PIERONI, Marco

PIERONI, Marco  

Dipartimento di Scienze degli Alimenti e del Farmaco  

Mostra records
Risultati 1 - 20 di 63 (tempo di esecuzione: 0.059 secondi).
Titolo Data di pubblicazione Autore(i) File
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry 1-gen-2020 Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M.
6-Hydrogen-8-Methylquinolones Active Against Replicating and Non-replicating Mycobacterium tuberculosis 1-gen-2012 Tabarrini, Oriana; Sabatini, Stefano; Massari, Serena; Pieroni, Marco; Franzblau, Scott G.; Cecchetti, Violetta
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin 1-gen-2016 Vucicevic, Jelica; Srdic Rajic, Tatjana; Pieroni, Marco; Laurila, Jonne M. M.; Perovic, Vladimir; Tassini, Sabrina; Azzali, Elisa; Costantino, Gabriele; Glisic, Sanja; Agbaba, Danica; Scheinin, Mika; Nikolic, Katarina; Radi, Marco; Veljkovic, Nevena
A competitive o‐acetylserine sulfhydrylase inhibitor modulates the formation of cysteine synthase complex 1-gen-2021 Marchetti, M.; De Angelis, F. S.; Annunziato, G.; Costantino, G.; Pieroni, M.; Ronda, L.; Mozzarelli, A.; Campanini, B.; Cannistraro, S.; Bizzarri, A. R.; Bettati, S.
Accepting the Invitation to Open Innovation in Malaria Drug Discovery: Synthesis, Biological Evaluation, and Investigation on the Structure-Activity Relationships of Benzo[b]thiophene-2-carboxamides as Antimalarial Agents 1-gen-2017 Pieroni, Marco; Azzali, Elisa; Basilico, Nicoletta; Parapini, Silvia; Zolkiewski, Michal; Beato, Claudia; Annunziato, Giannamaria; Bruno, Agostino; Vacondio, Federica; Costantino, Gabriele
Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting Mycobacterium tuberculosis energetics 1-gen-2018 Machado, Diana; Azzali, Elisa; Couto, Isabel; Costantino, Gabriele; Pieroni, Marco; Viveiros, Miguel
An Experimental Model for the Rapid Screening of Compounds with Potential Use Against Mycobacteria 1-gen-2016 Costa, Sofia Santos; Lopes, Elizeth; Azzali, Elisa; Machado, Diana; Coelho, Tatiane; Da Silva, Pedro Eduardo Almeida; Viveiros, Miguel; Pieroni, Marco; Couto, Isabel
Antituberculosis agents: Beyond medicinal chemistry rules 1-gen-2019 Pieroni, M.
Aspergillus fumigatus tryptophan metabolic route differently affects host immunity 1-gen-2021 Zelante, T.; Choera, T.; Beauvais, A.; Fallarino, F.; Paolicelli, G.; Pieraccini, G.; Pieroni, M.; Galosi, C.; Beato, C.; De Luca, A.; Boscaro, F.; Romoli, R.; Liu, X.; Warris, A.; Verweij, P. E.; Ballard, E.; Borghi, M.; Pariano, M.; Costantino, G.; Calvitti, M.; Vacca, C.; Oikonomou, V.; Gargaro, M.; Wong, A. Y. W.; Boon, L.; den Hartog, M.; Spacil, Z.; Puccetti, P.; Latge, J. -P.; Keller, N. P.; Romani, L.
Biochemical characterization of Aspergillus fumigatus AroH, a putative aromatic amino acid aminotransferase 1-gen-2018 Dindo, Mirco; Costanzi, Egidia; Pieroni, Marco; Costantini, Claudio; Annunziato, Giannamaria; Bruno, Agostino; Keller, Nancy P.; Romani, Luigina; Zelante, Teresa; Cellini, Barbara
Blocking cysteine biosynthesis in Salmonella typhimurium: the moonlighting enzyme CysK as a potential antibiotic target 1-gen-2014 Bettati, Stefano; Spyrakis, F.; Benoni, Roberto; Pieroni, Marco; Costantino, Gabriele; Pecchini, C.; Zani, Franca; Mozzarelli, Andrea
Challenging the drug-likeness dogma for new drug discovery in Tuberculosis 1-gen-2018 Machado, Diana; Girardini, Miriam; Viveiros, Miguel; Pieroni, Marco
Crystal structure of Aspergillus fumigatus AroH, an aromatic amino acid aminotransferase 1-gen-2021 Spizzichino, Sharon; Pampalone, Gioena; Dindo, Mirco; Bruno, Agostino; Romani, Luigina; Cutruzzolà, Francesca; Zelante, Teresa; Pieroni, Marco; Cellini, Barbara; Giardina, Giorgio
Cyclopropane derivatives as potential human serine racemase inhibitors: unveiling novel insights into a difficult target 1-gen-2016 Beato, Claudia; Pecchini, Chiara; Cocconcelli, Chiara; Campanini, Barbara; Marchetti, Marialaura; Pieroni, Marco; Mozzarelli, Andrea; Costantino, Gabriele
Cyclopropane-1,2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR 1-gen-2016 Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma; Pecchini, Chiara; Bruno, Agostino; Magalhães, Joana; Bettati, Stefano; Franko, Nina; Mozzarelli, Andrea; Costantino, Gabriele
Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: Implications for Primary Hyperoxaluria type 1 1-gen-2019 Dindo, M.; Grottelli, S.; Annunziato, G.; Giardina, G.; Pieroni, M.; Pampalone, G.; Faccini, A.; Cutruzzola, F.; Laurino, P.; Costantino, G.; Cellini, B.
Derivatives of 3-isoxazolecarboxylic acid esters - a potent and selective compound class against replicating and nonreplicating Mycobacterium tuberculosis 1-gen-2012 Lilienkampf, Annamaria; Pieroni, Marco; Franzblau, Scott G.; Bishai, William R.; Kozikowski, Alan P.
Design, Synthesis and Investigation onthe Structure–Activity Relationships of N-Substituted 2-Aminothiazole Derivatives as Antitubercular Agents 1-gen-2014 Pieroni, Marco; Wan, ; B., Cho S; Franzblau, Sg; Costantino, Gabriele
Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases 1-gen-2018 Annunziato, Giannamaria; Giovati, Laura; Andrea, Angeli; Pavone, Marialaura; Sonia Del Prete, ; Pieroni, Marco; Clemente, Capasso; Bruno, Agostino; Conti, Stefania; Magliani, Valter; Supuran, Claudiu T.; Costantino, Gabriele
Discovery of antitubercular 2,4-diphenyl-1H-imidazoles from chemical library repositioning and rational design 1-gen-2015 Pieroni, Marco; Wan, Baojie; Zuliani, Valentina; Franzblau, Scott G.; Costantino, Gabriele; Rivara, Mirko