Sfoglia per Autore Silva, Claudia
Recent advances in the discovery of ALKBH 1–8 inhibitors.
2025-01-01 Silva, Claudia; Zuliani, Valentina; Nicolini, Gabriella; Malacrida, Alessio; Rivara, Mirko
A Specific HPLC Method to Determine Residual HEPES in [68Ga]Ga-Radiopharmaceuticals: Development and Validation
2022-01-01 Migliari, Silvia; Scarlattei, Maura; Baldari, Giorgio; Silva, Claudia; Ruffini, Livia
Development and validation of an analytical hplc method to assess chemical and radiochemical purity of [68ga]ga-nodaga-exendin-4 produced by a fully automated method
2022-01-01 Migliari, S.; Sammartano, A.; Boss, M.; Gotthardt, M.; Scarlattei, M.; Baldari, G.; Silva, C.; Bonadonna, R. C.; Ruffini, L.
A Rapid and Specific HPLC Method to Determine Chemical and Radiochemical Purity of [68Ga] Ga-DOTA-Pentixafor (PET) Tracer: Development and Validation
2021-01-01 Migliari, Silvia; Sammartano, Antonino; Scarlattei, Maura; Baldari, Giorgio; Silva, Claudia; Ruffini, Livia
Balancing reactivity and antitumor activity: heteroarylthioacetamide derivatives as potent and time-dependent inhibitors of EGFR
2019-01-01 Castelli, R; Bozza, N; Cavazzoni, A; Bonelli, M; Vacondio, F; Ferlenghi, F; Callegari, D; Silva, C; Rivara, S; Lodola, A; Digiacomo, G; Fumarola, C; Alfieri, R; Petronini, Pg; Mor, M.
Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 7. Synthesis and Pharmacological Evaluation of 4-Quinolone-3-carboxamides and 4-Hydroxy-2-quinolone-3-carboxamides as High Affinity Cannabinoid Receptor 2 (CB2R) Ligands with Improved Aqueous Solubility
2016-01-01 Mugnaini, Claudia; Brizzi, Antonella; Ligresti, Alessia; Allarà, Marco; Lamponi, Stefania; Vacondio, Federica; Silva, Claudia; Mor, Marco; Di Marzo, Vincenzo; Corelli, Federico
Amino acid derivatives as palmitoylethanolamide prodrugs: Synthesis, in vitro metabolism and in vivo plasma profile in rats
2015-01-01 Vacondio, Federica; Bassi, Michele; Silva, Claudia; Castelli, Riccardo; Carmi, Caterina; Scalvini, Laura; Lodola, Alessio; Vivo, Valentina; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco; Rivara, Silvia
Predicting the reactivity of nitrile-carrying compounds with cysteine: a combined computational and experimental study.
2014-01-01 Berteotti, A; Vacondio, Federica; Lodola, Alessio; Bassi, M; Silva, Claudia; Mor, Marco; Cavalli, A.
Analysis of illicit dietary supplements sold in the Italian market: Identification of a sildenafil thioderivative as adulterant using UPLC-TOF/MS and GC/MS.
2014-01-01 Damiano, Fabio; Silva, Claudia; Gregori, Alberto; Vacondio, Federica; Mor, Marco; Menozzi, Marco; Di Giorgio, Domenico
Long-lasting inhibition of EGFR autophosphorylation in A549 tumor cells by intracellular accumulation of non-covalent inhibitors
2013-01-01 Vacondio, Federica; Carmi, Caterina; Elena, Galvani; Bassi, Michele; Silva, Claudia; Lodola, Alessio; Rivara, Silvia; Cavazzoni, Andrea; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco
N-(2-Oxo-3-oxetanyl)carbamic Acid Esters as N-Acylethanolamine Acid Amidase Inhibitors: Synthesis, Structure–Activity and Structure–Property Relationships.
2012-01-01 A., Duranti; A., Tontini; F., Antonietti; Vacondio, Federica; A., Fioni; Silva, Claudia; Lodola, Alessio; Rivara, Silvia; C., Solorzano; D., Piomelli; G., Tarzia; Mor, Marco
Brain Pharmacokinetics of Non-Imidazole Biphenyl H3 Receptor Antagonists: a Liquid Chromatography/Electrospray-Mass Spectrometry and ex vivo Binding Study in Rats
2012-01-01 Vacondio, Federica; Silva, Claudia; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco
Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma.
