Sfoglia per Autore
Three-Dimensional Quantitative Structure-Activity Relationship Studies on Selected MT1 and MT2 Melatonin Receptor Ligands: Requirements for Subtype Selectivity and Intrinsic Activity Modulation
2003-01-01 Rivara, Silvia; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Spadoni, G; Bedini, A; Tarzia, G; Lucini, V; Pannacci, M; Fraschini, F; Plazzi, Pier Vincenzo
Strategies leading to MT2 selective melatonin receptor antagonists
2003-01-01 Spadoni, G.; Bedini, A.; Piersanti, G.; Mor, Marco; Rivara, Silvia; Tarzia, G.
Design, synthesis and SAR of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors
2003-01-01 Tarzia, G; Duranti, A; Tontini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Park, C; Kathuria, S; Piomelli, D.
Antioxidant and cytoprotective activity of indole derivatives related to melatonin
2003-01-01 Mor, Marco; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Silva, Claudia; Vacondio, Federica; Rivara, Mirko; Plazzi, Pier Vincenzo; Franceschini, D.; Zusso, M.; Giusti, P.
Strategies leading to MT2 selective melatonin receptor antagonists.
2003-01-01 Spadoni, G; Bedini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Tarzia, G.
The 1,2-dichloroethane/water versus the n-octanol/water system: more about intra- or intermolecular H-bond interactions
2003-01-01 Galland, A; Bouchard, G; Caron, G; VAN BALEN, Gp; Martinet, Cam; Geynoz, S; Rey, S; Vacondio, Federica; Erimondi, G; Mor, Marco; Plazzi, Pier Vincenzo
pH-partition profiles of 4-(3-oxo-1,2-benzisothiazolin-2-yl)phenyl and phenoxyalkanoic acids
2003-01-01 Silva, Claudia; Mor, Marco; Vacondio, Federica; Zuliani, Valentina; Plazzi, P. V.
Synthesis and Structure-Activity Relationships of a Series of Pyrrole Cannabinoid Receptor Agonists
2003-01-01 Tarzia, G; Duranti, A; Tontini, A; Spadoni, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Kathuria, S; Piomelli, D.
Indole-based analogs of melatonin: in vitro antioxidant and cytoprotective activities
2004-01-01 Mor, Marco; Silva, Claudia; Vacondio, Federica; Plazzi, Pier Vincenzo; Bertoni, Simona; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Zusso, M.; Franceschini, D.; Giusti, P.
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity
2004-01-01 Lucini, V.; Pannacci, M.; Scaglione, F.; Fraschini, F.; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Piersanti, G.; Diamantini, G.; Tarzia, G.
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors
2004-01-01 Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B.
Cyclohexylcarbamic Acid 3'- or 4'-Substituted Biphenyl-3-yl Esters of as Fatty Acid Amide Hydrolase Inhibitors: Synthesis, Quantitative Structure-Activity Relationships and Molecular Modelling Studies
2004-01-01 Mor, Marco; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Tarzia, G.; Duranti, A.; Tontini, A.; Piersanti, G.; Kathuria, S.; Piomelli, D.
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists
2004-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Synthesis, Pharmacological Evaluation and Structure-Activity Relationships of Benzopyran Derivatives with Potent SERM Activity
2004-01-01 Amari, G.; Armani, E.; Ghirardi, S.; Delcanale, M.; Civelli, M.; Caruso, P. L.; Galbiati, E.; Lipreri, M.; Rivara, Silvia; Lodola, Alessio; Mor, Marco
MS/MS data-FAAH inhibitory activity relationships of some carbamic acid O-aryl esters
2004-01-01 Basso, E.; Duranti, A.; Mor, Marco; Piomelli, D.; Tontini, A.; Tarzia, G.
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors
2005-01-01 Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G.
Antidepressant-like activity and modulation of brain monoaminergic transmission by blockade of anandamide hydrolysis
2005-01-01 G., Gobbi; F. R., Bambico; R., Mangieri; M., Bortolato; P., Campolongo; M., Solinas; T., Cassano; M. G., Morgese; G., Debonnel; A., Duranti; A., Tontini; G., Tarzia; Mor, Marco; V., Trezza; S. R., Goldberg; V., Cuomo; D., Piomelli
QM/MM modelling of oleamide hydrolysis in fatty acid amide hydrolase (FAAH) reveals a new mechanism of nucleophile activation
2005-01-01 Lodola, Alessio; Mor, Marco; Hermann, Jc; Tarzia, G; Piomelli, D; Mulholland, A. J.
An endocannabinoid mechanism for stress-induced analgesia
2005-01-01 Hohmann, A. G.; Suplita, R. L.; Bolton, N. M.; Neely, M. H.; Fegley, D.; Mangieri, R.; Krey, J.; Walker, J. M.; Holmes, P. V.; Crystal, J. D.; Duranti, A.; Tontini, A.; Mor, Marco; Tarzia, G.; Piomelli, D.
