MARTINA, MARIA GRAZIA
MARTINA, MARIA GRAZIA
Dipartimento di Scienze degli Alimenti e del Farmaco
4-Trifluoromethyl bithiazoles as broad-spectrum antimicrobial agents for virus-related bacterial infections or co-infections
2024-01-01 Barbieri, Francesca; Carlen, Vincent; Martina, Maria Grazia; Sannio, Filomena; Cancade, Sacha; Perini, Cecilia; Restori, Margherita; Crespan, Emmanuele; Maga, Giovanni; Docquier, Jean-Denis; Cagno, Valeria; Radi, Marco
A Microwave‐Assisted One‐Pot Three‐Step Metal‐Free [4+2] Annulation for the Sustainable Synthesis of Highly Substituted 1,2,4‐Triazines
2024-01-01 Rubini, Daniele; Grazia Martina, Maria; Incerti, Matteo; Barbieri, Francesca; Radi, Marco
Benzofuran-2-Carboxamide Derivatives as Immunomodulatory Agents Blocking the CCL20-Induced Chemotaxis and Colon Cancer Growth
2024-01-01 Barbieri, Francesca; Martina, MARIA GRAZIA; Giorgio, Carmine; Chiara, MARIA LINDA; Allodi, Marika; Durante, Joseph; Bertoni, Simona; Radi, Marco
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses
2021-01-01 Martina Maria, Grazia.; Vicenti, I.; Bauer, L.; Crespan, E.; Rango, E.; Boccuto, A.; Olivieri, N.; Incerti, M.; Zwaagstra, M.; Allodi, M.; Bertoni, S.; Dreassi, E.; Zazzi, M.; van Kuppeveld, F. J. M.; Maga, G.; Radi, M.
Bithiazole inhibitors of PI4KB show broad-spectrum antiviral activity against different viral families
2024-01-01 Martina, Maria Grazia; Carlen, Vincent; Van der Reysen, Sarah; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Radi, Marco; Cagno, Valeria
CHEMISTRY-DRIVEN OPTIMIZATION OF PURINE-BASED ANTIVIRALS FOR THE IDENTIFICATION OF NEW BROAD-SPECTRUM AGENTS
2025-01-01 Valenti, Martina Eleonora; Martina, Maria Grazia; Vincetti, Paolo; Vicenti, Ilaria; Crespan, Emmanuele; Nencioni, Lucia; Kaptein, Suzanne J. F.; Neyts, Johan; Vanderlinden, Evelien; Schols, Dominique; De Forni, Davide; Lori, Franco; Zazzi, Maurizio; Maga, Giovanni; Radi, Marco
Combining Phenotypic and Targeted Approaches for the Identification of New Broad-Spectrum Antiviral Agents (BSAAs)
2023-01-01 Martina, Maria Grazia
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses
2025-01-01 Barbieri, Francesca; Martina, Maria Grazia; Pesce, Emanuela; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Rossi, Sara; Gemma, Sandra; Campiani, Giuseppe; Milite, Ciro; Pepe, Giacomo; Campiglia, Pietro; Sbardella, Gianluca; Maga, Giovanni; Cagno, Valeria; Pedemonte, Nicoletta; Radi, Marco
DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X
2025-01-01 Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco
DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X
2025-01-01 Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco
Development of Novel PCSK9 Inhibitors as Potential Broad-Spectrum Antivirals
2025-01-01 Savian, Chiara; Giannessi, Lisa; Martina, Maria Grazia; Ugolotti, Martina; Papotti, Bianca; Palumbo, Marcella; Giovanna Lupo, Maria; Mattina, Beatrice; Padula, Cristina; Nicoli, Sara; Ferri, Nicola; De Forni, Davide; Lori, Franco; Cagno, Valeria; Zimetti, Francesca; Radi, Marco
DISCOVERY OF NEW TSG101 INHIBITORS BLOCKING THE BUDDING OF EBOLA AND OTHER HIGHLY PATHOGENIC VIRUSES
2026-01-01 Valenti, Martina Eleonora; Rubini, Daniele; Parra-López, Marisa; Holzerland, Julia; Rodríguez-Martínez, Alejandro; Martina, Maria Grazia; Ramos, Maria C.; Castillo, Francisco; Harty, Ronald N.; Pérez-Sanchez, Horacio; Diederich, Sandra; Luque, Irene; Radi, Marco
Discovery of small-molecule targeting the CCL20/CCR6 axis as first-in-class inhibitors for inflammatory bowel diseases
2022-01-01 Martina, Maria Grazia; Giorgio, Carmine; Allodi, Marika; Palese, Simone; Barocelli, Elisabetta; Ballabeni, Vigilio; Szpakowska, Martyna; Chevigné, Andy; Piet Van Hamburg, Jan; Davelaar, Nadine; Lubberts, Erik; Bertoni, Simona; Radi, Marco
Effects of CCL20/CCR6 modulators in a T cell adoptive transfer model of colitis
2025-01-01 Allodi, M.; Flammini, L.; Giorgio, C.; Martina, M. G.; Barbieri, F.; Ballabeni, V.; Barocelli, E.; Radi, M.; Bertoni, S.
