Sfoglia per Autore
Creatine as a compatible osmolyte in muscle cells exposed to hypertonic stress
2006-01-01 Alfieri, R; Bonelli, M; Cavazzoni, A; Brigotti, Maurizio; Fumarola, C; Sestili, Piero; Mozzoni, P; DE PALMA, Giuseppe; Mutti, A; Carnicelli, D; Vacondio, F; Silva, C; Borghetti, A. F; Wheeler, K. P; Petronini, P.
Quantitative structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors.
2008-01-01 Fioni, A.; Vacondio, Federica; Mor, Marco; Silva, Claudia; Lodola, Alessio; Duranti, A.; Tontini, A.; Tarzia, G.; Piomelli, D.
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma.
2008-01-01 Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta
Synthesis and Quantitative Structure-Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates.
2008-01-01 Mor, Marco; Lodola, Alessio; Rivara, Silvia; Vacondio, Federica; Duranti, A.; Tontini, A.; Sanchini, S.; Piersanti, G.; Clapper, J. R.; King, A. R.; Tarzia, G.; Piomelli, D.
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor.
2008-01-01 Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
Structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors: chemical and biological stability
2009-01-01 Vacondio, Federica; Silva, Claudia; Lodola, Alessio; A., Fioni; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; Mor, Marco; G., Tarzia
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line
2009-01-01 Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships
2009-01-01 Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K.
A second generation of carbamate-based fatty acid amide hydrolase inhibitors with improved activity in vivo
2009-01-01 Clapper, Jason R.; Vacondio, Federica; King, Alvin R.; Duranti, Andrea; Tontini, Andrea; Silva, Claudia; Sanchini, Silvano; Tarzia, Giorgio; Mor, Marco; Piomelli, Daniele
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands
2009-01-01 Rivara, Silvia; Vacondio, Federica; Fioni, A; Silva, Claudia; Carmi, Caterina; Mor, Marco; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, G; Bedini, A; Orlando, P; Lucarini, S; Tarzia, G.
Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism.
2010-01-01 J. R., Clapper; G., Moreno Sanz; R., Russo; A., Guijarro; Vacondio, Federica; A., Duranti; A., Tontini; S., Sanchini; N. R., Sciolino; J. M., Spradley; A. G., Hohmann; A., Calignano; Mor, Marco; G., Tarzia; D., Piomelli
Synthesis and structure-activity relationships of N-(2-oxo-3-oxetanyl)amides as N-acylethanolamine-hydrolyzing acid amidase inhibitors.
2010-01-01 C., Solorzano; F., Antonietti; A., Duranti; A., Tontini; Rivara, Silvia; Lodola, Alessio; Vacondio, Federica; G., Tarzia; D., Piomelli; Mor, Marco
Qualitative structure-metabolism relationships in the hydrolysis of carbamates
2010-01-01 Vacondio, Federica; Silva, Claudia; Mor, Marco; B., Testa
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion
2010-01-01 Carmi, C.; Cavazzoni, A.; Vezzosi, S.; Bordi, F.; Vacondio, F.; Silva, C.; Rivara, S.; Lodola, A.; Alfieri, R.; La Monica, S; Galetti, M.; Ardizzoni, A.; Petronini, P. G.; Mor, M.
Mannich base derivatives as novel EGFR irreversible inhibitors
2011-01-01 Russo, Simonetta; Mor, Marco; Carmi, Caterina; Vacondio, Federica; Petronini, Pier Giorgio; Cavazzoni, Andrea
Epidermal Growth Factor Receptor Irreversible Inhibitors: Chemical Exploration of the Cysteine-Trap Portion
2011-01-01 Carmi, Caterina; Lodola, Alessio; Rivara, Silvia; Vacondio, Federica; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, Andrea; Petronini, Pier Giorgio; Mor, Marco
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: steric effects of N-alkyl chain on rat plasma and liver stability
2011-01-01 Vacondio, Federica; Silva, Claudia; Lodola, Alessio; Carmi, Caterina; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; G., Tarzia; Mor, Marco
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma.
2011-01-01 Vacondio, Federica; Silva, Claudia; Morini, Giovanni; Bordi, Fabrizio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain.
