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Lithocholic acid competitively inhibitis EphA2-ephrinA1 binding: pharmacological and structural considerations. 1-gen-2010 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta
Discovery of natural extracts interfering with EphA2-ephrinA1 system 1-gen-2010 Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Bruni, Renato; Domenichini, Giuseppe; Barocelli, Elisabetta; Tognolini, Massimiliano
Lithocholic acid competitively inhibits EphA2-ephrinA1 binding: pharmacological and structural considerations. 1-gen-2010 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta
Lithocholic acid is an Eph-ephrin ligand interfering with Eph-kinase activation 1-gen-2011 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Flammini, Lisa; Barocelli, Elisabetta; Incerti, Matteo; Lodola, Alessio; Tognolini, Massimiliano
Botanicals used as food supplements interfering with EphA2-ephrinA1 system: a screening study 1-gen-2011 Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Bruni, Renato; Flammini, Lisa; Barocelli, Elisabetta; A., Guerrini; Bertoni, Simona; Tognolini, Massimiliano
Structure activity relationship of new EphA2 ligands 1-gen-2011 Tognolini, Massimiliano; Incerti, Matteo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Barocelli, Elisabetta; Russo, Simonetta; B., Lelli; L., Bracci; Lodola, Alessio
Polyphenol rich botanicals used as food supplements interfere with EphA2-ephrinA1 system. 1-gen-2011 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Bruni, Renato; Flammini, Lisa; Barocelli, Elisabetta; D., Rossi; Domenichini, Giuseppe; F., Poli; Tognolini, Massimiliano
Design and structure-activity relationship of amino acid derivatives of lithocholic acid as novel EphA2 antagonists 1-gen-2012 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Vicini, Paola; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Structure–Activity Relationships and Mechanism of Action of Eph–ephrin Antagonists: Interaction of Cholanic Acid with the EphA2 Receptor 1-gen-2012 Tognolini, Massimiliano; Incerti, Matteo; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Bruni, Renato; Barbara, Lelli; Luisa, Bracci; Roberta, Noberini; Elena, B. Pasquale; Barocelli, Elisabetta; Vicini, Paola; Mor, Marco; Lodola, Alessio
Perturbation of The EphA2-EphrinA1 System in Human Prostate Cancer Cells by Colonic (Poly)phenol Catabolites 1-gen-2012 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Barocelli, Elisabetta; L., Calani; E., Reynaud; O., Dangles; G., Borges; A., Crozier; Brighenti, Furio; DEL RIO, Daniele
Target-hopping: a useful approach to identify novel Eph receptor antagonists 1-gen-2013 Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Pala, Daniele; Russo, Simonetta; Lodola, Alessio; Incerti, Matteo; Barocelli, Elisabetta; Tognolini, Massimiliano
Discovery and development of Eph-ephrin antagonists endowed with antiangiogenic properties 1-gen-2013 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Lodola, Alessio; Barocelli, Elisabetta; Tognolini, Massimiliano
Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor. 1-gen-2013 Incerti, Matteo; Tognolini, Massimiliano; Russo, Simonetta; Pala, Daniele; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Noberini, R; Pasquale, Eb; Vicini, Paola; Piersanti, Silvia; Rivara, Silvia; Barocelli, Elisabetta; Mor, Marco; Lodola, Alessio
Synthesis and Structure-Activity Relationships of Amino Acid Conjugates of Cholanic Acid as Antagonists of the EphA2 Receptor. 1-gen-2013 Russo, Simonetta; Incerti, Matteo; Tognolini, Massimiliano; Castelli, Riccardo; Pala, Daniele; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; De Franco, F; Gioiello, A; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio
Discovery and development of low molecular weight Eph-ephrin protein-protein inhbi-tors endowed with antiangiogenic activity 1-gen-2014 Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Barocelli, Elisabetta; Bertoni, Simona; Pala, Daniele; Mor, Marco; Russo, Simonetta; Lodola, Alessio
Combining pharmacology, target hopping and computational medicinal chemistry to discover novel scaffold targeting EPH-ephrin interaction. 1-gen-2014 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Castelli, Riccardo; Pala, Daniele; Mor, Marco; Barocelli, Elisabetta; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
Development of 3-oxo-cholenic derivatives as Eph antagonists able to block in vitro angiogenesis 1-gen-2014 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Castelli, Riccardo; Lodola, Alessio; Barocelli, Elisabetta; Mor, Marco; Russo, Simonetta; Incerti, Matteo; Pala, Daniele; Tognolini, Massimiliano
Therapeutic perspectives of Eph–ephrin system modulation 1-gen-2014 Tognolini, Massimiliano; HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Zanotti, Ilaria; Lodola, Alessio
270 Discovery, development and optimization of low molecular weight EPH–ephrin protein–protein inhibitors 1-gen-2014 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Barocelli, Elisabetta; Mor, Marco; Pala, Daniele; Russo, Simonetta; Incerti, Matteo; Lodola, Alessio
UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations. 1-gen-2014 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Incerti, Matteo; Russo, Simonetta; Pala, Daniele; Pasquale, Eb; Zanotti, Ilaria; Vicini, Paola; Barocelli, Elisabetta; Rivara, Silvia; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano
Mostrati risultati da 1 a 20 di 24
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