Sfoglia per Autore Radi, Marco
Optimization of 4‐Amino‐2‐Pyridone Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9: Integrating Structure–Activity and Structure–Metabolism Relationships
2026-01-01 Giannessi, Lisa; Lupo, Maria Giovanna; Ugolotti, Martina; Papotti, Bianca; Mattina, Beatrice; Martina, Maria Grazia; Demurtas, Anna; Padula, Cristina; Nicoli, Sara; Crescenzio, Marco; Ferri, Nicola; Zimetti, Francesca; Radi, Marco
DISCOVERY OF NEW TSG101 INHIBITORS BLOCKING THE BUDDING OF EBOLA AND OTHER HIGHLY PATHOGENIC VIRUSES
2026-01-01 Valenti, Martina Eleonora; Rubini, Daniele; Parra-López, Marisa; Holzerland, Julia; Rodríguez-Martínez, Alejandro; Martina, Maria Grazia; Ramos, Maria C.; Castillo, Francisco; Harty, Ronald N.; Pérez-Sanchez, Horacio; Diederich, Sandra; Luque, Irene; Radi, Marco
Investigating PCSK9 as a therapeutic target in Alzheimer's disease: evidence from patient-derived astrocytes
2025-01-01 Ugolotti, M.; Papotti, B.; Adorni, M. P.; Martina, M. G.; Giannessi, L.; Olejnik, A.; Bell, S. M.; Mortiboys, H.; Radi, M.; Zimetti, F.
Targeting the ESCRT machinery: a promising strategy for the development of novel Broad-Spectrum Antivirals (BSAs).
2025-01-01 Rubini, Daniele; Martina, Maria Grazia; Valenti, Martina Eleonora; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Harty, Ronald N.; Parra-López, Marisa; Holzerland, Julia; Diederich, Sandra; Luque, Irene; Radi, Marco
WO2026017799A1 - SUBSTITUTED 3-CYANOQUINOLINES FOR THE PREVENTION AND TREATMENT OF SEXUALLY TRANSMITTED DISEASES
2025-01-01 Cagno, Valeria; Radi, Marco; Rubini, Daniele; Martina, Maria Grazia
Targeting PI4KB and Src/Abl host kinases as broad-spectrum antiviral strategy: Myth or real opportunity?
2025-01-01 Martina, Maria Grazia; Rubini, Daniele; Radi, Marco; Cagno, Valeria
Discovery of p-Trifluoromethylbenzohydrazide Derivatives as Potent Antiviral Agents against Monkeypox Virus
2025-01-01 Rossi, Sara; Pozzetti, Luca; Carullo, Gabriele; Dichiara, Maria; Butini, Stefania; Radi, Marco; Ramunno, Anna; Terrosi, Chiara; Barra, Giovanni; Berisio, Rita; Gemma, Sandra; Cusi, Maria Grazia; Campiani, Giuseppe
Exploring the druggability of the UEV domain of human TSG101 in search for broad-spectrum antivirals
2025-01-01 Montero, Fernando; Parra-López, Marisa; Rodríguez-Martínez, Alejandro; Murciano-Calles, Javier; Buzon, Pedro; Han, Ziying; Lin, L-Y; Ramos, Maria C; Ruiz-Sanz, Javier; Martinez, Jose C; Radi, Marco; Moog, Christiane; Diederich, Sandra; Harty, Ronald N; Pérez-Sánchez, Horacio; Vicente, Francisca; Castillo, Francisco; Luque, Irene
Effects of CCL20/CCR6 modulators in a T cell adoptive transfer model of colitis
2025-01-01 Allodi, M.; Flammini, L.; Giorgio, C.; Martina, M. G.; Barbieri, F.; Ballabeni, V.; Barocelli, E.; Radi, M.; Bertoni, S.
Harnessing prebiotic formamide chemistry: a novel platform for antiviral exploration
2025-01-01 Martina, Maria Grazia; Vagaggini, Chiara; Dreassi, Elena; De Angelis, Marta; Nencioni, Lucia; Dragoni, Filippo; Giammarino, Federica; Boccuto, Adele; Zazzi, Maurizio; Vicenti, Ilaria; Radi, Marco
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses
2025-01-01 Barbieri, Francesca; Martina, Maria Grazia; Pesce, Emanuela; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Rossi, Sara; Gemma, Sandra; Campiani, Giuseppe; Milite, Ciro; Pepe, Giacomo; Campiglia, Pietro; Sbardella, Gianluca; Maga, Giovanni; Cagno, Valeria; Pedemonte, Nicoletta; Radi, Marco
CHEMISTRY-DRIVEN OPTIMIZATION OF PURINE-BASED ANTIVIRALS FOR THE IDENTIFICATION OF NEW BROAD-SPECTRUM AGENTS
2025-01-01 Valenti, Martina Eleonora; Martina, Maria Grazia; Vincetti, Paolo; Vicenti, Ilaria; Crespan, Emmanuele; Nencioni, Lucia; Kaptein, Suzanne J. F.; Neyts, Johan; Vanderlinden, Evelien; Schols, Dominique; De Forni, Davide; Lori, Franco; Zazzi, Maurizio; Maga, Giovanni; Radi, Marco
DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X
2025-01-01 Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco
DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X
2025-01-01 Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco
“Investigating PCSK9 inhibition as potential strategy in Alzheimer’s disease”
2025-01-01 Ugolotti, M.; Papotti, B.; Adorni, M. P.; Giannessi, L.; Lupo, M. G.; Ferri, N.; Radi, M.; Bernini, F.; Zimetti, F.
