Sfoglia per Autore
Design, synthesis and SAR of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors
2003-01-01 Tarzia, G; Duranti, A; Tontini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Park, C; Kathuria, S; Piomelli, D.
Strategies leading to MT2 selective melatonin receptor antagonists.
2003-01-01 Spadoni, G; Bedini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Tarzia, G.
Strategies leading to MT2 selective melatonin receptor antagonists
2003-01-01 Spadoni, G.; Bedini, A.; Piersanti, G.; Mor, Marco; Rivara, Silvia; Tarzia, G.
Three-Dimensional Quantitative Structure-Activity Relationship Studies on Selected MT1 and MT2 Melatonin Receptor Ligands: Requirements for Subtype Selectivity and Intrinsic Activity Modulation
2003-01-01 Rivara, Silvia; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Spadoni, G; Bedini, A; Tarzia, G; Lucini, V; Pannacci, M; Fraschini, F; Plazzi, Pier Vincenzo
Synthesis and Structure-Activity Relationships of a Series of Pyrrole Cannabinoid Receptor Agonists
2003-01-01 Tarzia, G; Duranti, A; Tontini, A; Spadoni, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Kathuria, S; Piomelli, D.
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors
2004-01-01 Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B.
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity
2004-01-01 Lucini, V.; Pannacci, M.; Scaglione, F.; Fraschini, F.; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Piersanti, G.; Diamantini, G.; Tarzia, G.
Synthesis, Pharmacological Evaluation and Structure-Activity Relationships of Benzopyran Derivatives with Potent SERM Activity
2004-01-01 Amari, G.; Armani, E.; Ghirardi, S.; Delcanale, M.; Civelli, M.; Caruso, P. L.; Galbiati, E.; Lipreri, M.; Rivara, Silvia; Lodola, Alessio; Mor, Marco
Cyclohexylcarbamic Acid 3'- or 4'-Substituted Biphenyl-3-yl Esters of as Fatty Acid Amide Hydrolase Inhibitors: Synthesis, Quantitative Structure-Activity Relationships and Molecular Modelling Studies
2004-01-01 Mor, Marco; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Tarzia, G.; Duranti, A.; Tontini, A.; Piersanti, G.; Kathuria, S.; Piomelli, D.
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists
2004-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors
2005-01-01 Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G.
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists
2005-01-01 Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Analysis of Structure-Activity Relationships for MT2 Selective Antagonists by Melatonin MT1 and MT2 Receptor Models
2005-01-01 Rivara, Silvia; Lorenzi, Simone; Mor, Marco; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Tarzia, G.
Selective inhibition of 2-AG hydrolysis enhances endocannabinoid signaling in hippocampus
2005-01-01 Makara, J. K.; Mor, Marco; Fegley, D.; Szab, S. I.; Kathuria, S.; Astarita, G.; Duranti, A.; Tontini, A.; Tarzia, G.; Rivara, Silvia; Freund, T. F.; Piomelli, D.
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series
2006-01-01 Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo
Synthesis and Structure-Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring
2006-01-01 Tarzia, G; Duranti, A; Gatti, G; Piersanti, G; Tontini, A; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Mor, Marco; Kathuria, S; Piomelli, D.
Pharmacological characterization of hydrolysis-resistant analogs of oleoylethanolamide with potent anorexiant properties.
2006-01-01 Astarita, G; DI GIACOMO, B; Gaetani, S; Oveisi, F; Compton, T. R.; Rivara, Silvia; Tarzia, G; Mor, Marco; Piomelli, D.
MT2 selective melatonin receptor antagonists: design and structure-activity relationships
2006-01-01 Rivara, Silvia; Mor, Marco; Lorenzi, Simone; Lodola, Alessio; Spadoni, G.; Bedini, A.; Tarzia, G.
Reassessing the melatonin pharmacophore- Enantiomeric resolution pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue.
2006-01-01 Rivara, Silvia; Diamantini, G.; DI GIACOMO, B.; Lamba, D.; Gatti, G.; Lucini, V.; Pannacci, M.; Mor, Marco; Spadoni, G.; Tarzia, G.
Design and synthesis of N-(3,3-diphenylpropenyl)alkanamides as a novel class of high-affinity MT2-selective melatonin receptor ligands.
