Sfoglia per Autore
Cognition enhancing effect in rats of a selected histamine H3 receptor antagonist with good brain penetration
2005-01-01 Barocelli, Elisabetta; Ballabeni, Vigilio; Flammini, Lisa; Bertoni, Simona; Tognolini, Massimiliano; Chiavarini, Milena; Zuliani, Valentina; Rivara, Mirko; Vacondio, Federica; Impicciatore, Mariannina
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold.
2006-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Discovery of histamine H3 receptor antagonistic property of simple imidazole-free derivatives: preliminary pharmacological investigation.
2006-01-01 Barocelli, Elisabetta; Ballabeni, Vigilio; Manenti, V; Flammini, Lisa; Bertoni, Simona; Morini, Giovanni; Comini, Mara; Impicciatore, Mariannina
In vitro pharmacology at human histamine H(3) receptors and brain access of non-imidazole alkylpiperidine derivatives.
2007-01-01 Bertoni, Simona; Flammini, Lisa; Manenti, V.; Ballabeni, Vigilio; Morini, Giovanni; Comini, Mara; Barocelli, Elisabetta
Pharmacological characterization of a new non-himidazole histamine H3 antagonist
2007-01-01 Flammini, Lisa; Bertoni, Simona; Saccani, Francesca; Ballabeni, Vigilio; Impicciatore, Mariannina; Barocelli, Elisabetta
Intestinal chronic obstruction affects motor responsiveness of rat hypertrophic longitudinal and circular muscles
2008-01-01 Bertoni, Simona; Ghizzardi, Paola; Flammini, Lisa; Saccani, Francesca; Gobbetti, Thomas; Cattaruzza, Fiore; Impicciatore, Mariannina; Ballabeni, Vigilio; Barocelli, Elisabetta
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity.
2008-01-01 Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Saccani, Francesca; Domenichini, Giuseppe; Morini, Giovanni; Comini, Mara; Rivara, Mirko; Barocelli, Elisabetta
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma.
2008-01-01 Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity.
2008-01-01 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor.
2008-01-01 Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
A promising imidazole-free histamine H3 receptor antagonist with good brain penetration and anticholinesterase activity.
2008-01-01 Barocelli, Elisabetta; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ghizzardi, Paola; Gobbetti, Thomas; Morini, Giovanni; Ballabeni, Vigilio
Aminopyridine derivatives with anticholinesterase and antiamnesic activity
2008-01-01 Scipione, L; DE VITA, D; Musella, A; Flammini, Lisa; Bertoni, Simona; Barocelli, Elisabetta
Multi-target-directed ligands: new histamine H3 receptor antagonists with anticholinesterase activity
2009-01-01 Flammini, Lisa; Bertoni, Simona; Saccani, Francesca; Incerti, Matteo; Morini, Giovanni; Ballabeni, Vigilio; Barocelli, Elisabetta
Histamine H4 receptor antagonism and mesenteric ischemia/reperfusion injury in mice
2009-01-01 Ghizzardi, Paola; Gobbetti, Thomas; Bertoni, Simona; Saccani, Francesca; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta
Accommodation and peristalsis are functional responses to chronic obstruction in rat hypertrophic ileum
2010-01-01 Bertoni, Simona; Flammini, Lisa; Saccani, Francesca; Ballabeni, Vigilio; G., Vegezzi; Tognolini, Massimiliano; Barocelli, Elisabetta
Lithocholic acid competitively inhibits EphA2-ephrinA1 binding: pharmacological and structural considerations.
2010-01-01 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta
Preventive effect of 5-HT1A receptor agonist Buspirone on mesenteric ischemia/reperfusion-induced inflammatory injuries in mice
2010-01-01 Saccani, Francesca; Flammini, Lisa; Gobbetti, Thomas; G., Vegezzi; Ghizzardi, Paola; Bertoni, Simona; Tognolini, Massimiliano; Ballabeni, Vigilio; Barocelli, Elisabetta
Lithocholic acid competitively inhibitis EphA2-ephrinA1 binding: pharmacological and structural considerations.
