PIOMELLI, DANIELE
PIOMELLI, DANIELE
Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines
2020-01-01 Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele.
Chapter 9: Natural and Synthetic Agents That Target Intracellular Monoacylglycerol Lipase (MGL) Activity
2021-01-01 Scalvini, L.; Rivara, S.; Jung, K. -M.; Mor, M.; Piomelli, D.
Different roles for the acyl chain and the amine leaving group in the substrate selectivity of N-Acylethanolamine acid amidase
2021-01-01 Ghidini, A.; Scalvini, L.; Palese, F.; Lodola, A.; Mor, M.; Piomelli, D.
Enhancement of peripheral fatty acyl ethanolamide signaling prevents stress‑induced social avoidance and anxiety‑like behaviors in male rats
2023-01-01 Carnevali, Luca; Barbetti, Margherita; Fotio, Yannick; Ferlenghi, Francesca; Vacondio, Federica; Mor, Marco; Piomelli, Daniele; Sgoifo, Andrea
Identification of bivalent ligands with melatonin receptor agonist and fatty acid amide hydrolase (FAAH) inhibitory activity that exhibit ocular hypotensive effect in the rabbit
2018-01-01 Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, Andrea; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S.
N-Acylethanolamine Acid Amidase (NAAA): Mechanism of Palmitoylethanolamide Hydrolysis Revealed by Mechanistic Simulations
2020-01-01 Scalvini, L.; Ghidini, A.; Lodola, A.; Callegari, D.; Rivara, S.; Piomelli, D.; Mor, M.
N-Acylethanolamine Acid Amidase (NAAA): Structure, Function, and Inhibition
2020-01-01 Piomelli, D; Scalvini, L; Fotio, Y; Lodola, A; Spadoni, G; Tarzia, G; Mor, M.
NAAA-regulated lipid signaling governs the transition from acute to chronic pain
2021-01-01 Fotio, Y.; Jung, K. -M.; Palese, F.; Obenaus, A.; Tagne, A. M.; Lin, L.; Rashid, T. I.; Pacheco, R.; Jullienne, A.; Ramirez, J.; Mor, M.; Spadoni, G.; Jang, C.; Hohmann, A. G.; Piomelli, D.
Pharmacokinetics, pharmacodynamics and safety studies on URB937, a peripherally restricted fatty acid amide hydrolase inhibitor, in rats
2019-01-01 Vozella, V.; Ahmed, F.; Choobchian, P.; Merrill, C. B.; Zibardi, C.; Tarzia, G.; Mor, M.; Duranti, A.; Tontini, A.; Rivara, S.; Piomelli, D.
Synthesis and characterization of the first inhibitor of: N -acylphosphatidylethanolamine phospholipase D (NAPE-PLD)
2017-01-01 Castellani, Beatrice; Diamanti, Eleonora; Pizzirani, Daniela; Tardia, Piero; Maccesi, Martina; Realini, Natalia; Magotti, Paola; Garau, Gianpiero; Bakkum, Thomas; Rivara, Silvia; Mor, Marco; Piomelli, Daniele
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines | 1-gen-2020 | Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele. | |
| Chapter 9: Natural and Synthetic Agents That Target Intracellular Monoacylglycerol Lipase (MGL) Activity | 1-gen-2021 | Scalvini, L.; Rivara, S.; Jung, K. -M.; Mor, M.; Piomelli, D. | |
| Different roles for the acyl chain and the amine leaving group in the substrate selectivity of N-Acylethanolamine acid amidase | 1-gen-2021 | Ghidini, A.; Scalvini, L.; Palese, F.; Lodola, A.; Mor, M.; Piomelli, D. | |
| Enhancement of peripheral fatty acyl ethanolamide signaling prevents stress‑induced social avoidance and anxiety‑like behaviors in male rats | 1-gen-2023 | Carnevali, Luca; Barbetti, Margherita; Fotio, Yannick; Ferlenghi, Francesca; Vacondio, Federica; Mor, Marco; Piomelli, Daniele; Sgoifo, Andrea | |
| Identification of bivalent ligands with melatonin receptor agonist and fatty acid amide hydrolase (FAAH) inhibitory activity that exhibit ocular hypotensive effect in the rabbit | 1-gen-2018 | Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, Andrea; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S. | |
| N-Acylethanolamine Acid Amidase (NAAA): Mechanism of Palmitoylethanolamide Hydrolysis Revealed by Mechanistic Simulations | 1-gen-2020 | Scalvini, L.; Ghidini, A.; Lodola, A.; Callegari, D.; Rivara, S.; Piomelli, D.; Mor, M. | |
| N-Acylethanolamine Acid Amidase (NAAA): Structure, Function, and Inhibition | 1-gen-2020 | Piomelli, D; Scalvini, L; Fotio, Y; Lodola, A; Spadoni, G; Tarzia, G; Mor, M. | |
| NAAA-regulated lipid signaling governs the transition from acute to chronic pain | 1-gen-2021 | Fotio, Y.; Jung, K. -M.; Palese, F.; Obenaus, A.; Tagne, A. M.; Lin, L.; Rashid, T. I.; Pacheco, R.; Jullienne, A.; Ramirez, J.; Mor, M.; Spadoni, G.; Jang, C.; Hohmann, A. G.; Piomelli, D. | |
| Pharmacokinetics, pharmacodynamics and safety studies on URB937, a peripherally restricted fatty acid amide hydrolase inhibitor, in rats | 1-gen-2019 | Vozella, V.; Ahmed, F.; Choobchian, P.; Merrill, C. B.; Zibardi, C.; Tarzia, G.; Mor, M.; Duranti, A.; Tontini, A.; Rivara, S.; Piomelli, D. | |
| Synthesis and characterization of the first inhibitor of: N -acylphosphatidylethanolamine phospholipase D (NAPE-PLD) | 1-gen-2017 | Castellani, Beatrice; Diamanti, Eleonora; Pizzirani, Daniela; Tardia, Piero; Maccesi, Martina; Realini, Natalia; Magotti, Paola; Garau, Gianpiero; Bakkum, Thomas; Rivara, Silvia; Mor, Marco; Piomelli, Daniele |