Sfoglia per Autore
QSAR study of 2-aminobenzimidazole derivatives as H3 antagonists
2001-01-01 Zuliani, Valentina; Mor, Marco; Rivara, Silvia; F., Bordi; Rivara, Mirko; D., Anceschi; Vacondio, Federica; Ballabeni, Vigilio; Bertoni, Simona; Barocelli, Elisabetta; P. V. P. L. A. Z. Z., I.
Development of a GPCR model for SAR interpretation of classical and new H3 antagonists
2003-01-01 S., Lorenzi; Mor, Marco; F., Bordi; Rivara, Silvia; Zuliani, Valentina; Rivara, Mirko; Bertoni, Simona; P. V., Plazzi
Antioxidant and cytoprotective activity of indole derivatives related to melatonin
2003-01-01 Mor, Marco; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Silva, Claudia; Vacondio, Federica; Rivara, Mirko; Plazzi, Pier Vincenzo; Franceschini, D.; Zusso, M.; Giusti, P.
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays
2003-01-01 Zuliani, Valentina; Bordi, Fabrizio; Rivara, Mirko; Silva, Claudia; Vacondio, Federica; Morini, Giovanni; Rivara, Silvia; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Magnanini, F.; Plazzi, Pier Vincenzo
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists
2004-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors
2004-01-01 Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B.
Cognition enhancing effect in rats of a selected histamine H3 receptor antagonist with good brain penetration
2005-01-01 Barocelli, Elisabetta; Ballabeni, Vigilio; Flammini, Lisa; Bertoni, Simona; Tognolini, Massimiliano; Chiavarini, Milena; Zuliani, Valentina; Rivara, Mirko; Vacondio, Federica; Impicciatore, Mariannina
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists
2005-01-01 Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series
2006-01-01 Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold.
2006-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity
2006-01-01 Spadoni, G; Diamantini, G; Bedini, A; Tarzia, G; Vacondio, Federica; Silva, Claudia; Rivara, Mirko; Mor, Marco; Plazzi, Pier Vincenzo; Zusso, M; Franceschini, D; Giusti, P.
A Practical Synthesis of 2,4(5)-Diarylimidazoles from Simple Building Blocks
2007-01-01 Zuliani, Valentina; Cocconcelli, G.; Fantini, M.; Ghiron, C.; Rivara, Mirko
2,4(5)-Diarylimidazoles: Synthesis and Biological Evaluation of a New Class of Sodium Channel Blockers against hNav1.2
2008-01-01 Rivara, Mirko; Baheti, A. R.; Fantini, M.; Cocconcelli, G.; Ghiron, C.; Kalmar, C. L.; Singh, N.; Merrick, E. C.; Patel, M. K.; Zuliani, Valentina
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity.
2008-01-01 Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Saccani, Francesca; Domenichini, Giuseppe; Morini, Giovanni; Comini, Mara; Rivara, Mirko; Barocelli, Elisabetta
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity.
2008-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor.
2008-01-01 Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma.
2008-01-01 Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships
2009-01-01 Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K.
Chiral NMR discrimination of the diastereoisomeric salts of the H(3)-antagonist 2-[3-(1H-imidazol-4-ylmethyl)piperidin-1-yl]-1H-benzimidazole.
2009-01-01 Rivara, Mirko; Zuliani, Valentina; Fantini, M; Dallaturca, E; Mor, Marco
Anticonvulsant Activity of 2,4(5)-Diarylimidazoles in Mice and Rat Models
2009-01-01 Rivara, Mirko; M., Fantini; Zuliani, Valentina; M. K., Patel
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
QSAR study of 2-aminobenzimidazole derivatives as H3 antagonists | 1-gen-2001 | Zuliani, Valentina; Mor, Marco; Rivara, Silvia; F., Bordi; Rivara, Mirko; D., Anceschi; Vacondio, Federica; Ballabeni, Vigilio; Bertoni, Simona; Barocelli, Elisabetta; P. V. P. L. A. Z. Z., I. | |
Development of a GPCR model for SAR interpretation of classical and new H3 antagonists | 1-gen-2003 | S., Lorenzi; Mor, Marco; F., Bordi; Rivara, Silvia; Zuliani, Valentina; Rivara, Mirko; Bertoni, Simona; P. V., Plazzi | |
Antioxidant and cytoprotective activity of indole derivatives related to melatonin | 1-gen-2003 | Mor, Marco; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Silva, Claudia; Vacondio, Federica; Rivara, Mirko; Plazzi, Pier Vincenzo; Franceschini, D.; Zusso, M.; Giusti, P. | |
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays | 1-gen-2003 | Zuliani, Valentina; Bordi, Fabrizio; Rivara, Mirko; Silva, Claudia; Vacondio, Federica; Morini, Giovanni; Rivara, Silvia; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Magnanini, F.; Plazzi, Pier Vincenzo | |
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists | 1-gen-2004 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo | |
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors | 1-gen-2004 | Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B. | |
Cognition enhancing effect in rats of a selected histamine H3 receptor antagonist with good brain penetration | 1-gen-2005 | Barocelli, Elisabetta; Ballabeni, Vigilio; Flammini, Lisa; Bertoni, Simona; Tognolini, Massimiliano; Chiavarini, Milena; Zuliani, Valentina; Rivara, Mirko; Vacondio, Federica; Impicciatore, Mariannina | |
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists | 1-gen-2005 | Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series | 1-gen-2006 | Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo | |
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. | 1-gen-2006 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity | 1-gen-2006 | Spadoni, G; Diamantini, G; Bedini, A; Tarzia, G; Vacondio, Federica; Silva, Claudia; Rivara, Mirko; Mor, Marco; Plazzi, Pier Vincenzo; Zusso, M; Franceschini, D; Giusti, P. | |
A Practical Synthesis of 2,4(5)-Diarylimidazoles from Simple Building Blocks | 1-gen-2007 | Zuliani, Valentina; Cocconcelli, G.; Fantini, M.; Ghiron, C.; Rivara, Mirko | |
2,4(5)-Diarylimidazoles: Synthesis and Biological Evaluation of a New Class of Sodium Channel Blockers against hNav1.2 | 1-gen-2008 | Rivara, Mirko; Baheti, A. R.; Fantini, M.; Cocconcelli, G.; Ghiron, C.; Kalmar, C. L.; Singh, N.; Merrick, E. C.; Patel, M. K.; Zuliani, Valentina | |
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity. | 1-gen-2008 | Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Saccani, Francesca; Domenichini, Giuseppe; Morini, Giovanni; Comini, Mara; Rivara, Mirko; Barocelli, Elisabetta | |
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. | 1-gen-2008 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. | 1-gen-2008 | Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. | 1-gen-2008 | Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta | |
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships | 1-gen-2009 | Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K. | |
Chiral NMR discrimination of the diastereoisomeric salts of the H(3)-antagonist 2-[3-(1H-imidazol-4-ylmethyl)piperidin-1-yl]-1H-benzimidazole. | 1-gen-2009 | Rivara, Mirko; Zuliani, Valentina; Fantini, M; Dallaturca, E; Mor, Marco | |
Anticonvulsant Activity of 2,4(5)-Diarylimidazoles in Mice and Rat Models | 1-gen-2009 | Rivara, Mirko; M., Fantini; Zuliani, Valentina; M. K., Patel |
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