2011-01-01 Vacondio, Federica; Silva, Claudia; Morini, Giovanni; Bordi, Fabrizio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco
Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: steric effects of N-alkyl chain on rat plasma and liver stability
2011-01-01 Vacondio, Federica; Silva, Claudia; Lodola, Alessio; Carmi, Caterina; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; G., Tarzia; Mor, Marco
Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion
2010-01-01 Carmi, C.; Cavazzoni, A.; Vezzosi, S.; Bordi, F.; Vacondio, F.; Silva, C.; Rivara, S.; Lodola, A.; Alfieri, R.; La Monica, S; Galetti, M.; Ardizzoni, A.; Petronini, P. G.; Mor, M.
Qualitative structure-metabolism relationships in the hydrolysis of carbamates
2010-01-01 Vacondio, Federica; Silva, Claudia; Mor, Marco; B., Testa
N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands
2009-01-01 Rivara, Silvia; Vacondio, Federica; Fioni, A; Silva, Claudia; Carmi, Caterina; Mor, Marco; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, G; Bedini, A; Orlando, P; Lucarini, S; Tarzia, G.
2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships
2009-01-01 Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K.
Structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors: chemical and biological stability
2009-01-01 Vacondio, Federica; Silva, Claudia; Lodola, Alessio; A., Fioni; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; Mor, Marco; G., Tarzia
A second generation of carbamate-based fatty acid amide hydrolase inhibitors with improved activity in vivo
2009-01-01 Clapper, Jason R.; Vacondio, Federica; King, Alvin R.; Duranti, Andrea; Tontini, Andrea; Silva, Claudia; Sanchini, Silvano; Tarzia, Giorgio; Mor, Marco; Piomelli, Daniele
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Recent advances in the discovery of ALKBH 1–8 inhibitors. | 1-gen-2025 | Silva, Claudia; Zuliani, Valentina; Nicolini, Gabriella; Malacrida, Alessio; Rivara, Mirko | |
| A Specific HPLC Method to Determine Residual HEPES in [68Ga]Ga-Radiopharmaceuticals: Development and Validation | 1-gen-2022 | Migliari, Silvia; Scarlattei, Maura; Baldari, Giorgio; Silva, Claudia; Ruffini, Livia | |
| Development and validation of an analytical hplc method to assess chemical and radiochemical purity of [68ga]ga-nodaga-exendin-4 produced by a fully automated method | 1-gen-2022 | Migliari, S.; Sammartano, A.; Boss, M.; Gotthardt, M.; Scarlattei, M.; Baldari, G.; Silva, C.; Bonadonna, R. C.; Ruffini, L. | |
| A Rapid and Specific HPLC Method to Determine Chemical and Radiochemical Purity of [68Ga] Ga-DOTA-Pentixafor (PET) Tracer: Development and Validation | 1-gen-2021 | Migliari, Silvia; Sammartano, Antonino; Scarlattei, Maura; Baldari, Giorgio; Silva, Claudia; Ruffini, Livia | |
| Balancing reactivity and antitumor activity: heteroarylthioacetamide derivatives as potent and time-dependent inhibitors of EGFR | 1-gen-2019 | Castelli, R; Bozza, N; Cavazzoni, A; Bonelli, M; Vacondio, F; Ferlenghi, F; Callegari, D; Silva, C; Rivara, S; Lodola, A; Digiacomo, G; Fumarola, C; Alfieri, R; Petronini, Pg; Mor, M. | |
| Investigations on the 4-Quinolone-3-carboxylic Acid Motif. 7. Synthesis and Pharmacological Evaluation of 4-Quinolone-3-carboxamides and 4-Hydroxy-2-quinolone-3-carboxamides as High Affinity Cannabinoid Receptor 2 (CB2R) Ligands with Improved Aqueous Solubility | 1-gen-2016 | Mugnaini, Claudia; Brizzi, Antonella; Ligresti, Alessia; Allarà, Marco; Lamponi, Stefania; Vacondio, Federica; Silva, Claudia; Mor, Marco; Di Marzo, Vincenzo; Corelli, Federico | |
| Amino acid derivatives as palmitoylethanolamide prodrugs: Synthesis, in vitro metabolism and in vivo plasma profile in rats | 1-gen-2015 | Vacondio, Federica; Bassi, Michele; Silva, Claudia; Castelli, Riccardo; Carmi, Caterina; Scalvini, Laura; Lodola, Alessio; Vivo, Valentina; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco; Rivara, Silvia | |
