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UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations. 1-gen-2014 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Russo, Simonetta; Pala, Daniele; Pasquale, Eb; Zanotti, Ilaria; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano
Target Hopping as a Useful Tool for the Identification of Novel EphA2 Protein–Protein Antagonists 1-gen-2014 Tognolini, Massimiliano; Incerti, Matteo; Pala, Daniele; Russo, Simonetta; Castelli, Riccardo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Lodola, Alessio
Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties 1-gen-2014 Spadoni, G.; Bedini, A.; Bartolucci, S.; Pala, Daniele; Mor, Marco; Riccioni, T.; Borsini, F.; Cabri, W.; Celona, D.; Marzi, M.; Tarzia, G.; Rivara, Silvia; Minetti, P.
Synthesis and characterization of new bivalent agents as melatonin- and histamine h3-ligands. 1-gen-2014 Pala, Daniele; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Flammini, Lisa; Barocelli, Elisabetta; Lucini, V; Scaglione, F; Bartolucci, S; Bedini, A; Rivara, Silvia; Spadoni, G.
ST7612AA1, a thioacetate-ω(γ-lactam carboxamide) derivative selected from a novel generation of oral HDAC inhibitors 1-gen-2014 Giannini, Giuseppe; Vesci, Loredana; Battistuzzi, Gianfranco; Vignola, Davide; Milazzo, Ferdinando M; Guglielmi, Mario Berardino; Barbarino, Marcella; Santaniello, Mosè; Fantò, Nicola; Mor, Marco; Rivara, Silvia; Pala, Daniele; Taddei, Maurizio; Pisano, Claudio; Cabri, Walter
Synthesis, structure and inhibitory activity of a stereoisomer of oseltamivir carboxylate 1-gen-2014 Sartori, Andrea; L., Dell’Amico; Battistini, Lucia; Curti, Claudio; Rivara, Silvia; Pala, Daniele; P. S., Kerry; Pelosi, Giorgio; Casiraghi, Giovanni; G., Rassu; Zanardi, Franca
Development of an orally bioavailable small molecule targeting Eph-ephrin system: in vitro and in vivo anticancer activity. 1-gen-2015 Tognolini, Massimiliano; Giorgio, Carmine; Festuccia, C; Rusnati, M; Chiodelli, P; Incerti, Matteo; Pala, Daniele; Callegari, Donatella; Bertoni, Simona; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta
In vitro and in vivo efficacy of an orally bioavailable antagonist of Eph-ephrin system in tumor angiogenesis and growth 1-gen-2015 Giorgio, Carmine; Castelli, Riccardo; Hassan Mohamed, I.; Incerti, Matteo; Vacondio, Federica; Bertoni, Simona; Festuccia, C.; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano
Multiple approaches for the discovery and development of small molecules targeting Eph-ephrin protein-protein interaction 1-gen-2015 Tognolini, Massimiliano; Giorgio, Carmine; Incerti, Matteo; Castelli, Riccardo; Festuccia, C.; Rusnati, M.; Vacondio, Federica; Russo, Simonetta; Pala, Daniele; Callegari, Donatella; Mor, Marco; Bertoni, Simona; Ballabeni, Vigilio; Lodola, Alessio; Barocelli, Elisabetta
Therapeutic uses of melatonin and melatonin derivatives: a patent review (2012 - 2014) 1-gen-2015 Rivara, Silvia; Pala, Daniele; Bedini, Annalida; Spadoni, Gilberto
Comparative Analysis of Virtual Screening Approaches in the Search for Novel EphA2 Receptor Antagonists 1-gen-2015 Callegari, Donatella; Pala, Daniele; Scalvini, Laura; Tognolini, Massimiliano; Incerti, Matteo; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines 1-gen-2015 Spadoni, Gilberto; Bedini, Annalida; Lucarini, Simone; Mari, Michele; Caignard, Daniel Henri; Boutin, Jean A.; Delagrange, Philippe; Lucini, Valeria; Scaglione, Francesco; Lodola, Alessio; Zanardi, Franca; Pala, Daniele; Mor, Marco; Rivara, Silvia
Δ5-Cholenoyl-amino acids as selective and orally available antagonists of the Eph-ephrin system 1-gen-2015 Castelli, Riccardo; Tognolini, Massimiliano; Vacondio, Federica; Incerti, Matteo; Pala, Daniele; Callegari, Donatella; Bertoni, Simona; Giorgio, Carmine; Hassan Mohamed, I; Zanotti, Ilaria; Bugatti, A; Rusnati, M; Festuccia, C; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Kinetic analysis and molecular modeling of the inhibition mechanism of roneparstat (SST0001) on human heparanase 1-gen-2016 Pala, Daniele; Rivara, Silvia; Mor, Marco; Milazzo, Ferdinando Maria; Roscilli, Giuseppe; Pavoni, Emiliano; Giannini, Giuseppe
Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return 1-gen-2016 Russo, Simonetta; Callegari, Donatella; Incerti, Matteo; Pala, Daniele; Giorgio, Carmine; Brunetti, Jlenia; Bracci, Luisa; Vicini, Paola; Barocelli, Elisabetta; Capoferri, Luigi; Rivara, Silvia; Tognolini, Massimiliano; Mor, Marco; Lodola, Alessio
Biochemical characterization of EphA2 antagonists with improved physico-chemical properties by cell-based assays and surface plasmon resonance analysis 1-gen-2016 Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Bugatti, Antonella; Vacondio, Federica; Barocelli, Elisabetta; Mor, Marco; Pala, Daniele; Hassan Mohamed, Iftiin; Gioiello, Antimo; Rusnati, Marco; Lodola, Alessio; Tognolini, Massimiliano
Free-energy studies reveal a possible mechanism for oxidation-dependent inhibition of MGL 1-gen-2016 Scalvini, Laura; Vacondio, Federica; Bassi, Michele; Pala, Daniele; Lodola, Alessio; Rivara, Silvia; Jung, Kwang Mook; Piomelli, Daniele; Mor, Marco
Metadynamics Simulations Distinguish Short- and Long-Residence-Time Inhibitors of Cyclin-Dependent Kinase 8. 1-gen-2017 Callegari, Donatella; Lodola, Alessio; Pala, Daniele; Rivara, Silvia; Mor, Marco; Rizzi, A; Capelli A., M.
Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs 1-gen-2017 Lodola, Alessio; Bertolini, S; Biagetti, M; Capacchi, S; Facchinetti, F; Gallo, Pm; Pappani, A; Mor, Marco; Pala, Daniele; Rivara, Silvia; Visentini, F; Corsi, M; Capelli A., M.
Metadynamics for perspective drug design: Computationally driven synthesis of new protein-protein interaction inhibitors targeting the EphA2 receptor 1-gen-2017 Incerti, Matteo; Russo, Simonetta; Callegari, Donatella; Pala, Daniele; Giorgio, Carmine; Zanotti, Ilaria; Barocelli, Elisabetta; Vicini, Paola; Vacondio, Federica; Rivara, Silvia; Castelli, Riccardo; Tognolini, Massimiliano; Lodola, Alessio
Mostrati risultati da 21 a 40 di 42
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