Sfoglia per Autore
Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups
2000-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Cytokinin-like activity of N,N'-diphenylureas. N,N'-bis-(2,3-methylenedioxyphenyl)urea and N,N'-bis-(3,4-methylenedioxyphenyl)urea enhance adventitious root formation in apple rootstock M26 (Malus pumila Mill)
2001-01-01 Ricci, Ada; Carra, A.; Torelli, Anna; Maggiali, Cesare Augusto; Morini, Giovanni; Branca, Camillo
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays
2003-01-01 Zuliani, Valentina; Bordi, Fabrizio; Rivara, Mirko; Silva, Claudia; Vacondio, Federica; Morini, Giovanni; Rivara, Silvia; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Magnanini, F.; Plazzi, Pier Vincenzo
Synthesis and 3D-QSAR Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group
2003-01-01 Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Plazzi, Pier Vincenzo; Carrupt, P. A.; Testa, B.
Synthesis of benzisoxazole and benzisothiazole derivatives with potential antitumor activity
2004-01-01 Incerti, Matteo; Vicini, Paola; Morini, Giovanni; Comini, Mara
Effect of Cl-Substitution on Rooting- or Cytokinin-like Activity of Diphenylurea Derivatives
2005-01-01 Ricci, Ada; Carra, A.; Rolli, Enrico; Bertoletti, C.; Morini, Giovanni; Incerti, Matteo; Vicini, Paola
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists
2005-01-01 Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series
2006-01-01 Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo
Discovery of histamine H3 receptor antagonistic property of simple imidazole-free derivatives: preliminary pharmacological investigation.
2006-01-01 Barocelli, Elisabetta; Ballabeni, Vigilio; Manenti, V; Flammini, Lisa; Bertoni, Simona; Morini, Giovanni; Comini, Mara; Impicciatore, Mariannina
Diheteroarylurea derivatives as adventitious rooting adjuvants in mung bean shoots and M26 apple rootstock.
2006-01-01 Ricci, Ada; Incerti, Matteo; Rolli, Enrico; Vicini, Paola; Morini, Giovanni; Comini, M; Branca, Camillo
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold.
2006-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
In vitro pharmacology at human histamine H(3) receptors and brain access of non-imidazole alkylpiperidine derivatives.
2007-01-01 Bertoni, Simona; Flammini, Lisa; Manenti, V.; Ballabeni, Vigilio; Morini, Giovanni; Comini, Mara; Barocelli, Elisabetta
A promising imidazole-free histamine H3 receptor antagonist with good brain penetration and anticholinesterase activity.
2008-01-01 Barocelli, Elisabetta; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ghizzardi, Paola; Gobbetti, Thomas; Morini, Giovanni; Ballabeni, Vigilio
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity.
2008-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity.
2008-01-01 Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Saccani, Francesca; Domenichini, Giuseppe; Morini, Giovanni; Comini, Mara; Rivara, Mirko; Barocelli, Elisabetta
Multi-target-directed ligands: new histamine H3 receptor antagonists with anticholinesterase activity
2009-01-01 Flammini, Lisa; Bertoni, Simona; Saccani, Francesca; Incerti, Matteo; Morini, Giovanni; Ballabeni, Vigilio; Barocelli, Elisabetta
Dual-Acting Drugs: an in vitro Study of Nonimidazole Histamine H(3) Receptor Antagonists Combining Anticholinesterase Activity
2010-01-01 Incerti, Matteo; Flammini, Lisa; Saccani, Francesca; Morini, Giovanni; Comini, Mara; Coruzzi, Massimo; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma.
2011-01-01 Vacondio, Federica; Silva, Claudia; Morini, Giovanni; Bordi, Fabrizio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups | 1-gen-2000 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo | |
Cytokinin-like activity of N,N'-diphenylureas. N,N'-bis-(2,3-methylenedioxyphenyl)urea and N,N'-bis-(3,4-methylenedioxyphenyl)urea enhance adventitious root formation in apple rootstock M26 (Malus pumila Mill) | 1-gen-2001 | Ricci, Ada; Carra, A.; Torelli, Anna; Maggiali, Cesare Augusto; Morini, Giovanni; Branca, Camillo | |
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays | 1-gen-2003 | Zuliani, Valentina; Bordi, Fabrizio; Rivara, Mirko; Silva, Claudia; Vacondio, Federica; Morini, Giovanni; Rivara, Silvia; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Magnanini, F.; Plazzi, Pier Vincenzo | |
Synthesis and 3D-QSAR Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group | 1-gen-2003 | Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Plazzi, Pier Vincenzo; Carrupt, P. A.; Testa, B. | |
Synthesis of benzisoxazole and benzisothiazole derivatives with potential antitumor activity | 1-gen-2004 | Incerti, Matteo; Vicini, Paola; Morini, Giovanni; Comini, Mara | |
Effect of Cl-Substitution on Rooting- or Cytokinin-like Activity of Diphenylurea Derivatives | 1-gen-2005 | Ricci, Ada; Carra, A.; Rolli, Enrico; Bertoletti, C.; Morini, Giovanni; Incerti, Matteo; Vicini, Paola | |
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists | 1-gen-2005 | Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series | 1-gen-2006 | Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo | |
Discovery of histamine H3 receptor antagonistic property of simple imidazole-free derivatives: preliminary pharmacological investigation. | 1-gen-2006 | Barocelli, Elisabetta; Ballabeni, Vigilio; Manenti, V; Flammini, Lisa; Bertoni, Simona; Morini, Giovanni; Comini, Mara; Impicciatore, Mariannina | |
Diheteroarylurea derivatives as adventitious rooting adjuvants in mung bean shoots and M26 apple rootstock. | 1-gen-2006 | Ricci, Ada; Incerti, Matteo; Rolli, Enrico; Vicini, Paola; Morini, Giovanni; Comini, M; Branca, Camillo | |
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. | 1-gen-2006 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
In vitro pharmacology at human histamine H(3) receptors and brain access of non-imidazole alkylpiperidine derivatives. | 1-gen-2007 | Bertoni, Simona; Flammini, Lisa; Manenti, V.; Ballabeni, Vigilio; Morini, Giovanni; Comini, Mara; Barocelli, Elisabetta | |
A promising imidazole-free histamine H3 receptor antagonist with good brain penetration and anticholinesterase activity. | 1-gen-2008 | Barocelli, Elisabetta; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ghizzardi, Paola; Gobbetti, Thomas; Morini, Giovanni; Ballabeni, Vigilio | |
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. | 1-gen-2008 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity. | 1-gen-2008 | Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Saccani, Francesca; Domenichini, Giuseppe; Morini, Giovanni; Comini, Mara; Rivara, Mirko; Barocelli, Elisabetta | |
Multi-target-directed ligands: new histamine H3 receptor antagonists with anticholinesterase activity | 1-gen-2009 | Flammini, Lisa; Bertoni, Simona; Saccani, Francesca; Incerti, Matteo; Morini, Giovanni; Ballabeni, Vigilio; Barocelli, Elisabetta | |
Dual-Acting Drugs: an in vitro Study of Nonimidazole Histamine H(3) Receptor Antagonists Combining Anticholinesterase Activity | 1-gen-2010 | Incerti, Matteo; Flammini, Lisa; Saccani, Francesca; Morini, Giovanni; Comini, Mara; Coruzzi, Massimo; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona | |
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma. | 1-gen-2011 | Vacondio, Federica; Silva, Claudia; Morini, Giovanni; Bordi, Fabrizio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco |
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