Sfoglia per Autore
Human serine racemase is allosterically modulated by NADH and reduced nicotinamide derivatives
2016-01-01 Bruno, Stefano; Marchesani, Francesco; Dellafiora, Luca; Margiotta, Marilena; Faggiano, Serena; Campanini, Barbara; Mozzarelli, Andrea
Structural insight into the interaction of O-acetylserine sulfhydrylase with competitive, peptidic inhibitors by Saturation Transfer Difference-NMR
2016-01-01 Benoni, Roberto; Pertinhez, Thelma; Spyrakis, Francesca; Davalli, S; Pellegrino, S; Paredi, Gianluca; Pezzotti, A; Bettati, Stefano; Campanini, Barbara; Mozzarelli, Andrea
Insights on O-acetylserine Sulfhydrylase Structure, Function and Biopharmaceutical Applications
2017-01-01 Campanini, Barbara; Mozzarelli, Andrea
Study of DNA binding and bending by Bacillus subtilis GabR, a PLP-dependent transcription factor
2017-01-01 Amidani, Davide; Tramonti, Angela; Canosa, ANDREA VALERIA; Campanini, Barbara; Maggi, Stefano; Milano, Teresa; DI SALVO, MARTINO LUIGI; Pascarella, Stefano; Contestabile, Roberto; Bettati, Stefano; Rivetti, Claudio
Activation of an anti-bacterial toxin by the biosynthetic enzyme CysK: mechanism of binding, interaction specificity and competition with cysteine synthase
2017-01-01 Benoni, Roberto; Beck, Christina M.; Garza-Sánchez, Fernando; Bettati, Stefano; Mozzarelli, Andrea; Hayes, Christopher S.; Campanini, Barbara
Modulation of Escherichia coli serine acetyltransferase catalytic activity in the cysteine synthase complex
2017-01-01 Benoni, Roberto; DE BEI, Omar; Paredi, Gianluca; Hayes, Christopher S.; Franko, Nina; Mozzarelli, Andrea; Bettati, Stefano; Campanini, Barbara
Magnesium and calcium ions differentially affect human serine racemase activity and modulate its quaternary equilibrium toward a tetrameric form
2017-01-01 Bruno, Stefano; Margiotta, Marilena; Marchesani, Francesco; Paredi, Gianluca; Orlandi, Valentina; Faggiano, Serena; Ronda, Luca; Campanini, Barbara; Mozzarelli, Andrea
Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets
2018-01-01 Magalhães, Joana; Annunziato, Giannamaria; Franko, Nina; Pieroni, Marco; Campanini, Barbara; Bruno, Agostino; Costantino, Gabriele
Glutamine 89 is a key residue in the allosteric modulation of human serine racemase activity by ATP
2018-01-01 Canosa, Andrea V; Faggiano, Serena; Marchetti, Marialaura; Armao, Stefano; Bettati, Stefano; Bruno, Stefano; Percudani, Riccardo; Campanini, Barbara; Mozzarelli, Andrea
Insight into GFPmut2 pH Dependence by Single Crystal Microspectrophotometry and X-ray Crystallography
2018-01-01 Lolli, Graziano; Raboni, Samanta; Pasqualetto, Elisa; Benoni, Roberto; Campanini, Barbara; Ronda, Luca; Mozzarelli, Andrea; Bettati, Stefano; Battistutta, Roberto
Inhibition of O-acetylserine sulfhydrylase by fluoroalanine derivatives
2018-01-01 Franko, N.; Grammatoglou, K.; Campanini, B.; Costantino, G.; Jirgensons, A.; Mozzarelli, A.
