Sfoglia per Autore
Recent advances in the development of melatonin MT(1) and MT(2) receptor agonists.
2010-01-01 Mor, Marco; Rivara, Silvia; Pala, Daniele; A., Bedini; G., Spadoni; G., Tarzia
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives.
2011-01-01 A., Bedini; S., Lucarini; G., Spadoni; G., Tarzia; F., Scaglione; S., Dugnani; M., Pannacci; V., Lucini; Carmi, Caterina; Pala, Daniele; Rivara, Silvia; Mor, Marco
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists
2012-01-01 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Design and structure-activity relationships of amino acid derivatives of lithocholic acid as novel EphA2 receptor antagonists.
2012-01-01 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Iftiin Hassan Mohamed, ; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-[[(3-O-Substituted)anilino]alkyl]amides.
2012-01-01 Rivara, Silvia; Pala, Daniele; Lodola, Alessio; Mor, Marco; Lucini, V.; Dugnani, S.; Scaglione, F.; Bedini, A.; Lucarini, S.; Tarzia, G.; Spadoni, G.
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain.
2012-01-01 Bordi, Fabrizio; Rivara, Silvia; E., Dallaturca; Carmi, Caterina; Pala, Daniele; Lodola, Alessio; Vacondio, Federica; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Computer-Aided Design of Novel Antagonists of the EphA2 Receptor
2013-01-01 Pala, Daniele; Rivara, Silvia; Incerti, Matteo; Tognolini, Massimiliano; Mor, Marco
Target-hopping: a useful approach to identify novel Eph receptor antagonists
2013-01-01 Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Pala, Daniele; Russo, Simonetta; Lodola, Alessio; Incerti, Matteo; Barocelli, Elisabetta; Tognolini, Massimiliano
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties
2013-01-01 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano
Structure-based virtual screening of MT2 melatonin receptor: influence of template choice and structural refinement.
2013-01-01 Pala, Daniele; Beuming, T; Sherman, W; Lodola, Alessio; Rivara, Silvia; Mor, Marco
Synthesis of (E)-8-(3-chlorostyryl)caffeine analogs leading to 9-deazaxanthine derivatives as dual A2A antagonists /MAO-B inhibitors.
2013-01-01 Rivara, Silvia; Piersanti, G.; Bartoccini, F.; Diamantini, G.; Pala, Daniele; Riccioni, T.; Stasi, M. A.; Cabri, W.; Borsini, F.; Mor, Marco; Tarzia, G.; Minetti, P.
Homology models of melatonin receptors: challenges and recent advances.
2013-01-01 Pala, Daniele; Lodola, Alessio; Bedini, A.; Spadoni, G.; Rivara, Silvia
Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor.
2013-01-01 Russo, Simonetta; Incerti, Matteo; Tognolini, Massimiliano; Castelli, Riccardo; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; De Franco, F; Gioiello, A; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Complex product composition generates risks for generic substitution also with dosage forms for intravenous administration
2013-01-01 Rossi, Alessandra; Buttini, Francesca; Colombo, Paolo; Mor, Marco; Pala, Daniele; F., Bortolotti; Colombo, Gaia
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor.
2013-01-01 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity
2014-01-01 Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Barocelli, Elisabetta; Bertoni, Simona; Pala, Daniele; Mor, Marco; Russo, Simonetta; Lodola, Alessio
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction.
2014-01-01 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Castelli, Riccardo; Pala, Daniele; Mor, Marco; Barocelli, Elisabetta; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis
2014-01-01 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta; Mor, Marco; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Tognolini, Massimiliano
Combining ligand- and structure-based approaches for the discovery of new inhibitors of the EPHA2-ephrin-A1 interaction
2014-01-01 Pala, Daniele; Castelli, Riccardo; Incerti, Matteo; Russo, Simonetta; Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Zanotti, Ilaria; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Synthesis and characterization of new bivalent agents as melatonin- and histamine h3-ligands.
