Sfoglia per Autore
N-(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability
2021-01-01 Ferlenghi, F.; Mari, M.; Gobbi, G.; Elisi, G. M.; Mor, M.; Rivara, S.; Vacondio, F.; Bartolucci, S.; Bedini, A.; Fanini, F.; Spadoni, G.
MT1 and MT2 melatonin receptors play opposite roles in brain cancer progression
2021-01-01 Kinker, G. S.; Ostrowski, L. H.; Ribeiro, P. A. C.; Chanoch, R.; Muxel, S. M.; Tirosh, I.; Spadoni, G.; Rivara, S.; Martins, V. R.; Santos, T. G.; Markus, R. P.; Fernandes, P. A. C. M.
New Coumarin derivatives as cholinergic and cannabinoid system modulators
2021-01-01 Montanari, S.; Allara, M.; Scalvini, L.; Kostrzewa, M.; Belluti, F.; Gobbi, S.; Naldi, M.; Rivara, S.; Bartolini, M.; Ligresti, A.; Bisi, A.; Rampa, A.
Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma
2021-01-01 Castelli, R.; Taranto, S.; Furiassi, L.; Bozza, N.; Marseglia, G.; Ferlenghi, F.; Rivara, S.; Retini, M.; Bedini, A.; Spadoni, G.; Matarazzo, S.; Ronca, R.; Presta, M.; Mor, M.; Giacomini, A.
New classes of potent heparanase inhibitors from ligand-based virtual screening
2020-01-01 Pala, D.; Scalvini, L.; Elisi, G. M.; Lodola, A.; Mor, M.; Spadoni, G.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Milazzo, F. M.; Battistuzzi, G.; Rivara, S.; Giannini, G.
Antidepressant-like effects of pharmacological inhibition of FAAH activity in socially isolated female rats
2020-01-01 Carnevali, L.; Statello, R.; Vacondio, F.; Ferlenghi, F.; Spadoni, G.; Rivara, S.; Mor, M.; Sgoifo, A.
N-Acylethanolamine Acid Amidase (NAAA): Mechanism of Palmitoylethanolamide Hydrolysis Revealed by Mechanistic Simulations
2020-01-01 Scalvini, L.; Ghidini, A.; Lodola, A.; Callegari, D.; Rivara, S.; Piomelli, D.; Mor, M.
Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines
2020-01-01 Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele.
The Control of Heparanase Through the Use of Small Molecules
2020-01-01 Giannini, G.; Battistuzzi, G.; Rivara, S.
Design and SAR Analysis of Covalent Inhibitors Driven by Hybrid QM/MM Simulations
2020-01-01 Lodola, A.; Callegari, D.; Scalvini, L.; Rivara, S.; Mor, M.
Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria
2020-01-01 Elisi, GIAN MARCO; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto
Pharmacokinetics, pharmacodynamics and safety studies on URB937, a peripherally restricted fatty acid amide hydrolase inhibitor, in rats
2019-01-01 Vozella, V.; Ahmed, F.; Choobchian, P.; Merrill, C. B.; Zibardi, C.; Tarzia, G.; Mor, M.; Duranti, A.; Tontini, A.; Rivara, S.; Piomelli, D.
Balancing reactivity and antitumor activity: heteroarylthioacetamide derivatives as potent and time-dependent inhibitors of EGFR
2019-01-01 Castelli, R; Bozza, N; Cavazzoni, A; Bonelli, M; Vacondio, F; Ferlenghi, F; Callegari, D; Silva, C; Rivara, S; Lodola, A; Digiacomo, G; Fumarola, C; Alfieri, R; Petronini, Pg; Mor, M.
New Antimicrobials Targeting Bacterial RNA Polymerase Holoenzyme Assembly Identified with an in Vivo BRET-Based Discovery Platform
2019-01-01 Sartini, S.; Levati, E.; Maccesi, M.; Guerra, M.; Spadoni, G.; Bach, S.; Benincasa, M.; Scocchi, M.; Ottonello, S.; Rivara, S.; Montanini, B.
Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity
2018-01-01 Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; Scipione, Luigi; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Ferrara, Fabiana Fosca; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; Milazzo, Ferdinando M.; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannini, Giuseppe
Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity
2018-01-01 Messore, A.; Madia, V. N.; Pescatori, L.; Saccoliti, F.; Tudino, V.; De Leo, A.; Bortolami, M.; De Vita, D.; Scipione, L.; Pepi, F.; Costi, R.; Rivara, S.; Scalvini, L.; Mor, M.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Cassinelli, G.; Milazzo, F. M.; Battistuzzi, G.; Di Santo, R.; Giannini, G.
Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands
2018-01-01 Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto
Identification of bivalent ligands with melatonin receptor agonist and fatty acid amide hydrolase (FAAH) inhibitory activity that exhibit ocular hypotensive effect in the rabbit
2018-01-01 Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, Andrea; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S.
Social stress contagion in rats: Behavioural, autonomic and neuroendocrine correlates
2017-01-01 Carnevali, Luca; Montano, Nicola; Statello, ROSARIO IGNAZIO; Coude', Gino; Vacondio, Federica; Rivara, Silvia; Ferrari, Pier Francesco; Sgoifo, Andrea
Metadynamics Simulations Distinguish Short- and Long-Residence-Time Inhibitors of Cyclin-Dependent Kinase 8.
2017-01-01 Callegari, Donatella; Lodola, Alessio; Pala, Daniele; Rivara, Silvia; Mor, Marco; Rizzi, A; Capelli A., M.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| N-(Anilinoethyl)amide Melatonergic Ligands with Improved Water Solubility and Metabolic Stability | 1-gen-2021 | Ferlenghi, F.; Mari, M.; Gobbi, G.; Elisi, G. M.; Mor, M.; Rivara, S.; Vacondio, F.; Bartolucci, S.; Bedini, A.; Fanini, F.; Spadoni, G. | |
| MT1 and MT2 melatonin receptors play opposite roles in brain cancer progression | 1-gen-2021 | Kinker, G. S.; Ostrowski, L. H.; Ribeiro, P. A. C.; Chanoch, R.; Muxel, S. M.; Tirosh, I.; Spadoni, G.; Rivara, S.; Martins, V. R.; Santos, T. G.; Markus, R. P.; Fernandes, P. A. C. M. | |
| New Coumarin derivatives as cholinergic and cannabinoid system modulators | 1-gen-2021 | Montanari, S.; Allara, M.; Scalvini, L.; Kostrzewa, M.; Belluti, F.; Gobbi, S.; Naldi, M.; Rivara, S.; Bartolini, M.; Ligresti, A.; Bisi, A.; Rampa, A. | |
| Chemical modification of NSC12 leads to a specific FGF-trap with antitumor activity in multiple myeloma | 1-gen-2021 | Castelli, R.; Taranto, S.; Furiassi, L.; Bozza, N.; Marseglia, G.; Ferlenghi, F.; Rivara, S.; Retini, M.; Bedini, A.; Spadoni, G.; Matarazzo, S.; Ronca, R.; Presta, M.; Mor, M.; Giacomini, A. | |
| New classes of potent heparanase inhibitors from ligand-based virtual screening | 1-gen-2020 | Pala, D.; Scalvini, L.; Elisi, G. M.; Lodola, A.; Mor, M.; Spadoni, G.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Milazzo, F. M.; Battistuzzi, G.; Rivara, S.; Giannini, G. | |
| Antidepressant-like effects of pharmacological inhibition of FAAH activity in socially isolated female rats | 1-gen-2020 | Carnevali, L.; Statello, R.; Vacondio, F.; Ferlenghi, F.; Spadoni, G.; Rivara, S.; Mor, M.; Sgoifo, A. | |
| N-Acylethanolamine Acid Amidase (NAAA): Mechanism of Palmitoylethanolamide Hydrolysis Revealed by Mechanistic Simulations | 1-gen-2020 | Scalvini, L.; Ghidini, A.; Lodola, A.; Callegari, D.; Rivara, S.; Piomelli, D.; Mor, M. | |
| Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines | 1-gen-2020 | Castelli, Riccardo; Scalvini, Laura; Vacondio, Federica; Lodola, Alessio; Anselmi, Mattia; Vezzosi, Stefano; Carmi, Caterina; Bassi, Michele; Ferlenghi, Francesca; Rivara, Silvia; Moller Ingvar, R.; Rand Kasper, D.; Daglian, Jennifer; Wei, Don; Dotsey Emmanuel, Y.; Ahmed, Faizy; Jung, Kwang-Mook; Stella, Nephi; Singh, Simar; Mor, Marco; Piomelli, Daniele. | |
| The Control of Heparanase Through the Use of Small Molecules | 1-gen-2020 | Giannini, G.; Battistuzzi, G.; Rivara, S. | |