2012-01-01 Bordi, Fabrizio; Rivara, Silvia; E., Dallaturca; Carmi, Caterina; Pala, Daniele; Lodola, Alessio; Vacondio, Federica; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Brain Pharmacokinetics of Non-Imidazole Biphenyl H3 Receptor Antagonists: a Liquid Chromatography/Electrospray-Mass Spectrometry and ex vivo Binding Study in Rats
2012-01-01 Vacondio, Federica; Silva, Claudia; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Creatine as a compatible osmolyte in muscle cells exposed to hypertonic stress | 1-gen-2006 | Alfieri, R; Bonelli, M; Cavazzoni, A; Brigotti, Maurizio; Fumarola, C; Sestili, Piero; Mozzoni, P; DE PALMA, Giuseppe; Mutti, A; Carnicelli, D; Vacondio, F; Silva, C; Borghetti, A. F; Wheeler, K. P; Petronini, P. | |
Quantitative structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors. | 1-gen-2008 | Fioni, A.; Vacondio, Federica; Mor, Marco; Silva, Claudia; Lodola, Alessio; Duranti, A.; Tontini, A.; Tarzia, G.; Piomelli, D. | |
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. | 1-gen-2008 | Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta | |
Synthesis and Quantitative Structure-Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates. | 1-gen-2008 | Mor, Marco; Lodola, Alessio; Rivara, Silvia; Vacondio, Federica; Duranti, A.; Tontini, A.; Sanchini, S.; Piersanti, G.; Clapper, J. R.; King, A. R.; Tarzia, G.; Piomelli, D. | |
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. | 1-gen-2008 | Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
Structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors: chemical and biological stability | 1-gen-2009 | Vacondio, Federica; Silva, Claudia; Lodola, Alessio; A., Fioni; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; Mor, Marco; G., Tarzia | |
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line | 1-gen-2009 | Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco | |
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships | 1-gen-2009 | Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K. | |
A second generation of carbamate-based fatty acid amide hydrolase inhibitors with improved activity in vivo | 1-gen-2009 | Clapper, Jason R.; Vacondio, Federica; King, Alvin R.; Duranti, Andrea; Tontini, Andrea; Silva, Claudia; Sanchini, Silvano; Tarzia, Giorgio; Mor, Marco; Piomelli, Daniele | |
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands | 1-gen-2009 | Rivara, Silvia; Vacondio, Federica; Fioni, A; Silva, Claudia; Carmi, Caterina; Mor, Marco; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, G; Bedini, A; Orlando, P; Lucarini, S; Tarzia, G. | |
Anandamide suppresses pain initiation through a peripheral endocannabinoid mechanism. | 1-gen-2010 | J. R., Clapper; G., Moreno Sanz; R., Russo; A., Guijarro; Vacondio, Federica; A., Duranti; A., Tontini; S., Sanchini; N. R., Sciolino; J. M., Spradley; A. G., Hohmann; A., Calignano; Mor, Marco; G., Tarzia; D., Piomelli | |
Synthesis and structure-activity relationships of N-(2-oxo-3-oxetanyl)amides as N-acylethanolamine-hydrolyzing acid amidase inhibitors. | 1-gen-2010 | C., Solorzano; F., Antonietti; A., Duranti; A., Tontini; Rivara, Silvia; Lodola, Alessio; Vacondio, Federica; G., Tarzia; D., Piomelli; Mor, Marco | |
Qualitative structure-metabolism relationships in the hydrolysis of carbamates | 1-gen-2010 | Vacondio, Federica; Silva, Claudia; Mor, Marco; B., Testa | |
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion | 1-gen-2010 | Carmi, C.; Cavazzoni, A.; Vezzosi, S.; Bordi, F.; Vacondio, F.; Silva, C.; Rivara, S.; Lodola, A.; Alfieri, R.; La Monica, S; Galetti, M.; Ardizzoni, A.; Petronini, P. G.; Mor, M. | |
Mannich base derivatives as novel EGFR irreversible inhibitors | 1-gen-2011 | Russo, Simonetta; Mor, Marco; Carmi, Caterina; Vacondio, Federica; Petronini, Pier Giorgio; Cavazzoni, Andrea | |
Epidermal Growth Factor Receptor Irreversible Inhibitors: Chemical Exploration of the Cysteine-Trap Portion | 1-gen-2011 | Carmi, Caterina; Lodola, Alessio; Rivara, Silvia; Vacondio, Federica; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, Andrea; Petronini, Pier Giorgio; Mor, Marco | |
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: steric effects of N-alkyl chain on rat plasma and liver stability | 1-gen-2011 | Vacondio, Federica; Silva, Claudia; Lodola, Alessio; Carmi, Caterina; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; G., Tarzia; Mor, Marco | |
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma. | 1-gen-2011 | Vacondio, Federica; Silva, Claudia; Morini, Giovanni; Bordi, Fabrizio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain. | 1-gen-2012 | Bordi, Fabrizio; Rivara, Silvia; E., Dallaturca; Carmi, Caterina; Pala, Daniele; Lodola, Alessio; Vacondio, Federica; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
Brain Pharmacokinetics of Non-Imidazole Biphenyl H3 Receptor Antagonists: a Liquid Chromatography/Electrospray-Mass Spectrometry and ex vivo Binding Study in Rats | 1-gen-2012 | Vacondio, Federica; Silva, Claudia; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco |
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