Harnessing prebiotic formamide chemistry: a novel platform for antiviral exploration
2025-01-01 Martina, Maria Grazia; Vagaggini, Chiara; Dreassi, Elena; De Angelis, Marta; Nencioni, Lucia; Dragoni, Filippo; Giammarino, Federica; Boccuto, Adele; Zazzi, Maurizio; Vicenti, Ilaria; Radi, Marco
Identification of 4-amino-2-Pyridones as new potent PCSK9 inhibitors: From phenotypic hit discovery to in vivo tolerability
2024-01-01 Giannessi, L; Lupo, Mg; Rossi, I; Martina, Mg; Vilella, A; Bodria, M; Giuliani, D; Zimetti, F; Zanotti, I; Potì, F; Bernini, F; Ferri, N; Radi, M
Investigating PCSK9 as a therapeutic target in Alzheimer's disease: evidence from patient-derived astrocytes
2025-01-01 Ugolotti, M.; Papotti, B.; Adorni, M. P.; Martina, M. G.; Giannessi, L.; Olejnik, A.; Bell, S. M.; Mortiboys, H.; Radi, M.; Zimetti, F.
Multicomponent Synthesis of Purines and Pyrimidines: From the Origin of Life to New Sustainable Approaches for Drug-Discovery Applications
2023-01-01 Martina, M. G.; Giannessi, L.; Radi, M.
Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties
2023-01-01 Grazia Martina, Maria; Giammarino, Federica; Vicenti, Ilaria; Groaz, Elisabetta; Rozenski, Jef; Incerti, Matteo; Sannio, Filomena; Docquier, Jean Denis; Zazzi, Maurizio; Radi, Marco
Optimization of 4‐Amino‐2‐Pyridone Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9: Integrating Structure–Activity and Structure–Metabolism Relationships
2026-01-01 Giannessi, Lisa; Lupo, Maria Giovanna; Ugolotti, Martina; Papotti, Bianca; Mattina, Beatrice; Martina, Maria Grazia; Demurtas, Anna; Padula, Cristina; Nicoli, Sara; Crescenzio, Marco; Ferri, Nicola; Zimetti, Francesca; Radi, Marco
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 4-Trifluoromethyl bithiazoles as broad-spectrum antimicrobial agents for virus-related bacterial infections or co-infections | 1-gen-2024 | Barbieri, Francesca; Carlen, Vincent; Martina, Maria Grazia; Sannio, Filomena; Cancade, Sacha; Perini, Cecilia; Restori, Margherita; Crespan, Emmanuele; Maga, Giovanni; Docquier, Jean-Denis; Cagno, Valeria; Radi, Marco | |
| A Microwave‐Assisted One‐Pot Three‐Step Metal‐Free [4+2] Annulation for the Sustainable Synthesis of Highly Substituted 1,2,4‐Triazines | 1-gen-2024 | Rubini, Daniele; Grazia Martina, Maria; Incerti, Matteo; Barbieri, Francesca; Radi, Marco | |
| Benzofuran-2-Carboxamide Derivatives as Immunomodulatory Agents Blocking the CCL20-Induced Chemotaxis and Colon Cancer Growth | 1-gen-2024 | Barbieri, Francesca; Martina, MARIA GRAZIA; Giorgio, Carmine; Chiara, MARIA LINDA; Allodi, Marika; Durante, Joseph; Bertoni, Simona; Radi, Marco | |
| Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses | 1-gen-2021 | Martina Maria, Grazia.; Vicenti, I.; Bauer, L.; Crespan, E.; Rango, E.; Boccuto, A.; Olivieri, N.; Incerti, M.; Zwaagstra, M.; Allodi, M.; Bertoni, S.; Dreassi, E.; Zazzi, M.; van Kuppeveld, F. J. M.; Maga, G.; Radi, M. | |
| Bithiazole inhibitors of PI4KB show broad-spectrum antiviral activity against different viral families | 1-gen-2024 | Martina, Maria Grazia; Carlen, Vincent; Van der Reysen, Sarah; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Radi, Marco; Cagno, Valeria | |
| CHEMISTRY-DRIVEN OPTIMIZATION OF PURINE-BASED ANTIVIRALS FOR THE IDENTIFICATION OF NEW BROAD-SPECTRUM AGENTS | 1-gen-2025 | Valenti, Martina Eleonora; Martina, Maria Grazia; Vincetti, Paolo; Vicenti, Ilaria; Crespan, Emmanuele; Nencioni, Lucia; Kaptein, Suzanne J. F.; Neyts, Johan; Vanderlinden, Evelien; Schols, Dominique; De Forni, Davide; Lori, Franco; Zazzi, Maurizio; Maga, Giovanni; Radi, Marco | |
| Combining Phenotypic and Targeted Approaches for the Identification of New Broad-Spectrum Antiviral Agents (BSAAs) | 1-gen-2023 | Martina, Maria Grazia | |
| Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses | 1-gen-2025 | Barbieri, Francesca; Martina, Maria Grazia; Pesce, Emanuela; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Rossi, Sara; Gemma, Sandra; Campiani, Giuseppe; Milite, Ciro; Pepe, Giacomo; Campiglia, Pietro; Sbardella, Gianluca; Maga, Giovanni; Cagno, Valeria; Pedemonte, Nicoletta; Radi, Marco | |
| DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X | 1-gen-2025 | Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco | |
| DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X | 1-gen-2025 | Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco | |
| Development of Novel PCSK9 Inhibitors as Potential Broad-Spectrum Antivirals | 1-gen-2025 | Savian, Chiara; Giannessi, Lisa; Martina, Maria Grazia; Ugolotti, Martina; Papotti, Bianca; Palumbo, Marcella; Giovanna Lupo, Maria; Mattina, Beatrice; Padula, Cristina; Nicoli, Sara; Ferri, Nicola; De Forni, Davide; Lori, Franco; Cagno, Valeria; Zimetti, Francesca; Radi, Marco | |
| DISCOVERY OF NEW TSG101 INHIBITORS BLOCKING THE BUDDING OF EBOLA AND OTHER HIGHLY PATHOGENIC VIRUSES | 1-gen-2026 | Valenti, Martina Eleonora; Rubini, Daniele; Parra-López, Marisa; Holzerland, Julia; Rodríguez-Martínez, Alejandro; Martina, Maria Grazia; Ramos, Maria C.; Castillo, Francisco; Harty, Ronald N.; Pérez-Sanchez, Horacio; Diederich, Sandra; Luque, Irene; Radi, Marco | |
| Discovery of small-molecule targeting the CCL20/CCR6 axis as first-in-class inhibitors for inflammatory bowel diseases | 1-gen-2022 | Martina, Maria Grazia; Giorgio, Carmine; Allodi, Marika; Palese, Simone; Barocelli, Elisabetta; Ballabeni, Vigilio; Szpakowska, Martyna; Chevigné, Andy; Piet Van Hamburg, Jan; Davelaar, Nadine; Lubberts, Erik; Bertoni, Simona; Radi, Marco | |
| Effects of CCL20/CCR6 modulators in a T cell adoptive transfer model of colitis | 1-gen-2025 | Allodi, M.; Flammini, L.; Giorgio, C.; Martina, M. G.; Barbieri, F.; Ballabeni, V.; Barocelli, E.; Radi, M.; Bertoni, S. | |
| Harnessing prebiotic formamide chemistry: a novel platform for antiviral exploration | 1-gen-2025 | Martina, Maria Grazia; Vagaggini, Chiara; Dreassi, Elena; De Angelis, Marta; Nencioni, Lucia; Dragoni, Filippo; Giammarino, Federica; Boccuto, Adele; Zazzi, Maurizio; Vicenti, Ilaria; Radi, Marco | |
| Identification of 4-amino-2-Pyridones as new potent PCSK9 inhibitors: From phenotypic hit discovery to in vivo tolerability | 1-gen-2024 | Giannessi, L; Lupo, Mg; Rossi, I; Martina, Mg; Vilella, A; Bodria, M; Giuliani, D; Zimetti, F; Zanotti, I; Potì, F; Bernini, F; Ferri, N; Radi, M | |
| Investigating PCSK9 as a therapeutic target in Alzheimer's disease: evidence from patient-derived astrocytes | 1-gen-2025 | Ugolotti, M.; Papotti, B.; Adorni, M. P.; Martina, M. G.; Giannessi, L.; Olejnik, A.; Bell, S. M.; Mortiboys, H.; Radi, M.; Zimetti, F. | |
| Multicomponent Synthesis of Purines and Pyrimidines: From the Origin of Life to New Sustainable Approaches for Drug-Discovery Applications | 1-gen-2023 | Martina, M. G.; Giannessi, L.; Radi, M. | |
| Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties | 1-gen-2023 | Grazia Martina, Maria; Giammarino, Federica; Vicenti, Ilaria; Groaz, Elisabetta; Rozenski, Jef; Incerti, Matteo; Sannio, Filomena; Docquier, Jean Denis; Zazzi, Maurizio; Radi, Marco | |
| Optimization of 4‐Amino‐2‐Pyridone Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9: Integrating Structure–Activity and Structure–Metabolism Relationships | 1-gen-2026 | Giannessi, Lisa; Lupo, Maria Giovanna; Ugolotti, Martina; Papotti, Bianca; Mattina, Beatrice; Martina, Maria Grazia; Demurtas, Anna; Padula, Cristina; Nicoli, Sara; Crescenzio, Marco; Ferri, Nicola; Zimetti, Francesca; Radi, Marco |