2010-01-01 Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta
Dual-Acting Drugs: an in vitro Study of Nonimidazole Histamine H(3) Receptor Antagonists Combining Anticholinesterase Activity
2010-01-01 Incerti, Matteo; Flammini, Lisa; Saccani, Francesca; Morini, Giovanni; Comini, Mara; Coruzzi, Massimo; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona
Lithocholic acid is an Eph-ephrin ligand interfering with Eph-kinase activation
2011-01-01 HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Flammini, Lisa; Barocelli, Elisabetta; Incerti, Matteo; Lodola, Alessio; Tognolini, Massimiliano
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Cognition enhancing effect in rats of a selected histamine H3 receptor antagonist with good brain penetration | 1-gen-2005 | Barocelli, Elisabetta; Ballabeni, Vigilio; Flammini, Lisa; Bertoni, Simona; Tognolini, Massimiliano; Chiavarini, Milena; Zuliani, Valentina; Rivara, Mirko; Vacondio, Federica; Impicciatore, Mariannina | |
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. | 1-gen-2006 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo | |
Discovery of histamine H3 receptor antagonistic property of simple imidazole-free derivatives: preliminary pharmacological investigation. | 1-gen-2006 | Barocelli, Elisabetta; Ballabeni, Vigilio; Manenti, V; Flammini, Lisa; Bertoni, Simona; Morini, Giovanni; Comini, Mara; Impicciatore, Mariannina | |
In vitro pharmacology at human histamine H(3) receptors and brain access of non-imidazole alkylpiperidine derivatives. | 1-gen-2007 | Bertoni, Simona; Flammini, Lisa; Manenti, V.; Ballabeni, Vigilio; Morini, Giovanni; Comini, Mara; Barocelli, Elisabetta | |
Pharmacological characterization of a new non-himidazole histamine H3 antagonist | 1-gen-2007 | Flammini, Lisa; Bertoni, Simona; Saccani, Francesca; Ballabeni, Vigilio; Impicciatore, Mariannina; Barocelli, Elisabetta | |
Intestinal chronic obstruction affects motor responsiveness of rat hypertrophic longitudinal and circular muscles | 1-gen-2008 | Bertoni, Simona; Ghizzardi, Paola; Flammini, Lisa; Saccani, Francesca; Gobbetti, Thomas; Cattaruzza, Fiore; Impicciatore, Mariannina; Ballabeni, Vigilio; Barocelli, Elisabetta | |
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity. | 1-gen-2008 | Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Saccani, Francesca; Domenichini, Giuseppe; Morini, Giovanni; Comini, Mara; Rivara, Mirko; Barocelli, Elisabetta | |
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. | 1-gen-2008 | Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta | |
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. | 1-gen-2008 | Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. | 1-gen-2008 | Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
A promising imidazole-free histamine H3 receptor antagonist with good brain penetration and anticholinesterase activity. | 1-gen-2008 | Barocelli, Elisabetta; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ghizzardi, Paola; Gobbetti, Thomas; Morini, Giovanni; Ballabeni, Vigilio | |
Aminopyridine derivatives with anticholinesterase and antiamnesic activity | 1-gen-2008 | Scipione, L; DE VITA, D; Musella, A; Flammini, Lisa; Bertoni, Simona; Barocelli, Elisabetta | |
Multi-target-directed ligands: new histamine H3 receptor antagonists with anticholinesterase activity | 1-gen-2009 | Flammini, Lisa; Bertoni, Simona; Saccani, Francesca; Incerti, Matteo; Morini, Giovanni; Ballabeni, Vigilio; Barocelli, Elisabetta | |
Histamine H4 receptor antagonism and mesenteric ischemia/reperfusion injury in mice | 1-gen-2009 | Ghizzardi, Paola; Gobbetti, Thomas; Bertoni, Simona; Saccani, Francesca; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta | |
Accommodation and peristalsis are functional responses to chronic obstruction in rat hypertrophic ileum | 1-gen-2010 | Bertoni, Simona; Flammini, Lisa; Saccani, Francesca; Ballabeni, Vigilio; G., Vegezzi; Tognolini, Massimiliano; Barocelli, Elisabetta | |
Lithocholic acid competitively inhibits EphA2-ephrinA1 binding: pharmacological and structural considerations. | 1-gen-2010 | Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta | |
Preventive effect of 5-HT1A receptor agonist Buspirone on mesenteric ischemia/reperfusion-induced inflammatory injuries in mice | 1-gen-2010 | Saccani, Francesca; Flammini, Lisa; Gobbetti, Thomas; G., Vegezzi; Ghizzardi, Paola; Bertoni, Simona; Tognolini, Massimiliano; Ballabeni, Vigilio; Barocelli, Elisabetta | |
Lithocholic acid competitively inhibitis EphA2-ephrinA1 binding: pharmacological and structural considerations. | 1-gen-2010 | Tognolini, Massimiliano; Giorgio, Carmine; HASSAN MOHAMED, Iftiin; Flammini, Lisa; Incerti, Matteo; Lodola, Alessio; Barocelli, Elisabetta | |
Dual-Acting Drugs: an in vitro Study of Nonimidazole Histamine H(3) Receptor Antagonists Combining Anticholinesterase Activity | 1-gen-2010 | Incerti, Matteo; Flammini, Lisa; Saccani, Francesca; Morini, Giovanni; Comini, Mara; Coruzzi, Massimo; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona | |
Lithocholic acid is an Eph-ephrin ligand interfering with Eph-kinase activation | 1-gen-2011 | HASSAN MOHAMED, Iftiin; Giorgio, Carmine; Flammini, Lisa; Barocelli, Elisabetta; Incerti, Matteo; Lodola, Alessio; Tognolini, Massimiliano |
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