A microwave-assisted synthesis of solid-supported reagents for the acylation of amines has been developed, and the same methodology has been successfully applied to the preparation of acylating agents anchored on different solid supports. Similarly, alcohols, phenols, and thiophenols have been easily acylated using these reagents under microwave irradiation.
Microwave-Assisted Acylation of Amines, Alcohols, and Phenols by the Use of Solid-Supported Reagents (SSRs) / Elena Petricci;Claudia Mugnaini;Marco Radi;Federico Corelli;Maurizio Botta. - In: JOURNAL OF ORGANIC CHEMISTRY. - ISSN 0022-3263. - 69(2004), pp. 7880-7887. [10.1021/jo048837q]