RADI, Marco
RADI, Marco
Dipartimento di Scienze degli Alimenti e del Farmaco
6-Vinyl pyrimidine and pyrimidinone derivatives and the use thereof
2005-01-01 Maurizio, Botta; Federico, Corelli; Elena, Petricci; Radi, Marco; Giovanni, Maga; Josè A., Estè; Antonello, Mai
A cascade screening approach for the identification of Bcr-Abl myristate pocket binders active against wild type and T315I mutant
2016-01-01 Radi, Marco; Schneider, Ralf; Fallacara, Anna Lucia; Botta, Lorenzo; Crespan, Emmanuele; Tintori, Cristina; Maga, Giovanni; Kissova, Miroslava; Calgani, Alessia; Richters, André; Musumeci, Franesca; Rauh, Daniel; Schenone, Silvia
A Combination Strategy to Inhibit Pim-1: Synergism between Noncompetitive and ATP-Competitive Inhibitors
2013-01-01 Mattia, Mori; Cristina, Tintori; Robert Selwyne Arul, Christopher; Radi, Marco; Silvia, Schenone; Francesca, Musumeci; Chiara, Brullo; Patrizia, Sanità; Simona, Delle monache; Adriano, Angelucci; Miroslava, Kissova; Emmanuele, Crespan; Giovanni, Maga; Maurizio, Botta
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin
2016-01-01 Vucicevic, Jelica; Srdic Rajic, Tatjana; Pieroni, Marco; Laurila, Jonne M. M.; Perovic, Vladimir; Tassini, Sabrina; Azzali, Elisa; Costantino, Gabriele; Glisic, Sanja; Agbaba, Danica; Scheinin, Mika; Nikolic, Katarina; Radi, Marco; Veljkovic, Nevena
A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: From in silico screening to cyclodextrin formulation
2012-01-01 Radi, Marco; Lasse, Evensen; Elena, Dreassi; Claudio, Zamperini; Marialessandra, Caporicci; Federico, Falchi; Francesca, Musumeci; Silvia, Schenone; James B., Lorens; Maurizio, Botta
A Convergent Approach for the Synthesis of Ara-Neplanocin a Analogues Under Subzero Microwave Assisted Conditions
2009-01-01 Radi, Marco; Jagadeeshwar R., Rao; Ashok K., Jha; Chu, Chung K.
A Domino Microwave-Assisted Protocol for the Synthesis of 2,6-Disubstituted Pyrimidinones
2011-01-01 Radi, Marco; Gianni, Casaluce; Maurizio, Botta
A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides
2016-01-01 Vincetti, Paolo; Brianza, Anna; Scalacci, Nicolò; Costantino, Gabriele; Castagnolo, Daniele; Radi, Marco
A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes
2016-01-01 Tassini, Sabrina; Castagnolo, Daniele; Scalacci, Nicolò; Kissova, Miroslava; Armijos Rivera, Jorge I.; Giagnorio, Federica; Maga, Giovanni; Costantino, Gabriele; Crespan, Emmanuele; Radi, Marco
A Multidisciplinary Approach for the Identification of Novel HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: S-DABOCs and DAVPs
2008-01-01 Radi, Marco; Chiara, Falciani; Lorenzo, Contemori; Elena, Petricci; Giovanni, Maga; Alberta, Samuele; Samantha, Zanoli; Montserrat, Terrazas; Marinunzia, Castria; Andrea, Togninelli; Esté, J. o. s. é. . A.; Imma Clotet, Codina; Mercedes Armand, Ugón; Maurizio, Botta
A one-pot two-step microwave-assisted synthesis of N1-substituted 5,6-ring-fused 2-pyridones
2013-01-01 Radi, Marco; Gian Paolo, Vallerini; Alessia, Petrelli; Paolo, Vincetti; Costantino, Gabriele
A one-pot, two-step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs)
2008-01-01 Radi, Marco; Sara, Saletti; Maurizio, Botta
A Versatile Route to C-6 Arylmethyl-FunctionalizedS-DABO and Related Analogues
2007-01-01 Radi, Marco; Lorenzo, Contemori; Daniele, Castagnolo; Raffaella, Spinosa; José A., Esté; Silvio, Massa; Maurizio, Botta
Allosteric Inhibitors of Bcr-Abl: Towards Novel Myristate-Pocket Binders
2013-01-01 Radi, Marco; Silvia, Schenone; Maurizio, Botta
Arylation of 2-Furyl 4-Fluorophenyl Ketone: An Extension of Heck Chemistry towards Novel Integrase Inhibitors
2010-01-01 Luigi, Franchi; Marta, Rinaldi; Giulia, Vignaroli; Anna, Innitzer; Radi, Marco; Maurizio, Botta
ATP-Competitive Inhibitors of mTOR: An Update
2011-01-01 Silvia, Schenone; Chiara, Brullo; Francesca, Musumeci; Radi, Marco; Maurizio, Botta
Biologically Driven Synthesis of Pyrazolo[3,4-d]pyrimidines As Protein Kinase Inhibitors: An Old Scaffold As a New Tool for Medicinal Chemistry and Chemical Biology Studies
2014-01-01 Silvia, Schenone; Radi, Marco; Francesca, Musumeci; Chiara, Brullo; Maurizio, Botta
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses
2021-01-01 Martina Maria, Grazia.; Vicenti, I.; Bauer, L.; Crespan, E.; Rango, E.; Boccuto, A.; Olivieri, N.; Incerti, M.; Zwaagstra, M.; Allodi, M.; Bertoni, S.; Dreassi, E.; Zazzi, M.; van Kuppeveld, F. J. M.; Maga, G.; Radi, M.
