RUSSO, Simonetta

RUSSO, Simonetta  

Dipartimento di Scienze degli Alimenti e del Farmaco  

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Titolo Data di pubblicazione Autore(i) File
270 Discovery, development and optimization of low molecular weight EPH–ephrin protein–protein inhibitors 1-gen-2014 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Barocelli, Elisabetta; Mor, Marco; Pala, Daniele; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. 1-gen-2013 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Biochemical characterization of EphA2 antagonists with improved physico-chemical properties by cell-based assays and surface plasmon resonance analysis 1-gen-2016 Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Bugatti, Antonella; Vacondio, Federica; Barocelli, Elisabetta; Mor, Marco; Pala, Daniele; Hassan Mohamed, Iftiin; Gioiello, Antimo; Rusnati, Marco; Lodola, Alessio; Tognolini, Massimiliano
Changes in digestive cancer diagnosis during the SARS-CoV-2 pandemic in Italy: A nationwide survey 1-gen-2021 Buscarini, E.; Benedetti, A.; Monica, F.; Pasquale, L.; Buttitta, F.; Cameletti, M.; Ferrari, C.; Ricciardiello, L.; Massironi, S.; Bianco, M. A.; Germana, B.; Rodino, S.; Anderloni, A.; Mussetto, A.; Nipote, B.; Russo, S.; Manta, R.; Lauri, A.; Occhipinti, V.; Marco, M. D.; Giovannone, M.; Binda, C.; Sbrancia, M.; Paolo, M. C. D.; de'-Angelis, G. L.; Fiori, G.; Dal-Fante, M.; Caro, G. D.; Usai-Satta, P.; Cesarini, M.; Piras, E.; Stasi, E.; Serio, G.; Montalbano, L. M.; Mirante, V. G.; Burattini, O.; Attardo, S.; Bargiggia, S.; Dinca, M.; Missale, G.; Alvisi, C.; Broglia, F.; Ferraris, L.; Conti-Bellocchi, M. C.; Luigiano, C.; Pallio, S.; Brunacci, M.; Manfrini, C.; Bozzi, R.; Checchin, D.; Togliani, T.; D'Errico, A.; Bazzoli, F.; La Bianca, O.; Berretti, D.; Alvaro, D.
Combining ligand- and structure-based approaches for the discovery of new inhibitors of the EPHA2-ephrin-A1 interaction 1-gen-2014 Pala, Daniele; Castelli, Riccardo; Incerti, Matteo; Russo, Simonetta; Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Zanotti, Ilaria; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction. 1-gen-2014 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Castelli, Riccardo; Pala, Daniele; Mor, Marco; Barocelli, Elisabetta; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists 1-gen-2012 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Design and structure-activity relationships of amino acid derivatives of lithocholic acid as novel EphA2 receptor antagonists. 1-gen-2012 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Iftiin Hassan Mohamed, ; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis 1-gen-2014 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta; Mor, Marco; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Tognolini, Massimiliano
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties 1-gen-2013 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity 1-gen-2014 Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Barocelli, Elisabetta; Bertoni, Simona; Pala, Daniele; Mor, Marco; Russo, Simonetta; Lodola, Alessio
Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return 1-gen-2016 Russo, Simonetta; Callegari, Donatella; Incerti, Matteo; Pala, Daniele; Giorgio, Carmine; Brunetti, Jlenia; Bracci, Luisa; Vicini, Paola; Barocelli, Elisabetta; Capoferri, Luigi; Rivara, Silvia; Tognolini, Massimiliano; Mor, Marco; Lodola, Alessio
Global Prevalence of Protein-Energy Wasting in Kidney Disease: A Meta-analysis of Contemporary Observational Studies From the International Society of Renal Nutrition and Metabolism 1-gen-2018 Carrero, J. J.; Thomas, F.; Nagy, K.; Arogundade, F.; Avesani, C. M.; Chan, M.; Chmielewski, M.; Cordeiro, A. C.; Espinosa-Cuevas, A.; Fiaccadori, E.; Guebre-Egziabher, F.; Hand, R. K.; Hung, A. M.; Ikizler, T. A.; Johansson, L. R.; Kalantar-Zadeh, K.; Karupaiah, T.; Lindholm, B.; Marckmann, P.; Mafra, D.; Parekh, R. S.; Park, J.; Russo, S.; Saxena, A.; Sezer, S.; Teta, D.; Ter Wee, P. M.; Verseput, C.; Wang, A. Y. M.; Xu, H.; Lu, Y.; Molnar, M. Z.; Kovesdy, C. P.
Inhibition of Eph/ephrin interaction with the small molecule UniPR500 improves glucose tolerance in healthy and insulin-resistant mice 1-gen-2019 Giorgio, C; Incerti, M; Pala, D; Russo, S; Chiodelli, P; Rusnati, M; Cantoni, Am; Di Lecce, R; Barocelli, E; Bertoni, S; Ravassard, P; Manenti, F; Piemonti, L; Ferlenghi, F; Lodola, A; Tognolini, M.
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides. 1-gen-2012 Carmi, Caterina; Galvani, Elena; Vacondio, Federica; Rivara, Silvia; Lodola, Alessio; Russo, Simonetta; Bordi, Fabrizio; Costantino, Gianluca; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, A.; Petronini, P. G.; Mor, Marco; Costantino, Gabriele
Mannich base derivatives as novel EGFR irreversible inhibitors 1-gen-2011 Russo, Simonetta; Mor, Marco; Carmi, Caterina; Vacondio, Federica; Petronini, Pier Giorgio; Cavazzoni, Andrea
Mechanical vibrations applied to nondestructive evaluation of materials and structures 1-gen-2017 Collini, L.; Gasparini, G.; Palermo, M.; Russo, S.
Metadynamics for perspective drug design: Computationally driven synthesis of new protein-protein interaction inhibitors targeting the EphA2 receptor 1-gen-2017 Incerti, Matteo; Russo, Simonetta; Callegari, Donatella; Pala, Daniele; Giorgio, Carmine; Zanotti, Ilaria; Barocelli, Elisabetta; Vicini, Paola; Vacondio, Federica; Rivara, Silvia; Castelli, Riccardo; Tognolini, Massimiliano; Lodola, Alessio
Multiple approaches for the discovery and development of small molecules targeting Eph-ephrin protein-protein interaction 1-gen-2015 Tognolini, Massimiliano; Giorgio, Carmine; Incerti, Matteo; Castelli, Riccardo; Festuccia, C.; Rusnati, M.; Vacondio, Federica; Russo, Simonetta; Pala, Daniele; Callegari, Donatella; Mor, Marco; Bertoni, Simona; Ballabeni, Vigilio; Lodola, Alessio; Barocelli, Elisabetta
Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3α-carbamoyloxy derivative with antiangiogenetic properties 1-gen-2020 Incerti, M.; Russo, S.; Corrado, M.; Giorgio, C.; Ballabeni, V.; Chiodelli, P.; Rusnati, M.; Scalvini, L.; Callegari, D.; Castelli, R.; Vacondio, F.; Ferlenghi, F.; Tognolini, M.; Lodola, A.