COSTANTINO, Gabriele

COSTANTINO, Gabriele  

Dipartimento di Scienze degli Alimenti e del Farmaco  

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Titolo Data di pubblicazione Autore(i) File
(2R,1'S,2'R,3'S)-2-(2'-Carboxy-3'-phenylcyclopropyl)glycine (PCCG-13), the first potent and selective competitive antagonist of phospholipase D-coupled metabotropic glutamate receptors: asymmetric synthesis and preliminary biological properties 1-gen-1999 Pellicciari, R; Marinozzi, M; Costantino, Gabriele; Natalini, B; Moroni, F; PELLEGRINI GIAMPIETRO, D.
1,4-Benzothiazine and 1,4-benzoxazine imidazole derivatives with antifungal activity: a docking study 1-gen-2002 Macchiarulo, A; Fringuelli, D; Vecchiarelli, A; Schiaffella, F; Costantino, Gabriele
1-Aminoindane-1,5-dicarboxylic Acid: a Novel Antagonist at Phospholipase C Linked Metabotropic Glutamate Receptors 1-gen-1995 R., Pellicciari; R., Luneia; Costantino, Gabriele; M., Marinozzi; B., Natalini; P., Jackobsen; A., Kanstrup; G., Lombardi; F., Moroni; C., Thomsen
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry 1-gen-2020 Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M.
6alpha-ethyl-chenodeoxycholic acid (6-ECDCA), a potent and selective FXR agonist endowed with anticholestatic activity. 1-gen-2002 Pellicciari, R; Fiorucci, S; Camaioni, E; Clerici, C; Maloney, Pr; Morelli, A; Parks, Dj; Costantino, Gabriele
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin 1-gen-2016 Vucicevic, Jelica; Srdic Rajic, Tatjana; Pieroni, Marco; Laurila, Jonne M. M.; Perovic, Vladimir; Tassini, Sabrina; Azzali, Elisa; Costantino, Gabriele; Glisic, Sanja; Agbaba, Danica; Scheinin, Mika; Nikolic, Katarina; Radi, Marco; Veljkovic, Nevena
A competitive o‐acetylserine sulfhydrylase inhibitor modulates the formation of cysteine synthase complex 1-gen-2021 Marchetti, M.; De Angelis, F. S.; Annunziato, G.; Costantino, G.; Pieroni, M.; Ronda, L.; Mozzarelli, A.; Campanini, B.; Cannistraro, S.; Bizzarri, A. R.; Bettati, S.
A High Performance Workflow for Chemistry Driven de Novo Design 1-gen-2013 Beccari, Ar; Cavazzoni, C; Beato, Claudia; Costantino, Gabriele
A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides 1-gen-2016 Vincetti, Paolo; Brianza, Anna; Scalacci, Nicolò; Costantino, Gabriele; Castagnolo, Daniele; Radi, Marco
A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes 1-gen-2016 Tassini, Sabrina; Castagnolo, Daniele; Scalacci, Nicolò; Kissova, Miroslava; Armijos Rivera, Jorge I.; Giagnorio, Federica; Maga, Giovanni; Costantino, Gabriele; Crespan, Emmanuele; Radi, Marco
A one-pot two-step microwave-assisted synthesis of N1-substituted 5,6-ring-fused 2-pyridones 1-gen-2013 Radi, Marco; Gian Paolo, Vallerini; Alessia, Petrelli; Paolo, Vincetti; Costantino, Gabriele
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents 1-gen-2017 Pieroni, Marco; Azzali, Elisa; Basilico, Nicoletta; Parapini, Silvia; Zolkiewski, Michal; Beato, Claudia; Annunziato, Giannamaria; Bruno, Agostino; Vacondio, Federica; Costantino, Gabriele
Addressing the Conformational Flexibility of Serine Racemase by Combining Targeted Molecular Dynamics, Conformational Sampling and Docking Studies 1-gen-2011 A., Bruno; Amori, Laura; Costantino, Gabriele
Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting Mycobacterium tuberculosis energetics 1-gen-2018 Machado, Diana; Azzali, Elisa; Couto, Isabel; Costantino, Gabriele; Pieroni, Marco; Viveiros, Miguel
alfa-Diazocarbonyl Chemistry - Target Driven Applications 1-gen-1998 R., Pellicciari; Costantino, Gabriele; M., Marinozzi; L., Mattoli; B., Natalini
Aminonicotinic acid 1-oxides are chemically stable inhibitors of quinolinic acid synthesis in the mammalian brain: a step towards new anti-excitotoxic agents 1-gen-2013 Vallerini, Gp; Amori, Laura; Beato, Claudia; Tararina, M; Wang, Xd; Schwarcz, R; Costantino, Gabriele
Antifungal properties of newly designed carbonic anhydrases inhibitors selective for microbial enzymes 1-gen-2018 Giovati, Laura; Annunziato, Giannamaria; Ciociola, Tecla; Magliani, Valter; Polonelli, Luciano; Conti, Stefania; Supuran, Claudiu T.; Costantino, Gabriele
Antimicrobial peptides (AMPs): a patent review (2015-2020) 1-gen-2020 Annunziato, Giannamaria; Costantino, Gabriele
Aspergillus fumigatus tryptophan metabolic route differently affects host immunity 1-gen-2021 Zelante, T.; Choera, T.; Beauvais, A.; Fallarino, F.; Paolicelli, G.; Pieraccini, G.; Pieroni, M.; Galosi, C.; Beato, C.; De Luca, A.; Boscaro, F.; Romoli, R.; Liu, X.; Warris, A.; Verweij, P. E.; Ballard, E.; Borghi, M.; Pariano, M.; Costantino, G.; Calvitti, M.; Vacca, C.; Oikonomou, V.; Gargaro, M.; Wong, A. Y. W.; Boon, L.; den Hartog, M.; Spacil, Z.; Puccetti, P.; Latge, J. -P.; Keller, N. P.; Romani, L.
Asymmetric Synthesis of Enantiomerically Pure (2S,1'S,2'S,3'R)-phenylcarboxycyclopropylglycine (PCCG-4): A Potent and Selective Ligand at Group II Metabotropic Glutamate Receptors 1-gen-1996 M., Marinozzi; B., Natalini; Costantino, Gabriele; P., Tijskens; C., Thomsen; R., Pellicciari