GOVERNA, Paolo
GOVERNA, Paolo
Dipartimento di Scienze degli Alimenti e del Farmaco
Antiviral activity of cannabidiolic acid and its methyl ester against SARS-CoV-2
2023-01-01 Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica
Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma
2024-01-01 Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity
2024-01-01 Aslan, Hakan; Renzi, Gioele; Angeli, Andrea; D'Agostino, Ilaria; Ronca, Roberto; Massardi, Maria Luisa; Tavani, Camilla; Carradori, Simone; Ferraroni, Marta; Governa, Paolo; Manetti, Fabrizio; Carta, Fabrizio; Supuran, Claudiu T.
Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation
2023-01-01 Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta
Chemical hybridization approaches applied to natural and synthetic compounds for the discovery of drugs active against neglected tropical diseases
2019-01-01 Petricci, Elena; Governa, Paolo; Manetti, Fabrizio
Enhanced mapping of small-molecule binding sites in cells
2024-01-01 Wozniak, Jacob M.; Li, Weichao; Governa, Paolo; Chen, Li-Yun; Jadhav, Appaso; Dongre, Ashok; Forli, Stefano; Parker, Christopher G.
FFAR1/GPR40: One target, different binding sites, many agonists, no drugs, but a continuous and unprofitable tug-of-war between ligand lipophilicity, activity, and toxicity
2021-01-01 Governa, Paolo; Caroleo, Maria Cristina; Carullo, Gabriele; Aiello, Francesca; Cione, Erika; Manetti, Fabrizio
Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol
2023-01-01 Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta
Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor
2025-01-01 Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco
Mantonico and pecorello grape seed extracts: chemical characterization and evaluation of in vitro wound-healing and anti-inflammatory activities
2020-01-01 Carullo, G.; Sciubba, F.; Governa, P.; Mazzotta, S.; Frattaruolo, L.; Grillo, G.; Cappello, A. R.; Cravotto, G.; Di Cocco, M. E.; Aiello, F.
Morita−Baylis−Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands
2025-01-01 Paolino, Marco; Tassone, Giusy; Governa, Paolo; Saletti, Mario; Lami, Matteo; Carletti, Riccardo; Sacchetta, Filippo; Pozzi, Cecilia; Orlandini, Maurizio; Manetti, Fabrizio; Olivucci, Massimo; Cappelli, Andrea
Phytochemical characterization and gastroprotective activity of Copaifera langsdorffii Desf. oleoresin and fruit methanolic extract
2019-01-01 Biagi, Marco; Governa, Paolo; Miraldi, Elisabetta; Magnano, Anna Rosa; Giachetti, Daniela
Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway
2021-01-01 Mazzotta, Sarah; Governa, Paolo; Borgonetti, Vittoria; Marcolongo, Paola; Nanni, Claudio; Gamberucci, Alessandra; Manetti, Fabrizio; Pessina, Federica; Carullo, Gabriele; Brizzi, Antonella; Aiello, Francesca
Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening
2022-01-01 Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena
Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view
2022-01-01 Governa, Paolo; Manetti, Fabrizio
Survey on the recent advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) inhibition by diketone and triketone derivatives and congeneric compounds: structural analysis of HPPD/inhibitor complexes and structure-activity relationship considerations
2022-01-01 Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena
The veterinary anti-parasitic selamectin Is a novel inhibitor of the mycobacterium tuberculosis DprE1 enzyme
2022-01-01 Ezquerra-Aznárez, José Manuel; Degiacomi, Giulia; Gašparovič, Henrich; Stelitano, Giovanni; Sammartino, Josè Camilla; Korduláková, Jana; Governa, Paolo; Manetti, Fabrizio; Pasca, Maria Rosalia; Chiarelli, Laurent Roberto; Ramón-García, Santiago
Zingiberene, a non-zinc-binding class I HDAC inhibitor: a novel strategy for the management of neuropathic pain
2023-01-01 Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Antiviral activity of cannabidiolic acid and its methyl ester against SARS-CoV-2 | 1-gen-2023 | Tamburello, Martina; Salamone, Stefano; Anceschi, Lisa; Governa, Paolo; Brighenti, Virginia; Morellini, Alice; Rossini, Giada; Manetti, Fabrizio; Gallinella, Giorgio; Pollastro, Federica; Pellati, Federica | |
| Applying molecular hybridization to design a new class of pyrazolo[3,4-d]pyrimidines as Src inhibitors active in hepatocellular carcinoma | 1-gen-2024 | Di Maria, Salvatore; Passannanti, Raffaele; Poggialini, Federica; Vagaggini, Chiara; Serafinelli, Alessia; Bianchi, Elena; Governa, Paolo; Botta, Lorenzo; Maga, Giovanni; Crespan, Emmanuele; Manetti, Fabrizio; Dreassi, Elena; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia | |
| Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activity | 1-gen-2024 | Aslan, Hakan; Renzi, Gioele; Angeli, Andrea; D'Agostino, Ilaria; Ronca, Roberto; Massardi, Maria Luisa; Tavani, Camilla; Carradori, Simone; Ferraroni, Marta; Governa, Paolo; Manetti, Fabrizio; Carta, Fabrizio; Supuran, Claudiu T. | |
