Sfoglia per Autore
Quantitative structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors.
2008-01-01 Fioni, A.; Vacondio, Federica; Mor, Marco; Silva, Claudia; Lodola, Alessio; Duranti, A.; Tontini, A.; Tarzia, G.; Piomelli, D.
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma.
2008-01-01 Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor.
2008-01-01 Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity
2006-01-01 Spadoni, G; Diamantini, G; Bedini, A; Tarzia, G; Vacondio, Federica; Silva, Claudia; Rivara, Mirko; Mor, Marco; Plazzi, Pier Vincenzo; Zusso, M; Franceschini, D; Giusti, P.
Creatine as a compatible osmolyte in muscle cells exposed to hypertonic stress
2006-01-01 Alfieri, R; Bonelli, M; Cavazzoni, A; Brigotti, Maurizio; Fumarola, C; Sestili, Piero; Mozzoni, P; DE PALMA, Giuseppe; Mutti, A; Carnicelli, D; Vacondio, F; Silva, C; Borghetti, A. F; Wheeler, K. P; Petronini, P.
Indole-based analogs of melatonin: in vitro antioxidant and cytoprotective activities
2004-01-01 Mor, Marco; Silva, Claudia; Vacondio, Federica; Plazzi, Pier Vincenzo; Bertoni, Simona; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Zusso, M.; Franceschini, D.; Giusti, P.
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists
2004-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors
2004-01-01 Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B.
Antioxidant and cytoprotective activity of indole derivatives related to melatonin
2003-01-01 Mor, Marco; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Silva, Claudia; Vacondio, Federica; Rivara, Mirko; Plazzi, Pier Vincenzo; Franceschini, D.; Zusso, M.; Giusti, P.
Synthesis and 3D-QSAR Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group
2003-01-01 Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Plazzi, Pier Vincenzo; Carrupt, P. A.; Testa, B.
pH-partition profiles of 4-(3-oxo-1,2-benzisothiazolin-2-yl)phenyl and phenoxyalkanoic acids
2003-01-01 Silva, Claudia; Mor, Marco; Vacondio, Federica; Zuliani, Valentina; Plazzi, P. V.
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays
2003-01-01 Zuliani, Valentina; Bordi, Fabrizio; Rivara, Mirko; Silva, Claudia; Vacondio, Federica; Morini, Giovanni; Rivara, Silvia; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Magnanini, F.; Plazzi, Pier Vincenzo
Three-Dimensional Quantitative Structure-Activity Relationship Studies on Selected MT1 and MT2 Melatonin Receptor Ligands: Requirements for Subtype Selectivity and Intrinsic Activity Modulation
2003-01-01 Rivara, Silvia; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Spadoni, G; Bedini, A; Tarzia, G; Lucini, V; Pannacci, M; Fraschini, F; Plazzi, Pier Vincenzo
Relationship between structure and ex-vivo binding of imidazole H3 antagonists to rat brain H3 receptors
2001-01-01 Vacondio, Federica; Zuliani, Valentina; Mor, Marco; Silva, Claudia; F., Bordi; F., Vacondio; Ballabeni, Vigilio; F., Magnanini; Barocelli, Elisabetta; P. V., Plazzi; P. A., Carrupt; B., Testa
Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups
2000-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Structure-Property Relationships on Histamine H3-Antagonists: Binding of Phenyl-substituted Alkylthioimidazole Derivatives to Rat Plasma Proteins
2000-01-01 Silva, Claudia; Plazzi, Pier Vincenzo; Bordi, Fabrizio; Rivara, Silvia; Vacondio, Federica; Zuliani, Valentina; Caretta, Antonio; Mor, Marco
Aminobenzimidazoles as new potent H3-antagonists
1999-01-01 Zuliani, Valentina; F., Bordi; Mor, Marco; Silva, Claudia; Rivara, Silvia; Vacondio, Federica; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; P. V., Plazzi
2-Aminobenzimidazoles as new potent H3-antagonists
1999-01-01 Zuliani, Valentina; F., Bordi; Mor, Marco; Silva, Claudia; Rivara, Silvia; Vacondio, Federica; Barocelli, Elisabetta; Ballabeni, Vigilio; M., Impicciatore; P. V., Plazzi
Interactions of new and conventional H3-blockers with non-histaminergic receptors involved in neurogenic and myogenic contractile responses of guinea-pig ileum
1999-01-01 Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Silva, Claudia; Impicciatore, Mariannina
Histamine H3-antagonists: the basicity of the polar group in quantitative structure-activity and structure-property relationship
1998-01-01 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Morini, Giovanni; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Quantitative structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors. | 1-gen-2008 | Fioni, A.; Vacondio, Federica; Mor, Marco; Silva, Claudia; Lodola, Alessio; Duranti, A.; Tontini, A.; Tarzia, G.; Piomelli, D. | |
| Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. | 1-gen-2008 | Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta | |
| Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. | 1-gen-2008 | Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
| Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity | 1-gen-2006 | Spadoni, G; Diamantini, G; Bedini, A; Tarzia, G; Vacondio, Federica; Silva, Claudia; Rivara, Mirko; Mor, Marco; Plazzi, Pier Vincenzo; Zusso, M; Franceschini, D; Giusti, P. | |
| Creatine as a compatible osmolyte in muscle cells exposed to hypertonic stress | 1-gen-2006 | Alfieri, R; Bonelli, M; Cavazzoni, A; Brigotti, Maurizio; Fumarola, C; Sestili, Piero; Mozzoni, P; DE PALMA, Giuseppe; Mutti, A; Carnicelli, D; Vacondio, F; Silva, C; Borghetti, A. F; Wheeler, K. P; Petronini, P. | |
| Indole-based analogs of melatonin: in vitro antioxidant and cytoprotective activities | 1-gen-2004 | Mor, Marco; Silva, Claudia; Vacondio, Federica; Plazzi, Pier Vincenzo; Bertoni, Simona; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Zusso, M.; Franceschini, D.; Giusti, P. | |
| Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists | 1-gen-2004 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo | |
| Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors | 1-gen-2004 | Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B. | |
| Antioxidant and cytoprotective activity of indole derivatives related to melatonin | 1-gen-2003 | Mor, Marco; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Silva, Claudia; Vacondio, Federica; Rivara, Mirko; Plazzi, Pier Vincenzo; Franceschini, D.; Zusso, M.; Giusti, P. | |
| Synthesis and 3D-QSAR Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group | 1-gen-2003 | Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Plazzi, Pier Vincenzo; Carrupt, P. A.; Testa, B. | |
| pH-partition profiles of 4-(3-oxo-1,2-benzisothiazolin-2-yl)phenyl and phenoxyalkanoic acids | 1-gen-2003 | Silva, Claudia; Mor, Marco; Vacondio, Federica; Zuliani, Valentina; Plazzi, P. V. | |
| The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays | 1-gen-2003 | Zuliani, Valentina; Bordi, Fabrizio; Rivara, Mirko; Silva, Claudia; Vacondio, Federica; Morini, Giovanni; Rivara, Silvia; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Magnanini, F.; Plazzi, Pier Vincenzo | |
| Three-Dimensional Quantitative Structure-Activity Relationship Studies on Selected MT1 and MT2 Melatonin Receptor Ligands: Requirements for Subtype Selectivity and Intrinsic Activity Modulation | 1-gen-2003 | Rivara, Silvia; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Vacondio, Federica; Spadoni, G; Bedini, A; Tarzia, G; Lucini, V; Pannacci, M; Fraschini, F; Plazzi, Pier Vincenzo | |
| Relationship between structure and ex-vivo binding of imidazole H3 antagonists to rat brain H3 receptors | 1-gen-2001 | Vacondio, Federica; Zuliani, Valentina; Mor, Marco; Silva, Claudia; F., Bordi; F., Vacondio; Ballabeni, Vigilio; F., Magnanini; Barocelli, Elisabetta; P. V., Plazzi; P. A., Carrupt; B., Testa | |
| Synthesis and biological assays of new H3-antagonists with imidazole and imidazoline polar groups | 1-gen-2000 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Morini, Giovanni; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo | |
| Structure-Property Relationships on Histamine H3-Antagonists: Binding of Phenyl-substituted Alkylthioimidazole Derivatives to Rat Plasma Proteins | 1-gen-2000 | Silva, Claudia; Plazzi, Pier Vincenzo; Bordi, Fabrizio; Rivara, Silvia; Vacondio, Federica; Zuliani, Valentina; Caretta, Antonio; Mor, Marco | |
| Aminobenzimidazoles as new potent H3-antagonists | 1-gen-1999 | Zuliani, Valentina; F., Bordi; Mor, Marco; Silva, Claudia; Rivara, Silvia; Vacondio, Federica; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; P. V., Plazzi | |
| 2-Aminobenzimidazoles as new potent H3-antagonists | 1-gen-1999 | Zuliani, Valentina; F., Bordi; Mor, Marco; Silva, Claudia; Rivara, Silvia; Vacondio, Federica; Barocelli, Elisabetta; Ballabeni, Vigilio; M., Impicciatore; P. V., Plazzi | |
| Interactions of new and conventional H3-blockers with non-histaminergic receptors involved in neurogenic and myogenic contractile responses of guinea-pig ileum | 1-gen-1999 | Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Silva, Claudia; Impicciatore, Mariannina | |
| Histamine H3-antagonists: the basicity of the polar group in quantitative structure-activity and structure-property relationship | 1-gen-1998 | Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Morini, Giovanni; Barocelli, Elisabetta; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo |
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