Sfoglia per Autore
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor
2020-01-01 Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G.
Birth of a pathway for sulfur metabolism in early amniote evolution
2020-01-01 Malatesta, M; Mori, G; Acquotti, D; Campanini, B; Peracchi, A; Antin, P B; Percudani, R
The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase
2020-01-01 Marchesani, F.; Gianquinto, E.; Autiero, I.; Michielon, A.; Campanini, B.; Faggiano, S.; Bettati, S.; Mozzarelli, A.; Spyrakis, F.; Bruno, S.
Nuovi composti antimicrobici
2021-01-01 Annunziato, Giannamaria; Costantino, Gabriele; Cabassi, Clotilde Silvia; Pieroni, Marco; Bruno, Agostino; Campanini, Barbara; Bettati, Stefano; Mozzarelli, Andrea
Investigational Studies on a Hit Compound Cyclopropane-Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin Adjuvant
2021-01-01 Annunziato, G.; Spadini, C.; Franko, N.; Storici, P.; Demitri, N.; Pieroni, M.; Flisi, S.; Rosati, L.; Iannarelli, M.; Marchetti, M.; Magalhaes, J.; Bettati, S.; Mozzarelli, A.; Cabassi, C. S.; Campanini, B.; Costantino, G.
The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase
2021-01-01 Marchesani, F.; Gianquinto, E.; Autiero, I.; Michielon, A.; Campanini, B.; Faggiano, S.; Bettati, S.; Mozzarelli, A.; Spyrakis, F.; Bruno, S.
Revealing the dynamic allosteric changes required for formation of the cysteine synthase complex by hydrogen-deuterium exchange MS
2021-01-01 Rosa, B.; Dickinson, E. R.; Marchetti, M.; Campanini, B.; Pioselli, B.; Bettati, S.; Rand, K. D.
Human serine racemase is inhibited by glyceraldehyde 3-phosphate, but not by glyceraldehyde 3-phosphate dehydrogenase
2021-01-01 Michielon, A.; Marchesani, F.; Faggiano, S.; Giaccari, R.; Campanini, B.; Bettati, S.; Mozzarelli, A.; Bruno, S.
A competitive o‐acetylserine sulfhydrylase inhibitor modulates the formation of cysteine synthase complex
2021-01-01 Marchetti, M.; De Angelis, F. S.; Annunziato, G.; Costantino, G.; Pieroni, M.; Ronda, L.; Mozzarelli, A.; Campanini, B.; Cannistraro, S.; Bizzarri, A. R.; Bettati, S.
A novel assay for phosphoserine phosphatase exploiting serine acetyltransferase as the coupling enzyme
2021-01-01 Marchesani, F.; Zangelmi, E.; Bruno, S.; Bettati, S.; Peracchi, A.; Campanini, B.
Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants
2021-01-01 Magalhães, Joana; Franko, Nina; Raboni, Samanta; Annunziato, Giannamaria; Tammela, Päivi; Bruno, Agostino; Bettati, Stefano; Armao, Stefano; Spadini, Costanza; Cabassi, Clotilde Silvia; Mozzarelli, Andrea; Pieroni, Marco; Campanini, Barbara; Costantino, Gabriele
Understanding iron hijacking by Staphylococcus aureus: a structural and mechanistic insight into the interaction of IsdB hemophore with human hemoglobin
2022-01-01 De Bei, O; Marchetti, M; Ronda, L; Gianquinto, E; Levantino, M; Lazzarato, L; Chirgadze, Dy; Hardwick, Sw; Cooper, Lr; Cozzi, M; Faggiano, S; Spyrakis, F; Luisi, Bf; Campanini, B; Bettati, S
Cryo-EM structures of staphylococcal IsdB bound to human hemoglobin reveal the process of heme extraction
2022-01-01 DE BEI, Omar; Marchetti, Marialaura; Ronda, Luca; Gianquinto, Eleonora; Lazzarato, Loretta; Chirgadze, Dimitri Y.; Hadwick, Steven W.; Cooper, Lee R.; Spyrakis, Francesca; Luisi, Ben F.; Campanini, Barbara; Bettati, Stefano
Exploring the chemical space around N-(5-nitrothiazol-2-yl)-1,2,3-thiadiazole-4-carboxamide, a hit compound with serine acetyltransferase (SAT) inhibitory properties
2022-01-01 Pavone, M.; Raboni, S.; Marchetti, M.; Annunziato, G.; Bettati, S.; Papotti, B.; Marchi, C.; Carosati, E.; Pieroni, M.; Campanini, B.; Costantino, G.
Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria
2022-01-01 Annunziato, Giannamaria; Spadini, Costanza; Marchetti, Marialaura; Franko, Nina; Pavone, Marialaura; Iannarelli, Mattia; Bruno, Agostino; Pieroni, Marco; Bettati, Stefano; Cabassi, Clotilde Silvia; Campanini, Barbara; Costantino, Gabriele
Human Serine Racemase Weakly Binds the Third PDZ Domain of PSD-95
2022-01-01 Giaccari, R.; Marchesani, F.; Compari, C.; Fisicaro, E.; Mozzarelli, A.; Campanini, B.; Bettati, S.; Bruno, S.; Faggiano, S.
Use of Exogenous Enzymes in Human Therapy: Approved Drugs and Potential Applications
2022-01-01 Cioni, P.; Gabellieri, E.; Campanini, B.; Bettati, S.; Raboni, S.
Phosphoserine Aminotransferase Pathogenetic Variants in Serine Deficiency Disorders: A Functional Characterization
2023-01-01 Marchesani, F.; Michielon, A.; Viale, E.; Bianchera, A.; Cavazzini, D.; Pollegioni, L.; Murtas, G.; Mozzarelli, A.; Bettati, S.; Peracchi, A.; Campanini, B.; Bruno, S.
The human phosphorylated pathway: a multienzyme metabolic assembly for l-serine biosynthesis
2023-01-01 Rabattoni, V.; Marchesani, F.; Murtas, G.; Sacchi, S.; Mozzarelli, A.; Bruno, S.; Peracchi, A.; Pollegioni, L.; Campanini, B.
L-serine biosynthesis in the human central nervous system: Structure and function of phosphoserine aminotransferase
2023-01-01 Marchesani, Francesco; Zangelmi, Erika; Murtas, Giulia; Costanzi, Elisa; Ullah, Raheem; Peracchi, Alessio; Bruno, Stefano; Pollegioni, Loredano; Mozzarelli, Andrea; Storici, Paola; Campanini, Barbara
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor | 1-gen-2020 | Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G. | |
Birth of a pathway for sulfur metabolism in early amniote evolution | 1-gen-2020 | Malatesta, M; Mori, G; Acquotti, D; Campanini, B; Peracchi, A; Antin, P B; Percudani, R | |
The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase | 1-gen-2020 | Marchesani, F.; Gianquinto, E.; Autiero, I.; Michielon, A.; Campanini, B.; Faggiano, S.; Bettati, S.; Mozzarelli, A.; Spyrakis, F.; Bruno, S. | |
Nuovi composti antimicrobici | 1-gen-2021 | Annunziato, Giannamaria; Costantino, Gabriele; Cabassi, Clotilde Silvia; Pieroni, Marco; Bruno, Agostino; Campanini, Barbara; Bettati, Stefano; Mozzarelli, Andrea | |
Investigational Studies on a Hit Compound Cyclopropane-Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin Adjuvant | 1-gen-2021 | Annunziato, G.; Spadini, C.; Franko, N.; Storici, P.; Demitri, N.; Pieroni, M.; Flisi, S.; Rosati, L.; Iannarelli, M.; Marchetti, M.; Magalhaes, J.; Bettati, S.; Mozzarelli, A.; Cabassi, C. S.; Campanini, B.; Costantino, G. | |
The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase | 1-gen-2021 | Marchesani, F.; Gianquinto, E.; Autiero, I.; Michielon, A.; Campanini, B.; Faggiano, S.; Bettati, S.; Mozzarelli, A.; Spyrakis, F.; Bruno, S. | |
Revealing the dynamic allosteric changes required for formation of the cysteine synthase complex by hydrogen-deuterium exchange MS | 1-gen-2021 | Rosa, B.; Dickinson, E. R.; Marchetti, M.; Campanini, B.; Pioselli, B.; Bettati, S.; Rand, K. D. | |
Human serine racemase is inhibited by glyceraldehyde 3-phosphate, but not by glyceraldehyde 3-phosphate dehydrogenase | 1-gen-2021 | Michielon, A.; Marchesani, F.; Faggiano, S.; Giaccari, R.; Campanini, B.; Bettati, S.; Mozzarelli, A.; Bruno, S. | |
