| Nome |
# |
|
Advances in Exploring Heterocyclic Dienoxysilane Nucleophiles in Asymmetric Synthesis, file e177fbc4-1a25-50b0-e053-d805fe0adaee
|
32
|
|
Grafting Aminocyclopentane Carboxylic Acids onto the RGD Tripeptide Sequence Generates Low Nanomolar alfaVbeta3/alfaVbeta5 Integrin Dual Binders, file e177fbc4-0aad-50b0-e053-d805fe0adaee
|
22
|
|
Catalytic, Asymmetric Vinylogous Mukaiyama Aldol Reactions of Pyrrole- and Furan-Based Dienoxy Silanes: How the Diene Heteroatom Impacts Stereocontrol, file e177fbc4-250f-50b0-e053-d805fe0adaee
|
21
|
|
Integrin-targeted AmpRGD sunitinib liposomes as integrated antiangiogenic tools, file e177fbc6-de29-50b0-e053-d805fe0adaee
|
20
|
|
Discovery of Subnanomolar Arginine-Glycine-Aspartate-Based alphaVbeta3/alphaVbeta5 Integrin Binders Embedding 4-Aminoproline Residues, file e177fbc4-261a-50b0-e053-d805fe0adaee
|
17
|
|
Efficacy of a Selective Binder of αVβ3 Integrin Linked to the Tyrosine Kinase Inhibitor Sunitinib in Ovarian Carcinoma Preclinical Models, file e177fbc6-7051-50b0-e053-d805fe0adaee
|
16
|
|
Total Synthesis of Both Enantiomers of trans-beta-Hydroxypipecolic Acid, file e177fbc4-247f-50b0-e053-d805fe0adaee
|
15
|
|
Streamlined, Asymmetric Synthesis of 8,4'-Oxyneolignans, file e177fbc4-0f65-50b0-e053-d805fe0adaee
|
14
|
|
Asymmetric Total Synthesis of 1-Deoxy-7,8-di-epi-castanospermine, file e177fbc4-1b4c-50b0-e053-d805fe0adaee
|
14
|
|
4-Aminoproline-Based Arginine-Glycine-Aspartate Integrin Binders with Exposed Ligation Points: Practical in-Solution Synthesis, Conjugation and Binding Affinity Evaluation, file e177fbc4-1ba9-50b0-e053-d805fe0adaee
|
14
|
|
(E)-3-(Alkoxycarbonyl-2-Alkyliden)-2-Oxindoles: Multidentate Pronucleophiles for the Organocatalytic, Vinylogous Michael Addition to Nitroolefins, file e177fbc7-6052-50b0-e053-d805fe0adaee
|
14
|
|
Cell-targeted c(AmpRGD)-sunitinib molecular conjugates impair tumor growth of melanoma, file e177fbc7-4d33-50b0-e053-d805fe0adaee
|
13
|
|
Grafting Aminocyclopentane Carboxylic Acids onto the RGD Tripeptide Sequence Generates Low Nanomolar alfaVbeta3/alfaVbeta5 Integrin Dual Binders, file e177fbc4-0aab-50b0-e053-d805fe0adaee
|
12
|
|
Uncatalyzed, Diastereoselective Vinylogous Mukaiyama Aldol Reactions on Aqueous Media: Pyrrole vs Furan 2-Silyloxy Dienes, file e177fbc4-276b-50b0-e053-d805fe0adaee
|
12
|
|
Divergent Synthesis of 3-Amino-3-deoxy- and 4-Amino-4-deoxyhexoses, file e177fbc4-241a-50b0-e053-d805fe0adaee
|
11
|
|
Uncatalyzed, Diastereoselective Vinylogous Mukaiyama Aldol Reactions on Aqueous Media: Pyrrole vs Furan 2-Silyloxy Dienes, file e177fbc4-276c-50b0-e053-d805fe0adaee
|
11
|
|
Streamlined, Asymmetric Synthesis of 8,4'-Oxyneolignans, file e177fbc4-0f64-50b0-e053-d805fe0adaee
|
10
|
|
Asymmetric, catalytic, vinylogous aldol reactions using pyrrole-based dienoxy silanes. Enantioselective synthesis of alpha,beta-unsaturated gamma-butyrolactam synthons, file e177fbc4-1b2a-50b0-e053-d805fe0adaee
|
9
|
|
Targeting alphaVbeta3 Integrin: Design and Applications of Mono- and Multifunctional RGD-Based Peptides and Semipeptides, file e177fbc4-1baf-50b0-e053-d805fe0adaee
|
9
|
|