C6-Unsubstituted Pyrazolo[3,4-d]pyrimidines Are Dual Src/Abl Inhibitors Effective against Imatinib Mesylate Resistant Chronic Myeloid Leukemia Cell Lines
2009-01-01 Maria Alessandra, Santucci; Valentina, Corradi; Manuela, Mancini; Fabrizio, Manetti; Radi, Marco; Silvia, Schenone; Maurizio, Botta
Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d ]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma
2015-01-01 Tintori, Cristina; Fallacara, Anna Lucia; Radi, Marco; Zamperini, Claudio; Dreassi, Elena; Crespan, Emmanuele; Maga, Giovanni; Schenone, Silvia; Musumeci, Francesca; Brullo, Chiara; Richters, André; Gasparrini, Francesca; Angelucci, Adriano; Festuccia, Claudio; Delle Monache, Simona; Rauh, Daniel; Botta, Maurizio
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 6-Vinyl pyrimidine and pyrimidinone derivatives and the use thereof | 1-gen-2005 | Maurizio, Botta; Federico, Corelli; Elena, Petricci; Radi, Marco; Giovanni, Maga; Josè A., Estè; Antonello, Mai | |
| A cascade screening approach for the identification of Bcr-Abl myristate pocket binders active against wild type and T315I mutant | 1-gen-2016 | Radi, Marco; Schneider, Ralf; Fallacara, Anna Lucia; Botta, Lorenzo; Crespan, Emmanuele; Tintori, Cristina; Maga, Giovanni; Kissova, Miroslava; Calgani, Alessia; Richters, André; Musumeci, Franesca; Rauh, Daniel; Schenone, Silvia | |
| A Combination Strategy to Inhibit Pim-1: Synergism between Noncompetitive and ATP-Competitive Inhibitors | 1-gen-2013 | Mattia, Mori; Cristina, Tintori; Robert Selwyne Arul, Christopher; Radi, Marco; Silvia, Schenone; Francesca, Musumeci; Chiara, Brullo; Patrizia, Sanità; Simona, Delle monache; Adriano, Angelucci; Miroslava, Kissova; Emmanuele, Crespan; Giovanni, Maga; Maurizio, Botta | |
| A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin | 1-gen-2016 | Vucicevic, Jelica; Srdic Rajic, Tatjana; Pieroni, Marco; Laurila, Jonne M. M.; Perovic, Vladimir; Tassini, Sabrina; Azzali, Elisa; Costantino, Gabriele; Glisic, Sanja; Agbaba, Danica; Scheinin, Mika; Nikolic, Katarina; Radi, Marco; Veljkovic, Nevena | |
| A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: From in silico screening to cyclodextrin formulation | 1-gen-2012 | Radi, Marco; Lasse, Evensen; Elena, Dreassi; Claudio, Zamperini; Marialessandra, Caporicci; Federico, Falchi; Francesca, Musumeci; Silvia, Schenone; James B., Lorens; Maurizio, Botta | |
| A Convergent Approach for the Synthesis of Ara-Neplanocin a Analogues Under Subzero Microwave Assisted Conditions | 1-gen-2009 | Radi, Marco; Jagadeeshwar R., Rao; Ashok K., Jha; Chu, Chung K. | |
| A Domino Microwave-Assisted Protocol for the Synthesis of 2,6-Disubstituted Pyrimidinones | 1-gen-2011 | Radi, Marco; Gianni, Casaluce; Maurizio, Botta | |
| A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides | 1-gen-2016 | Vincetti, Paolo; Brianza, Anna; Scalacci, Nicolò; Costantino, Gabriele; Castagnolo, Daniele; Radi, Marco | |
