Sfoglia per Autore
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity
2006-01-01 Carmi, Caterina; Cavazzoni, Andrea; Zuliani, Valentina; Lodola, Alessio; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series
2006-01-01 Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo
Antiproliferative and proapototic effects of a new combi-molecule on non small cell lung cancer cell lines
2007-01-01 Alfieri, Roberta; Cavazzoni, Andrea; Carmi, Caterina; M., Galetti; Zuliani, Valentina; Fumarola, Claudia; Mor, Marco; Petronini, Pier Giorgio
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano
2007-01-01 Cavazzoni, Andrea; Galetti, Maricla; LA MONICA, S; Fumarola, C; Bonelli, Mara; Carmi, C; Zuliani, Valentina; Lodola, Alessio; Bordi, F; Plazzi, P. V.; Mor, Marco; Petronini, Pg
5-benzylidene-hydantoin UPR 1024 acts as EGFR inhibitor and induces DNA damage in A549 NSCLC cell line
2007-01-01 Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Carmi, C; Zuliani, Valentina; Fumarola, C; Bonelli, Mara; Frazzi, R; Mor, Marco; Petronini, Pier Giorgio
A Practical Synthesis of 2,4(5)-Diarylimidazoles from Simple Building Blocks
2007-01-01 Zuliani, Valentina; Cocconcelli, G.; Fantini, M.; Ghiron, C.; Rivara, Mirko
2,4(5)-Diarylimidazoles: Synthesis and Biological Evaluation of a New Class of Sodium Channel Blockers against hNav1.2
2008-01-01 Rivara, Mirko; Baheti, A. R.; Fantini, M.; Cocconcelli, G.; Ghiron, C.; Kalmar, C. L.; Singh, N.; Merrick, E. C.; Patel, M. K.; Zuliani, Valentina
Dual mechanisms of action of the 5-benzylidene-hydantoin UPR1024 on lung cancer cell lines
2008-01-01 Cavazzoni, Andrea; Alfieri, Roberta; Carmi, C.; Zuliani, Valentina; Galetti, Maricla; Fumarola, Claudia; Frazzi, Raffaele; Bonelli, Mara; Bordi, Fabrizio; Lodola, Alessio; Mor, Marco; Petronini, Pier Giorgio
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor.
2008-01-01 Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships
2009-01-01 Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K.
Anticonvulsant Activity of 2,4(5)-Diarylimidazoles in Mice and Rat Models
2009-01-01 Rivara, Mirko; M., Fantini; Zuliani, Valentina; M. K., Patel
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line
2009-01-01 Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
Recent Advances in the Medicinal Chemistry of Sodium Channel Blockers and their Therapeutic Potential
2009-01-01 Zuliani, Valentina; Patel, M. K.; Fantini, M.; Rivara, Mirko
Chiral NMR discrimination of the diastereoisomeric salts of the H(3)-antagonist 2-[3-(1H-imidazol-4-ylmethyl)piperidin-1-yl]-1H-benzimidazole.
2009-01-01 Rivara, Mirko; Zuliani, Valentina; Fantini, M; Dallaturca, E; Mor, Marco
A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine
2009-01-01 Rivara, Mirko; Zuliani, Valentina; Plazzi, Pier Vincenzo; Bordi, Fabrizio
Anticonvulsant Activity of 2,4(1H)-Diarylimidazoles in Mice and Rats Acute Seizure Models
2010-01-01 Zuliani, Valentina; M., Fantini; A., Nigam; J. P., Stables; M. K., Patel; Rivara, Mirko
NMR Analysis of a Series of Imidazobenzoxazines
2010-01-01 Rivara, Mirko; M., Fantini; Acquotti, Domenico; Zuliani, Valentina
Sodium channel blockers for neuropathic pain.
2010-01-01 Zuliani, Valentina; Rivara, Mirko; M., Fantini; Costantino, Gabriele
Microwave Assisted Efficient Synthesis of Imidazole-based Privileged Structure
2010-01-01 M., Fantini; Zuliani, Valentina; M. A., Spotti; Rivara, Mirko
Advances in Design and Development of Sodium Channel Blockers.
