Sfoglia per Autore Rivara, Silvia
N-Acylaminoethyltetrahydroquinolines: A new class of melatonin receptor ligands with in vivo activity on glioblastoma
2026-01-01 Bedini, Annalida; Galvani, Francesca; Elisi, Gian Marco; Scalvini, Laura; Mari, Michele; Recchia, Adriano; Fernandes, Pedro Augusto C. M.; Kinker, Gabriela S.; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Markus, Regina P.; Rivara, Silvia; Spadoni, Gilberto; Mor, Marco
JAK3 Inhibitors: Covalent and Noncovalent Interactions of a Cyanamide Group Investigated by Multiscale Free-Energy Simulations
2025-01-01 Scalvini, L.; Pala, D.; Cuzzolin, A.; Galvani, F.; Lodola, A.; Rivara, S.; Mor, M.; Rizzi, A.
Small molecules targeting the eubacterial β-sliding clamp discovered by combined in silico and in vitro screening approaches
2025-01-01 Caputo, Alessia; Elisi, Gian Marco; Levati, Elisabetta; Barotti, Giulia; Sartini, Sara; Wagner, Jerome; Burnouf, Dominique Y; Ottonello, Simone; Rivara, Silvia; Montanini, Barbara
Investigating drug-gut microbiota interactions: reductive and hydrolytic metabolism of oral glucocorticoids by in vitro artificial gut microbiota
2024-01-01 Viglioli, Martina; Rizzo, Sonia Mirjam; Alessandri, Giulia; Fontana, Federico; Milani, Christian; Turroni, Francesca; Mancabelli, Leonardo; Croci, Nicole; Rivara, Silvia; Vacondio, Federica; Ventura, Marco; Mor, Marco
Protective Activity of Melatonin Combinations and Melatonin-Based Hybrid Molecules in Neurodegenerative Diseases
2024-01-01 Galvani, F.; Cammarota, M.; Vacondio, F.; Rivara, S.; Boscia, F.
Discovery of a new 1-(phenylsulfonyl)-1H-indole derivative targeting the EphA2 receptor with antiproliferative activity on U251 glioblastoma cell line
2024-01-01 Guidetti, Lorenzo; Castelli, Riccardo; Zappia, Alfonso; Ferrari, Francesca Romana; Giorgio, Carmine; Barocelli, Elisabetta; Pagliaro, Luca; Vento, Federica; Roti, Giovanni; Scalvini, Laura; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano
Melatonin receptor structure and signaling
2024-01-01 Okamoto, H. H.; Cecon, E.; Nureki, O.; Rivara, S.; Jockers, R.
Social stress-induced depressive-like symptoms and changes in gut microbial and lipidomic profiles are prevented by pharmacological inhibition of FAAH activity in male rats
2024-01-01 Barbetti, Margherita; Mancabelli, Leonardo; Vacondio, Federica; Longhi, Giulia; Ferlenghi, Francesca; Viglioli, Martina; Turroni, Francesca; Carnevali, Luca; Mor, Marco; Ventura, Marco; Sgoifo, Andrea; Rivara, Silvia
Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence
2024-01-01 Bedini, A.; Elisi, G. M.; Fanini, F.; Retini, M.; Scalvini, L.; Pasquini, S.; Contri, C.; Varani, K.; Spadoni, G.; Mor, M.; Vincenzi, F.; Rivara, S.
Discovery of novel FGF trap small molecules endowed with anti-myeloma activity
2024-01-01 Taranto, Sara; Castelli, Riccardo; Marseglia, Giuseppe; Scalvini, Laura; Vacondio, Federica; Gianoncelli, Alessandra; Ribaudo, Giovanni; Faletti, Jessica; Gazzaroli, Giorgia; Rocca, Edoardo; Ronca, Roberto; Rusnati, Marco; Sacco, Antonio; Roccaro, Aldo Maria; Presta, Marco; Mor, Marco; Giacomini, Arianna; Rivara, Silvia
Molecular Determinants of EphA2 and EphB2 Antagonism Enable the Design of Ligands with Improved Selectivity
2023-01-01 Guidetti, Lorenzo; Zappia, Alfonso; Scalvini, Laura; Ferrari, Francesca Romana; Giorgio, Carmine; Castelli, Riccardo; Galvani, Francesca; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Urbinati, Chiara; Rusnati, Marco; Tognolini, Massimiliano; Lodola, Alessio
Combined targeting of fatty acid amide hydrolase and melatonin receptors promotes neuroprotection and stimulates inflammation resolution in rats
2023-01-01 Cammarota, Mariarosaria; Ferlenghi, Francesca; Vacondio, Federica; Vincenzi, Fabrizio; Varani, Katia; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Boscia, Francesca
2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors
2022-01-01 Mari, M.; Elisi, G. M.; Bedini, A.; Lucarini, S.; Retini, M.; Lucini, V.; Scaglione, F.; Vincenzi, F.; Varani, K.; Castelli, R.; Mor, M.; Rivara, S.; Spadoni, G.