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design
2018-01-01 Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara
Human serine racemase is nitrosylated at multiple sites
2018-01-01 Marchesani, Francesco; Bruno, Stefano; Paredi, Gianluca; Raboni, Samanta; Campanini, Barbara; Mozzarelli, Andrea
The Energy Landscape of Human Serine Racemase
2019-01-01 Raboni, Samanta; Marchetti, Marialaura; Faggiano, Serena; Campanini, Barbara; Bruno, Stefano; Marchesani, Francesco; Margiotta, Marilena; Mozzarelli, Andrea
Interaction of human hemoglobin and semi-hemoglobins with the Staphylococcus aureus hemophore IsdB: a kinetic and mechanistic insight
2019-01-01 Gianquinto, E.; Moscetti, I.; De Bei, O.; Campanini, B.; Marchetti, M.; Luque, F. J.; Cannistraro, S.; Ronda, L.; Bizzarri, A. R.; Spyrakis, F.; Bettati, S.
Combination of SAXS and protein painting discloses the three-dimensional organization of the bacterial cysteine synthase complex, a potential target for enhancers of antibiotic action
2019-01-01 Rosa, B.; Marchetti, M.; Paredi, G.; Amenitsch, H.; Franko, N.; Benoni, R.; Giabbai, B.; De Marino, M. G.; Mozzarelli, A.; Ronda, L.; Storici, P.; Campanini, B.; Bettati, S.
Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms
2019-01-01 Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Nikitjuka, Anna; Mozzarelli, Andrea; Bettati, Stefano; Karawajczyk, Anna; Jirgensons, Aigars; Campanini, Barbara; Costantino, Gabriele
More than a Confinement: “Soft” and “Hard” Enzyme Entrapment Modulates Biological Catalyst Function
2019-01-01 Cottone, Grazia; Giuffrida, Sergio; Bettati, Stefano; Bruno, Stefano; Campanini, Barbara; Marchetti, Marialaura; Abbruzzetti, Stefania; Viappiani, Cristiano; Cupane, Antonio; Mozzarelli, Andrea; Ronda, Luca
The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase
2020-01-01 Marchesani, F.; Gianquinto, E.; Autiero, I.; Michielon, A.; Campanini, B.; Faggiano, S.; Bettati, S.; Mozzarelli, A.; Spyrakis, F.; Bruno, S.
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor
2020-01-01 Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Human serine racemase is allosterically modulated by NADH and reduced nicotinamide derivatives | 1-gen-2016 | Bruno, Stefano; Marchesani, Francesco; Dellafiora, Luca; Margiotta, Marilena; Faggiano, Serena; Campanini, Barbara; Mozzarelli, Andrea | |
Structural insight into the interaction of O-acetylserine sulfhydrylase with competitive, peptidic inhibitors by Saturation Transfer Difference-NMR | 1-gen-2016 | Benoni, Roberto; Pertinhez, Thelma; Spyrakis, Francesca; Davalli, S; Pellegrino, S; Paredi, Gianluca; Pezzotti, A; Bettati, Stefano; Campanini, Barbara; Mozzarelli, Andrea | |
Insights on O-acetylserine Sulfhydrylase Structure, Function and Biopharmaceutical Applications | 1-gen-2017 | Campanini, Barbara; Mozzarelli, Andrea | |
Study of DNA binding and bending by Bacillus subtilis GabR, a PLP-dependent transcription factor | 1-gen-2017 | Amidani, Davide; Tramonti, Angela; Canosa, ANDREA VALERIA; Campanini, Barbara; Maggi, Stefano; Milano, Teresa; DI SALVO, MARTINO LUIGI; Pascarella, Stefano; Contestabile, Roberto; Bettati, Stefano; Rivetti, Claudio | |
Activation of an anti-bacterial toxin by the biosynthetic enzyme CysK: mechanism of binding, interaction specificity and competition with cysteine synthase | 1-gen-2017 | Benoni, Roberto; Beck, Christina M.; Garza-Sánchez, Fernando; Bettati, Stefano; Mozzarelli, Andrea; Hayes, Christopher S.; Campanini, Barbara | |
Modulation of Escherichia coli serine acetyltransferase catalytic activity in the cysteine synthase complex | 1-gen-2017 | Benoni, Roberto; DE BEI, Omar; Paredi, Gianluca; Hayes, Christopher S.; Franko, Nina; Mozzarelli, Andrea; Bettati, Stefano; Campanini, Barbara | |