2011-01-01 Zuliani, Valentina; L., Amori; Rivara, Mirko
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity | 1-gen-2006 | Carmi, Caterina; Cavazzoni, Andrea; Zuliani, Valentina; Lodola, Alessio; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco | |
| Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series | 1-gen-2006 | Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo | |
| Antiproliferative and proapototic effects of a new combi-molecule on non small cell lung cancer cell lines | 1-gen-2007 | Alfieri, Roberta; Cavazzoni, Andrea; Carmi, Caterina; M., Galetti; Zuliani, Valentina; Fumarola, Claudia; Mor, Marco; Petronini, Pier Giorgio | |
| Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano | 1-gen-2007 | Cavazzoni, Andrea; Galetti, Maricla; LA MONICA, S; Fumarola, C; Bonelli, Mara; Carmi, C; Zuliani, Valentina; Lodola, Alessio; Bordi, F; Plazzi, P. V.; Mor, Marco; Petronini, Pg | |
| 5-benzylidene-hydantoin UPR 1024 acts as EGFR inhibitor and induces DNA damage in A549 NSCLC cell line | 1-gen-2007 | Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Carmi, C; Zuliani, Valentina; Fumarola, C; Bonelli, Mara; Frazzi, R; Mor, Marco; Petronini, Pier Giorgio | |
| A Practical Synthesis of 2,4(5)-Diarylimidazoles from Simple Building Blocks | 1-gen-2007 | Zuliani, Valentina; Cocconcelli, G.; Fantini, M.; Ghiron, C.; Rivara, Mirko | |
| 2,4(5)-Diarylimidazoles: Synthesis and Biological Evaluation of a New Class of Sodium Channel Blockers against hNav1.2 | 1-gen-2008 | Rivara, Mirko; Baheti, A. R.; Fantini, M.; Cocconcelli, G.; Ghiron, C.; Kalmar, C. L.; Singh, N.; Merrick, E. C.; Patel, M. K.; Zuliani, Valentina | |
| Dual mechanisms of action of the 5-benzylidene-hydantoin UPR1024 on lung cancer cell lines | 1-gen-2008 | Cavazzoni, Andrea; Alfieri, Roberta; Carmi, C.; Zuliani, Valentina; Galetti, Maricla; Fumarola, Claudia; Frazzi, Raffaele; Bonelli, Mara; Bordi, Fabrizio; Lodola, Alessio; Mor, Marco; Petronini, Pier Giorgio | |
| Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. | 1-gen-2008 | Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
| 2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships | 1-gen-2009 | Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K. | |
| Anticonvulsant Activity of 2,4(5)-Diarylimidazoles in Mice and Rat Models | 1-gen-2009 | Rivara, Mirko; M., Fantini; Zuliani, Valentina; M. K., Patel | |
| 5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line | 1-gen-2009 | Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco | |
| Recent Advances in the Medicinal Chemistry of Sodium Channel Blockers and their Therapeutic Potential | 1-gen-2009 | Zuliani, Valentina; Patel, M. K.; Fantini, M.; Rivara, Mirko | |
| Chiral NMR discrimination of the diastereoisomeric salts of the H(3)-antagonist 2-[3-(1H-imidazol-4-ylmethyl)piperidin-1-yl]-1H-benzimidazole. | 1-gen-2009 | Rivara, Mirko; Zuliani, Valentina; Fantini, M; Dallaturca, E; Mor, Marco | |
| A Short and Efficient Synthesis of the Selective H4 Receptor Agonist 4-Methylhistamine | 1-gen-2009 | Rivara, Mirko; Zuliani, Valentina; Plazzi, Pier Vincenzo; Bordi, Fabrizio | |
| Anticonvulsant Activity of 2,4(1H)-Diarylimidazoles in Mice and Rats Acute Seizure Models | 1-gen-2010 | Zuliani, Valentina; M., Fantini; A., Nigam; J. P., Stables; M. K., Patel; Rivara, Mirko | |
| NMR Analysis of a Series of Imidazobenzoxazines | 1-gen-2010 | Rivara, Mirko; M., Fantini; Acquotti, Domenico; Zuliani, Valentina | |
| Sodium channel blockers for neuropathic pain. | 1-gen-2010 | Zuliani, Valentina; Rivara, Mirko; M., Fantini; Costantino, Gabriele | |
| Microwave Assisted Efficient Synthesis of Imidazole-based Privileged Structure | 1-gen-2010 | M., Fantini; Zuliani, Valentina; M. A., Spotti; Rivara, Mirko | |
| Advances in Design and Development of Sodium Channel Blockers. | 1-gen-2011 | Zuliani, Valentina; L., Amori; Rivara, Mirko |
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