An Optimized Workflow for the Discovery of New Antimicrobial Compounds Targeting Bacterial RNA Polymerase Complex Formation
2022-01-01 Caputo, Alessia; Sartini, Sara; Levati, Elisabetta; Minato, Ilaria; Elisi, Gian Marco; Di Stasi, Adriana; Guillou, Catherine; Goekjian, Peter G; Garcia, Pierre; Gueyrard, David; Bach, Stéphane; Comte, Arnaud; Ottonello, Simone; Rivara, Silvia; Montanini, Barbara
In silico drug discovery of melatonin receptor ligands with therapeutic potential
2022-01-01 Elisi, G. M.; Scalvini, L.; Lodola, A.; Bedini, A.; Spadoni, G.; Rivara, S.
Mechanistic Modeling of Monoglyceride Lipase Covalent Modification Elucidates the Role of Leaving Group Expulsion and Discriminates Inhibitors with High and Low Potency
2022-01-01 Galvani, F.; Scalvini, L.; Rivara, S.; Lodola, A.; Mor, M.
Free-Energy Simulations Support a Lipophilic Binding Route for Melatonin Receptors
2022-01-01 Elisi, GIAN MARCO; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Rivara, Silvia
Chapter 9: Natural and Synthetic Agents That Target Intracellular Monoacylglycerol Lipase (MGL) Activity
2021-01-01 Scalvini, L.; Rivara, S.; Jung, K. -M.; Mor, M.; Piomelli, D.
A sulfonyl fluoride derivative inhibits EGFR L858R/T790M/C797S by covalent modification of the catalytic lysine
2021-01-01 Ferlenghi, F; Scalvini, L; Vacondio, F; Castelli, R; Bozza, N; Marseglia, G; Rivara, S; Lodola, A; La Monica, S; Minari, R; Petronini, Pg; Alfieri, R; Tiseo, M; Mor, M.
New Coumarin derivatives as cholinergic and cannabinoid system modulators
2021-01-01 Montanari, S.; Allara, M.; Scalvini, L.; Kostrzewa, M.; Belluti, F.; Gobbi, S.; Naldi, M.; Rivara, S.; Bartolini, M.; Ligresti, A.; Bisi, A.; Rampa, A.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| N-Acylaminoethyltetrahydroquinolines: A new class of melatonin receptor ligands with in vivo activity on glioblastoma | 1-gen-2026 | Bedini, Annalida; Galvani, Francesca; Elisi, Gian Marco; Scalvini, Laura; Mari, Michele; Recchia, Adriano; Fernandes, Pedro Augusto C. M.; Kinker, Gabriela S.; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Markus, Regina P.; Rivara, Silvia; Spadoni, Gilberto; Mor, Marco | |
| JAK3 Inhibitors: Covalent and Noncovalent Interactions of a Cyanamide Group Investigated by Multiscale Free-Energy Simulations | 1-gen-2025 | Scalvini, L.; Pala, D.; Cuzzolin, A.; Galvani, F.; Lodola, A.; Rivara, S.; Mor, M.; Rizzi, A. | |
| Small molecules targeting the eubacterial β-sliding clamp discovered by combined in silico and in vitro screening approaches | 1-gen-2025 | Caputo, Alessia; Elisi, Gian Marco; Levati, Elisabetta; Barotti, Giulia; Sartini, Sara; Wagner, Jerome; Burnouf, Dominique Y; Ottonello, Simone; Rivara, Silvia; Montanini, Barbara | |
| Investigating drug-gut microbiota interactions: reductive and hydrolytic metabolism of oral glucocorticoids by in vitro artificial gut microbiota | 1-gen-2024 | Viglioli, Martina; Rizzo, Sonia Mirjam; Alessandri, Giulia; Fontana, Federico; Milani, Christian; Turroni, Francesca; Mancabelli, Leonardo; Croci, Nicole; Rivara, Silvia; Vacondio, Federica; Ventura, Marco; Mor, Marco | |
| Protective Activity of Melatonin Combinations and Melatonin-Based Hybrid Molecules in Neurodegenerative Diseases | 1-gen-2024 | Galvani, F.; Cammarota, M.; Vacondio, F.; Rivara, S.; Boscia, F. | |
| Discovery of a new 1-(phenylsulfonyl)-1H-indole derivative targeting the EphA2 receptor with antiproliferative activity on U251 glioblastoma cell line | 1-gen-2024 | Guidetti, Lorenzo; Castelli, Riccardo; Zappia, Alfonso; Ferrari, Francesca Romana; Giorgio, Carmine; Barocelli, Elisabetta; Pagliaro, Luca; Vento, Federica; Roti, Giovanni; Scalvini, Laura; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano | |
| Melatonin receptor structure and signaling | 1-gen-2024 | Okamoto, H. H.; Cecon, E.; Nureki, O.; Rivara, S.; Jockers, R. | |
