MARTINA, MARIA GRAZIA

MARTINA, MARIA GRAZIA  

Dipartimento di Scienze degli Alimenti e del Farmaco  

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4-Trifluoromethyl bithiazoles as broad-spectrum antimicrobial agents for virus-related bacterial infections or co-infections 1-gen-2024 Barbieri, Francesca; Carlen, Vincent; Martina, Maria Grazia; Sannio, Filomena; Cancade, Sacha; Perini, Cecilia; Restori, Margherita; Crespan, Emmanuele; Maga, Giovanni; Docquier, Jean-Denis; Cagno, Valeria; Radi, Marco
A Microwave‐Assisted One‐Pot Three‐Step Metal‐Free [4+2] Annulation for the Sustainable Synthesis of Highly Substituted 1,2,4‐Triazines 1-gen-2024 Rubini, Daniele; Grazia Martina, Maria; Incerti, Matteo; Barbieri, Francesca; Radi, Marco
A sustainable metal-free microwave-assisted one-pot step [4+2] annulation for the synthesis of 3,5-disubstituted 1,2,4-triazines. 1-gen-2023 Rubini, Daniele; Martina, Maria Grazia; Incerti, Matteo; Barbieri, Francesca; Radi, Marco
A sustainable one-pot three step approach for the synthesis of 3,5-disubstituted 1,2,4-triazines as versatile pharmacological tools. 1-gen-2024 Rubini, D.; Martina, M. G.; Incerti, M.; Barbieri, F.; Radi, M.
Benzofuran-2-Carboxamide Derivatives as Immunomodulatory Agents Blocking the CCL20-Induced Chemotaxis and Colon Cancer Growth 1-gen-2024 Barbieri, Francesca; Martina, MARIA GRAZIA; Giorgio, Carmine; Chiara, MARIA LINDA; Allodi, Marika; Durante, Joseph; Bertoni, Simona; Radi, Marco
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses 1-gen-2021 Martina Maria, Grazia.; Vicenti, I.; Bauer, L.; Crespan, E.; Rango, E.; Boccuto, A.; Olivieri, N.; Incerti, M.; Zwaagstra, M.; Allodi, M.; Bertoni, S.; Dreassi, E.; Zazzi, M.; van Kuppeveld, F. J. M.; Maga, G.; Radi, M.
Bithiazole inhibitors of PI4KB show broad-spectrum antiviral activity against different viral families 1-gen-2024 Martina, Maria Grazia; Carlen, Vincent; Van der Reysen, Sarah; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Radi, Marco; Cagno, Valeria
CHEMISTRY-DRIVEN OPTIMIZATION OF PURINE-BASED ANTIVIRALS FOR THE IDENTIFICATION OF NEW BROAD-SPECTRUM AGENTS 1-gen-2025 Valenti, Martina Eleonora; Martina, Maria Grazia; Vincetti, Paolo; Vicenti, Ilaria; Crespan, Emmanuele; Nencioni, Lucia; Kaptein, Suzanne J. F.; Neyts, Johan; Vanderlinden, Evelien; Schols, Dominique; De Forni, Davide; Lori, Franco; Zazzi, Maurizio; Maga, Giovanni; Radi, Marco
Combining Phenotypic and Targeted Approaches for the Identification of New Broad-Spectrum Antiviral Agents (BSAAs) 1-gen-2023 Martina, Maria Grazia
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses 1-gen-2025 Barbieri, Francesca; Martina, Maria Grazia; Pesce, Emanuela; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Rossi, Sara; Gemma, Sandra; Campiani, Giuseppe; Milite, Ciro; Pepe, Giacomo; Campiglia, Pietro; Sbardella, Gianluca; Maga, Giovanni; Cagno, Valeria; Pedemonte, Nicoletta; Radi, Marco
DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X 1-gen-2025 Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco
DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X 1-gen-2025 Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco
Development of Novel PCSK9 Inhibitors as Potential Broad-Spectrum Antivirals 1-gen-2025 Savian, Chiara; Giannessi, Lisa; Martina, Maria Grazia; Ugolotti, Martina; Papotti, Bianca; Palumbo, Marcella; Giovanna Lupo, Maria; Mattina, Beatrice; Padula, Cristina; Nicoli, Sara; Ferri, Nicola; De Forni, Davide; Lori, Franco; Cagno, Valeria; Zimetti, Francesca; Radi, Marco
DISCOVERY OF NEW TSG101 INHIBITORS BLOCKING THE BUDDING OF EBOLA AND OTHER HIGHLY PATHOGENIC VIRUSES 1-gen-2026 Valenti, Martina Eleonora; Rubini, Daniele; Parra-López, Marisa; Holzerland, Julia; Rodríguez-Martínez, Alejandro; Martina, Maria Grazia; Ramos, Maria C.; Castillo, Francisco; Harty, Ronald N.; Pérez-Sanchez, Horacio; Diederich, Sandra; Luque, Irene; Radi, Marco
Discovery of small molecule inhibitors of the Tsg101-PTAP interaction as potential host-targeted broad-spectrum antivirals. 1-gen-2024 Rubini, Daniele; Martina, Maria Grazia; Valenti, Martina Eleonora; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Harty, Ronald N.; Parra-López, Marisa; Luque, Irene; Radi, Marco
Discovery of small-molecule targeting the CCL20/CCR6 axis as first-in-class inhibitors for inflammatory bowel diseases 1-gen-2022 Martina, Maria Grazia; Giorgio, Carmine; Allodi, Marika; Palese, Simone; Barocelli, Elisabetta; Ballabeni, Vigilio; Szpakowska, Martyna; Chevigné, Andy; Piet Van Hamburg, Jan; Davelaar, Nadine; Lubberts, Erik; Bertoni, Simona; Radi, Marco
Effects of CCL20/CCR6 modulators in a T cell adoptive transfer model of colitis 1-gen-2025 Allodi, M.; Flammini, L.; Giorgio, C.; Martina, M. G.; Barbieri, F.; Ballabeni, V.; Barocelli, E.; Radi, M.; Bertoni, S.
Harnessing prebiotic formamide chemistry: a novel platform for antiviral exploration 1-gen-2025 Martina, Maria Grazia; Vagaggini, Chiara; Dreassi, Elena; De Angelis, Marta; Nencioni, Lucia; Dragoni, Filippo; Giammarino, Federica; Boccuto, Adele; Zazzi, Maurizio; Vicenti, Ilaria; Radi, Marco
Identification of 4-amino-2-Pyridones as new potent PCSK9 inhibitors: From phenotypic hit discovery to in vivo tolerability 1-gen-2024 Giannessi, L; Lupo, Mg; Rossi, I; Martina, Mg; Vilella, A; Bodria, M; Giuliani, D; Zimetti, F; Zanotti, I; Potì, F; Bernini, F; Ferri, N; Radi, M
Investigating PCSK9 as a therapeutic target in Alzheimer's disease: evidence from patient-derived astrocytes 1-gen-2025 Ugolotti, M.; Papotti, B.; Adorni, M. P.; Martina, M. G.; Giannessi, L.; Olejnik, A.; Bell, S. M.; Mortiboys, H.; Radi, M.; Zimetti, F.