2014-01-01 Pala, Daniele; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Flammini, Lisa; Barocelli, Elisabetta; Lucini, V; Scaglione, F; Bartolucci, S; Bedini, A; Rivara, Silvia; Spadoni, G.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Recent advances in the development of melatonin MT(1) and MT(2) receptor agonists. | 1-gen-2010 | Mor, Marco; Rivara, Silvia; Pala, Daniele; A., Bedini; G., Spadoni; G., Tarzia | |
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives. | 1-gen-2011 | A., Bedini; S., Lucarini; G., Spadoni; G., Tarzia; F., Scaglione; S., Dugnani; M., Pannacci; V., Lucini; Carmi, Caterina; Pala, Daniele; Rivara, Silvia; Mor, Marco | |
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists | 1-gen-2012 | Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio | |
Design and structure-activity relationships of amino acid derivatives of lithocholic acid as novel EphA2 receptor antagonists. | 1-gen-2012 | Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Iftiin Hassan Mohamed, ; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio | |
MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-[[(3-O-Substituted)anilino]alkyl]amides. | 1-gen-2012 | Rivara, Silvia; Pala, Daniele; Lodola, Alessio; Mor, Marco; Lucini, V.; Dugnani, S.; Scaglione, F.; Bedini, A.; Lucarini, S.; Tarzia, G.; Spadoni, G. | |
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain. | 1-gen-2012 | Bordi, Fabrizio; Rivara, Silvia; E., Dallaturca; Carmi, Caterina; Pala, Daniele; Lodola, Alessio; Vacondio, Federica; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
Computer-Aided Design of Novel Antagonists of the EphA2 Receptor | 1-gen-2013 | Pala, Daniele; Rivara, Silvia; Incerti, Matteo; Tognolini, Massimiliano; Mor, Marco | |
Target-hopping: a useful approach to identify novel Eph receptor antagonists | 1-gen-2013 | Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Pala, Daniele; Russo, Simonetta; Lodola, Alessio; Incerti, Matteo; Barocelli, Elisabetta; Tognolini, Massimiliano | |
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties | 1-gen-2013 | HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano | |
Structure-based virtual screening of MT2 melatonin receptor: influence of template choice and structural refinement. | 1-gen-2013 | Pala, Daniele; Beuming, T; Sherman, W; Lodola, Alessio; Rivara, Silvia; Mor, Marco | |
Synthesis of (E)-8-(3-chlorostyryl)caffeine analogs leading to 9-deazaxanthine derivatives as dual A2A antagonists /MAO-B inhibitors. | 1-gen-2013 | Rivara, Silvia; Piersanti, G.; Bartoccini, F.; Diamantini, G.; Pala, Daniele; Riccioni, T.; Stasi, M. A.; Cabri, W.; Borsini, F.; Mor, Marco; Tarzia, G.; Minetti, P. | |
Homology models of melatonin receptors: challenges and recent advances. | 1-gen-2013 | Pala, Daniele; Lodola, Alessio; Bedini, A.; Spadoni, G.; Rivara, Silvia | |
Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor. | 1-gen-2013 | Russo, Simonetta; Incerti, Matteo; Tognolini, Massimiliano; Castelli, Riccardo; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; De Franco, F; Gioiello, A; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio | |
Complex product composition generates risks for generic substitution also with dosage forms for intravenous administration | 1-gen-2013 | Rossi, Alessandra; Buttini, Francesca; Colombo, Paolo; Mor, Marco; Pala, Daniele; F., Bortolotti; Colombo, Gaia | |
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. | 1-gen-2013 | Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio | |
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity | 1-gen-2014 | Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Barocelli, Elisabetta; Bertoni, Simona; Pala, Daniele; Mor, Marco; Russo, Simonetta; Lodola, Alessio | |
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction. | 1-gen-2014 | Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Castelli, Riccardo; Pala, Daniele; Mor, Marco; Barocelli, Elisabetta; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio | |
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis | 1-gen-2014 | HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta; Mor, Marco; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Tognolini, Massimiliano | |
Combining ligand- and structure-based approaches for the discovery of new inhibitors of the EPHA2-ephrin-A1 interaction | 1-gen-2014 | Pala, Daniele; Castelli, Riccardo; Incerti, Matteo; Russo, Simonetta; Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Zanotti, Ilaria; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio | |
Synthesis and characterization of new bivalent agents as melatonin- and histamine h3-ligands. | 1-gen-2014 | Pala, Daniele; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Flammini, Lisa; Barocelli, Elisabetta; Lucini, V; Scaglione, F; Bartolucci, S; Bedini, A; Rivara, Silvia; Spadoni, G. |
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