviluppo e caratterizzazione farmacologica di un nuovo potente e selettivo H3-bloccante istaminico non-tioureico 107
Pharmacological profile of original potent H3 receptor antagonists 107
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors 107
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma. 107
Structure-Property Relationships on Histamine H3-Antagonists: Binding of Phenyl-substituted Alkylthioimidazole Derivatives to Rat Plasma Proteins 106
Ligands for the histamine H3-receptor: new potent antagonists of the 2-thioimidazole type 106
Antipyreticactivity of new compounds 4-(3-oxo-l,2-benzisothiazolin-2-yl)puenyialkanoicacids, their esters, amides and 1,1 dioxide derivatives 105
Studio di sostanze analoghe alDimaprit sulla secrezione gastrica "in vitro" 101
Rat protein binding and cerebral phospholipid affinity of the H3-receptor antagonist thioperamide 100
Pharmacological characterization of H3 receptor antagonists with imidazole, thioimidazole and thioimidazoline polar groups in the side chain 99
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. 98
Synthesis and binding assays of H3-receptor ligands. 95
Pharmacological profile of new thioperamide derivatives at histamine peripheral H1-, H2, H3-receptors in guinea-pig 93
Are histamine receptors involved in the stimulant activities ofthiazolylethylamines supposed as cyclic models of dimaprit? 86
Melatonin Receptor Ligands: Synthesis of New Melatonin Derivatives and Comprehensive Comparative Molecular Field Analysis (CoMFA) Study. 75
Pharmacological activities of two new histamine analogs 65
THIAZOLYLALKYLAMINES - SYNTHESIS OF ANALOGS OF IMIDAZOLYLETHYLAMINES AND THEIR INFLUENCE ON GASTRIC-SECRETION 65
Influence of urea-equivalent groups in position 5 of 2-amino, 2-(1-aminoethylidenamino) and 2-guanidino thiazole derivatives on H2-receptor antagonist activity in gastric fistula cat. 63
null 61
null 37
Totale 8.637
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Categoria #
all - tutte 28.409
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 28.409
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021101 0 0 0 0 0 0 0 0 0 8 91 2
2021/2022344 7 3 3 30 17 33 45 49 19 24 21 93
2022/20231.308 156 143 89 86 121 162 18 74 411 10 30 8
2023/2024410 22 45 3 10 31 137 39 17 14 19 27 46
2024/20251.468 51 78 89 93 105 183 42 60 197 144 132 294
2025/20262.882 276 300 287 291 433 208 304 120 473 190 0 0
Totale 8.637