2006-01-01 Bedini, A; Spadoni, G; Gatti, G; Lucarini, S; Tarzia, G; Rivara, Silvia; Lorenzi, Simone; Lodola, Alessio; Mor, Marco; Lucini, V; Pannacci, M; Scaglione, F.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Design, synthesis and SAR of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors | 1-gen-2003 | Tarzia, G; Duranti, A; Tontini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Park, C; Kathuria, S; Piomelli, D. | |
Strategies leading to MT2 selective melatonin receptor antagonists. | 1-gen-2003 | Spadoni, G; Bedini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Tarzia, G. | |
Strategies leading to MT2 selective melatonin receptor antagonists | 1-gen-2003 | Spadoni, G.; Bedini, A.; Piersanti, G.; Mor, Marco; Rivara, Silvia; Tarzia, G. | |
Three-Dimensional Quantitative Structure-Activity Relationship Studies on Selected MT1 and MT2 Melatonin Receptor Ligands: Requirements for Subtype Selectivity and Intrinsic Activity Modulation | 1-gen-2003 | Rivara, Silvia; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Spadoni, G; Bedini, A; Tarzia, G; Lucini, V; Pannacci, M; Fraschini, F; Plazzi, Pier Vincenzo | |
Synthesis and Structure-Activity Relationships of a Series of Pyrrole Cannabinoid Receptor Agonists | 1-gen-2003 | Tarzia, G; Duranti, A; Tontini, A; Spadoni, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Kathuria, S; Piomelli, D. | |
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors | 1-gen-2004 | Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B. | |
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity | 1-gen-2004 | Lucini, V.; Pannacci, M.; Scaglione, F.; Fraschini, F.; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Piersanti, G.; Diamantini, G.; Tarzia, G. | |
Synthesis, Pharmacological Evaluation and Structure-Activity Relationships of Benzopyran Derivatives with Potent SERM Activity | 1-gen-2004 | Amari, G.; Armani, E.; Ghirardi, S.; Delcanale, M.; Civelli, M.; Caruso, P. L.; Galbiati, E.; Lipreri, M.; Rivara, Silvia; Lodola, Alessio; Mor, Marco | |
Cyclohexylcarbamic Acid 3'- or 4'-Substituted Biphenyl-3-yl Esters of as Fatty Acid Amide Hydrolase Inhibitors: Synthesis, Quantitative Structure-Activity Relationships and Molecular Modelling Studies | 1-gen-2004 | Mor, Marco; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Tarzia, G.; Duranti, A.; Tontini, A.; Piersanti, G.; Kathuria, S.; Piomelli, D. | |
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists | 1-gen-2004 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo | |
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors | 1-gen-2005 | Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G. | |
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists | 1-gen-2005 | Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
Analysis of Structure-Activity Relationships for MT2 Selective Antagonists by Melatonin MT1 and MT2 Receptor Models | 1-gen-2005 | Rivara, Silvia; Lorenzi, Simone; Mor, Marco; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Tarzia, G. | |
Selective inhibition of 2-AG hydrolysis enhances endocannabinoid signaling in hippocampus | 1-gen-2005 | Makara, J. K.; Mor, Marco; Fegley, D.; Szab, S. I.; Kathuria, S.; Astarita, G.; Duranti, A.; Tontini, A.; Tarzia, G.; Rivara, Silvia; Freund, T. F.; Piomelli, D. | |
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series | 1-gen-2006 | Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo | |
Synthesis and Structure-Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring | 1-gen-2006 | Tarzia, G; Duranti, A; Gatti, G; Piersanti, G; Tontini, A; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Mor, Marco; Kathuria, S; Piomelli, D. | |
Pharmacological characterization of hydrolysis-resistant analogs of oleoylethanolamide with potent anorexiant properties. | 1-gen-2006 | Astarita, G; DI GIACOMO, B; Gaetani, S; Oveisi, F; Compton, T. R.; Rivara, Silvia; Tarzia, G; Mor, Marco; Piomelli, D. | |
MT2 selective melatonin receptor antagonists: design and structure-activity relationships | 1-gen-2006 | Rivara, Silvia; Mor, Marco; Lorenzi, Simone; Lodola, Alessio; Spadoni, G.; Bedini, A.; Tarzia, G. | |
Reassessing the melatonin pharmacophore- Enantiomeric resolution pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue. | 1-gen-2006 | Rivara, Silvia; Diamantini, G.; DI GIACOMO, B.; Lamba, D.; Gatti, G.; Lucini, V.; Pannacci, M.; Mor, Marco; Spadoni, G.; Tarzia, G. | |
Design and synthesis of N-(3,3-diphenylpropenyl)alkanamides as a novel class of high-affinity MT2-selective melatonin receptor ligands. | 1-gen-2006 | Bedini, A; Spadoni, G; Gatti, G; Lucarini, S; Tarzia, G; Rivara, Silvia; Lorenzi, Simone; Lodola, Alessio; Mor, Marco; Lucini, V; Pannacci, M; Scaglione, F. |
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