Sfoglia per Autore
Synthesis and characterization of new bivalent agents as melatonin- and histamine h3-ligands.
2014-01-01 Pala, Daniele; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Flammini, Lisa; Barocelli, Elisabetta; Lucini, V; Scaglione, F; Bartolucci, S; Bedini, A; Rivara, Silvia; Spadoni, G.
Comparative Analysis of Virtual Screening Approaches in the Search for Novel EphA2 Receptor Antagonists
2015-01-01 Callegari, Donatella; Pala, Daniele; Scalvini, Laura; Tognolini, Massimiliano; Incerti, Matteo; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Amino acid derivatives as palmitoylethanolamide prodrugs: Synthesis, in vitro metabolism and in vivo plasma profile in rats
2015-01-01 Vacondio, Federica; Bassi, Michele; Silva, Claudia; Castelli, Riccardo; Carmi, Caterina; Scalvini, Laura; Lodola, Alessio; Vivo, Valentina; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco; Rivara, Silvia
The Hippo Pathway and YAP/TAZ-TEAD Protein-Protein Interaction as Targets for Regenerative Medicine and Cancer Treatment
2015-01-01 Santucci, Matteo; Vignudelli, Tatiana; Ferrari, Stefania; Mor, Marco; Scalvini, Laura; Bolognesi, Maria Laura; Uliassi, Elisa; Costi, Maria Paola
Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer's Disease Agents
2016-01-01 Montanari, Serena; Scalvini, Laura; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Andrisano, Vincenza; Ligresti, Alessia; Di Marzo, Vincenzo; Rivara, Silvia; Mor, Marco; Bisi, Alessandra; Rampa, Angela
Free-energy studies reveal a possible mechanism for oxidation-dependent inhibition of MGL
2016-01-01 Scalvini, Laura; Vacondio, Federica; Bassi, Michele; Pala, Daniele; Lodola, Alessio; Rivara, Silvia; Jung, Kwang Mook; Piomelli, Daniele; Mor, Marco
Monoglyceride lipase: Structure and inhibitors
2016-01-01 Scalvini, Laura; Piomelli, Daniele; Mor, Marco
Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity
2018-01-01 Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; Scipione, Luigi; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Ferrara, Fabiana Fosca; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; Milazzo, Ferdinando M.; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannini, Giuseppe
Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth
2018-01-01 Saxena, P; Severi, L; Santucci, M; Taddia, ; Ferrari, S; Luciani, R; Marverti, G; Marraccini, C; Tondi, D; Mor, M; Scalvini, L; Vitiello, S; Losi, L; Fonda, S; Pacifico, S; Guerrini, R; D'Arca, D; Ponterini, G; Costi, Mp
Repurposing of drugs targeting yap-tead functions
2018-01-01 Elisi, GIAN MARCO; Santucci, M.; D'Arca, D.; Lauriola, A.; Marverti, G.; Losi, L.; Scalvini, L.; Bolognesi, M. L.; Mor, M.; Costi, M. P.
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands
2018-01-01 Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
Identification of bivalent ligands with melatonin receptor agonist and fatty acid amide hydrolase (FAAH) inhibitory activity that exhibit ocular hypotensive effect in the rabbit
2018-01-01 Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, Andrea; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S.
Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity
2018-01-01 Messore, A.; Madia, V. N.; Pescatori, L.; Saccoliti, F.; Tudino, V.; De Leo, A.; Bortolami, M.; De Vita, D.; Scipione, L.; Pepi, F.; Costi, R.; Rivara, S.; Scalvini, L.; Mor, M.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Cassinelli, G.; Milazzo, F. M.; Battistuzzi, G.; Di Santo, R.; Giannini, G.
N-Acylethanolamine Acid Amidase (NAAA): Mechanism of Palmitoylethanolamide Hydrolysis Revealed by Mechanistic Simulations
2020-01-01 Scalvini, L.; Ghidini, A.; Lodola, A.; Callegari, D.; Rivara, S.; Piomelli, D.; Mor, M.
Design and SAR Analysis of Covalent Inhibitors Driven by Hybrid QM/MM Simulations
2020-01-01 Lodola, A.; Callegari, D.; Scalvini, L.; Rivara, S.; Mor, M.
Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria
2020-01-01 Elisi, GIAN MARCO; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines
2020-01-01 Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele.
Drug-gut microbiota metabolic interactions: the case of UniPR1331, selective antagonist of the Eph-ephrin system, in mice
2020-01-01 Ferlenghi, F.; Castelli, R.; Scalvini, L.; Giorgio, C.; Corrado, M.; Tognolini, M.; Mor, M.; Lodola, A.; Vacondio, F.
New classes of potent heparanase inhibitors from ligand-based virtual screening
2020-01-01 Pala, D.; Scalvini, L.; Elisi, G. M.; Lodola, A.; Mor, M.; Spadoni, G.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Milazzo, F. M.; Battistuzzi, G.; Rivara, S.; Giannini, G.
Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3α-carbamoyloxy derivative with antiangiogenetic properties
2020-01-01 Incerti, M.; Russo, S.; Corrado, M.; Giorgio, C.; Ballabeni, V.; Chiodelli, P.; Rusnati, M.; Scalvini, L.; Callegari, D.; Castelli, R.; Vacondio, F.; Ferlenghi, F.; Tognolini, M.; Lodola, A.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Synthesis and characterization of new bivalent agents as melatonin- and histamine h3-ligands. | 1-gen-2014 | Pala, Daniele; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Flammini, Lisa; Barocelli, Elisabetta; Lucini, V; Scaglione, F; Bartolucci, S; Bedini, A; Rivara, Silvia; Spadoni, G. | |
| Comparative Analysis of Virtual Screening Approaches in the Search for Novel EphA2 Receptor Antagonists | 1-gen-2015 | Callegari, Donatella; Pala, Daniele; Scalvini, Laura; Tognolini, Massimiliano; Incerti, Matteo; Rivara, Silvia; Mor, Marco; Lodola, Alessio | |
| Amino acid derivatives as palmitoylethanolamide prodrugs: Synthesis, in vitro metabolism and in vivo plasma profile in rats | 1-gen-2015 | Vacondio, Federica; Bassi, Michele; Silva, Claudia; Castelli, Riccardo; Carmi, Caterina; Scalvini, Laura; Lodola, Alessio; Vivo, Valentina; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco; Rivara, Silvia | |
| The Hippo Pathway and YAP/TAZ-TEAD Protein-Protein Interaction as Targets for Regenerative Medicine and Cancer Treatment | 1-gen-2015 | Santucci, Matteo; Vignudelli, Tatiana; Ferrari, Stefania; Mor, Marco; Scalvini, Laura; Bolognesi, Maria Laura; Uliassi, Elisa; Costi, Maria Paola | |
| Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer's Disease Agents | 1-gen-2016 | Montanari, Serena; Scalvini, Laura; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Andrisano, Vincenza; Ligresti, Alessia; Di Marzo, Vincenzo; Rivara, Silvia; Mor, Marco; Bisi, Alessandra; Rampa, Angela | |
| Free-energy studies reveal a possible mechanism for oxidation-dependent inhibition of MGL | 1-gen-2016 | Scalvini, Laura; Vacondio, Federica; Bassi, Michele; Pala, Daniele; Lodola, Alessio; Rivara, Silvia; Jung, Kwang Mook; Piomelli, Daniele; Mor, Marco | |
| Monoglyceride lipase: Structure and inhibitors | 1-gen-2016 | Scalvini, Laura; Piomelli, Daniele; Mor, Marco | |
| Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity | 1-gen-2018 | Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; Scipione, Luigi; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Ferrara, Fabiana Fosca; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; Milazzo, Ferdinando M.; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannini, Giuseppe | |
| Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth | 1-gen-2018 | Saxena, P; Severi, L; Santucci, M; Taddia, ; Ferrari, S; Luciani, R; Marverti, G; Marraccini, C; Tondi, D; Mor, M; Scalvini, L; Vitiello, S; Losi, L; Fonda, S; Pacifico, S; Guerrini, R; D'Arca, D; Ponterini, G; Costi, Mp | |
| Repurposing of drugs targeting yap-tead functions | 1-gen-2018 | Elisi, GIAN MARCO; Santucci, M.; D'Arca, D.; Lauriola, A.; Marverti, G.; Losi, L.; Scalvini, L.; Bolognesi, M. L.; Mor, M.; Costi, M. P. | |
| Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands | 1-gen-2018 | Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto | |
| Identification of bivalent ligands with melatonin receptor agonist and fatty acid amide hydrolase (FAAH) inhibitory activity that exhibit ocular hypotensive effect in the rabbit | 1-gen-2018 | Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, Andrea; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S. | |
| Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity | 1-gen-2018 | Messore, A.; Madia, V. N.; Pescatori, L.; Saccoliti, F.; Tudino, V.; De Leo, A.; Bortolami, M.; De Vita, D.; Scipione, L.; Pepi, F.; Costi, R.; Rivara, S.; Scalvini, L.; Mor, M.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Cassinelli, G.; Milazzo, F. M.; Battistuzzi, G.; Di Santo, R.; Giannini, G. | |
| N-Acylethanolamine Acid Amidase (NAAA): Mechanism of Palmitoylethanolamide Hydrolysis Revealed by Mechanistic Simulations | 1-gen-2020 | Scalvini, L.; Ghidini, A.; Lodola, A.; Callegari, D.; Rivara, S.; Piomelli, D.; Mor, M. | |
| Design and SAR Analysis of Covalent Inhibitors Driven by Hybrid QM/MM Simulations | 1-gen-2020 | Lodola, A.; Callegari, D.; Scalvini, L.; Rivara, S.; Mor, M. | |
| Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria | 1-gen-2020 | Elisi, GIAN MARCO; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
| Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines | 1-gen-2020 | Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele. | |
| Drug-gut microbiota metabolic interactions: the case of UniPR1331, selective antagonist of the Eph-ephrin system, in mice | 1-gen-2020 | Ferlenghi, F.; Castelli, R.; Scalvini, L.; Giorgio, C.; Corrado, M.; Tognolini, M.; Mor, M.; Lodola, A.; Vacondio, F. | |
| New classes of potent heparanase inhibitors from ligand-based virtual screening | 1-gen-2020 | Pala, D.; Scalvini, L.; Elisi, G. M.; Lodola, A.; Mor, M.; Spadoni, G.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Milazzo, F. M.; Battistuzzi, G.; Rivara, S.; Giannini, G. | |
| Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3α-carbamoyloxy derivative with antiangiogenetic properties | 1-gen-2020 | Incerti, M.; Russo, S.; Corrado, M.; Giorgio, C.; Ballabeni, V.; Chiodelli, P.; Rusnati, M.; Scalvini, L.; Callegari, D.; Castelli, R.; Vacondio, F.; Ferlenghi, F.; Tognolini, M.; Lodola, A. |
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