LODOLA, Alessio

LODOLA, Alessio  

Dipartimento di Scienze degli Alimenti e del Farmaco  

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Risultati 1 - 20 di 155 (tempo di esecuzione: 0.364 secondi).
Titolo Data di pubblicazione Autore(i) File
270 Discovery, development and optimization of low molecular weight EPH–ephrin protein–protein inhibitors 1-gen-2014 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Barocelli, Elisabetta; Mor, Marco; Pala, Daniele; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity 1-gen-2006 Carmi, Caterina; Cavazzoni, Andrea; Zuliani, Valentina; Lodola, Alessio; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line 1-gen-2009 Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
A catalytic mechanism for cysteine N-terminal nucleophile hydrolases, as revealed by free energy simulations 1-gen-2012 Lodola, Alessio; D., Branduardi; M., De Vivo; L., Capoferri; Mor, Marco; D., Piomelli; A., Cavalli
A catalytically silent FAAH-1 variant drives anandamide transport in neurons 1-gen-2012 Jin, Fu; Giovanni, Bottegoni; Oscar, Sasso; Rosalia, Bertorelli; Walter, Rocchia; Matteo, Masetti; Ana, Guijarro; Lodola, Alessio; Andrea, Armirotti; Gianpiero, Garau; Tiziano, Bandiera; Angelo, Reggiani; Mor, Marco; Andrea, Cavalli; Daniele, Piomelli
A critical cysteine residue in monoacylglycerol lipase is targeted by a new class of isothiazolinone-based enzyme inhibitors. 1-gen-2009 King, A. R.; Lodola, Alessio; Carmi, Caterina; Fu, J.; Mor, Marco; Piomelli, D.
A Pharmacological Investigation of Eph-Ephrin Antagonism in Prostate Cancer: UniPR1331 Efficacy Evidence 1-gen-2023 Festuccia, Claudio; Corrado, Miriam; Rossetti, Alessandra; Castelli, Riccardo; Lodola, Alessio; Gravina, Giovanni Luca; Tognolini, Massimiliano; Giorgio, Carmine
A sulfonyl fluoride derivative inhibits EGFR L858R/T790M/C797S by covalent modification of the catalytic lysine 1-gen-2021 Ferlenghi, F; Scalvini, L; Vacondio, F; Castelli, R; Bozza, N; Marseglia, G; Rivara, S; Lodola, A; La Monica, S; Minari, R; Petronini, Pg; Alfieri, R; Tiseo, M; Mor, M.
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. 1-gen-2013 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Amino acid derivatives as palmitoylethanolamide prodrugs: Synthesis, in vitro metabolism and in vivo plasma profile in rats 1-gen-2015 Vacondio, Federica; Bassi, Michele; Silva, Claudia; Castelli, Riccardo; Carmi, Caterina; Scalvini, Laura; Lodola, Alessio; Vivo, Valentina; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco; Rivara, Silvia
Analysis of adam12-mediated ephrin-a1 cleavage and its biological functions 1-gen-2021 Ieguchi, K.; Tomita, T.; Takao, T.; Omori, T.; Mishima, T.; Shimizu, I.; Tognolini, M.; Lodola, A.; Tsunoda, T.; Kobayashi, S.; Wada, S.; Maru, Y.
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors 1-gen-2005 Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G.
Application of a SCC-DFTB QM/MM approach to the investigation of the catalytic mechanism of fatty acid amide hydrolase. 1-gen-2011 L., Capoferri; Mor, Marco; J., Sirirak; E., Chudyk; Aj, Mulholland; Lodola, Alessio
APPLICATION OF COMPUTATIONAL METHODSTO THE DESIGN OF FATTY ACID AMIDE HYDROLASE(FAAH) INHIBITORS BASED ON A CARBAMICTEMPLATE STRUCTURE 1-gen-2011 Lodola, Alessio; Rivara, Silvia; Mor, Marco
Applications and Advances of QM/MM methods in Computational Enzymology 1-gen-2008 Lodola, Alessio; Woods, C.; Mulholland, A. J.
Are we using the right pharmacological tools to target EphA4? 1-gen-2014 Tognolini, Massimiliano; Incerti, Matteo; Lodola, Alessio
Aromatic interactions and rotational strengths within protein environment: An electronic structural study on beta-lactamases from class A 1-gen-2008 Christov, C.; Karabencheva, T.; Lodola, Alessio
Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs 1-gen-2017 Lodola, Alessio; Bertolini, S; Biagetti, M; Capacchi, S; Facchinetti, F; Gallo, Pm; Pappani, A; Mor, Marco; Pala, Daniele; Rivara, Silvia; Visentini, F; Corsi, M; Capelli A., M.
Balancing reactivity and antitumor activity: heteroarylthioacetamide derivatives as potent and time-dependent inhibitors of EGFR 1-gen-2019 Castelli, R; Bozza, N; Cavazzoni, A; Bonelli, M; Vacondio, F; Ferlenghi, F; Callegari, D; Silva, C; Rivara, S; Lodola, A; Digiacomo, G; Fumarola, C; Alfieri, R; Petronini, Pg; Mor, M.
Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines 1-gen-2020 Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele.