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In pursuit of natural product leads: Synthesis and biological evaluation of 2-[3-hydroxy-2-[(3-hydroxypyridine-2-carbonyl)amino]phenyl]benzoxazole-4- carboxylic acid (A-33853) and its analogues: Discovery of N-(2-benzoxazol-2- ylphenyl)benzamides as novel antileishmanial chemotypes 1-gen-2008 Tipparaju, Suresh K.; Joyasawal, Sipak; Pieroni, Marco; Kaiser, Marcel; Brun, Reto; Kozikowski, Alan P.
Synthesis, biological evaluation, and structure-activity relationships for 5-[(E)-2-arylethenyl]-3-isoxazolecarboxylic acid alkyl ester derivatives as valuable antitubercular chemotypes 1-gen-2009 Pieroni, Marco; Lilienkampf, Annamaria; Baojie, Wan; Yuehong, Wang; Franzblau, Scott G.; Kozikowski, Alan P.
From serendipity to rational antituberculosis drug discovery of mefloquine-isoxazole carboxylic acid esters 1-gen-2009 Mao, Jialin; Yuan, Hai; Wang, Yuehong; Wan, Baojie; Pieroni, Marco; Huang, Qingqing; Van Breemen, Richard B.; Kozikowski, Alan P; Franzblau, Scott G.
From 6-aminoquinolone antibacterials to 6-amino-7- thiopyranopyridinylquinolone ethyl esters as inhibitors of staphylococcus aureus multidrug efflux pumps 1-gen-2010 Pieroni, Marco; Dimovska, Mirjana; Brincat, Jean Pierre; Sabatini, Stefano; Carosati, Emanuele; Massari, Serena; Kaatz, Glenn W.; Fravolini, Arnaldo
NOC chemistry for tuberculosis - Further investigations on the structure-activity relationships of antitubercular isoxazole-3-carboxylic acid ester derivatives 1-gen-2010 Pieroni, Marco; Lilienkampf, Annamaria; Wang, Yuehong; Wan, Baojie; Cho, Sanghyun; Franzblau, Scott G.; Kozikowski, Alan P.
Rational design of 5-phenyl-3-isoxazolecarboxylic acid ethyl esters as growth inhibitors of Mycobacterium tuberculosis. A potent and selective series for further drug development 1-gen-2010 Lilienkampf, Annamaria; Pieroni, Marco; Wan, Baojie; Wang, Yuehong; Franzblau, Scott G.; Kozikowski, Alan P.
Pyrido[1,2-a]benzimidazole-Based Agents Active Against Tuberculosis (TB), Multidrug-Resistant (MDR) TB and Extensively Drug-Resistant (XDR) TB 1-gen-2011 Pieroni, Marco; Tipparaju, Suresh K.; Lun, Shichun; Song, Yang; Sturm, A. Willem; Bishai, William R; Kozikowski, Alan P.
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis 1-gen-2012 Tabarrini, Oriana; Sabatini, Stefano; Massari, Serena; Pieroni, Marco; Franzblau, Scott G.; Cecchetti, Violetta
Synthesis, biological evaluation, and structure-activity relationships of N -benzoyl-2-hydroxybenzamides as agents active against P. falciparum (K1 strain), trypanosomes, and leishmania 1-gen-2012 Stec, Jozef; Huang, Qingqing; Pieroni, Marco; Kaiser, Marcel; Fomovska, Alina; Mui, Ernest; Witola, William H.; Bettis, Samuel; Mcleod, Rima; Brun, Reto; Kozikowski, Alan P.
Synthesis and Structure-Activity Relationships of Lansine Analogues as Antileishmanial Agents 1-gen-2012 Pieroni, Marco; Girmay, Sisay; Sun, Dianqing; Sahu, Rajnish; Tekwani, Babu L.; Tan, Ghee T.
Searching for innovative quinolone-like scaffolds: Synthesis and biological evaluation of 2,1-benzothiazine 2,2-dioxide derivatives 1-gen-2012 Pieroni, Marco; Sabatini, Stefano; Massari, Serena; Kaatz, Glenn W.; Cecchetti, Violetta; Tabarrini, Oriana
Derivatives of 3-isoxazolecarboxylic acid esters - a potent and selective compound class against replicating and nonreplicating Mycobacterium tuberculosis 1-gen-2012 Lilienkampf, Annamaria; Pieroni, Marco; Franzblau, Scott G.; Bishai, William R.; Kozikowski, Alan P.
Novel N-benzoyl-2-hydroxybenzamide disrupts unique parasite secretory pathway 1-gen-2012 Fomovska, Alina; Huang, Qingqing; El Bissati, Kamal; Mui, Ernest J.; Witola, William H.; Cheng, Gang; Zhou, Ying; Sommerville, Caroline; Roberts, Craig W.; Bettis, Sam; Prigge, Sean T.; Afanador, Gustavo A.; Hickman, Mark R.; Lee, Patty J.; Leed, Susan E.; Auschwitz, Jennifer M.; Pieroni, Marco; Stec, Jozef; Muench, Stephen P.; Rice, David W.; Kozikowski, Alan P.; Mcleod, Rima
Indoleamides are active against drug-resistant mycobacterium tuberculosis 1-gen-2013 Lun, Shichun; Guo, Haidan; Onajole, Oluseye K.; Pieroni, Marco; Gunosewoyo, Hendra; Chen, Gang; Tipparaju, Suresh K.; Ammerman, Nicole C.; Kozikowski, Alan P.; Bishai, William R.
Structural analogs of huperzine A improve survival in guinea pigs exposed to soman 1-gen-2013 Gunosewoyo, Hendra; Tipparaju, Suresh K.; Pieroni, Marco; Wang, Ying; Doctor, Bhupendra P.; Nambiar, Madhusoodana P.; Kozikowski, Alan P.
Preliminary structure - Activity relationships and biological evaluation of novel antitubercular indolecarboxamide derivatives against drug-susceptible and drug-resistant Mycobacterium tuberculosis strains 1-gen-2013 Onajole, Oluseye K.; Pieroni, Marco; Tipparaju, Suresh K.; Lun, Shichun; Stec, Jozef; Chen, Gang; Gunosewoyo, Hendra; Guo, Haidan; Ammerman, Nicole C.; Bishai, William R.; Kozikowski, Alan P.
Blocking cysteine biosynthesis in Salmonella typhimurium: the moonlighting enzyme CysK as a potential antibiotic target 1-gen-2014 Bettati, Stefano; Spyrakis, F.; Benoni, Roberto; Pieroni, Marco; Costantino, Gabriele; Pecchini, C.; Zani, Franca; Mozzarelli, Andrea
Spectinamides: A challenge, a proof, and a suggestion 1-gen-2014 Viveiros, Miguel; Pieroni, Marco
Design, Synthesis and Investigation onthe Structure–Activity Relationships of N-Substituted 2-Aminothiazole Derivatives as Antitubercular Agents 1-gen-2014 Pieroni, Marco; Wan, ; B., Cho S; Franzblau, Sg; Costantino, Gabriele
Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design 1-gen-2015 Pieroni, Marco; Wan, Baojie; Zuliani, Valentina; Franzblau, Scott G.; Costantino, Gabriele; Rivara, Mirko
Mostrati risultati da 1 a 20 di 65
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