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists
2005-01-01 Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Three-Dimensional Quantitative Structure-Activity Relationship Studies on Selected MT1 and MT2 Melatonin Receptor Ligands: Requirements for Subtype Selectivity and Intrinsic Activity Modulation | 1-gen-2003 | Rivara, Silvia; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Spadoni, G; Bedini, A; Tarzia, G; Lucini, V; Pannacci, M; Fraschini, F; Plazzi, Pier Vincenzo | |
Strategies leading to MT2 selective melatonin receptor antagonists | 1-gen-2003 | Spadoni, G.; Bedini, A.; Piersanti, G.; Mor, Marco; Rivara, Silvia; Tarzia, G. | |
Design, synthesis and SAR of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors | 1-gen-2003 | Tarzia, G; Duranti, A; Tontini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Park, C; Kathuria, S; Piomelli, D. | |
Antioxidant and cytoprotective activity of indole derivatives related to melatonin | 1-gen-2003 | Mor, Marco; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Silva, Claudia; Vacondio, Federica; Rivara, Mirko; Plazzi, Pier Vincenzo; Franceschini, D.; Zusso, M.; Giusti, P. | |
Strategies leading to MT2 selective melatonin receptor antagonists. | 1-gen-2003 | Spadoni, G; Bedini, A; Piersanti, G; Mor, Marco; Rivara, Silvia; Tarzia, G. | |
The 1,2-dichloroethane/water versus the n-octanol/water system: more about intra- or intermolecular H-bond interactions | 1-gen-2003 | Galland, A; Bouchard, G; Caron, G; VAN BALEN, Gp; Martinet, Cam; Geynoz, S; Rey, S; Vacondio, Federica; Erimondi, G; Mor, Marco; Plazzi, Pier Vincenzo | |
pH-partition profiles of 4-(3-oxo-1,2-benzisothiazolin-2-yl)phenyl and phenoxyalkanoic acids | 1-gen-2003 | Silva, Claudia; Mor, Marco; Vacondio, Federica; Zuliani, Valentina; Plazzi, P. V. | |
Synthesis and Structure-Activity Relationships of a Series of Pyrrole Cannabinoid Receptor Agonists | 1-gen-2003 | Tarzia, G; Duranti, A; Tontini, A; Spadoni, G; Mor, Marco; Rivara, Silvia; Plazzi, Pier Vincenzo; Kathuria, S; Piomelli, D. | |
Indole-based analogs of melatonin: in vitro antioxidant and cytoprotective activities | 1-gen-2004 | Mor, Marco; Silva, Claudia; Vacondio, Federica; Plazzi, Pier Vincenzo; Bertoni, Simona; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Zusso, M.; Franceschini, D.; Giusti, P. | |
Tricyclic Alkylamides as Melatonin Receptor Ligands with Antagonist or Inverse Agonist Activity | 1-gen-2004 | Lucini, V.; Pannacci, M.; Scaglione, F.; Fraschini, F.; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Piersanti, G.; Diamantini, G.; Tarzia, G. | |
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors | 1-gen-2004 | Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B. | |
Cyclohexylcarbamic Acid 3'- or 4'-Substituted Biphenyl-3-yl Esters of as Fatty Acid Amide Hydrolase Inhibitors: Synthesis, Quantitative Structure-Activity Relationships and Molecular Modelling Studies | 1-gen-2004 | Mor, Marco; Rivara, Silvia; Lodola, Alessio; Plazzi, Pier Vincenzo; Tarzia, G.; Duranti, A.; Tontini, A.; Piersanti, G.; Kathuria, S.; Piomelli, D. | |
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists | 1-gen-2004 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo | |
Synthesis, Pharmacological Evaluation and Structure-Activity Relationships of Benzopyran Derivatives with Potent SERM Activity | 1-gen-2004 | Amari, G.; Armani, E.; Ghirardi, S.; Delcanale, M.; Civelli, M.; Caruso, P. L.; Galbiati, E.; Lipreri, M.; Rivara, Silvia; Lodola, Alessio; Mor, Marco | |
MS/MS data-FAAH inhibitory activity relationships of some carbamic acid O-aryl esters | 1-gen-2004 | Basso, E.; Duranti, A.; Mor, Marco; Piomelli, D.; Tontini, A.; Tarzia, G. | |
Application of 3D-QSAR in the Rational Design of Receptor Ligands and Enzyme Inhibitors | 1-gen-2005 | Mor, Marco; Rivara, Silvia; Lodola, Alessio; Lorenzi, Simone; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Spadoni, G.; Bedini, A.; Duranti, A.; Tontini, A.; Tarzia, G. | |
Antidepressant-like activity and modulation of brain monoaminergic transmission by blockade of anandamide hydrolysis | 1-gen-2005 | G., Gobbi; F. R., Bambico; R., Mangieri; M., Bortolato; P., Campolongo; M., Solinas; T., Cassano; M. G., Morgese; G., Debonnel; A., Duranti; A., Tontini; G., Tarzia; Mor, Marco; V., Trezza; S. R., Goldberg; V., Cuomo; D., Piomelli | |
QM/MM modelling of oleamide hydrolysis in fatty acid amide hydrolase (FAAH) reveals a new mechanism of nucleophile activation | 1-gen-2005 | Lodola, Alessio; Mor, Marco; Hermann, Jc; Tarzia, G; Piomelli, D; Mulholland, A. J. | |
An endocannabinoid mechanism for stress-induced analgesia | 1-gen-2005 | Hohmann, A. G.; Suplita, R. L.; Bolton, N. M.; Neely, M. H.; Fegley, D.; Mangieri, R.; Krey, J.; Walker, J. M.; Holmes, P. V.; Crystal, J. D.; Duranti, A.; Tontini, A.; Mor, Marco; Tarzia, G.; Piomelli, D. | |
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists | 1-gen-2005 | Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile