Sfoglia per Autore
Parallel Solution-phase and Microwave-assisted Synthesis of New S-DABO Derivatives Endowed with Subnanomolar Anti-HIV-1 Activity
2005-01-01 Manetti, F; Est, Ja; CLOTET CODINA, I; ARMAND UGON, M; Maga, G; Crespan, E; Cancio, R; Mugnaini, C; Bernardini, C; Togninelli, A; Carmi, Caterina; Alongi, M; Petricci, E; Massa, S; Corelli, F; Botta, M.
Parallel Solution-Phase Synthesis of 1,5-disubstitued Hydantoins as New Protein Tyrosine Kinase Inhibitors
2005-01-01 Carmi, Caterina
Solution Phase Parallel Synthesis of S-DABO Analogues
2006-01-01 Togninelli, A; Carmi, Caterina; Petricci, E; Mugnaini, C; Massa, S; Corelli, F; Botta, M.
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity
2006-01-01 Carmi, Caterina; Cavazzoni, Andrea; Zuliani, Valentina; Lodola, Alessio; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
Antiproliferative and proapototic effects of a new combi-molecule on non small cell lung cancer cell lines
2007-01-01 Alfieri, Roberta; Cavazzoni, Andrea; Carmi, Caterina; M., Galetti; Zuliani, Valentina; Fumarola, Claudia; Mor, Marco; Petronini, Pier Giorgio
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano
2007-01-01 Cavazzoni, Andrea; Galetti, Maricla; LA MONICA, S; Fumarola, C; Bonelli, Mara; Carmi, C; Zuliani, Valentina; Lodola, Alessio; Bordi, F; Plazzi, P. V.; Mor, Marco; Petronini, Pg
Irreversible EGFR inhibitor compounds with antiproliferative activity
2008-01-01 Mor, Marco; Bordi, Fabrizio; Carmi, Caterina; S., Vezzosi; Lodola, Alessio; Petronini, Pier Giorgio; Alfieri, Roberta; Cavazzoni, Andrea
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands
2009-01-01 Rivara, Silvia; Vacondio, Federica; Fioni, A; Silva, Claudia; Carmi, Caterina; Mor, Marco; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, G; Bedini, A; Orlando, P; Lucarini, S; Tarzia, G.
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line
2009-01-01 Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
A critical cysteine residue in monoacylglycerol lipase is targeted by a new class of isothiazolinone-based enzyme inhibitors.
2009-01-01 King, A. R.; Lodola, Alessio; Carmi, Caterina; Fu, J.; Mor, Marco; Piomelli, D.
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion
2010-01-01 Carmi, C.; Cavazzoni, A.; Vezzosi, S.; Bordi, F.; Vacondio, F.; Silva, C.; Rivara, S.; Lodola, A.; Alfieri, R.; La Monica, S; Galetti, M.; Ardizzoni, A.; Petronini, P. G.; Mor, M.
New strategies to overcome resistance to EGFR tyrosine kinase inhibitors in non small cell lung cancer
2010-01-01 Alfieri, Roberta; Cavazzoni, Andrea; Galetti, Maricla; Andreoli, Roberta; Carmi, Caterina; Mor, Marco; Petronini, Pier Giorgio
Mannich base derivatives as novel EGFR irreversible inhibitors
2011-01-01 Russo, Simonetta; Mor, Marco; Carmi, Caterina; Vacondio, Federica; Petronini, Pier Giorgio; Cavazzoni, Andrea
Epidermal Growth Factor Receptor Irreversible Inhibitors: Chemical Exploration of the Cysteine-Trap Portion
2011-01-01 Carmi, Caterina; Lodola, Alessio; Rivara, Silvia; Vacondio, Federica; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, Andrea; Petronini, Pier Giorgio; Mor, Marco
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: steric effects of N-alkyl chain on rat plasma and liver stability
2011-01-01 Vacondio, Federica; Silva, Claudia; Lodola, Alessio; Carmi, Caterina; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; G., Tarzia; Mor, Marco
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives.
