COSTANTINO, Gabriele

COSTANTINO, Gabriele  

Dipartimento di Scienze degli Alimenti e del Farmaco  

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Titolo Data di pubblicazione Autore(i) File
1,4-Benzothiazine and 1,4-benzoxazine imidazole derivatives with antifungal activity: a docking study 1-gen-2002 Macchiarulo, A; Fringuelli, D; Vecchiarelli, A; Schiaffella, F; Costantino, Gabriele
1-Aminoindane-1,5-dicarboxylic Acid: a Novel Antagonist at Phospholipase C Linked Metabotropic Glutamate Receptors 1-gen-1995 R., Pellicciari; R., Luneia; Costantino, Gabriele; M., Marinozzi; B., Natalini; P., Jackobsen; A., Kanstrup; G., Lombardi; F., Moroni; C., Thomsen
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry 1-gen-2020 Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M.
(2R,1'S,2'R,3'S)-2-(2'-Carboxy-3'-phenylcyclopropyl)glycine (PCCG-13), the first potent and selective competitive antagonist of phospholipase D-coupled metabotropic glutamate receptors: asymmetric synthesis and preliminary biological properties 1-gen-1999 Pellicciari, R; Marinozzi, M; Costantino, Gabriele; Natalini, B; Moroni, F; PELLEGRINI GIAMPIETRO, D.
6alpha-ethyl-chenodeoxycholic acid (6-ECDCA), a potent and selective FXR agonist endowed with anticholestatic activity. 1-gen-2002 Pellicciari, R; Fiorucci, S; Camaioni, E; Clerici, C; Maloney, Pr; Morelli, A; Parks, Dj; Costantino, Gabriele
A High Performance Workflow for Chemistry Driven de Novo Design 1-gen-2013 Beccari, Ar; Cavazzoni, C; Beato, Claudia; Costantino, Gabriele
A one-pot two-step microwave-assisted synthesis of N1-substituted 5,6-ring-fused 2-pyridones. 1-gen-2013 Radi, M.; Vallerini, G. P.; Petrelli, A.; Vincetti, P.; Costantino, Gabriele
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents 1-gen-2017 Pieroni, Marco; Azzali, Elisa; Basilico, Nicoletta; Parapini, Silvia; Zolkiewski, Michal; Beato, Claudia; Annunziato, Giannamaria; Bruno, Agostino; Vacondio, Federica; Costantino, Gabriele
Addressing the Conformational Flexibility of Serine Racemase by Combining Targeted Molecular Dynamics, Conformational Sampling and Docking Studies 1-gen-2011 A., Bruno; Amori, Laura; Costantino, Gabriele
Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting Mycobacterium tuberculosis energetics 1-gen-2018 Machado, Diana; Azzali, Elisa; Couto, Isabel; Costantino, Gabriele; Pieroni, Marco; Viveiros, Miguel
alfa-Diazocarbonyl Chemistry - Target Driven Applications 1-gen-1998 R., Pellicciari; Costantino, Gabriele; M., Marinozzi; L., Mattoli; B., Natalini
Aminonicotinic acid 1-oxides are chemically stable inhibitors of quinolinic acid synthesis in the mammalian brain: a step towards new anti-excitotoxic agents 1-gen-2013 Vallerini, Gp; Amori, Laura; Beato, Claudia; Tararina, M; Wang, Xd; Schwarcz, R; Costantino, Gabriele
Antifungal properties of newly designed carbonic anhydrases inhibitors selective for microbial enzymes 1-gen-2018 Giovati, Laura; Annunziato, Giannamaria; Ciociola, Tecla; Magliani, Valter; Polonelli, Luciano; Conti, Stefania; Supuran, Claudiu T.; Costantino, Gabriele
The aryl hydrocarbon receptor (AhR) mediates the counter-regulatory effects of pelargonidins in models of inflammation and metabolic dysfunctions 1-gen-2019 Biagioli, M.; Carino, A.; Fiorucci, C.; Annunziato, G.; Marchiano, S.; Bordoni, M.; Roselli, R.; Giorgio, C. D.; Castiglione, F.; Ricci, P.; Bruno, A.; Faccini, A.; Distrutti, E.; Baldoni, M.; Costantino, G.; Fiorucci, S.
Aspergillus fumigatus tryptophan metabolic route differently affects host immunity 1-gen-2021 Zelante, T.; Choera, T.; Beauvais, A.; Fallarino, F.; Paolicelli, G.; Pieraccini, G.; Pieroni, M.; Galosi, C.; Beato, C.; De Luca, A.; Boscaro, F.; Romoli, R.; Liu, X.; Warris, A.; Verweij, P. E.; Ballard, E.; Borghi, M.; Pariano, M.; Costantino, G.; Calvitti, M.; Vacca, C.; Oikonomou, V.; Gargaro, M.; Wong, A. Y. W.; Boon, L.; den Hartog, M.; Spacil, Z.; Puccetti, P.; Latge, J. -P.; Keller, N. P.; Romani, L.
Asymmetric Synthesis of Enantiomerically Pure (2S,1'S,2'S,3'R)-phenylcarboxycyclopropylglycine (PCCG-4): A Potent and Selective Ligand at Group II Metabotropic Glutamate Receptors 1-gen-1996 M., Marinozzi; B., Natalini; Costantino, Gabriele; P., Tijskens; C., Thomsen; R., Pellicciari
Autocorrelation as a tool for a congruent description of molecules in 3D-QSAR studies 1-gen-1993 S., Clementi; G., Cruciani; D., Riganelli; R., Valigi; Costantino, Gabriele; M., Baroni; S., Wold
Back door modulation of the farnesoid X receptor: design, synthesis, and biological evaluation of a series of side chain modified chenodeoxycholic acid derivatives. 1-gen-2006 Pellicciari, R.; Gioiello, A.; Sadeghpour, B. M.; Rizzo, G.; Meyer, U.; Parks, D. J.; ENTRENA GUADIX, A.; Costantino, Gabriele
Bile acid derivatives as ligands of the farnesoid X receptor. Synthesis, evaluation, and structure-activity relationship of a series of body and side chain modified analogues of chenodeoxycholic acid. 1-gen-2004 Pellicciari, R; Costantino, Gabriele; Camaioni, E; Sadeghpour, Bm; Entrena, A; Willson, Tm; Fiorucci, S; Clerici, C; Gioiello, A.
Binding mode of 6ECDCA, a potent bile acid agonist of the farnesoid X receptor (FXR) 1-gen-2003 Costantino, Gabriele; Macchiarulo, A; ENTRENA GUADIX, A; Camaioni, E; Pellicciari, R.