Sfoglia per Autore
Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A
2015-01-01 Pieroni, Marco; Annunziato, Giannamaria; Azzali, Elisa; Dessanti, Paola; Mercurio, Ciro; Meroni, Giuseppe; Trifiró, Paolo; Vianello, Paola; Villa, Manuela; Beato, Claudia; Varasi, Mario; Costantino, Gabriele
Rational Design, Synthesis and Preliminary Structure-Activity Relationships of α-Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella Typhimurium O-Acetylserine Sulfhydrylase
2016-01-01 Pieroni, Marco; Annunziato, Giannamaria; Beato, Claudia; Wouters, R.; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma; Bettati, Stefano; Mozzarelli, Andrea; Costantino, Gabriele
Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches
2016-01-01 Annunziato, Giannamaria; Angeli, Andrea; D'Alba, Francesca; Bruno, Agostino; Pieroni, Marco; Vullo, Daniela; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T.; Costantino, Gabriele
Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR
2016-01-01 Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma; Pecchini, Chiara; Bruno, Agostino; Magalhães, Joana; Bettati, Stefano; Franko, Nina; Mozzarelli, Andrea; Costantino, Gabriele
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents
2017-01-01 Pieroni, Marco; Azzali, Elisa; Basilico, Nicoletta; Parapini, Silvia; Zolkiewski, Michal; Beato, Claudia; Annunziato, Giannamaria; Bruno, Agostino; Vacondio, Federica; Costantino, Gabriele
Antifungal properties of newly designed carbonic anhydrases inhibitors selective for microbial enzymes
2018-01-01 Giovati, Laura; Annunziato, Giannamaria; Ciociola, Tecla; Magliani, Valter; Polonelli, Luciano; Conti, Stefania; Supuran, Claudiu T.; Costantino, Gabriele
Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets
2018-01-01 Magalhães, Joana; Annunziato, Giannamaria; Franko, Nina; Pieroni, Marco; Campanini, Barbara; Bruno, Agostino; Costantino, Gabriele
Biochemical characterization of Aspergillus fumigatus AroH, a putative aromatic amino acid aminotransferase
2018-01-01 Dindo, Mirco; Costanzi, Egidia; Pieroni, Marco; Costantini, Claudio; Annunziato, Giannamaria; Bruno, Agostino; Keller, Nancy P.; Romani, Luigina; Zelante, Teresa; Cellini, Barbara
Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases
2018-01-01 Annunziato, Giannamaria; Giovati, Laura; Andrea, Angeli; Pavone, Marialaura; Sonia Del Prete, ; Pieroni, Marco; Clemente, Capasso; Bruno, Agostino; Conti, Stefania; Magliani, Valter; Supuran, Claudiu T.; Costantino, Gabriele
In vitro digestion of zingiber officinale extract and evaluation of stability as a first step to determine its bioaccesibility
2018-01-01 Annunziato, Giannamaria; Falavigna, Claudia; Pieroni, Marco; Faccini, Andrea; Micheli, Fabrizio; Costantino, Gabriele
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design
2018-01-01 Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara
Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: Implications for Primary Hyperoxaluria type 1
2019-01-01 Dindo, M.; Grottelli, S.; Annunziato, G.; Giardina, G.; Pieroni, M.; Pampalone, G.; Faccini, A.; Cutruzzola, F.; Laurino, P.; Costantino, G.; Cellini, B.
Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections
2019-01-01 Rossi, Irene; Buttini, Francesca; Sonvico, Fabio; Affaticati, Filippo; Martinelli, Francesco; Annunziato, Giannamaria; Machado, Diana; Viveiros, Miguel; Pieroni, Marco; Bettini, Ruggero
Strategies to overcome antimicrobial resistance (AMR) making use of non-essential target inhibitors: A review
2019-01-01 Annunziato, G.
Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms
2019-01-01 Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Nikitjuka, Anna; Mozzarelli, Andrea; Bettati, Stefano; Karawajczyk, Anna; Jirgensons, Aigars; Campanini, Barbara; Costantino, Gabriele
The aryl hydrocarbon receptor (AhR) mediates the counter-regulatory effects of pelargonidins in models of inflammation and metabolic dysfunctions
2019-01-01 Biagioli, M.; Carino, A.; Fiorucci, C.; Annunziato, G.; Marchiano, S.; Bordoni, M.; Roselli, R.; Giorgio, C. D.; Castiglione, F.; Ricci, P.; Bruno, A.; Faccini, A.; Distrutti, E.; Baldoni, M.; Costantino, G.; Fiorucci, S.
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor
2020-01-01 Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G.
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry
2020-01-01 Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M.
