Sfoglia per Autore
Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains
2018-01-01 Machado, Diana; Perdigão, João; Portugal, Isabel; Pieroni, Marco; Silva, Pedro A.; Couto and Miguel Viveiros, Isabel
Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets
2018-01-01 Magalhães, Joana; Annunziato, Giannamaria; Franko, Nina; Pieroni, Marco; Campanini, Barbara; Bruno, Agostino; Costantino, Gabriele
Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design
2018-01-01 Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara
In vitro digestion of zingiber officinale extract and evaluation of stability as a first step to determine its bioaccesibility
2018-01-01 Annunziato, Giannamaria; Falavigna, Claudia; Pieroni, Marco; Faccini, Andrea; Micheli, Fabrizio; Costantino, Gabriele
Modulation of bacterial metabolism by the microenvironment controls MAIT cell stimulation article
2018-01-01 Schmaler, M.; Colone, A.; Spagnuolo, J.; Zimmermann, M.; Lepore, M.; Kalinichenko, A.; Bhatia, S.; Cottier, F.; Rutishauser, T.; Pavelka, N.; Egli, A.; Azzali, E.; Pieroni, M.; Costantino, G.; Hruz, P.; Sauer, U.; Mori, L.; De Libero, G.
Antituberculosis agents: Beyond medicinal chemistry rules
2019-01-01 Pieroni, M.
Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections
2019-01-01 Rossi, Irene; Buttini, Francesca; Sonvico, Fabio; Affaticati, Filippo; Martinelli, Francesco; Annunziato, Giannamaria; Machado, Diana; Viveiros, Miguel; Pieroni, Marco; Bettini, Ruggero
Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: Implications for Primary Hyperoxaluria type 1
2019-01-01 Dindo, M.; Grottelli, S.; Annunziato, G.; Giardina, G.; Pieroni, M.; Pampalone, G.; Faccini, A.; Cutruzzola, F.; Laurino, P.; Costantino, G.; Cellini, B.
Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms
2019-01-01 Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Nikitjuka, Anna; Mozzarelli, Andrea; Bettati, Stefano; Karawajczyk, Anna; Jirgensons, Aigars; Campanini, Barbara; Costantino, Gabriele
Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor
2020-01-01 Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G.
2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry
2020-01-01 Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M.
Nitric oxide-releasing cyclodextrins as biodegradable antibacterial scaffolds: a patent evaluation of US2019343869(A1)
2020-01-01 Pieroni, M.
Nuovi composti antimicrobici
2021-01-01 Annunziato, Giannamaria; Costantino, Gabriele; Cabassi, Clotilde Silvia; Pieroni, Marco; Bruno, Agostino; Campanini, Barbara; Bettati, Stefano; Mozzarelli, Andrea
A competitive o‐acetylserine sulfhydrylase inhibitor modulates the formation of cysteine synthase complex
2021-01-01 Marchetti, M.; De Angelis, F. S.; Annunziato, G.; Costantino, G.; Pieroni, M.; Ronda, L.; Mozzarelli, A.; Campanini, B.; Cannistraro, S.; Bizzarri, A. R.; Bettati, S.
Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants
2021-01-01 Magalhães, Joana; Franko, Nina; Raboni, Samanta; Annunziato, Giannamaria; Tammela, Päivi; Bruno, Agostino; Bettati, Stefano; Armao, Stefano; Spadini, Costanza; Cabassi, Clotilde Silvia; Mozzarelli, Andrea; Pieroni, Marco; Campanini, Barbara; Costantino, Gabriele
Aspergillus fumigatus tryptophan metabolic route differently affects host immunity
2021-01-01 Zelante, T.; Choera, T.; Beauvais, A.; Fallarino, F.; Paolicelli, G.; Pieraccini, G.; Pieroni, M.; Galosi, C.; Beato, C.; De Luca, A.; Boscaro, F.; Romoli, R.; Liu, X.; Warris, A.; Verweij, P. E.; Ballard, E.; Borghi, M.; Pariano, M.; Costantino, G.; Calvitti, M.; Vacca, C.; Oikonomou, V.; Gargaro, M.; Wong, A. Y. W.; Boon, L.; den Hartog, M.; Spacil, Z.; Puccetti, P.; Latge, J. -P.; Keller, N. P.; Romani, L.
Investigational Studies on a Hit Compound Cyclopropane-Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin Adjuvant
2021-01-01 Annunziato, G.; Spadini, C.; Franko, N.; Storici, P.; Demitri, N.; Pieroni, M.; Flisi, S.; Rosati, L.; Iannarelli, M.; Marchetti, M.; Magalhaes, J.; Bettati, S.; Mozzarelli, A.; Cabassi, C. S.; Campanini, B.; Costantino, G.