Vicarious Silylative Mukaiyama Aldol Reaction: A Vinylogous Extension, file e177fbc4-1de7-50b0-e053-d805fe0adaee
|
9
|
|
Discovery of Subnanomolar Arginine-Glycine-Aspartate-Based alphaVbeta3/alphaVbeta5 Integrin Binders Embedding 4-Aminoproline Residues, file e177fbc4-2619-50b0-e053-d805fe0adaee
|
8
|
|
Variable Strategy toward Carbasugars and Relatives. 4. Viable Access to (4a-Carbapentofuranosyl)amines, (5a-Carbahexopyranosyl)amines, and Amino Acids Thereof, file e177fbc4-229d-50b0-e053-d805fe0adaee
|
7
|
|
Direct, Organocatalytic, Enantioseletcive Michael Reactions: Turning Common Michael Acceptors Into Vinylogous Carbon Nucleophiles, file e177fbc4-4299-50b0-e053-d805fe0adaee
|
7
|
|
Unlocking Access to Enantiopure Fused Uracils by Chemodivergent [4+2] Cross‐Cycloadditions: DFT‐Supported Homo‐Synergistic Organocatalytic Approach, file e177fbc6-e834-50b0-e053-d805fe0adaee
|
7
|
|
RGD Peptide-Drug Conjugates as Effective Dual Targeting Platforms: Recent Advances, file e177fbc7-5459-50b0-e053-d805fe0adaee
|
7
|
|
Synthesis and Applications of Pyrrolidine-Based RGD Integrin Binders and Conjugates, file e177fbc4-2aff-50b0-e053-d805fe0adaee
|
6
|
|
Variable Strategy towards Carbasugars and Relatives. 6. Diastereoselective Synthesis of 2-Deoxy-2-amino-5a-carba-beta-L-mannopyranuronic Acid and 2-Deoxy-2-amino-5a-carba-beta-L-mannopyranose, file e177fbc4-0943-50b0-e053-d805fe0adaee
|
5
|
|
Expeditious Syntheses of Sugar-Modified Nucleosides and Collections Thereof Exploiting Furan-, Pyrrole-, and Thiophene-Based Siloxy Dienes, file e177fbc4-2416-50b0-e053-d805fe0adaee
|
5
|
|
Direct-type vinylogous Mukaiyama-Michael addition reactions involving pyrrolinone donors, file e177fbc4-2475-50b0-e053-d805fe0adaee
|
5
|
|
Catalytic Enantioselective Three-Component Vinylogous Mukaiyama Mannich Reactions with Pyrrole-Based Dienoxy Silanes, file e177fbc4-2b00-50b0-e053-d805fe0adaee
|
5
|
|
Direct, Asymmetric Synthesis of Carbocycle-Fused Uracils via [4+2] Cycloadditions: a Noncovalent Organocatalysis Approach, file e177fbc7-2a46-50b0-e053-d805fe0adaee
|
5
|
|
New 4-aminoproline-based small molecule cyclopeptidomimetics as potential modulators of α4β1 integrin, file e177fbc7-66cc-50b0-e053-d805fe0adaee
|
5
|
|
Enantioselective Total Synthesis of (1R,3S,4R,5R)-1-Amino-4,5-dihydroxycyclopentane-1,3-dicarboxylic Acid. A Full-Aldol Access to Carbaketose Derivatives, file e177fbc4-0944-50b0-e053-d805fe0adaee
|
4
|
|
Nintedanib-Containing Dual Conjugates Targeting αVβ6 Integrin and Tyrosine Kinase Receptors as Potential Antifibrotic Agents, file e177fbc8-1c85-50b0-e053-d805fe0adaee
|
4
|
|
New Enantioselective Entry to Cycloheptane Amino Acid Polyols, file e177fbc4-0f66-50b0-e053-d805fe0adaee
|
3
|
|
Further Uses of Pyrrole-Based Dienoxysilane Synthons: A Full Aldol Approach to Azabicyclo[x.2.1]alkane Systems, file e177fbc4-192d-50b0-e053-d805fe0adaee
|
3
|
|
Vicarious Silylative Mukaiyama Aldol Reaction: A Vinylogous Extension, file e177fbc4-1de8-50b0-e053-d805fe0adaee
|
3
|
|
Modular Approach toward the Construction of the Core Motifs of Annonaceous Acetogenins and Variants Thereof, file e177fbc4-2419-50b0-e053-d805fe0adaee
|
3
|
|
DIRECT ENANTIOSELECTIVE VINYLOGOUS MICHAEL ADDITION OF