Antimicrobial peptides (AMPs): a patent review (2015-2020)
2020-01-01 Annunziato, Giannamaria; Costantino, Gabriele
Nuovi composti antimicrobici
2021-01-01 Annunziato, Giannamaria; Costantino, Gabriele; Cabassi, Clotilde Silvia; Pieroni, Marco; Bruno, Agostino; Campanini, Barbara; Bettati, Stefano; Mozzarelli, Andrea
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Further insights into the SAR of α-substituted cyclopropylamine derivatives as inhibitors of histone demethylase KDM1A | 1-gen-2015 | Pieroni, Marco; Annunziato, Giannamaria; Azzali, Elisa; Dessanti, Paola; Mercurio, Ciro; Meroni, Giuseppe; Trifiró, Paolo; Vianello, Paola; Villa, Manuela; Beato, Claudia; Varasi, Mario; Costantino, Gabriele | |
| Rational Design, Synthesis and Preliminary Structure-Activity Relationships of α-Substituted-2-Phenylcyclopropane Carboxylic Acids as Inhibitors of Salmonella Typhimurium O-Acetylserine Sulfhydrylase | 1-gen-2016 | Pieroni, Marco; Annunziato, Giannamaria; Beato, Claudia; Wouters, R.; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma; Bettati, Stefano; Mozzarelli, Andrea; Costantino, Gabriele | |
| Discovery of New Potential Anti-Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target-Focused Repurposing Approaches | 1-gen-2016 | Annunziato, Giannamaria; Angeli, Andrea; D'Alba, Francesca; Bruno, Agostino; Pieroni, Marco; Vullo, Daniela; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T.; Costantino, Gabriele | |
| Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR | 1-gen-2016 | Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma; Pecchini, Chiara; Bruno, Agostino; Magalhães, Joana; Bettati, Stefano; Franko, Nina; Mozzarelli, Andrea; Costantino, Gabriele | |
| Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents | 1-gen-2017 | Pieroni, Marco; Azzali, Elisa; Basilico, Nicoletta; Parapini, Silvia; Zolkiewski, Michal; Beato, Claudia; Annunziato, Giannamaria; Bruno, Agostino; Vacondio, Federica; Costantino, Gabriele | |
| Antifungal properties of newly designed carbonic anhydrases inhibitors selective for microbial enzymes | 1-gen-2018 | Giovati, Laura; Annunziato, Giannamaria; Ciociola, Tecla; Magliani, Valter; Polonelli, Luciano; Conti, Stefania; Supuran, Claudiu T.; Costantino, Gabriele | |
| Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets | 1-gen-2018 | Magalhães, Joana; Annunziato, Giannamaria; Franko, Nina; Pieroni, Marco; Campanini, Barbara; Bruno, Agostino; Costantino, Gabriele | |
| Biochemical characterization of Aspergillus fumigatus AroH, a putative aromatic amino acid aminotransferase | 1-gen-2018 | Dindo, Mirco; Costanzi, Egidia; Pieroni, Marco; Costantini, Claudio; Annunziato, Giannamaria; Bruno, Agostino; Keller, Nancy P.; Romani, Luigina; Zelante, Teresa; Cellini, Barbara | |
| Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases | 1-gen-2018 | Annunziato, Giannamaria; Giovati, Laura; Andrea, Angeli; Pavone, Marialaura; Sonia Del Prete, ; Pieroni, Marco; Clemente, Capasso; Bruno, Agostino; Conti, Stefania; Magliani, Valter; Supuran, Claudiu T.; Costantino, Gabriele | |
| In vitro digestion of zingiber officinale extract and evaluation of stability as a first step to determine its bioaccesibility | 1-gen-2018 | Annunziato, Giannamaria; Falavigna, Claudia; Pieroni, Marco; Faccini, Andrea; Micheli, Fabrizio; Costantino, Gabriele | |
| Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design | 1-gen-2018 | Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara | |
| Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: Implications for Primary Hyperoxaluria type 1 | 1-gen-2019 | Dindo, M.; Grottelli, S.; Annunziato, G.; Giardina, G.; Pieroni, M.; Pampalone, G.; Faccini, A.; Cutruzzola, F.; Laurino, P.; Costantino, G.; Cellini, B. | |
| Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections | 1-gen-2019 | Rossi, Irene; Buttini, Francesca; Sonvico, Fabio; Affaticati, Filippo; Martinelli, Francesco; Annunziato, Giannamaria; Machado, Diana; Viveiros, Miguel; Pieroni, Marco; Bettini, Ruggero | |
| Strategies to overcome antimicrobial resistance (AMR) making use of non-essential target inhibitors: A review | 1-gen-2019 | Annunziato, G. | |
| Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms | 1-gen-2019 | Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Nikitjuka, Anna; Mozzarelli, Andrea; Bettati, Stefano; Karawajczyk, Anna; Jirgensons, Aigars; Campanini, Barbara; Costantino, Gabriele | |
| The aryl hydrocarbon receptor (AhR) mediates the counter-regulatory effects of pelargonidins in models of inflammation and metabolic dysfunctions | 1-gen-2019 | Biagioli, M.; Carino, A.; Fiorucci, C.; Annunziato, G.; Marchiano, S.; Bordoni, M.; Roselli, R.; Giorgio, C. D.; Castiglione, F.; Ricci, P.; Bruno, A.; Faccini, A.; Distrutti, E.; Baldoni, M.; Costantino, G.; Fiorucci, S. | |
| Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor | 1-gen-2020 | Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G. | |
| 2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry | 1-gen-2020 | Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M. | |
| Antimicrobial peptides (AMPs): a patent review (2015-2020) | 1-gen-2020 | Annunziato, Giannamaria; Costantino, Gabriele | |
| Nuovi composti antimicrobici | 1-gen-2021 | Annunziato, Giannamaria; Costantino, Gabriele; Cabassi, Clotilde Silvia; Pieroni, Marco; Bruno, Agostino; Campanini, Barbara; Bettati, Stefano; Mozzarelli, Andrea |
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