| Social stress-induced depressive-like symptoms and changes in gut microbial and lipidomic profiles are prevented by pharmacological inhibition of FAAH activity in male rats | 1-gen-2024 | Barbetti, Margherita; Mancabelli, Leonardo; Vacondio, Federica; Longhi, Giulia; Ferlenghi, Francesca; Viglioli, Martina; Turroni, Francesca; Carnevali, Luca; Mor, Marco; Ventura, Marco; Sgoifo, Andrea; Rivara, Silvia | |
| Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence | 1-gen-2024 | Bedini, A.; Elisi, G. M.; Fanini, F.; Retini, M.; Scalvini, L.; Pasquini, S.; Contri, C.; Varani, K.; Spadoni, G.; Mor, M.; Vincenzi, F.; Rivara, S. | |
| Discovery of novel FGF trap small molecules endowed with anti-myeloma activity | 1-gen-2024 | Taranto, Sara; Castelli, Riccardo; Marseglia, Giuseppe; Scalvini, Laura; Vacondio, Federica; Gianoncelli, Alessandra; Ribaudo, Giovanni; Faletti, Jessica; Gazzaroli, Giorgia; Rocca, Edoardo; Ronca, Roberto; Rusnati, Marco; Sacco, Antonio; Roccaro, Aldo Maria; Presta, Marco; Mor, Marco; Giacomini, Arianna; Rivara, Silvia | |
| Molecular Determinants of EphA2 and EphB2 Antagonism Enable the Design of Ligands with Improved Selectivity | 1-gen-2023 | Guidetti, Lorenzo; Zappia, Alfonso; Scalvini, Laura; Ferrari, Francesca Romana; Giorgio, Carmine; Castelli, Riccardo; Galvani, Francesca; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Urbinati, Chiara; Rusnati, Marco; Tognolini, Massimiliano; Lodola, Alessio | |
| Combined targeting of fatty acid amide hydrolase and melatonin receptors promotes neuroprotection and stimulates inflammation resolution in rats | 1-gen-2023 | Cammarota, Mariarosaria; Ferlenghi, Francesca; Vacondio, Federica; Vincenzi, Fabrizio; Varani, Katia; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Boscia, Francesca | |
| 2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors | 1-gen-2022 | Mari, M.; Elisi, G. M.; Bedini, A.; Lucarini, S.; Retini, M.; Lucini, V.; Scaglione, F.; Vincenzi, F.; Varani, K.; Castelli, R.; Mor, M.; Rivara, S.; Spadoni, G. | |
| An Optimized Workflow for the Discovery of New Antimicrobial Compounds Targeting Bacterial RNA Polymerase Complex Formation | 1-gen-2022 | Caputo, Alessia; Sartini, Sara; Levati, Elisabetta; Minato, Ilaria; Elisi, Gian Marco; Di Stasi, Adriana; Guillou, Catherine; Goekjian, Peter G; Garcia, Pierre; Gueyrard, David; Bach, Stéphane; Comte, Arnaud; Ottonello, Simone; Rivara, Silvia; Montanini, Barbara | |
| In silico drug discovery of melatonin receptor ligands with therapeutic potential | 1-gen-2022 | Elisi, G. M.; Scalvini, L.; Lodola, A.; Bedini, A.; Spadoni, G.; Rivara, S. | |
| Mechanistic Modeling of Monoglyceride Lipase Covalent Modification Elucidates the Role of Leaving Group Expulsion and Discriminates Inhibitors with High and Low Potency | 1-gen-2022 | Galvani, F.; Scalvini, L.; Rivara, S.; Lodola, A.; Mor, M. | |
| Free-Energy Simulations Support a Lipophilic Binding Route for Melatonin Receptors | 1-gen-2022 | Elisi, GIAN MARCO; Scalvini, Laura; Lodola, Alessio; Mor, Marco; Rivara, Silvia | |
| Chapter 9: Natural and Synthetic Agents That Target Intracellular Monoacylglycerol Lipase (MGL) Activity | 1-gen-2021 | Scalvini, L.; Rivara, S.; Jung, K. -M.; Mor, M.; Piomelli, D. | |
| A sulfonyl fluoride derivative inhibits EGFR L858R/T790M/C797S by covalent modification of the catalytic lysine | 1-gen-2021 | Ferlenghi, F; Scalvini, L; Vacondio, F; Castelli, R; Bozza, N; Marseglia, G; Rivara, S; Lodola, A; La Monica, S; Minari, R; Petronini, Pg; Alfieri, R; Tiseo, M; Mor, M. | |
| New Coumarin derivatives as cholinergic and cannabinoid system modulators | 1-gen-2021 | Montanari, S.; Allara, M.; Scalvini, L.; Kostrzewa, M.; Belluti, F.; Gobbi, S.; Naldi, M.; Rivara, S.; Bartolini, M.; Ligresti, A.; Bisi, A.; Rampa, A. |
Legenda icone
- file ad accesso aperto
- file disponibili sulla rete interna
- file disponibili agli utenti autorizzati
- file disponibili solo agli amministratori
- file sotto embargo
- nessun file disponibile