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QSAR study of 2-aminobenzimidazole derivatives as H3 antagonists 1-gen-2001 Zuliani, Valentina; Mor, Marco; Rivara, Silvia; F., Bordi; Rivara, Mirko; D., Anceschi; Vacondio, Federica; Ballabeni, Vigilio; Bertoni, Simona; Barocelli, Elisabetta; P. V. P. L. A. Z. Z., I.
Development of a GPCR model for SAR interpretation of classical and new H3 antagonists 1-gen-2003 S., Lorenzi; Mor, Marco; F., Bordi; Rivara, Silvia; Zuliani, Valentina; Rivara, Mirko; Bertoni, Simona; P. V., Plazzi
The Role of HB-Donor Groups in the Heterocyclic Polar Fragment of H3-Antagonists. I. Synthesis and Biological Assays 1-gen-2003 Zuliani, Valentina; Bordi, Fabrizio; Rivara, Mirko; Silva, Claudia; Vacondio, Federica; Morini, Giovanni; Rivara, Silvia; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Magnanini, F.; Plazzi, Pier Vincenzo
Antioxidant and cytoprotective activity of indole derivatives related to melatonin 1-gen-2003 Mor, Marco; Spadoni, G.; Diamantini, G.; Bedini, A.; Tarzia, G.; Silva, Claudia; Vacondio, Federica; Rivara, Mirko; Plazzi, Pier Vincenzo; Franceschini, D.; Zusso, M.; Giusti, P.
Imidazole H3-antagonists: Relationship between Structure and Ex-vivo binding to Rat Brain H3-Receptors 1-gen-2004 Vacondio, Federica; Mor, Marco; Silva, Claudia; Zuliani, Valentina; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Magnanini, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Carrupt, P. A.; Testa, B.
Synthesis, biological activity, QSAR and QSPR study of 2/aminobenzimidazole derivatives as potent H3-antagonists 1-gen-2004 Mor, Marco; Bordi, Fabrizio; Silva, Claudia; Rivara, Silvia; Zuliani, Valentina; Vacondio, Federica; Rivara, Mirko; Barocelli, Elisabetta; Bertoni, Simona; Ballabeni, Vigilio; Impicciatore, Mariannina; Plazzi, Pier Vincenzo
Cognition enhancing effect in rats of a selected histamine H3 receptor antagonist with good brain penetration 1-gen-2005 Barocelli, Elisabetta; Ballabeni, Vigilio; Flammini, Lisa; Bertoni, Simona; Tognolini, Massimiliano; Chiavarini, Milena; Zuliani, Valentina; Rivara, Mirko; Vacondio, Federica; Impicciatore, Mariannina
Validation of a histamine H3 receptor model through structure–activity relationships for classical H3 antagonists 1-gen-2005 Lorenzi, Simone; Mor, Marco; Bordi, Fabrizio; Rivara, Silvia; Rivara, Mirko; Morini, Giovanni; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Dibasic non-imidazole histamine H3 receptor antagonists with a rigid byphenyl scaffold. 1-gen-2006 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Lorenzi, Simone; Bordi, Fabrizio; Mor, Marco; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Plazzi, Pier Vincenzo
Synthesis and biological evaluation of new non-imidazole H(3)-receptor antagonists of the 2-aminobenzimidazole series 1-gen-2006 Rivara, Mirko; Zuliani, Valentina; Cocconcelli, G; Morini, Giovanni; Comini, Mara; Rivara, Silvia; Mor, Marco; Bordi, Fabrizio; Barocelli, Elisabetta; Ballabeni, Vigilio; Bertoni, Simona; Plazzi, Pier Vincenzo
Synthesis, antioxidant activity and structure-activity relationships for a new series of 2-(N-acylaminoethyl)indoles with melatonin-like cytoprotective activity 1-gen-2006 Spadoni, G; Diamantini, G; Bedini, A; Tarzia, G; Vacondio, Federica; Silva, Claudia; Rivara, Mirko; Mor, Marco; Plazzi, Pier Vincenzo; Zusso, M; Franceschini, D; Giusti, P.
A Practical Synthesis of 2,4(5)-Diarylimidazoles from Simple Building Blocks 1-gen-2007 Zuliani, Valentina; Cocconcelli, G.; Fantini, M.; Ghiron, C.; Rivara, Mirko
Development and validation of a LC-MS method with electrospray ionization for the determination of the imidazole H(3) antagonist ROS203 in rat plasma. 1-gen-2008 Vacondio, Federica; Silva, Claudia; A., Fioni; Mor, Marco; Rivara, Mirko; Bordi, Fabrizio; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta
2,4(5)-Diarylimidazoles: Synthesis and Biological Evaluation of a New Class of Sodium Channel Blockers against hNav1.2 1-gen-2008 Rivara, Mirko; Baheti, A. R.; Fantini, M.; Cocconcelli, G.; Ghiron, C.; Kalmar, C. L.; Singh, N.; Merrick, E. C.; Patel, M. K.; Zuliani, Valentina
Synthesis and stability in biological media of 1H-imidazole-1-carboxylates of ROS203, an antagonist of the histamine H3 receptor. 1-gen-2008 Rivara, Mirko; Vacondio, Federica; Silva, Claudia; Zuliani, Valentina; Fantini, M.; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity. 1-gen-2008 Bertoni, Simona; Ballabeni, Vigilio; Flammini, Lisa; Saccani, Francesca; Domenichini, Giuseppe; Morini, Giovanni; Comini, Mara; Rivara, Mirko; Barocelli, Elisabetta
Synthesis and structure-activity relationships for biphenyl H3 receptor antagonists with moderate anti-cholinesterase activity. 1-gen-2008 Morini, Giovanni; Comini, Mara; Rivara, Mirko; Rivara, Silvia; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Flammini, Lisa; Saccani, Francesca; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships 1-gen-2009 Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K.
Recent Advances in the Medicinal Chemistry of Sodium Channel Blockers and their Therapeutic Potential 1-gen-2009 Zuliani, Valentina; Patel, M. K.; Fantini, M.; Rivara, Mirko
Anticonvulsant Activity of 2,4(5)-Diarylimidazoles in Mice and Rat Models 1-gen-2009 Rivara, Mirko; M., Fantini; Zuliani, Valentina; M. K., Patel
Mostrati risultati da 1 a 20 di 47
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