3-ALKYLIDENE OXINDOLES TO NITROOLEFINS CATALYZED BY
BIFUNCTIONAL CINCHONA ALKALOID THIOUREAS, file e177fbc4-3545-50b0-e053-d805fe0adaee
|
3
|
|
Nintedanib-αVβ6 Integrin Ligand Conjugates Reduce TGFβ-Induced EMT in Human Non-Small Cell Lung Cancer, file 0699949c-5aca-41de-b4f5-2c18beb088c1
|
2
|
|
Grafting Aminocyclopentane Carboxylic Acids onto the RGD Tripeptide Sequence Generates Low Nanomolar alfaVbeta3/alfaVbeta5 Integrin Dual Binders, file e177fbc4-0aaa-50b0-e053-d805fe0adaee
|
2
|
|
New Enantioselective Entry to Cycloheptane Amino Acid Polyols, file e177fbc4-0fcc-50b0-e053-d805fe0adaee
|
2
|
|
Diastereo- and Enantioselective Catalytic Vinylogous Mukaiyama-Mannich Reactions of Pyrrole-Based Silyl Dienolates with Alkyl-Substituted Aldehydes, file e177fbc4-2e32-50b0-e053-d805fe0adaee
|
2
|
|
The Principle of Vinylogy as Applied to Heterocyclic Donor Systems, file e177fbc4-af16-50b0-e053-d805fe0adaee
|
2
|
|
Pushing the Boundaries of Vinylogous Reactivity: Catalytic Enantioselective Mukaiyama Aldol Reactions of Highly Unsaturated 2-Silyloxyindoles, file e177fbc7-4f93-50b0-e053-d805fe0adaee
|
2
|
|
Shifting Towards αVβ6 Integrin Ligands Using Novel Aminoproline-Based Cyclic Peptidomimetics, file e177fbc7-4fc7-50b0-e053-d805fe0adaee
|
2
|
|
Turning the Imidazole Core into Three‐Dimensional Ring Systems: Mild Organocatalytic Entry to Enantiopure 6,7‐Dihydrobenzimidazoles, file 250860ff-04fe-4c58-822f-0b78b40d0268
|
1
|
|
Synthesis of a Small Repertoire of Non-Racemic 5a-Carbahexopyranoses and 1-Thio-5a-carbahexopyranoses, file e177fbc4-0c6b-50b0-e053-d805fe0adaee
|
1
|
|
Targeting alphaVbeta3 Integrin: Design and Applications of Mono- and Multifunctional RGD-Based Peptides and Semipeptides, file e177fbc4-1bae-50b0-e053-d805fe0adaee
|
1
|
|
Novel Carbasugar-Containing Cyclic RGD Peptides for Integrin Receptors Recognition, file e177fbc4-218b-50b0-e053-d805fe0adaee
|
1
|
|
Direct-type vinylogous Mukaiyama-Michael addition reactions involving pyrrolinone donors, file e177fbc4-2476-50b0-e053-d805fe0adaee
|
1
|
|
Catalytic, Asymmetric Vinylogous Mukaiyama Aldol Reactions of Pyrrole- and Furan-Based Dienoxy Silanes: How the Diene Heteroatom Impacts Stereocontrol, file e177fbc4-250e-50b0-e053-d805fe0adaee
|
1
|
|
Aqueous and Solvent-Free Uncatalyzed Vinylogous Mukaiyama-Mannich Reaction of Pyrrole Dienoxy Silanes, file e177fbc4-2ff0-50b0-e053-d805fe0adaee
|
1
|
|
Uncatalyzed, Diastereoselective Vinylogous Mukaiyama Aldol Reactions on Aqueous Media: Pyrrole vs Furan 2-Silyloxy Dienes, file e177fbc4-3613-50b0-e053-d805fe0adaee
|
1
|
|
Direct Regio-, Diastereo-, and Enantioselective Vinylogous Michael Addition of Prochiral 3-Alkylideneoxindoles to Nitroolefins, file e177fbc4-a895-50b0-e053-d805fe0adaee
|
1
|
|
Synthesis, structure and inhibitory activity of a stereoisomer of oseltamivir carboxylate, file e177fbc4-b0ca-50b0-e053-d805fe0adaee
|
1
|
|
Merging RGD/Sunitinib Chemotypes to Unique Hybrid Constructs is Useful to Impair Tumor Angiogenesis and Melanoma Growth, file e177fbc6-2b4c-50b0-e053-d805fe0adaee
|
1
|
|
Towards New Small-Molecule Peptidomimetics as Selective alphaVbeta6 Integrin Ligands, file e177fbc6-2b4e-50b0-e053-d805fe0adaee
|
1
|
| Totale |
416 |