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Recent advances in the development of melatonin MT(1) and MT(2) receptor agonists. 1-gen-2010 Mor, Marco; Rivara, Silvia; Pala, Daniele; A., Bedini; G., Spadoni; G., Tarzia
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives. 1-gen-2011 A., Bedini; S., Lucarini; G., Spadoni; G., Tarzia; F., Scaglione; S., Dugnani; M., Pannacci; V., Lucini; Carmi, Caterina; Pala, Daniele; Rivara, Silvia; Mor, Marco
Design and structure-activity relationships of amino acid derivatives of lithocholic acid as novel EphA2 receptor antagonists. 1-gen-2012 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Iftiin Hassan Mohamed, ; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists 1-gen-2012 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
MT1-Selective Melatonin Receptor Ligands: Synthesis, Pharmacological Evaluation, and Molecular Dynamics Investigation of N-[[(3-O-Substituted)anilino]alkyl]amides. 1-gen-2012 Rivara, Silvia; Pala, Daniele; Lodola, Alessio; Mor, Marco; Lucini, V.; Dugnani, S.; Scaglione, F.; Bedini, A.; Lucarini, S.; Tarzia, G.; Spadoni, G.
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain. 1-gen-2012 Bordi, Fabrizio; Rivara, Silvia; E., Dallaturca; Carmi, Caterina; Pala, Daniele; Lodola, Alessio; Vacondio, Federica; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Computer-Aided Design of Novel Antagonists of the EphA2 Receptor 1-gen-2013 Pala, Daniele; Rivara, Silvia; Incerti, Matteo; Tognolini, Massimiliano; Mor, Marco
Target-hopping: a useful approach to identify novel Eph receptor antagonists 1-gen-2013 Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Pala, Daniele; Russo, Simonetta; Lodola, Alessio; Incerti, Matteo; Barocelli, Elisabetta; Tognolini, Massimiliano
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties 1-gen-2013 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano
Homology models of melatonin receptors: challenges and recent advances. 1-gen-2013 Pala, Daniele; Lodola, Alessio; Bedini, A.; Spadoni, G.; Rivara, Silvia
Structure-based virtual screening of MT2 melatonin receptor: influence of template choice and structural refinement. 1-gen-2013 Pala, Daniele; Beuming, T; Sherman, W; Lodola, Alessio; Rivara, Silvia; Mor, Marco
Synthesis of (E)-8-(3-chlorostyryl)caffeine analogs leading to 9-deazaxanthine derivatives as dual A2A antagonists /MAO-B inhibitors. 1-gen-2013 Rivara, Silvia; Piersanti, G.; Bartoccini, F.; Diamantini, G.; Pala, Daniele; Riccioni, T.; Stasi, M. A.; Cabri, W.; Borsini, F.; Mor, Marco; Tarzia, G.; Minetti, P.
Complex product composition generates risks for generic substitution also with dosage forms for intravenous administration 1-gen-2013 Rossi, Alessandra; Buttini, Francesca; Colombo, Paolo; Mor, Marco; Pala, Daniele; F., Bortolotti; Colombo, Gaia
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. 1-gen-2013 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor. 1-gen-2013 Russo, Simonetta; Incerti, Matteo; Tognolini, Massimiliano; Castelli, Riccardo; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; De Franco, F; Gioiello, A; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity 1-gen-2014 Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Barocelli, Elisabetta; Bertoni, Simona; Pala, Daniele; Mor, Marco; Russo, Simonetta; Lodola, Alessio
Synthesis and characterization of new bivalent agents as melatonin- and histamine h3-ligands. 1-gen-2014 Pala, Daniele; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Flammini, Lisa; Barocelli, Elisabetta; Lucini, V; Scaglione, F; Bartolucci, S; Bedini, A; Rivara, Silvia; Spadoni, G.
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction. 1-gen-2014 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Castelli, Riccardo; Pala, Daniele; Mor, Marco; Barocelli, Elisabetta; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis 1-gen-2014 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta; Mor, Marco; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Tognolini, Massimiliano
Towards the development of 5-HT7 ligands combining serotonin-like and arylpiperazine moieties 1-gen-2014 Spadoni, G.; Bedini, A.; Bartolucci, S.; Pala, Daniele; Mor, Marco; Riccioni, T.; Borsini, F.; Cabri, W.; Celona, D.; Marzi, M.; Tarzia, G.; Rivara, Silvia; Minetti, P.
Mostrati risultati da 1 a 20 di 42
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