| A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes | 1-gen-2016 | Tassini, Sabrina; Castagnolo, Daniele; Scalacci, Nicolò; Kissova, Miroslava; Armijos Rivera, Jorge I.; Giagnorio, Federica; Maga, Giovanni; Costantino, Gabriele; Crespan, Emmanuele; Radi, Marco | |
| A Multidisciplinary Approach for the Identification of Novel HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: S-DABOCs and DAVPs | 1-gen-2008 | Radi, Marco; Chiara, Falciani; Lorenzo, Contemori; Elena, Petricci; Giovanni, Maga; Alberta, Samuele; Samantha, Zanoli; Montserrat, Terrazas; Marinunzia, Castria; Andrea, Togninelli; Esté, J. o. s. é. . A.; Imma Clotet, Codina; Mercedes Armand, Ugón; Maurizio, Botta | |
| A one-pot two-step microwave-assisted synthesis of N1-substituted 5,6-ring-fused 2-pyridones | 1-gen-2013 | Radi, Marco; Gian Paolo, Vallerini; Alessia, Petrelli; Paolo, Vincetti; Costantino, Gabriele | |
| A one-pot, two-step microwave-assisted synthesis of highly functionalized benzoxazoles using solid-supported reagents (SSRs) | 1-gen-2008 | Radi, Marco; Sara, Saletti; Maurizio, Botta | |
| A Versatile Route to C-6 Arylmethyl-FunctionalizedS-DABO and Related Analogues | 1-gen-2007 | Radi, Marco; Lorenzo, Contemori; Daniele, Castagnolo; Raffaella, Spinosa; José A., Esté; Silvio, Massa; Maurizio, Botta | |
| Allosteric Inhibitors of Bcr-Abl: Towards Novel Myristate-Pocket Binders | 1-gen-2013 | Radi, Marco; Silvia, Schenone; Maurizio, Botta | |
| Arylation of 2-Furyl 4-Fluorophenyl Ketone: An Extension of Heck Chemistry towards Novel Integrase Inhibitors | 1-gen-2010 | Luigi, Franchi; Marta, Rinaldi; Giulia, Vignaroli; Anna, Innitzer; Radi, Marco; Maurizio, Botta | |
| ATP-Competitive Inhibitors of mTOR: An Update | 1-gen-2011 | Silvia, Schenone; Chiara, Brullo; Francesca, Musumeci; Radi, Marco; Maurizio, Botta | |
| Biologically Driven Synthesis of Pyrazolo[3,4-d]pyrimidines As Protein Kinase Inhibitors: An Old Scaffold As a New Tool for Medicinal Chemistry and Chemical Biology Studies | 1-gen-2014 | Silvia, Schenone; Radi, Marco; Francesca, Musumeci; Chiara, Brullo; Maurizio, Botta | |
| Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses | 1-gen-2021 | Martina Maria, Grazia.; Vicenti, I.; Bauer, L.; Crespan, E.; Rango, E.; Boccuto, A.; Olivieri, N.; Incerti, M.; Zwaagstra, M.; Allodi, M.; Bertoni, S.; Dreassi, E.; Zazzi, M.; van Kuppeveld, F. J. M.; Maga, G.; Radi, M. | |
| C6-Unsubstituted Pyrazolo[3,4-d]pyrimidines Are Dual Src/Abl Inhibitors Effective against Imatinib Mesylate Resistant Chronic Myeloid Leukemia Cell Lines | 1-gen-2009 | Maria Alessandra, Santucci; Valentina, Corradi; Manuela, Mancini; Fabrizio, Manetti; Radi, Marco; Silvia, Schenone; Maurizio, Botta | |
| Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d ]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma | 1-gen-2015 | Tintori, Cristina; Fallacara, Anna Lucia; Radi, Marco; Zamperini, Claudio; Dreassi, Elena; Crespan, Emmanuele; Maga, Giovanni; Schenone, Silvia; Musumeci, Francesca; Brullo, Chiara; Richters, André; Gasparrini, Francesca; Angelucci, Adriano; Festuccia, Claudio; Delle Monache, Simona; Rauh, Daniel; Botta, Maurizio |