Sfoglia per Rivista ACS MEDICINAL CHEMISTRY LETTERS
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry
2020-01-01 Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M.
Covalent Inhibitors of Plasmodium falciparum Glyceraldehyde 3-Phosphate Dehydrogenase with Antimalarial Activity in Vitro
2019-01-01 Cullia, G.; Bruno, S.; Parapini, S.; Margiotta, M.; Tamborini, L.; Pinto, A.; Galbiati, A.; Mozzarelli, A.; Persico, M.; Paladino, A.; Fattorusso, C.; Taramelli, D.; Conti, P.
Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture
2020-01-01 Pala, N.; Esposito, F.; Tramontano, E.; Singh, P. K.; Sanna, V.; Carcelli, M.; Haigh, L. D.; Satta, S.; Sechi, M.
Exploring Heteroaryl-pyrazole Carboxylic Acids as Human Carbonic Anhydrase XII Inhibitors
2017-01-01 Cadoni, Roberta; Pala, Nicolino; Lomelino, Carrie; Mahon, Brian P.; Mckenna, Robert; Dallocchio, Roberto; Dessã¬, Alessandro; Carcelli, Mauro; Rogolino, Dominga; Sanna, Vanna; Rassu, Mauro; Iaccarino, Ciro; Vullo, Daniela; Supuran, Claudiu T.; Sechi, Mario
How a Blockchain Approach Can Improve Data Reliability in the COVID-19 Pandemic
2022-01-01 Cozzini, Pietro; Agosta, Federica; Dolcetti, Greta; Righi, Gianfranco
Identification of Isoform 2 Acid-Sensing Ion Channel Inhibitors as Tool Compounds for Target Validation Studies in CNS
2019-01-01 Bencheva, L. I.; De Matteo, M.; Ferrante, L.; Ferrara, M.; Prandi, A.; Randazzo, P.; Ronzoni, S.; Sinisi, R.; Seneci, P.; Summa, V.; Gallo, M.; Veneziano, M.; Cellucci, A.; Mazzocchi, N.; Menegon, A.; Di Fabio, R.
Inhibition of Human Immunodeficiency Virus-1 Integrase by β-Diketo Acid Coated Gold Nanoparticles
2020-01-01 Sanna, V.; Youssef, M. F.; Pala, N.; Rogolino, D.; Carcelli, M.; Singh, P. K.; Sanchez, T.; Neamati, N.; Sechi, M.
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor
2020-01-01 Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G.
Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches
2022-01-01 Pagnozzi, D.; Pala, N.; Biosa, G.; Dallocchio, R.; Dessi, A.; Singh, P. K.; Rogolino, D.; Di Fiore, A.; De Simone, G.; Supuran, C. T.; Sechi, M.
pippo
2012-01-01 Cantoni, Margherita
Predicting the reactivity of nitrile-carrying compounds with cysteine: a combined computational and experimental study.
2014-01-01 Berteotti, A; Vacondio, Federica; Lodola, Alessio; Bassi, M; Silva, Claudia; Mor, Marco; Cavalli, A.
Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors
2013-01-01 Giulia, Vignaroli; Claudio, Zamperini; Elena, Dreassi; Radi, Marco; Adriano, Angelucci; Patrizia, Sanità; Emmanuele, Crespan; Miroslava, Kissova; Giovanni, Maga; Silvia, Schenone; Francesca, Musumeci; Maurizio, Botta
Scaffold Morphing Approach To Expand the Toolbox of Broad-Spectrum Antivirals Blocking Dengue/Zika Replication
2019-01-01 Vincetti, Paolo; Kaptein, Suzanne J. F.; Costantino, Gabriele; Neyts, Johan; Radi, Marco
Synthesis of Novel 3,5-Disubstituted-2-oxindole Derivatives As Antitumor Agents against Human Nonsmall Cell Lung Cancer
2013-01-01 Nesi, G; Sestito, S; Mey, V; Ricciardi, S; Falasca, M; Danesi, R; Lapucci, A; Breschi, Mc; Fogli, S; Rapposelli, S
Virtual Screening and Biological Validation of Novel Influenza Virus PA Endonuclease Inhibitors
2015-01-01 Pala, Nicolino; Stevaert, Annelies; Dallocchio, Roberto; Dessì, Alessandro; Rogolino, Dominga; Carcelli, Mauro; Sanna, Vanna; Sechi, Mario; Naesens, Lieve
β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine
2012-01-01 A., Armirotti; E., Romeo; S., Ponzano; L., Mengatto; M., Dionisi; C., Karacsonyi; F., Bertozzi; G., Garau; G., Tarozzo; A., Reggiani; T., Bandiera; G., Tarzia; Mor, Marco; D., Piomelli
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry | 1-gen-2020 | Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M. | |