| Predicting the reactivity of nitrile-carrying compounds with cysteine: a combined computational and experimental study. | 1-gen-2014 | Berteotti, A; Vacondio, Federica; Lodola, Alessio; Bassi, M; Silva, Claudia; Mor, Marco; Cavalli, A. | |
| Analysis of illicit dietary supplements sold in the Italian market: Identification of a sildenafil thioderivative as adulterant using UPLC-TOF/MS and GC/MS. | 1-gen-2014 | Damiano, Fabio; Silva, Claudia; Gregori, Alberto; Vacondio, Federica; Mor, Marco; Menozzi, Marco; Di Giorgio, Domenico | |
| Long-lasting inhibition of EGFR autophosphorylation in A549 tumor cells by intracellular accumulation of non-covalent inhibitors | 1-gen-2013 | Vacondio, Federica; Carmi, Caterina; Elena, Galvani; Bassi, Michele; Silva, Claudia; Lodola, Alessio; Rivara, Silvia; Cavazzoni, Andrea; Alfieri, Roberta; Petronini, Pier Giorgio; Mor, Marco | |
| N-(2-Oxo-3-oxetanyl)carbamic Acid Esters as N-Acylethanolamine Acid Amidase Inhibitors: Synthesis, Structure–Activity and Structure–Property Relationships. | 1-gen-2012 | A., Duranti; A., Tontini; F., Antonietti; Vacondio, Federica; A., Fioni; Silva, Claudia; Lodola, Alessio; Rivara, Silvia; C., Solorzano; D., Piomelli; G., Tarzia; Mor, Marco | |
| Brain Pharmacokinetics of Non-Imidazole Biphenyl H3 Receptor Antagonists: a Liquid Chromatography/Electrospray-Mass Spectrometry and ex vivo Binding Study in Rats | 1-gen-2012 | Vacondio, Federica; Silva, Claudia; Flammini, Lisa; Ballabeni, Vigilio; Barocelli, Elisabetta; Mor, Marco | |
| Liquid chromatography-mass spectrometric method for determination of the non-imidazole H(3) -receptor antagonist UPR1056 in rat plasma. | 1-gen-2011 | Vacondio, Federica; Silva, Claudia; Morini, Giovanni; Bordi, Fabrizio; Flammini, Lisa; Barocelli, Elisabetta; Mor, Marco | |
| Biphenyl-3-yl alkylcarbamates as fatty acid amide hydrolase (FAAH) inhibitors: steric effects of N-alkyl chain on rat plasma and liver stability | 1-gen-2011 | Vacondio, Federica; Silva, Claudia; Lodola, Alessio; Carmi, Caterina; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; G., Tarzia; Mor, Marco | |
| Novel Irreversible Epidermal Growth Factor Receptor Inhibitors by Chemical Modulation of the Cysteine-Trap Portion | 1-gen-2010 | Carmi, C.; Cavazzoni, A.; Vezzosi, S.; Bordi, F.; Vacondio, F.; Silva, C.; Rivara, S.; Lodola, A.; Alfieri, R.; La Monica, S; Galetti, M.; Ardizzoni, A.; Petronini, P. G.; Mor, M. | |
| Qualitative structure-metabolism relationships in the hydrolysis of carbamates | 1-gen-2010 | Vacondio, Federica; Silva, Claudia; Mor, Marco; B., Testa | |
| N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands | 1-gen-2009 | Rivara, Silvia; Vacondio, Federica; Fioni, A; Silva, Claudia; Carmi, Caterina; Mor, Marco; Lucini, V; Pannacci, M; Caronno, A; Scaglione, F; Gobbi, G; Spadoni, G; Bedini, A; Orlando, P; Lucarini, S; Tarzia, G. | |
| 2,4(5)-Diarylimidazoles as Inhibitors of hNaV1.2 Sodium Channels: Pharmacological Evaluationand Structure-Property Relationships | 1-gen-2009 | Fantini, M.; Rivara, Mirko; Zuliani, Valentina; Kalmar, C. L.; Vacondio, Federica; Silva, Claudia; Baheti, A. R.; Singh, N.; Merrick, E. C.; Katari, R. S.; Cocconcelli, G.; Ghiron, C.; Patel, M. K. | |
| Structure-property relationships of a class of carbamate-based fatty acid amide hydrolase (FAAH) inhibitors: chemical and biological stability | 1-gen-2009 | Vacondio, Federica; Silva, Claudia; Lodola, Alessio; A., Fioni; Rivara, Silvia; A., Duranti; A., Tontini; S., Sanchini; J. R., Clapper; D., Piomelli; Mor, Marco; G., Tarzia | |
| A second generation of carbamate-based fatty acid amide hydrolase inhibitors with improved activity in vivo | 1-gen-2009 | Clapper, Jason R.; Vacondio, Federica; King, Alvin R.; Duranti, Andrea; Tontini, Andrea; Silva, Claudia; Sanchini, Silvano; Tarzia, Giorgio; Mor, Marco; Piomelli, Daniele |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile