Sfoglia per Autore
Structure activity relationship of new EphA2 ligands
2011-01-01 Tognolini, Massimiliano; Incerti, Matteo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Barocelli, Elisabetta; Russo, Simonetta; B., Lelli; L., Bracci; Lodola, Alessio
Mannich base derivatives as novel EGFR irreversible inhibitors
2011-01-01 Russo, Simonetta; Mor, Marco; Carmi, Caterina; Vacondio, Federica; Petronini, Pier Giorgio; Cavazzoni, Andrea
Design and structure-activity relationships of amino acid derivatives of lithocholic acid as novel EphA2 receptor antagonists.
2012-01-01 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Iftiin Hassan Mohamed, ; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists
2012-01-01 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Structure-activity realtionships of new EphaA2 ligands
2012-01-01 Russo, Simonetta
Structure–Activity Relationships and Mechanism of Action of Eph–ephrin Antagonists: Interaction of Cholanic Acid with the EphA2 Receptor
2012-01-01 Tognolini, Massimiliano; Incerti, Matteo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Bruni, Renato; Barbara, Lelli; Luisa, Bracci; Roberta, Noberini; Elena, B. Pasquale; Barocelli, Elisabetta; Vicini, Paola; Mor, Marco; Lodola, Alessio
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides.
2012-01-01 Carmi, Caterina; Galvani, Elena; Vacondio, Federica; Rivara, Silvia; Lodola, Alessio; Russo, Simonetta; Bordi, Fabrizio; Costantino, Gianluca; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, A.; Petronini, P. G.; Mor, Marco; Costantino, Gabriele
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor.
2013-01-01 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Target-hopping: a useful approach to identify novel Eph receptor antagonists
2013-01-01 Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Pala, Daniele; Russo, Simonetta; Lodola, Alessio; Incerti, Matteo; Barocelli, Elisabetta; Tognolini, Massimiliano
Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor.
2013-01-01 Russo, Simonetta; Incerti, Matteo; Tognolini, Massimiliano; Castelli, Riccardo; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; De Franco, F; Gioiello, A; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties
2013-01-01 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano
Target Hopping as a Useful Tool for the Identification of Novel EphA2 Protein–Protein Antagonists
2014-01-01 Tognolini, Massimiliano; Incerti, Matteo; Pala, Daniele; Russo, Simonetta; Castelli, Riccardo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Lodola, Alessio
Combining ligand- and structure-based approaches for the discovery of new inhibitors of the EPHA2-ephrin-A1 interaction
2014-01-01 Pala, Daniele; Castelli, Riccardo; Incerti, Matteo; Russo, Simonetta; Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Zanotti, Ilaria; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio
UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations.
2014-01-01 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Russo, Simonetta; Pala, Daniele; Pasquale, Eb; Zanotti, Ilaria; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano
270 Discovery, development and optimization of low molecular weight EPH–ephrin protein–protein inhibitors
2014-01-01 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Barocelli, Elisabetta; Mor, Marco; Pala, Daniele; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity
2014-01-01 Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Barocelli, Elisabetta; Bertoni, Simona; Pala, Daniele; Mor, Marco; Russo, Simonetta; Lodola, Alessio
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis
2014-01-01 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta; Mor, Marco; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Tognolini, Massimiliano
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction.