Magnesium and calcium ions differentially affect human serine racemase activity and modulate its quaternary equilibrium toward a tetrameric form | 1-gen-2017 | Bruno, Stefano; Margiotta, Marilena; Marchesani, Francesco; Paredi, Gianluca; Orlandi, Valentina; Faggiano, Serena; Ronda, Luca; Campanini, Barbara; Mozzarelli, Andrea | |
Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets | 1-gen-2018 | Magalhães, Joana; Annunziato, Giannamaria; Franko, Nina; Pieroni, Marco; Campanini, Barbara; Bruno, Agostino; Costantino, Gabriele | |
Glutamine 89 is a key residue in the allosteric modulation of human serine racemase activity by ATP | 1-gen-2018 | Canosa, Andrea V; Faggiano, Serena; Marchetti, Marialaura; Armao, Stefano; Bettati, Stefano; Bruno, Stefano; Percudani, Riccardo; Campanini, Barbara; Mozzarelli, Andrea | |
Insight into GFPmut2 pH Dependence by Single Crystal Microspectrophotometry and X-ray Crystallography | 1-gen-2018 | Lolli, Graziano; Raboni, Samanta; Pasqualetto, Elisa; Benoni, Roberto; Campanini, Barbara; Ronda, Luca; Mozzarelli, Andrea; Bettati, Stefano; Battistutta, Roberto | |
Inhibition of O-acetylserine sulfhydrylase by fluoroalanine derivatives | 1-gen-2018 | Franko, N.; Grammatoglou, K.; Campanini, B.; Costantino, G.; Jirgensons, A.; Mozzarelli, A. | |
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design | 1-gen-2018 | Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara | |
Human serine racemase is nitrosylated at multiple sites | 1-gen-2018 | Marchesani, Francesco; Bruno, Stefano; Paredi, Gianluca; Raboni, Samanta; Campanini, Barbara; Mozzarelli, Andrea | |
The Energy Landscape of Human Serine Racemase | 1-gen-2019 | Raboni, Samanta; Marchetti, Marialaura; Faggiano, Serena; Campanini, Barbara; Bruno, Stefano; Marchesani, Francesco; Margiotta, Marilena; Mozzarelli, Andrea | |
Interaction of human hemoglobin and semi-hemoglobins with the Staphylococcus aureus hemophore IsdB: a kinetic and mechanistic insight | 1-gen-2019 | Gianquinto, E.; Moscetti, I.; De Bei, O.; Campanini, B.; Marchetti, M.; Luque, F. J.; Cannistraro, S.; Ronda, L.; Bizzarri, A. R.; Spyrakis, F.; Bettati, S. | |
Combination of SAXS and protein painting discloses the three-dimensional organization of the bacterial cysteine synthase complex, a potential target for enhancers of antibiotic action | 1-gen-2019 | Rosa, B.; Marchetti, M.; Paredi, G.; Amenitsch, H.; Franko, N.; Benoni, R.; Giabbai, B.; De Marino, M. G.; Mozzarelli, A.; Ronda, L.; Storici, P.; Campanini, B.; Bettati, S. | |
Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms | 1-gen-2019 | Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Nikitjuka, Anna; Mozzarelli, Andrea; Bettati, Stefano; Karawajczyk, Anna; Jirgensons, Aigars; Campanini, Barbara; Costantino, Gabriele | |
More than a Confinement: “Soft” and “Hard” Enzyme Entrapment Modulates Biological Catalyst Function | 1-gen-2019 | Cottone, Grazia; Giuffrida, Sergio; Bettati, Stefano; Bruno, Stefano; Campanini, Barbara; Marchetti, Marialaura; Abbruzzetti, Stefania; Viappiani, Cristiano; Cupane, Antonio; Mozzarelli, Andrea; Ronda, Luca | |
The allosteric interplay between S-nitrosylation and glycine binding controls the activity of human serine racemase | 1-gen-2020 | Marchesani, F.; Gianquinto, E.; Autiero, I.; Michielon, A.; Campanini, B.; Faggiano, S.; Bettati, S.; Mozzarelli, A.; Spyrakis, F.; Bruno, S. | |
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor | 1-gen-2020 | Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G. |
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