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Mostrati risultati da 21 a 40 di 63
Titolo Data di pubblicazione Autore(i) File
Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design 1-gen-2015 Pieroni, Marco; Wan, Baojie; Zuliani, Valentina; Franzblau, Scott G.; Costantino, Gabriele; Rivara, Mirko
Rational Design and Synthesis of Thioridazine Analogues as Enhancers of the Antituberculosis Therapy 1-gen-2015 Pieroni, Marco; Machado, Diana; Azzali, Elisa; Santos Costa, Sofia; Couto, Isabel; Costantino, Gabriele; Viveiros, Miguel
Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A 1-gen-2015 Pieroni, Marco; Annunziato, Giannamaria; Azzali, Elisa; Dessanti, Paola; Mercurio, Ciro; Meroni, Giuseppe; Trifiró, Paolo; Vianello, Paola; Villa, Manuela; Beato, Claudia; Varasi, Mario; Costantino, Gabriele
Inhibitors of the sulfur assimilation pathway in bacterial pathogens as enhancers of antibiotic therapy 1-gen-2015 Campanini, Barbara; Pieroni, Marco; Raboni, Samanta; Bettati, Stefano; Benoni, Roberto; Pecchini, Chiara; Costantino, Gabriele; Mozzarelli, Andrea
Synthesis of 7-desmethyl analogs of (+)- and (-)-huperzine A 1-gen-2015 Pieroni, Marco; Tipparaju, Suresh K.
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin 1-gen-2016 Vucicevic, Jelica; Srdic Rajic, Tatjana; Pieroni, Marco; Laurila, Jonne M. M.; Perovic, Vladimir; Tassini, Sabrina; Azzali, Elisa; Costantino, Gabriele; Glisic, Sanja; Agbaba, Danica; Scheinin, Mika; Nikolic, Katarina; Radi, Marco; Veljkovic, Nevena
Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR 1-gen-2016 Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma; Pecchini, Chiara; Bruno, Agostino; Magalhães, Joana; Bettati, Stefano; Franko, Nina; Mozzarelli, Andrea; Costantino, Gabriele
Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches 1-gen-2016 Annunziato, Giannamaria; Angeli, Andrea; D'Alba, Francesca; Bruno, Agostino; Pieroni, Marco; Vullo, Daniela; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T.; Costantino, Gabriele
Cyclopropane derivatives as potential human serine racemase inhibitors: unveiling novel insights into a difficult target 1-gen-2016 Beato, Claudia; Pecchini, Chiara; Cocconcelli, Chiara; Campanini, Barbara; Marchetti, Marialaura; Pieroni, Marco; Mozzarelli, Andrea; Costantino, Gabriele
Rational Design, Synthesis and Preliminary Structure-Activity Relationships of α-Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella Typhimurium O-Acetylserine Sulfhydrylase 1-gen-2016 Pieroni, Marco; Annunziato, Giannamaria; Beato, Claudia; Wouters, R.; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma; Bettati, Stefano; Mozzarelli, Andrea; Costantino, Gabriele
An Experimental Model for the Rapid Screening of Compounds with Potential Use Against Mycobacteria 1-gen-2016 Costa, Sofia Santos; Lopes, Elizeth; Azzali, Elisa; Machado, Diana; Coelho, Tatiane; Da Silva, Pedro Eduardo Almeida; Viveiros, Miguel; Pieroni, Marco; Couto, Isabel
Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary Diseases 1-gen-2017 Tassini, Sabrina; Sun, Liang; Lanko, Kristina; Crespan, Emmanuele; Langron, Emily; Falchi, Federico; Kissova, Miroslava; Armijos Rivera, Jorge I.; Delang, Leen; Mirabelli, Carmen; Neyts, Johan; Pieroni, Marco; Cavalli, Andrea; Costantino, Gabriele; Maga, Giovanni; Vergani, Paola; Leyssen, Pieter; Radi, Marco
Substituted N-Phenyl-5-(2-(phenylamino)thiazol-4-yl)isoxazole-3-carboxamides Are Valuable Antitubercular Candidates that Evade Innate Efflux Machinery 1-gen-2017 Azzali, Elisa; Machado, Diana; Kaushik, Amit; Vacondio, Federica; Flisi, Sara; Cabassi, Clotilde Silvia; Lamichhane, Gyanu; Viveiros, Miguel; Costantino, Gabriele; Pieroni, Marco
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents 1-gen-2017 Pieroni, Marco; Azzali, Elisa; Basilico, Nicoletta; Parapini, Silvia; Zolkiewski, Michal; Beato, Claudia; Annunziato, Giannamaria; Bruno, Agostino; Vacondio, Federica; Costantino, Gabriele
Modulation of bacterial metabolism by the microenvironment controls MAIT cell stimulation 1-gen-2018 Schmaler, Mathias; Colone, Alessia; Spagnuolo, Julian; Lepore, Marco; Kalinichenko, Artem; Bhatia, Sumedha; Pavelka, Norman; Rutishauser, Tobias; Egli, Adrian; Azzali, Elisa; Pieroni, Marco; Costantino, Gabriele; Hruz, Petr; Mori, Lucia; de Libero, Gennaro
Sodium Hyaluronate Microparticles for Pulmonary Delivery of Anti-mycobacterial Drugs 1-gen-2018 Rossi, I.; Buttini, F.; Affaticati, Filippo; Sonvico, F.; Pieroni, M.; Bettini, R.
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design 1-gen-2018 Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara
Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting Mycobacterium tuberculosis energetics 1-gen-2018 Machado, Diana; Azzali, Elisa; Couto, Isabel; Costantino, Gabriele; Pieroni, Marco; Viveiros, Miguel
Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains 1-gen-2018 Machado, Diana; Perdigão, João; Portugal, Isabel; Pieroni, Marco; Silva, Pedro A.; Couto and Miguel Viveiros, Isabel
Modulation of bacterial metabolism by the microenvironment controls MAIT cell stimulation article 1-gen-2018 Schmaler, M.; Colone, A.; Spagnuolo, J.; Zimmermann, M.; Lepore, M.; Kalinichenko, A.; Bhatia, S.; Cottier, F.; Rutishauser, T.; Pavelka, N.; Egli, A.; Azzali, E.; Pieroni, M.; Costantino, G.; Hruz, P.; Sauer, U.; Mori, L.; De Libero, G.
Mostrati risultati da 21 a 40 di 63
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