| Design and SAR Analysis of Covalent Inhibitors Driven by Hybrid QM/MM Simulations | 1-gen-2020 | Lodola, A.; Callegari, D.; Scalvini, L.; Rivara, S.; Mor, M. | |
| Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria | 1-gen-2020 | Elisi, GIAN MARCO; Bedini, Annalida; Scalvini, Laura; Carmi, Caterina; Bartolucci, Silvia; Lucini, Valeria; Scaglione, Francesco; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto | |
| Pharmacokinetics, pharmacodynamics and safety studies on URB937, a peripherally restricted fatty acid amide hydrolase inhibitor, in rats | 1-gen-2019 | Vozella, V.; Ahmed, F.; Choobchian, P.; Merrill, C. B.; Zibardi, C.; Tarzia, G.; Mor, M.; Duranti, A.; Tontini, A.; Rivara, S.; Piomelli, D. | |
| Balancing reactivity and antitumor activity: heteroarylthioacetamide derivatives as potent and time-dependent inhibitors of EGFR | 1-gen-2019 | Castelli, R; Bozza, N; Cavazzoni, A; Bonelli, M; Vacondio, F; Ferlenghi, F; Callegari, D; Silva, C; Rivara, S; Lodola, A; Digiacomo, G; Fumarola, C; Alfieri, R; Petronini, Pg; Mor, M. | |
| New Antimicrobials Targeting Bacterial RNA Polymerase Holoenzyme Assembly Identified with an in Vivo BRET-Based Discovery Platform | 1-gen-2019 | Sartini, S.; Levati, E.; Maccesi, M.; Guerra, M.; Spadoni, G.; Bach, S.; Benincasa, M.; Scocchi, M.; Ottonello, S.; Rivara, S.; Montanini, B. | |
| Novel Benzazole Derivatives Endowed with Potent Antiheparanase Activity | 1-gen-2018 | Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; Scipione, Luigi; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Ferrara, Fabiana Fosca; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; Milazzo, Ferdinando M.; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannini, Giuseppe | |
| Novel Symmetrical Benzazolyl Derivatives Endowed with Potent Anti-Heparanase Activity | 1-gen-2018 | Messore, A.; Madia, V. N.; Pescatori, L.; Saccoliti, F.; Tudino, V.; De Leo, A.; Bortolami, M.; De Vita, D.; Scipione, L.; Pepi, F.; Costi, R.; Rivara, S.; Scalvini, L.; Mor, M.; Ferrara, F. F.; Pavoni, E.; Roscilli, G.; Cassinelli, G.; Milazzo, F. M.; Battistuzzi, G.; Di Santo, R.; Giannini, G. | |
| Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands | 1-gen-2018 | Rivara, Silvia; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Caignard, Daniel-Henri; Delagrange, Philippe; Collina, Simona; Lucini, Valeria; Scaglione, Francesco; Furiassi, Lucia; Mari, Michele; Lucarini, Simone; Bedini, Annalida; Spadoni, Gilberto | |
| Identification of bivalent ligands with melatonin receptor agonist and fatty acid amide hydrolase (FAAH) inhibitory activity that exhibit ocular hypotensive effect in the rabbit | 1-gen-2018 | Spadoni, G; Bedini, A; Furiassi, L; Mari, M; Mor, M; Scalvini, L; Lodola, A; Ghidini, Andrea; Lucini, V; Dugnani, S; Scaglione, F; Piomelli, D; Jung, Km; Supuran, Ct; Lucarini, L; Durante, M; Sgambellone, S; Masini, E; Rivara, S. | |
| Social stress contagion in rats: Behavioural, autonomic and neuroendocrine correlates | 1-gen-2017 | Carnevali, Luca; Montano, Nicola; Statello, ROSARIO IGNAZIO; Coude', Gino; Vacondio, Federica; Rivara, Silvia; Ferrari, Pier Francesco; Sgoifo, Andrea | |
| Metadynamics Simulations Distinguish Short- and Long-Residence-Time Inhibitors of Cyclin-Dependent Kinase 8. | 1-gen-2017 | Callegari, Donatella; Lodola, Alessio; Pala, Daniele; Rivara, Silvia; Mor, Marco; Rizzi, A; Capelli A., M. |
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