2011-01-01 A., Bedini; S., Lucarini; G., Spadoni; G., Tarzia; F., Scaglione; S., Dugnani; M., Pannacci; V., Lucini; Carmi, Caterina; Pala, Daniele; Rivara, Silvia; Mor, Marco
Clinical perspective for irreversible tyrosine kinase inhibitors in cancer
2012-01-01 Carmi, Caterina; Mor, Marco; Petronini, Pier Giorgio; Alfieri, Roberta
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain.
2012-01-01 Bordi, Fabrizio; Rivara, Silvia; E., Dallaturca; Carmi, Caterina; Pala, Daniele; Lodola, Alessio; Vacondio, Federica; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides.
2012-01-01 Carmi, Caterina; Galvani, Elena; Vacondio, Federica; Rivara, Silvia; Lodola, Alessio; Russo, Simonetta; Bordi, Fabrizio; Costantino, Gianluca; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, A.; Petronini, P. G.; Mor, Marco; Costantino, Gabriele
Molecular mechanisms underlying the antitumor activity of 3-aminopropanamide irreversible inhibitors of the epidermal growth factor receptor in non-small cell lung cancer
2013-01-01 Galvani, Elena; E., Giovannetti; Saccani, Francesca; Cavazzoni, Andrea; L. G., Leon; H., Dekker; Alfieri, Roberta; Carmi, Caterina; Mor, Marco; Ardizzoni, Andrea; Petronini, Pier Giorgio; G. J., Peters
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Parallel Solution-phase and Microwave-assisted Synthesis of New S-DABO Derivatives Endowed with Subnanomolar Anti-HIV-1 Activity | 1-gen-2005 | Manetti, F; Est, Ja; CLOTET CODINA, I; ARMAND UGON, M; Maga, G; Crespan, E; Cancio, R; Mugnaini, C; Bernardini, C; Togninelli, A; Carmi, Caterina; Alongi, M; Petricci, E; Massa, S; Corelli, F; Botta, M. | |
Parallel Solution-Phase Synthesis of 1,5-disubstitued Hydantoins as New Protein Tyrosine Kinase Inhibitors | 1-gen-2005 | Carmi, Caterina | |
Solution Phase Parallel Synthesis of S-DABO Analogues | 1-gen-2006 | Togninelli, A; Carmi, Caterina; Petricci, E; Mugnaini, C; Massa, S; Corelli, F; Botta, M. | |
5-Benzylidene-hydantoins as new EGFR inhibitors with antiproliferative activity | 1-gen-2006 | Carmi, Caterina; Cavazzoni, Andrea; Zuliani, Valentina; Lodola, Alessio; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco | |
Antiproliferative and proapototic effects of a new combi-molecule on non small cell lung cancer cell lines | 1-gen-2007 | Alfieri, Roberta; Cavazzoni, Andrea; Carmi, Caterina; M., Galetti; Zuliani, Valentina; Fumarola, Claudia; Mor, Marco; Petronini, Pier Giorgio | |
Meccanismo d’azione di UPR 1024: un nuovo farmaco con attività antiproliferativa in cellule di carcinoma polmonare umano | 1-gen-2007 | Cavazzoni, Andrea; Galetti, Maricla; LA MONICA, S; Fumarola, C; Bonelli, Mara; Carmi, C; Zuliani, Valentina; Lodola, Alessio; Bordi, F; Plazzi, P. V.; Mor, Marco; Petronini, Pg | |
Irreversible EGFR inhibitor compounds with antiproliferative activity | 1-gen-2008 | Mor, Marco; Bordi, Fabrizio; Carmi, Caterina; S., Vezzosi; Lodola, Alessio; Petronini, Pier Giorgio; Alfieri, Roberta; Cavazzoni, Andrea | |
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands | 1-gen-2009 | Rivara, Silvia; Vacondio, Federica; Fioni, A; Silva, Claudia; Carmi, Caterina; Mor, Marco; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, G; Bedini, A; Orlando, P; Lucarini, S; Tarzia, G. | |
