SCALVINI, Laura

SCALVINI, Laura  

Dipartimento di Scienze degli Alimenti e del Farmaco  

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A sulfonyl fluoride derivative inhibits EGFR L858R/T790M/C797S by covalent modification of the catalytic lysine 1-gen-2021 Ferlenghi, F; Scalvini, L; Vacondio, F; Castelli, R; Bozza, N; Marseglia, G; Rivara, S; Lodola, A; La Monica, S; Minari, R; Petronini, Pg; Alfieri, R; Tiseo, M; Mor, M.
Amino acid derivatives as palmitoylethanolamide prodrugs: Synthesis, in vitro metabolism and in vivo plasma profile in rats 1-gen-2015 Vacondio, Federica; Bassi, Michele; Silva, Claudia; Castelli, Riccardo; Carmi, Caterina; Scalvini, Laura; Lodola, Alessio; Vivo, Valentina; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco; Rivara, Silvia
Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines 1-gen-2020 Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele.
Chapter 9: Natural and Synthetic Agents That Target Intracellular Monoacylglycerol Lipase (MGL) Activity 1-gen-2021 Scalvini, L.; Rivara, S.; Jung, K. -M.; Mor, M.; Piomelli, D.
Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria 1-gen-2020 Elisi, GIAN MARCO; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Comparative Analysis of Virtual Screening Approaches in the Search for Novel EphA2 Receptor Antagonists 1-gen-2015 Callegari, Donatella; Pala, Daniele; Scalvini, Laura; Tognolini, Massimiliano; Incerti, Matteo; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Conformational Propensity and Biological Studies of Proline Mutated LR Peptides Inhibiting Human Thymidylate Synthase and Ovarian Cancer Cell Growth 1-gen-2018 Saxena, P; Severi, L; Santucci, M; Taddia, ; Ferrari, S; Luciani, R; Marverti, G; Marraccini, C; Tondi, D; Mor, M; Scalvini, L; Vitiello, S; Losi, L; Fonda, S; Pacifico, S; Guerrini, R; D'Arca, D; Ponterini, G; Costi, Mp
Design and SAR Analysis of Covalent Inhibitors Driven by Hybrid QM/MM Simulations 1-gen-2020 Lodola, A.; Callegari, D.; Scalvini, L.; Rivara, S.; Mor, M.
Different roles for the acyl chain and the amine leaving group in the substrate selectivity of N-Acylethanolamine acid amidase 1-gen-2021 Ghidini, A.; Scalvini, L.; Palese, F.; Lodola, A.; Mor, M.; Piomelli, D.
Drug-gut microbiota metabolic interactions: the case of UniPR1331, selective antagonist of the Eph-ephrin system, in mice 1-gen-2020 Ferlenghi, F.; Castelli, R.; Scalvini, L.; Giorgio, C.; Corrado, M.; Tognolini, M.; Mor, M.; Lodola, A.; Vacondio, F.
Fatty Acid Amide Hydrolase (FAAH), Acetylcholinesterase (AChE), and Butyrylcholinesterase (BuChE): Networked Targets for the Development of Carbamates as Potential Anti-Alzheimer's Disease Agents 1-gen-2016 Montanari, Serena; Scalvini, Laura; Bartolini, Manuela; Belluti, Federica; Gobbi, Silvia; Andrisano, Vincenza; Ligresti, Alessia; Di Marzo, Vincenzo; Rivara, Silvia; Mor, Marco; Bisi, Alessandra; Rampa, Angela
Fighting tertiary mutations in EGFR-driven lung-cancers: Current advances and future perspectives in medicinal chemistry 1-gen-2021 Scalvini, Laura; Castelli, Riccardo; La Monica, Silvia; Tiseo, Marcello; Alfieri, Roberta
Free-Energy Simulations Support a Lipophilic Binding Route for Melatonin Receptors 1-gen-2022 Elisi, GIAN MARCO; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Rivara, Silvia
Free-energy studies reveal a possible mechanism for oxidation-dependent inhibition of MGL 1-gen-2016 Scalvini, Laura; Vacondio, Federica; Bassi, Michele; Pala, Daniele; Lodola, Alessio; Rivara, Silvia; Jung, Kwang Mook; Piomelli, Daniele; Mor, Marco
Identification of a Quinone Derivative as a YAP/TEAD Activity Modulator from a Repurposing Library 1-gen-2022 Lauriola, Angela; Uliassi, Elisa; Santucci, Matteo; Laura Bolognesi, Maria; Mor, Marco; Scalvini, Laura; Elisi, GIAN MARCO; Gozzi, Gaia; Tagliazucchi, Lorenzo; Marverti, Gaetano; Ferrari, Stefania; Losi, Lorena; D’Arca, Domenico; Paola Costi, Maria
Identification of bivalent ligands with melatonin receptor agonist and fatty acid amide hydrolase (FAAH) inhibitory activity that exhibit ocular hypotensive effect in the rabbit 1-gen-2018 Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, Andrea; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S.
In silico drug discovery of melatonin receptor ligands with therapeutic potential 1-gen-2022 Elisi, G. M.; Scalvini, L.; Lodola, A.; Bedini, A.; Spadoni, G.; Rivara, S.
Mechanistic Modeling of Lys745 Sulfonylation in EGFR C797S Reveals Chemical Determinants for Inhibitor Activity and Discriminates Reversible from Irreversible Agents 1-gen-2023 Arafet, Kemel; Scalvini, Laura; Galvani, Francesca; Martí, Sergio; Moliner, Vicent; Mor, Marco; Lodola, Alessio
Mechanistic Modeling of Monoglyceride Lipase Covalent Modification Elucidates the Role of Leaving Group Expulsion and Discriminates Inhibitors with High and Low Potency 1-gen-2022 Galvani, F.; Scalvini, L.; Rivara, S.; Lodola, A.; Mor, M.
Molecular Determinants of EphA2 and EphB2 Antagonism Enable the Design of Ligands with Improved Selectivity 1-gen-2023 Guidetti, Lorenzo; Zappia, Alfonso; Scalvini, Laura; Ferrari, Francesca Romana; Giorgio, Carmine; Castelli, Riccardo; Galvani, Francesca; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Urbinati, Chiara; Rusnati, Marco; Tognolini, Massimiliano; Lodola, Alessio