| Cannabidiol-rich non-psychotropic Cannabis sativa L. oils attenuate peripheral neuropathy symptoms by regulation of CB2-mediated microglial neuroinflammation | 1-gen-2023 | Borgonetti, Vittoria; Anceschi, Lisa; Brighenti, Virginia; Corsi, Lorenzo; Governa, Paolo; Manetti, Fabrizio; Pellati, Federica; Galeotti, Nicoletta | |
| Chemical hybridization approaches applied to natural and synthetic compounds for the discovery of drugs active against neglected tropical diseases | 1-gen-2019 | Petricci, Elena; Governa, Paolo; Manetti, Fabrizio | |
| Enhanced mapping of small-molecule binding sites in cells | 1-gen-2024 | Wozniak, Jacob M.; Li, Weichao; Governa, Paolo; Chen, Li-Yun; Jadhav, Appaso; Dongre, Ashok; Forli, Stefano; Parker, Christopher G. | |
| FFAR1/GPR40: One target, different binding sites, many agonists, no drugs, but a continuous and unprofitable tug-of-war between ligand lipophilicity, activity, and toxicity | 1-gen-2021 | Governa, Paolo; Caroleo, Maria Cristina; Carullo, Gabriele; Aiello, Francesca; Cione, Erika; Manetti, Fabrizio | |
| Helichrysum stoechas (L.) Moench reduces body weight gain and modulates mood disorders via inhibition of silent information regulator 1 (SIRT1) by arzanol | 1-gen-2023 | Borgonetti, Vittoria; Caroli, Clarissa; Governa, Paolo; Virginia, Brighenti; Pollastro, Federica; Franchini, Silvia; Manetti, Fabrizio; Les, Francisco; López, Victor; Pellati, Federica; Galeotti, Nicoletta | |
| Light-mediated activation/deactivation control and in vitro ADME-Tox profiling of a donepezil-like Dual AChE/MAO-B Inhibitor | 1-gen-2025 | Poggialini, Federica; Governa, Paolo; Vagaggini, Chiara; Maramai, Samuele; Lamponi, Stefania; Mugnaini, Claudia; Brizzi, Antonella; Purgatorio, Rosa; De Candia, Modesto; Catto, Marco; Dreassi, Elena; Manetti, Fabrizio; Corelli, Federico; Altomare, Cosimo Damiano; Cappelli, Andrea; Paolino, Marco | |
| Mantonico and pecorello grape seed extracts: chemical characterization and evaluation of in vitro wound-healing and anti-inflammatory activities | 1-gen-2020 | Carullo, G.; Sciubba, F.; Governa, P.; Mazzotta, S.; Frattaruolo, L.; Grillo, G.; Cappello, A. R.; Cravotto, G.; Di Cocco, M. E.; Aiello, F. | |
| Morita−Baylis−Hillman Adduct Chemistry as a Tool for the Design of Lysine-Targeted Covalent Ligands | 1-gen-2025 | Paolino, Marco; Tassone, Giusy; Governa, Paolo; Saletti, Mario; Lami, Matteo; Carletti, Riccardo; Sacchetta, Filippo; Pozzi, Cecilia; Orlandini, Maurizio; Manetti, Fabrizio; Olivucci, Massimo; Cappelli, Andrea | |
| Phytochemical characterization and gastroprotective activity of Copaifera langsdorffii Desf. oleoresin and fruit methanolic extract | 1-gen-2019 | Biagi, Marco; Governa, Paolo; Miraldi, Elisabetta; Magnano, Anna Rosa; Giachetti, Daniela | |
| Pinocembrin and its linolenoyl ester derivative induce wound healing activity in HaCaT cell line potentially involving a GPR120/FFA4 mediated pathway | 1-gen-2021 | Mazzotta, Sarah; Governa, Paolo; Borgonetti, Vittoria; Marcolongo, Paola; Nanni, Claudio; Gamberucci, Alessandra; Manetti, Fabrizio; Pessina, Federica; Carullo, Gabriele; Brizzi, Antonella; Aiello, Francesca | |
| Quinolines and Oxazino-quinoline derivatives as small molecule GLI1 inhibitors identified by virtual screening | 1-gen-2022 | Manetti, Fabrizio; Maresca, Luisa; Crivaro, Enrica; Pepe, Sara; Cini, Elena; Singh, Snigdha; Governa, Paolo; Maramai, Samuele; Giannini, Giuseppe; Stecca, Barbara; Petricci, Elena | |
| Recent research results have converted gp120 binders to a therapeutic option for the treatment of HIV-1 infection. A medicinal chemistry point of view | 1-gen-2022 | Governa, Paolo; Manetti, Fabrizio | |
| Survey on the recent advances in 4-Hydroxyphenylpyruvate Dioxygenase (HPPD) inhibition by diketone and triketone derivatives and congeneric compounds: structural analysis of HPPD/inhibitor complexes and structure-activity relationship considerations | 1-gen-2022 | Governa, Paolo; Bernardini, Giulia; Braconi, Daniela; Manetti, Fabrizio; Santucci, Annalisa; Petricci, Elena | |
| The veterinary anti-parasitic selamectin Is a novel inhibitor of the mycobacterium tuberculosis DprE1 enzyme | 1-gen-2022 | Ezquerra-Aznárez, José Manuel; Degiacomi, Giulia; Gašparovič, Henrich; Stelitano, Giovanni; Sammartino, Josè Camilla; Korduláková, Jana; Governa, Paolo; Manetti, Fabrizio; Pasca, Maria Rosalia; Chiarelli, Laurent Roberto; Ramón-García, Santiago | |
| Zingiberene, a non-zinc-binding class I HDAC inhibitor: a novel strategy for the management of neuropathic pain | 1-gen-2023 | Borgonetti, Vittoria; Governa, Paolo; Manetti, Fabrizio; Galeotti, Nicoletta |