A competitive o‐acetylserine sulfhydrylase inhibitor modulates the formation of cysteine synthase complex | 1-gen-2021 | Marchetti, M.; De Angelis, F. S.; Annunziato, G.; Costantino, G.; Pieroni, M.; Ronda, L.; Mozzarelli, A.; Campanini, B.; Cannistraro, S.; Bizzarri, A. R.; Bettati, S. | |
A novel assay for phosphoserine phosphatase exploiting serine acetyltransferase as the coupling enzyme | 1-gen-2021 | Marchesani, F.; Zangelmi, E.; Bruno, S.; Bettati, S.; Peracchi, A.; Campanini, B. | |
Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants | 1-gen-2021 | Magalhães, Joana; Franko, Nina; Raboni, Samanta; Annunziato, Giannamaria; Tammela, Päivi; Bruno, Agostino; Bettati, Stefano; Armao, Stefano; Spadini, Costanza; Cabassi, Clotilde Silvia; Mozzarelli, Andrea; Pieroni, Marco; Campanini, Barbara; Costantino, Gabriele | |
Understanding iron hijacking by Staphylococcus aureus: a structural and mechanistic insight into the interaction of IsdB hemophore with human hemoglobin | 1-gen-2022 | De Bei, O; Marchetti, M; Ronda, L; Gianquinto, E; Levantino, M; Lazzarato, L; Chirgadze, Dy; Hardwick, Sw; Cooper, Lr; Cozzi, M; Faggiano, S; Spyrakis, F; Luisi, Bf; Campanini, B; Bettati, S | |
Cryo-EM structures of staphylococcal IsdB bound to human hemoglobin reveal the process of heme extraction | 1-gen-2022 | DE BEI, Omar; Marchetti, Marialaura; Ronda, Luca; Gianquinto, Eleonora; Lazzarato, Loretta; Chirgadze, Dimitri Y.; Hadwick, Steven W.; Cooper, Lee R.; Spyrakis, Francesca; Luisi, Ben F.; Campanini, Barbara; Bettati, Stefano | |
Exploring the chemical space around N-(5-nitrothiazol-2-yl)-1,2,3-thiadiazole-4-carboxamide, a hit compound with serine acetyltransferase (SAT) inhibitory properties | 1-gen-2022 | Pavone, M.; Raboni, S.; Marchetti, M.; Annunziato, G.; Bettati, S.; Papotti, B.; Marchi, C.; Carosati, E.; Pieroni, M.; Campanini, B.; Costantino, G. | |
Inhibitors of O-Acetylserine Sulfhydrylase with a Cyclopropane-Carboxylic Acid Scaffold Are Effective Colistin Adjuvants in Gram Negative Bacteria | 1-gen-2022 | Annunziato, Giannamaria; Spadini, Costanza; Marchetti, Marialaura; Franko, Nina; Pavone, Marialaura; Iannarelli, Mattia; Bruno, Agostino; Pieroni, Marco; Bettati, Stefano; Cabassi, Clotilde Silvia; Campanini, Barbara; Costantino, Gabriele | |
Human Serine Racemase Weakly Binds the Third PDZ Domain of PSD-95 | 1-gen-2022 | Giaccari, R.; Marchesani, F.; Compari, C.; Fisicaro, E.; Mozzarelli, A.; Campanini, B.; Bettati, S.; Bruno, S.; Faggiano, S. | |
Use of Exogenous Enzymes in Human Therapy: Approved Drugs and Potential Applications | 1-gen-2022 | Cioni, P.; Gabellieri, E.; Campanini, B.; Bettati, S.; Raboni, S. | |
Phosphoserine Aminotransferase Pathogenetic Variants in Serine Deficiency Disorders: A Functional Characterization | 1-gen-2023 | Marchesani, F.; Michielon, A.; Viale, E.; Bianchera, A.; Cavazzini, D.; Pollegioni, L.; Murtas, G.; Mozzarelli, A.; Bettati, S.; Peracchi, A.; Campanini, B.; Bruno, S. | |
The human phosphorylated pathway: a multienzyme metabolic assembly for l-serine biosynthesis | 1-gen-2023 | Rabattoni, V.; Marchesani, F.; Murtas, G.; Sacchi, S.; Mozzarelli, A.; Bruno, S.; Peracchi, A.; Pollegioni, L.; Campanini, B. | |
L-serine biosynthesis in the human central nervous system: Structure and function of phosphoserine aminotransferase | 1-gen-2023 | Marchesani, Francesco; Zangelmi, Erika; Murtas, Giulia; Costanzi, Elisa; Ullah, Raheem; Peracchi, Alessio; Bruno, Stefano; Pollegioni, Loredano; Mozzarelli, Andrea; Storici, Paola; Campanini, Barbara |
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