Covalent Inhibitors of Plasmodium falciparum Glyceraldehyde 3-Phosphate Dehydrogenase with Antimalarial Activity in Vitro | 1-gen-2019 | Cullia, G.; Bruno, S.; Parapini, S.; Margiotta, M.; Tamborini, L.; Pinto, A.; Galbiati, A.; Mozzarelli, A.; Persico, M.; Paladino, A.; Fattorusso, C.; Taramelli, D.; Conti, P. | |
Development of a Raltegravir-based Photoaffinity-Labeled Probe for Human Immunodeficiency Virus-1 Integrase Capture | 1-gen-2020 | Pala, N.; Esposito, F.; Tramontano, E.; Singh, P. K.; Sanna, V.; Carcelli, M.; Haigh, L. D.; Satta, S.; Sechi, M. | |
Exploring Heteroaryl-pyrazole Carboxylic Acids as Human Carbonic Anhydrase XII Inhibitors | 1-gen-2017 | Cadoni, Roberta; Pala, Nicolino; Lomelino, Carrie; Mahon, Brian P.; Mckenna, Robert; Dallocchio, Roberto; Dessã¬, Alessandro; Carcelli, Mauro; Rogolino, Dominga; Sanna, Vanna; Rassu, Mauro; Iaccarino, Ciro; Vullo, Daniela; Supuran, Claudiu T.; Sechi, Mario | |
How a Blockchain Approach Can Improve Data Reliability in the COVID-19 Pandemic | 1-gen-2022 | Cozzini, Pietro; Agosta, Federica; Dolcetti, Greta; Righi, Gianfranco | |
Identification of Isoform 2 Acid-Sensing Ion Channel Inhibitors as Tool Compounds for Target Validation Studies in CNS | 1-gen-2019 | Bencheva, L. I.; De Matteo, M.; Ferrante, L.; Ferrara, M.; Prandi, A.; Randazzo, P.; Ronzoni, S.; Sinisi, R.; Seneci, P.; Summa, V.; Gallo, M.; Veneziano, M.; Cellucci, A.; Mazzocchi, N.; Menegon, A.; Di Fabio, R. | |
Inhibition of Human Immunodeficiency Virus-1 Integrase by β-Diketo Acid Coated Gold Nanoparticles | 1-gen-2020 | Sanna, V.; Youssef, M. F.; Pala, N.; Rogolino, D.; Carcelli, M.; Singh, P. K.; Sanchez, T.; Neamati, N.; Sechi, M. | |
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor | 1-gen-2020 | Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G. | |
Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches | 1-gen-2022 | Pagnozzi, D.; Pala, N.; Biosa, G.; Dallocchio, R.; Dessi, A.; Singh, P. K.; Rogolino, D.; Di Fiore, A.; De Simone, G.; Supuran, C. T.; Sechi, M. | |
pippo | 1-gen-2012 | Cantoni, Margherita | |
Predicting the reactivity of nitrile-carrying compounds with cysteine: a combined computational and experimental study. | 1-gen-2014 | Berteotti, A; Vacondio, Federica; Lodola, Alessio; Bassi, M; Silva, Claudia; Mor, Marco; Cavalli, A. | |
Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors | 1-gen-2013 | Giulia, Vignaroli; Claudio, Zamperini; Elena, Dreassi; Radi, Marco; Adriano, Angelucci; Patrizia, Sanità; Emmanuele, Crespan; Miroslava, Kissova; Giovanni, Maga; Silvia, Schenone; Francesca, Musumeci; Maurizio, Botta | |
Scaffold Morphing Approach To Expand the Toolbox of Broad-Spectrum Antivirals Blocking Dengue/Zika Replication | 1-gen-2019 | Vincetti, Paolo; Kaptein, Suzanne J. F.; Costantino, Gabriele; Neyts, Johan; Radi, Marco | |
Synthesis of Novel 3,5-Disubstituted-2-oxindole Derivatives As Antitumor Agents against Human Nonsmall Cell Lung Cancer | 1-gen-2013 | Nesi, G; Sestito, S; Mey, V; Ricciardi, S; Falasca, M; Danesi, R; Lapucci, A; Breschi, Mc; Fogli, S; Rapposelli, S | |
Virtual Screening and Biological Validation of Novel Influenza Virus PA Endonuclease Inhibitors | 1-gen-2015 | Pala, Nicolino; Stevaert, Annelies; Dallocchio, Roberto; Dessì, Alessandro; Rogolino, Dominga; Carcelli, Mauro; Sanna, Vanna; Sechi, Mario; Naesens, Lieve | |
β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal Cysteine | 1-gen-2012 | A., Armirotti; E., Romeo; S., Ponzano; L., Mengatto; M., Dionisi; C., Karacsonyi; F., Bertozzi; G., Garau; G., Tarozzo; A., Reggiani; T., Bandiera; G., Tarzia; Mor, Marco; D., Piomelli |
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