Sfoglia per Autore  

Opzioni
Mostrati risultati da 21 a 40 di 155
Titolo Data di pubblicazione Autore(i) File
Synthesis and Quantitative Structure-Activity Relationship of Fatty Acid Amide Hydrolase Inhibitors: Modulation at the N-Portion of Biphenyl-3-yl Alkylcarbamates. 1-gen-2008 Mor, Marco; Lodola, Alessio; Rivara, Silvia; Vacondio, Federica; Duranti, A.; Tontini, A.; Sanchini, S.; Piersanti, G.; Clapper, J. R.; King, A. R.; Tarzia, G.; Piomelli, D.
Identification of productive inhibitor binding orientation in fatty acid amide hydrolase (FAAH) by QM/MM mechanistic modelling. 1-gen-2008 Lodola, Alessio; Mor, Marco; Rivara, Silvia; Christov, C.; Tarzia, G.; Piomelli, D.; Mulholland, A. J.
Optimizing EGFR inhibitor treatment in non small cell lung cancer 1-gen-2009 Alfieri, Roberta; Cavazzoni, Andrea; Galetti, Maricla; LA MONICA, S; Mor, Marco; Carmi, C; Lodola, Alessio; Tiseo, M; Ardizzoni, A; Petronini, P. G.
Insights into the mechanism and inhibition of fatty acid amide hydrolase from quantum mechanics/molecular mechanics (QM/MM) modelling. 1-gen-2009 Lodola, Alessio; Mor, Marco; Sirirak, J.; Mulholland, A. J.
Pharmacological Tools in Endocannabinoid Neurobiology 1-gen-2009 Mor, Marco; Lodola, Alessio
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line 1-gen-2009 Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
A critical cysteine residue in monoacylglycerol lipase is targeted by a new class of isothiazolinone-based enzyme inhibitors. 1-gen-2009 King, A. R.; Lodola, Alessio; Carmi, Caterina; Fu, J.; Mor, Marco; Piomelli, D.
Structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors: chemical and biological stability 1-gen-2009 Vacondio, Federica; Silva, Claudia; Lodola, Alessio; A., Fioni; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; Mor, Marco; G., Tarzia
Discovery of potent and reversible monoacylglycerol lipase inhibitors. 1-gen-2009 King, Ar; Dotsey, Ey; Lodola, Alessio; Jung, Km; Ghomian, A; Qiu, Y; Fu, J; Mor, Marco; Piomelli, D.
Selective N-acylethanolamine-hydrolyzing acid amidase inhibition reveals a key role for endogenous palmitoylethanolamide in inflammation 1-gen-2009 Carlos, Solorzano; Chenggang, Zhu; Natalia, Battistaa; Giuseppe, Astarita; Lodola, Alessio; Rivara, Silvia; Mor, Marco; Roberto, Russo; Mauro, Maccarrone; Francesca, Antonietti; Andrea, Duranti; Andrea, Tontini; Salvatore, Cuzzocrea; Giorgio, Tarzia; Daniele, Piomelli
Lithocholic acid competitively inhibitis EphA2-ephrinA1 binding: pharmacological and structural considerations. 1-gen-2010 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion 1-gen-2010 Carmi, C.; Cavazzoni, A.; Vezzosi, S.; Bordi, F.; Vacondio, F.; Silva, C.; Rivara, S.; Lodola, A.; Alfieri, R.; La Monica, S; Galetti, M.; Ardizzoni, A.; Petronini, P. G.; Mor, M.
Structural Fluctuations in Enzyme-Catalyzed Reactions:Determinants of Reactivity in Fatty Acid AmideHydrolase from Multivariate Statistical Analysis ofQuantum Mechanics/Molecular Mechanics Paths 1-gen-2010 Lodola, Alessio; J., Sirirak; N., Fey; Rivara, Silvia; Mor, Marco; A. J., Mulholland
Lithocholic acid competitively inhibits EphA2-ephrinA1 binding: pharmacological and structural considerations. 1-gen-2010 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta
Synthesis and structure-activity relationships of N-(2-oxo-3-oxetanyl)amides as N-acylethanolamine-hydrolyzing acid amidase inhibitors. 1-gen-2010 C., Solorzano; F., Antonietti; A., Duranti; A., Tontini; Rivara, Silvia; Lodola, Alessio; Vacondio, Federica; G., Tarzia; D., Piomelli; Mor, Marco
Lithocholic acid is an Eph-ephrin ligand interfering with Eph-kinase activation 1-gen-2011 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Flammini, Lisa; Barocelli, Elisabetta; Incerti, Matteo; Lodola, Alessio; Tognolini, Massimiliano
Structure activity relationship of new EphA2 ligands 1-gen-2011 Tognolini, Massimiliano; Incerti, Matteo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Barocelli, Elisabetta; Russo, Simonetta; B., Lelli; L., Bracci; Lodola, Alessio
Catalytic, Asymmetric Hypervinylogous Mukaiyama Aldol Reactions of Extended Furan-Based Silyl Enolates 1-gen-2011 Curti, Claudio; Battistini, Lucia; Sartori, Andrea; Lodola, Alessio; Mor, Marco; Rassu, G.; Pelosi, Giorgio; Zanardi, Franca; Casiraghi, Giovanni
Covalent Inhibitors of Fatty Acid Amide Hydrolase: A Rationale for the Activity of Piperidine and Piperazine Aryl Ureas 1-gen-2011 G., Palermo; D., Branduardi; M., Masetti; Lodola, Alessio; Mor, Marco; D., Piomelli; A., Cavalli; M., De Vivo
Understanding the role of carbamate reactivity in fatty acid amide hydrolase inhibition by QM/MM mechanistic modelling. 1-gen-2011 Lodola, Alessio; L., Capoferri; Rivara, Silvia; E., Chudyk; J., Sirirak; E., Dyguda Kazimierowicz; Wa, Sokalski; M., Mileni; G., Tarzia; D., Piomelli; Mor, Marco; Aj, Mulholland
Mostrati risultati da 21 a 40 di 155
Legenda icone

  •  file ad accesso aperto
  •  file disponibili sulla rete interna
  •  file disponibili agli utenti autorizzati
  •  file disponibili solo agli amministratori
  •  file sotto embargo
  •  nessun file disponibile