Towards the sustainable discovery and development of new antibiotics
2021-01-01 Miethke, M.; Pieroni, M.; Weber, T.; Bronstrup, M.; Hammann, P.; Halby, L.; Arimondo, P. B.; Glaser, P.; Aigle, B.; Bode, H. B.; Moreira, R.; Li, Y.; Luzhetskyy, A.; Medema, M. H.; Pernodet, J. -L.; Stadler, M.; Tormo, J. R.; Genilloud, O.; Truman, A. W.; Weissman, K. J.; Takano, E.; Sabatini, S.; Stegmann, E.; Brotz-Oesterhelt, H.; Wohlleben, W.; Seemann, M.; Empting, M.; Hirsch, A. K. H.; Loretz, B.; Lehr, C. -M.; Titz, A.; Herrmann, J.; Jaeger, T.; Alt, S.; Hesterkamp, T.; Winterhalter, M.; Schiefer, A.; Pfarr, K.; Hoerauf, A.; Graz, H.; Graz, M.; Lindvall, M.; Ramurthy, S.; Karlen, A.; van Dongen, M.; Petkovic, H.; Keller, A.; Peyrane, F.; Donadio, S.; Fraisse, L.; Piddock, L. J. V.; Gilbert, I. H.; Moser, H. E.; Muller, R.
Crystal structure of Aspergillus fumigatus AroH, an aromatic amino acid aminotransferase
2021-01-01 Spizzichino, Sharon; Pampalone, Gioena; Dindo, Mirco; Bruno, Agostino; Romani, Luigina; Cutruzzolà, Francesca; Zelante, Teresa; Pieroni, Marco; Cellini, Barbara; Giardina, Giorgio
Identification of Human Alanine-Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1
2022-01-01 Grottelli, Silvia; Annunziato, Giannamaria; Pampalone, Gioena; Pieroni, Marco; Dindo, Mirco; Ferlenghi, Francesca; Costantino, Gabriele; Cellini, Barbara
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains | 1-gen-2018 | Machado, Diana; Perdigão, João; Portugal, Isabel; Pieroni, Marco; Silva, Pedro A.; Couto and Miguel Viveiros, Isabel | |
| Integration of Enhanced Sampling Methods with Saturation Transfer Difference Experiments to Identify Protein Druggable Pockets | 1-gen-2018 | Magalhães, Joana; Annunziato, Giannamaria; Franko, Nina; Pieroni, Marco; Campanini, Barbara; Bruno, Agostino; Costantino, Gabriele | |
| Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design | 1-gen-2018 | Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara | |
| In vitro digestion of zingiber officinale extract and evaluation of stability as a first step to determine its bioaccesibility | 1-gen-2018 | Annunziato, Giannamaria; Falavigna, Claudia; Pieroni, Marco; Faccini, Andrea; Micheli, Fabrizio; Costantino, Gabriele | |
| Modulation of bacterial metabolism by the microenvironment controls MAIT cell stimulation article | 1-gen-2018 | Schmaler, M.; Colone, A.; Spagnuolo, J.; Zimmermann, M.; Lepore, M.; Kalinichenko, A.; Bhatia, S.; Cottier, F.; Rutishauser, T.; Pavelka, N.; Egli, A.; Azzali, E.; Pieroni, M.; Costantino, G.; Hruz, P.; Sauer, U.; Mori, L.; De Libero, G. | |
| Antituberculosis agents: Beyond medicinal chemistry rules | 1-gen-2019 | Pieroni, M. | |
| Sodium Hyaluronate Nanocomposite Respirable Microparticles to Tackle Antibiotic Resistance with Potential Application in Treatment of Mycobacterial Pulmonary Infections | 1-gen-2019 | Rossi, Irene; Buttini, Francesca; Sonvico, Fabio; Affaticati, Filippo; Martinelli, Francesco; Annunziato, Giannamaria; Machado, Diana; Viveiros, Miguel; Pieroni, Marco; Bettini, Ruggero | |
| Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: Implications for Primary Hyperoxaluria type 1 | 1-gen-2019 | Dindo, M.; Grottelli, S.; Annunziato, G.; Giardina, G.; Pieroni, M.; Pampalone, G.; Faccini, A.; Cutruzzola, F.; Laurino, P.; Costantino, G.; Cellini, B. | |
| Refining the structure−activity relationships of 2-phenylcyclopropane carboxylic acids as inhibitors of O-acetylserine sulfhydrylase isoforms | 1-gen-2019 | Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Nikitjuka, Anna; Mozzarelli, Andrea; Bettati, Stefano; Karawajczyk, Anna; Jirgensons, Aigars; Campanini, Barbara; Costantino, Gabriele | |
| Inhibition of Nonessential Bacterial Targets: Discovery of a Novel Serine O-Acetyltransferase Inhibitor | 1-gen-2020 | Magalhaes, J.; Franko, N.; Raboni, S.; Annunziato, G.; Tammela, P.; Bruno, A.; Bettati, S.; Mozzarelli, A.; Pieroni, M.; Campanini, B.; Costantino, G. | |
