Sfoglia per Autore
Synthesis of 6,6-Dicarboxy-3,4-methano-L-proline, a New Constrained Glutamate Analog Endowed with Neuroprotective Properties
1996-01-01 M., Marinozzi; B., Natalini; Costantino, Gabriele; R., Pellicciari; V., Bruno; F., Nicoletti
Dirhodium(II)-tetraacetate-Mediated Decomposition of Ethyldiazo- acetate and Ethyldiazomalonate in the Presence of Fullerene. A New Procedure for the Selective Synthesis of [6-6]-Closed Methanofullerenes
1997-01-01 R., Pellicciari; D., Annibali; Costantino, Gabriele; M., Marinozzi; B., Natalini
Synthesis, preliminary evaluation and molecular modeling studies of new, conformationally constrained analogues of the competitive NMDA receptor antagonist 4-(phosphonomethyl)-2-piperidinecarboxylic acid (CGS 19755).
1997-01-01 Pellicciari, R; Marinozzi, M; Natalini, B; Costantino, Gabriele; Lankin, Dc; Snyder, Jp; Monahan, Jb
Regulation of Biliary Bicarbonate Secretion by Bile Salts
1997-01-01 C., Clerici; G., Gentili; A., Errico; F., Camilleri; F., Brasacchio; R., Pellicciari; Costantino, Gabriele; L., Mattoli; D., Annibali; A., Morelli
alfa-Diazocarbonyl Chemistry - Target Driven Applications
1998-01-01 R., Pellicciari; Costantino, Gabriele; M., Marinozzi; L., Mattoli; B., Natalini
Metabotropic glutamate receptors: new ligads and molecular modelling studies
1998-01-01 R., Pellicciari; Costantino, Gabriele; M., Marinozzi; B., Natalini; C., Thomsen; F., Moroni
Synthesis and preliminary evaluation of (S)-2-(4'-carboxycubyl)glycine, a new selective mGluR1 antagonist.
1998-01-01 Pellicciari, R; Costantino, Gabriele; Giovagnoni, E; Mattoli, L; Brabet, I; Pin, Jp
Modulation of glutamate receptor pathways in the search for new neuroprotective agents.
1998-01-01 Pellicciari, R; Costantino, Gabriele; Marinozzi, M; Natalini, B.
Pharmacophore models of group I and group II metabotropic glutamate receptor agonists. Analysis of conformational, steric, and topological parameters affecting potency and selectivity
1999-01-01 Costantino, Gabriele; Pellicciari, R; Macchiarulo, A.
(2R,1'S,2'R,3'S)-2-(2'-Carboxy-3'-phenylcyclopropyl)glycine (PCCG-13), the first potent and selective competitive antagonist of phospholipase D-coupled metabotropic glutamate receptors: asymmetric synthesis and preliminary biological properties
1999-01-01 Pellicciari, R; Marinozzi, M; Costantino, Gabriele; Natalini, B; Moroni, F; PELLEGRINI GIAMPIETRO, D.
Chromatographic separation and evaluation of the lipophilicity by reversed phase HPLC chromatography of fullerene C60 derivatives
1999-01-01 Natalini, B; Capodiferro, V; Mattoli, L; Marinozzi, M; Costantino, Gabriele; Pellicciari, R.
Metabotropic G-protein-coupled glutamate receptors as therapeutic targets
1999-01-01 Pellicciari, R; Costantino, Gabriele
Modeling of amino-terminal domains of group I metabotropic glutamate receptors: structural motifs affecting ligand selectivity
1999-01-01 Costantino, Gabriele; Macchiarulo, A; Pellicciari, R.
Metabotropic glutamate receptors: a structural view point
2000-01-01 Pellicciari, R; Costantino, Gabriele; Macchiarulo, A.
Synthesis, molecular modeling and preliminary biological evaluation of 1-amino-3-phosphono-3-cyclopentene-1-carboxylic acid and 1-amino-3-phosphono-2-cyclopentene-1-carboxylic acid, two novel agonists of metabotropic glutamate receptors of group III.
2000-01-01 Amori, L; Marinozzi, M; Pellicciari, R; Gasparini, F; Flor, Pj; Kuhn, R; Costantino, Gabriele
Evaluation of hydrophobic/hydrophilic balance of bile acids by comparative molecular field analysis (CoMFA).
2000-01-01 Costantino, Gabriele; Natalini, B; Pellicciari, R.
Synthesis and preliminary biological evaluation at the glycineB site of (+) and (-)-oxetanylglycine, a novel non proteinogenic aminoacid
2001-01-01 Teran, Mc; Costantino, Gabriele; Marinozzi, M; Pellicciari, R.
QSAR and molecular modeling studies of baclofen analogues as GABA(B) agonists. Insights into the role of the aromatic moiety in GABA(B) binding and activation
2001-01-01 Macchiarulo, A; ENTRENA GUADIX, A; Costantino, Gabriele
Design, synthesis and preliminary evaluation of novel 3'-substituted carboxycyclopropylglycines as antagonists at group 2 metabotropic glutamate receptors
2001-01-01 Pellicciari, R; Marinozzi, M; Macchiarulo, A; Amori, L; JOSEF FLOR, P; Gasparini, F; Kuhn, R; Costantino, Gabriele
Design, Synthesis and Preliminary Evaluation of Novel 3’-Substituted Carboxycyclopropylglycines as Antagonists at Group 2 Metabotropic Glutamate Receptors
2001-01-01 R., Pellicciari; Costantino, Gabriele; M., Marinozzi; A., Macchiarulo; Amori, Laura; P. J., Flor; F., Gasparini; R., Kuhn; S., Urwyler
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