RIVARA, Silvia

RIVARA, Silvia  

Dipartimento di Scienze degli Alimenti e del Farmaco  

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Titolo Data di pubblicazione Autore(i) File
2-[N-Acylamino(C1-C3)alkyl]indoles as MT1 Melatonin Receptor Partial Agonists, Antagonists, and Putative Inverse Agonists. 1-gen-1998 Spadoni, G.; Balsamini, C.; Bedini, A.; Diamantini, G.; DI GIACOMO, B.; Tontini, A.; Tarzia, G.; Mor, Marco; Plazzi, P. V.; Rivara, Silvia; Nonno, R.; Pannacci, M.; Lucini, V.; Fraschini, F.; Stankov, B. M.
2-Aminobenzimidazoles as new potent H3-antagonists 1-gen-1999 Zuliani, Valentina; F., Bordi; Mor, Marco; Silva, Claudia; Rivara, Silvia; Vacondio, Federica; Barocelli, Elisabetta; Ballabeni, Vigilio; M., Impicciatore; P. V., Plazzi
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors 1-gen-2022 Mari, M.; Elisi, G. M.; Bedini, A.; Lucarini, S.; Retini, M.; Lucini, V.; Scaglione, F.; Vincenzi, F.; Varani, K.; Castelli, R.; Mor, M.; Rivara, S.; Spadoni, G.
2-N-Acylaminoalkylindoles: Design and Quantitative Structure-Activity Relationship Studies Leading to MT2-Selective Melatonin Antagonists 1-gen-2001 Spadoni, G.; Balsamini, C.; Diamantini, G.; Tontini, A.; Tarzia, G.; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Nonno, R.; Lucini, V.; Pannacci, M.; Fraschini, F.
A sulfonyl fluoride derivative inhibits EGFR L858R/T790M/C797S by covalent modification of the catalytic lysine 1-gen-2021 Ferlenghi, F; Scalvini, L; Vacondio, F; Castelli, R; Bozza, N; Marseglia, G; Rivara, S; Lodola, A; La Monica, S; Minari, R; Petronini, Pg; Alfieri, R; Tiseo, M; Mor, M.
Alchilammidi tricicliche: ligandi selettivi dei recettori melatoninergici MT1 e MT2 1-gen-2003 Spadoni, G; Bedini, A; Tarzia, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Fraschini, F.
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. 1-gen-2013 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Amino acid derivatives as palmitoylethanolamide prodrugs: Synthesis, in vitro metabolism and in vivo plasma profile in rats 1-gen-2015 Vacondio, Federica; Bassi, Michele; Silva, Claudia; Castelli, Riccardo; Carmi, Caterina; Scalvini, Laura; Lodola, Alessio; Vivo, Valentina; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco; Rivara, Silvia
Aminobenzimidazoles as new potent H3-antagonists 1-gen-1999 Zuliani, Valentina; F., Bordi; Mor, Marco; Silva, Claudia; Rivara, Silvia; Vacondio, Federica; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; P. V., Plazzi
An Optimized Workflow for the Discovery of New Antimicrobial Compounds Targeting Bacterial RNA Polymerase Complex Formation 1-gen-2022 Caputo, Alessia; Sartini, Sara; Levati, Elisabetta; Minato, Ilaria; Elisi, Gian Marco; Di Stasi, Adriana; Guillou, Catherine; Goekjian, Peter G; Garcia, Pierre; Gueyrard, David; Bach, Stéphane; Comte, Arnaud; Ottonello, Simone; Rivara, Silvia; Montanini, Barbara
Analysis of Structure-Activity Relationships for MT2 Selective Antagonists by Melatonin MT1 and MT2 Receptor Models 1-gen-2005 Rivara, Silvia; Lorenzi, Simone; Mor, Marco; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Tarzia, G.
Antidepressant-like activity and cardioprotective effects of fatty acid amide hydrolase inhibitor URB694 in socially stressed Wistar Kyoto rats 1-gen-2015 Carnevali, Luca; Vacondio, Federica; Rossi, Stefano; Callegari, Sergio; Macchi, Emilio; Spadoni, Gilberto; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Sgoifo, Andrea
Antidepressant-like effects of pharmacological inhibition of FAAH activity in socially isolated female rats 1-gen-2020 Carnevali, L.; Statello, R.; Vacondio, F.; Ferlenghi, F.; Spadoni, G.; Rivara, S.; Mor, M.; Sgoifo, A.
Antiproliferative and pro-apoptotic activity of melatonin analogues on melanoma and breast cancer cells 1-gen-2017 Gatti, Giuliana; Lucini, Valeria; Dugnani, Silvana; Calastretti, Angela; Spadoni, Gilberto; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Canti, Gianfranco; Scaglione, Francesco; Bevilacqua, Annamaria
Anxiolytic effects of the melatonin MT2 receptor partial agonist UCM765: Comparison with melatonin and diazepam. 1-gen-2012 Ochoa Sanchez, R.; Rainer, Q.; Comai, S.; Spadoni, G.; Bedini, A.; Rivara, Silvia; Fraschini, F.; Mor, Marco; Tarzia, G.; Gobbi, G.
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors 1-gen-2005 Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G.
APPLICATION OF COMPUTATIONAL METHODSTO THE DESIGN OF FATTY ACID AMIDE HYDROLASE(FAAH) INHIBITORS BASED ON A CARBAMICTEMPLATE STRUCTURE 1-gen-2011 Lodola, Alessio; Rivara, Silvia; Mor, Marco
Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs 1-gen-2017 Lodola, Alessio; Bertolini, S; Biagetti, M; Capacchi, S; Facchinetti, F; Gallo, Pm; Pappani, A; Mor, Marco; Pala, Daniele; Rivara, Silvia; Visentini, F; Corsi, M; Capelli A., M.
Balancing reactivity and antitumor activity: heteroarylthioacetamide derivatives as potent and time-dependent inhibitors of EGFR 1-gen-2019 Castelli, R; Bozza, N; Cavazzoni, A; Bonelli, M; Vacondio, F; Ferlenghi, F; Callegari, D; Silva, C; Rivara, S; Lodola, A; Digiacomo, G; Fumarola, C; Alfieri, R; Petronini, Pg; Mor, M.
Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines 1-gen-2020 Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele.