Sfoglia per Autore
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity
2004-01-01 Lucini, V.; Pannacci, M.; Scaglione, F.; Fraschini, F.; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Piersanti, G.; Diamantini, G.; Tarzia, G.
Indole-based analogs of melatonin: in vitro antioxidant and cytoprotective activities
2004-01-01 Mor, Marco; Silva, Claudia; Vacondio, Federica; Plazzi, Pier Vincenzo; Bertoni, Simona; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Zusso, M.; Franceschini, D.; Giusti, P.
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists
2004-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors
2005-01-01 Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G.
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists
2005-01-01 Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Analysis of Structure-Activity Relationships for MT2 Selective Antagonists by Melatonin MT1 and MT2 Receptor Models
2005-01-01 Rivara, Silvia; Lorenzi, Simone; Mor, Marco; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Tarzia, G.
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity
2006-01-01 Spadoni, G; Diamantini, G; Bedini, A; Tarzia, G; Vacondio, Federica; Silva, Claudia; Rivara, Mirko; Mor, Marco; Plazzi, Pier Vincenzo; Zusso, M; Franceschini, D; Giusti, P.
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series
2006-01-01 Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo
Synthesis and Structure-Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring
2006-01-01 Tarzia, G; Duranti, A; Gatti, G; Piersanti, G; Tontini, A; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Mor, Marco; Kathuria, S; Piomelli, D.
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold.
2006-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity
2006-01-01 Carmi, Caterina; Cavazzoni, Andrea; Zuliani, Valentina; Lodola, Alessio; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano
2007-01-01 Cavazzoni, Andrea; Galetti, Maricla; LA MONICA, S; Fumarola, C; Bonelli, Mara; Carmi, C; Zuliani, Valentina; Lodola, Alessio; Bordi, F; Plazzi, P. V.; Mor, Marco; Petronini, Pg
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor.
2008-01-01 Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity.
2008-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine
2009-01-01 Rivara, Mirko; Zuliani, Valentina; Plazzi, Pier Vincenzo; Bordi, Fabrizio
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line
2009-01-01 Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity | 1-gen-2004 | Lucini, V.; Pannacci, M.; Scaglione, F.; Fraschini, F.; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Piersanti, G.; Diamantini, G.; Tarzia, G. | |
Indole-based analogs of melatonin: in vitro antioxidant and cytoprotective activities | 1-gen-2004 | Mor, Marco; Silva, Claudia; Vacondio, Federica; Plazzi, Pier Vincenzo; Bertoni, Simona; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Zusso, M.; Franceschini, D.; Giusti, P. | |
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists | 1-gen-2004 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo | |
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors | 1-gen-2005 | Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G. | |
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists | 1-gen-2005 | Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
Analysis of Structure-Activity Relationships for MT2 Selective Antagonists by Melatonin MT1 and MT2 Receptor Models | 1-gen-2005 | Rivara, Silvia; Lorenzi, Simone; Mor, Marco; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Tarzia, G. | |
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity | 1-gen-2006 | Spadoni, G; Diamantini, G; Bedini, A; Tarzia, G; Vacondio, Federica; Silva, Claudia; Rivara, Mirko; Mor, Marco; Plazzi, Pier Vincenzo; Zusso, M; Franceschini, D; Giusti, P. | |
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series | 1-gen-2006 | Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo | |
Synthesis and Structure-Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring | 1-gen-2006 | Tarzia, G; Duranti, A; Gatti, G; Piersanti, G; Tontini, A; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Mor, Marco; Kathuria, S; Piomelli, D. | |
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. | 1-gen-2006 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity | 1-gen-2006 | Carmi, Caterina; Cavazzoni, Andrea; Zuliani, Valentina; Lodola, Alessio; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco | |
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano | 1-gen-2007 | Cavazzoni, Andrea; Galetti, Maricla; LA MONICA, S; Fumarola, C; Bonelli, Mara; Carmi, C; Zuliani, Valentina; Lodola, Alessio; Bordi, F; Plazzi, P. V.; Mor, Marco; Petronini, Pg | |
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. | 1-gen-2008 | Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. | 1-gen-2008 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine | 1-gen-2009 | Rivara, Mirko; Zuliani, Valentina; Plazzi, Pier Vincenzo; Bordi, Fabrizio | |
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line | 1-gen-2009 | Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco |
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