| 2-Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry | 1-gen-2020 | Azzali, E.; Girardini, M.; Annunziato, G.; Pavone, M.; Vacondio, F.; Mori, G.; Pasca, M. R.; Costantino, G.; Pieroni, M. | |
| Nitric oxide-releasing cyclodextrins as biodegradable antibacterial scaffolds: a patent evaluation of US2019343869(A1) | 1-gen-2020 | Pieroni, M. | |
| Nuovi composti antimicrobici | 1-gen-2021 | Annunziato, Giannamaria; Costantino, Gabriele; Cabassi, Clotilde Silvia; Pieroni, Marco; Bruno, Agostino; Campanini, Barbara; Bettati, Stefano; Mozzarelli, Andrea | |
| A competitive o‐acetylserine sulfhydrylase inhibitor modulates the formation of cysteine synthase complex | 1-gen-2021 | Marchetti, M.; De Angelis, F. S.; Annunziato, G.; Costantino, G.; Pieroni, M.; Ronda, L.; Mozzarelli, A.; Campanini, B.; Cannistraro, S.; Bizzarri, A. R.; Bettati, S. | |
| Discovery of Substituted (2-Aminooxazol-4-yl)Isoxazole-3-carboxylic Acids as Inhibitors of Bacterial Serine Acetyltransferase in the Quest for Novel Potential Antibacterial Adjuvants | 1-gen-2021 | Magalhães, Joana; Franko, Nina; Raboni, Samanta; Annunziato, Giannamaria; Tammela, Päivi; Bruno, Agostino; Bettati, Stefano; Armao, Stefano; Spadini, Costanza; Cabassi, Clotilde Silvia; Mozzarelli, Andrea; Pieroni, Marco; Campanini, Barbara; Costantino, Gabriele | |
| Aspergillus fumigatus tryptophan metabolic route differently affects host immunity | 1-gen-2021 | Zelante, T.; Choera, T.; Beauvais, A.; Fallarino, F.; Paolicelli, G.; Pieraccini, G.; Pieroni, M.; Galosi, C.; Beato, C.; De Luca, A.; Boscaro, F.; Romoli, R.; Liu, X.; Warris, A.; Verweij, P. E.; Ballard, E.; Borghi, M.; Pariano, M.; Costantino, G.; Calvitti, M.; Vacca, C.; Oikonomou, V.; Gargaro, M.; Wong, A. Y. W.; Boon, L.; den Hartog, M.; Spacil, Z.; Puccetti, P.; Latge, J. -P.; Keller, N. P.; Romani, L. | |
| Investigational Studies on a Hit Compound Cyclopropane-Carboxylic Acid Derivative Targeting O-Acetylserine Sulfhydrylase as a Colistin Adjuvant | 1-gen-2021 | Annunziato, G.; Spadini, C.; Franko, N.; Storici, P.; Demitri, N.; Pieroni, M.; Flisi, S.; Rosati, L.; Iannarelli, M.; Marchetti, M.; Magalhaes, J.; Bettati, S.; Mozzarelli, A.; Cabassi, C. S.; Campanini, B.; Costantino, G. | |
| Towards the sustainable discovery and development of new antibiotics | 1-gen-2021 | Miethke, M.; Pieroni, M.; Weber, T.; Bronstrup, M.; Hammann, P.; Halby, L.; Arimondo, P. B.; Glaser, P.; Aigle, B.; Bode, H. B.; Moreira, R.; Li, Y.; Luzhetskyy, A.; Medema, M. H.; Pernodet, J. -L.; Stadler, M.; Tormo, J. R.; Genilloud, O.; Truman, A. W.; Weissman, K. J.; Takano, E.; Sabatini, S.; Stegmann, E.; Brotz-Oesterhelt, H.; Wohlleben, W.; Seemann, M.; Empting, M.; Hirsch, A. K. H.; Loretz, B.; Lehr, C. -M.; Titz, A.; Herrmann, J.; Jaeger, T.; Alt, S.; Hesterkamp, T.; Winterhalter, M.; Schiefer, A.; Pfarr, K.; Hoerauf, A.; Graz, H.; Graz, M.; Lindvall, M.; Ramurthy, S.; Karlen, A.; van Dongen, M.; Petkovic, H.; Keller, A.; Peyrane, F.; Donadio, S.; Fraisse, L.; Piddock, L. J. V.; Gilbert, I. H.; Moser, H. E.; Muller, R. | |
| Crystal structure of Aspergillus fumigatus AroH, an aromatic amino acid aminotransferase | 1-gen-2021 | Spizzichino, Sharon; Pampalone, Gioena; Dindo, Mirco; Bruno, Agostino; Romani, Luigina; Cutruzzolà, Francesca; Zelante, Teresa; Pieroni, Marco; Cellini, Barbara; Giardina, Giorgio | |
| Identification of Human Alanine-Glyoxylate Aminotransferase Ligands as Pharmacological Chaperones for Variants Associated with Primary Hyperoxaluria Type 1 | 1-gen-2022 | Grottelli, Silvia; Annunziato, Giannamaria; Pampalone, Gioena; Pieroni, Marco; Dindo, Mirco; Ferlenghi, Francesca; Costantino, Gabriele; Cellini, Barbara |
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