5-Benzylidene-hydantoins: synthesis and antiproliferative activity on A549 lung cancer cell line | 1-gen-2009 | Zuliani, Valentina; Carmi, Caterina; Rivara, Mirko; Fantini, M; Lodola, Alessio; Vacondio, Federica; Bordi, Fabrizio; Plazzi, Pier Vincenzo; Cavazzoni, Andrea; Galetti, Maricla; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco | |
A critical cysteine residue in monoacylglycerol lipase is targeted by a new class of isothiazolinone-based enzyme inhibitors. | 1-gen-2009 | King, A. R.; Lodola, Alessio; Carmi, Caterina; Fu, J.; Mor, Marco; Piomelli, D. | |
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion | 1-gen-2010 | Carmi, C.; Cavazzoni, A.; Vezzosi, S.; Bordi, F.; Vacondio, F.; Silva, C.; Rivara, S.; Lodola, A.; Alfieri, R.; La Monica, S; Galetti, M.; Ardizzoni, A.; Petronini, P. G.; Mor, M. | |
New strategies to overcome resistance to EGFR tyrosine kinase inhibitors in non small cell lung cancer | 1-gen-2010 | Alfieri, Roberta; Cavazzoni, Andrea; Galetti, Maricla; Andreoli, Roberta; Carmi, Caterina; Mor, Marco; Petronini, Pier Giorgio | |
Mannich base derivatives as novel EGFR irreversible inhibitors | 1-gen-2011 | Russo, Simonetta; Mor, Marco; Carmi, Caterina; Vacondio, Federica; Petronini, Pier Giorgio; Cavazzoni, Andrea | |
Epidermal Growth Factor Receptor Irreversible Inhibitors: Chemical Exploration of the Cysteine-Trap Portion | 1-gen-2011 | Carmi, Caterina; Lodola, Alessio; Rivara, Silvia; Vacondio, Federica; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, Andrea; Petronini, Pier Giorgio; Mor, Marco | |
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: steric effects of N-alkyl chain on rat plasma and liver stability | 1-gen-2011 | Vacondio, Federica; Silva, Claudia; Lodola, Alessio; Carmi, Caterina; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; G., Tarzia; Mor, Marco | |
Toward the Definition of Stereochemical Requirements for MT(2)-Selective Antagonists and Partial Agonists by Studying 4-Phenyl-2-propionamidotetralin Derivatives. | 1-gen-2011 | A., Bedini; S., Lucarini; G., Spadoni; G., Tarzia; F., Scaglione; S., Dugnani; M., Pannacci; V., Lucini; Carmi, Caterina; Pala, Daniele; Rivara, Silvia; Mor, Marco | |
Clinical perspective for irreversible tyrosine kinase inhibitors in cancer | 1-gen-2012 | Carmi, Caterina; Mor, Marco; Petronini, Pier Giorgio; Alfieri, Roberta | |
Dibasic biphenyl H(3) receptor antagonists: Steric tolerance for a lipophilic side chain. | 1-gen-2012 | Bordi, Fabrizio; Rivara, Silvia; E., Dallaturca; Carmi, Caterina; Pala, Daniele; Lodola, Alessio; Vacondio, Federica; Flammini, Lisa; Bertoni, Simona; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
Irreversible Inhibition of Epidermal Growth Factor Receptor Activity by 3-Aminopropanamides. | 1-gen-2012 | Carmi, Caterina; Galvani, Elena; Vacondio, Federica; Rivara, Silvia; Lodola, Alessio; Russo, Simonetta; Bordi, Fabrizio; Costantino, Gianluca; Cavazzoni, Andrea; Alfieri, Roberta; Ardizzoni, A.; Petronini, P. G.; Mor, Marco; Costantino, Gabriele | |
Molecular mechanisms underlying the antitumor activity of 3-aminopropanamide irreversible inhibitors of the epidermal growth factor receptor in non-small cell lung cancer | 1-gen-2013 | Galvani, Elena; E., Giovannetti; Saccani, Francesca; Cavazzoni, Andrea; L. G., Leon; H., Dekker; Alfieri, Roberta; Carmi, Caterina; Mor, Marco; Ardizzoni, Andrea; Petronini, Pier Giorgio; G. J., Peters |
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