2014-01-01 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Castelli, Riccardo; Pala, Daniele; Mor, Marco; Barocelli, Elisabetta; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
Multiple approaches for the discovery and development of small molecules targeting Eph-ephrin protein-protein interaction
2015-01-01 Tognolini, Massimiliano; Giorgio, Carmine; Incerti, Matteo; Castelli, Riccardo; Festuccia, C.; Rusnati, M.; Vacondio, Federica; Russo, Simonetta; Pala, Daniele; Callegari, Donatella; Mor, Marco; Bertoni, Simona; Ballabeni, Vigilio; Lodola, Alessio; Barocelli, Elisabetta
Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return
2016-01-01 Russo, Simonetta; Callegari, Donatella; Incerti, Matteo; Pala, Daniele; Giorgio, Carmine; Brunetti, Jlenia; Bracci, Luisa; Vicini, Paola; Barocelli, Elisabetta; Capoferri, Luigi; Rivara, Silvia; Tognolini, Massimiliano; Mor, Marco; Lodola, Alessio
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Structure activity relationship of new EphA2 ligands | 1-gen-2011 | Tognolini, Massimiliano; Incerti, Matteo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Barocelli, Elisabetta; Russo, Simonetta; B., Lelli; L., Bracci; Lodola, Alessio | |
Mannich base derivatives as novel EGFR irreversible inhibitors | 1-gen-2011 | Russo, Simonetta; Mor, Marco; Carmi, Caterina; Vacondio, Federica; Petronini, Pier Giorgio; Cavazzoni, Andrea | |
Design and structure-activity relationships of amino acid derivatives of lithocholic acid as novel EphA2 receptor antagonists. | 1-gen-2012 | Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Iftiin Hassan Mohamed, ; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio | |
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists | 1-gen-2012 | Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio | |
Structure-activity realtionships of new EphaA2 ligands | 1-gen-2012 | Russo, Simonetta | |
Structure–Activity Relationships and Mechanism of Action of Eph–ephrin Antagonists: Interaction of Cholanic Acid with the EphA2 Receptor | 1-gen-2012 | Tognolini, Massimiliano; Incerti, Matteo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Bruni, Renato; Barbara, Lelli; Luisa, Bracci; Roberta, Noberini; Elena, B. Pasquale; Barocelli, Elisabetta; Vicini, Paola; Mor, Marco; Lodola, Alessio | |
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides. | 1-gen-2012 | Carmi, Caterina; Galvani, Elena; Vacondio, Federica; Rivara, Silvia; Lodola, Alessio; Russo, Simonetta; Bordi, Fabrizio; Costantino, Gianluca; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, A.; Petronini, P. G.; Mor, Marco; Costantino, Gabriele | |
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. | 1-gen-2013 | Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio | |
Target-hopping: a useful approach to identify novel Eph receptor antagonists | 1-gen-2013 | Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Pala, Daniele; Russo, Simonetta; Lodola, Alessio; Incerti, Matteo; Barocelli, Elisabetta; Tognolini, Massimiliano | |
Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor. | 1-gen-2013 | Russo, Simonetta; Incerti, Matteo; Tognolini, Massimiliano; Castelli, Riccardo; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; De Franco, F; Gioiello, A; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio | |
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties | 1-gen-2013 | HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano | |
Target Hopping as a Useful Tool for the Identification of Novel EphA2 Protein–Protein Antagonists | 1-gen-2014 | Tognolini, Massimiliano; Incerti, Matteo; Pala, Daniele; Russo, Simonetta; Castelli, Riccardo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Lodola, Alessio | |
Combining ligand- and structure-based approaches for the discovery of new inhibitors of the EPHA2-ephrin-A1 interaction | 1-gen-2014 | Pala, Daniele; Castelli, Riccardo; Incerti, Matteo; Russo, Simonetta; Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Zanotti, Ilaria; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio | |
UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations. | 1-gen-2014 | HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Russo, Simonetta; Pala, Daniele; Pasquale, Eb; Zanotti, Ilaria; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano | |
270 Discovery, development and optimization of low molecular weight EPH–ephrin protein–protein inhibitors | 1-gen-2014 | Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Barocelli, Elisabetta; Mor, Marco; Pala, Daniele; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio | |
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity | 1-gen-2014 | Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Barocelli, Elisabetta; Bertoni, Simona; Pala, Daniele; Mor, Marco; Russo, Simonetta; Lodola, Alessio | |
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis | 1-gen-2014 | HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta; Mor, Marco; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Tognolini, Massimiliano | |
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction. | 1-gen-2014 | Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Castelli, Riccardo; Pala, Daniele; Mor, Marco; Barocelli, Elisabetta; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio | |
Multiple approaches for the discovery and development of small molecules targeting Eph-ephrin protein-protein interaction | 1-gen-2015 | Tognolini, Massimiliano; Giorgio, Carmine; Incerti, Matteo; Castelli, Riccardo; Festuccia, C.; Rusnati, M.; Vacondio, Federica; Russo, Simonetta; Pala, Daniele; Callegari, Donatella; Mor, Marco; Bertoni, Simona; Ballabeni, Vigilio; Lodola, Alessio; Barocelli, Elisabetta | |
Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return | 1-gen-2016 | Russo, Simonetta; Callegari, Donatella; Incerti, Matteo; Pala, Daniele; Giorgio, Carmine; Brunetti, Jlenia; Bracci, Luisa; Vicini, Paola; Barocelli, Elisabetta; Capoferri, Luigi; Rivara, Silvia; Tognolini, Massimiliano; Mor, Marco; Lodola, Alessio |
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