Development of Novel PCSK9 Inhibitors as Potential Broad-Spectrum Antivirals
2025-01-01 Savian, Chiara; Giannessi, Lisa; Martina, Maria Grazia; Ugolotti, Martina; Papotti, Bianca; Palumbo, Marcella; Giovanna Lupo, Maria; Mattina, Beatrice; Padula, Cristina; Nicoli, Sara; Ferri, Nicola; De Forni, Davide; Lori, Franco; Cagno, Valeria; Zimetti, Francesca; Radi, Marco
A sustainable one-pot three step approach for the synthesis of 3,5-disubstituted 1,2,4-triazines as versatile pharmacological tools.
2024-01-01 Rubini, D.; Martina, M. G.; Incerti, M.; Barbieri, F.; Radi, M.
Discovery of small molecule inhibitors of the Tsg101-PTAP interaction as potential host-targeted broad-spectrum antivirals.
2024-01-01 Rubini, Daniele; Martina, Maria Grazia; Valenti, Martina Eleonora; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Harty, Ronald N.; Parra-López, Marisa; Luque, Irene; Radi, Marco
Targeting the ESCRT machinery: a promising strategy for the development of novel Broad-Spectrum Antivirals (BSAs).
2024-01-01 Rubini, Daniele; Martina, Maria Grazia; Valenti, Martina Eleonora; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Harty, Ronald N.; Parra-López, Marisa; Diederich, Sandra; Luque, Irene; Radi, Marco
Identification of 4-amino-2-Pyridones as new potent PCSK9 inhibitors: From phenotypic hit discovery to in vivo tolerability
2024-01-01 Giannessi, L; Lupo, Mg; Rossi, I; Martina, Mg; Vilella, A; Bodria, M; Giuliani, D; Zimetti, F; Zanotti, I; Potì, F; Bernini, F; Ferri, N; Radi, M
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Optimization of 4‐Amino‐2‐Pyridone Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9: Integrating Structure–Activity and Structure–Metabolism Relationships | 1-gen-2026 | Giannessi, Lisa; Lupo, Maria Giovanna; Ugolotti, Martina; Papotti, Bianca; Mattina, Beatrice; Martina, Maria Grazia; Demurtas, Anna; Padula, Cristina; Nicoli, Sara; Crescenzio, Marco; Ferri, Nicola; Zimetti, Francesca; Radi, Marco | |
| DISCOVERY OF NEW TSG101 INHIBITORS BLOCKING THE BUDDING OF EBOLA AND OTHER HIGHLY PATHOGENIC VIRUSES | 1-gen-2026 | Valenti, Martina Eleonora; Rubini, Daniele; Parra-López, Marisa; Holzerland, Julia; Rodríguez-Martínez, Alejandro; Martina, Maria Grazia; Ramos, Maria C.; Castillo, Francisco; Harty, Ronald N.; Pérez-Sanchez, Horacio; Diederich, Sandra; Luque, Irene; Radi, Marco | |
| Investigating PCSK9 as a therapeutic target in Alzheimer's disease: evidence from patient-derived astrocytes | 1-gen-2025 | Ugolotti, M.; Papotti, B.; Adorni, M. P.; Martina, M. G.; Giannessi, L.; Olejnik, A.; Bell, S. M.; Mortiboys, H.; Radi, M.; Zimetti, F. | |
| Targeting the ESCRT machinery: a promising strategy for the development of novel Broad-Spectrum Antivirals (BSAs). | 1-gen-2025 | Rubini, Daniele; Martina, Maria Grazia; Valenti, Martina Eleonora; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Harty, Ronald N.; Parra-López, Marisa; Holzerland, Julia; Diederich, Sandra; Luque, Irene; Radi, Marco | |
| WO2026017799A1 - SUBSTITUTED 3-CYANOQUINOLINES FOR THE PREVENTION AND TREATMENT OF SEXUALLY TRANSMITTED DISEASES | 1-gen-2025 | Cagno, Valeria; Radi, Marco; Rubini, Daniele; Martina, Maria Grazia | |
| Targeting PI4KB and Src/Abl host kinases as broad-spectrum antiviral strategy: Myth or real opportunity? | 1-gen-2025 | Martina, Maria Grazia; Rubini, Daniele; Radi, Marco; Cagno, Valeria | |
| Discovery of p-Trifluoromethylbenzohydrazide Derivatives as Potent Antiviral Agents against Monkeypox Virus | 1-gen-2025 | Rossi, Sara; Pozzetti, Luca; Carullo, Gabriele; Dichiara, Maria; Butini, Stefania; Radi, Marco; Ramunno, Anna; Terrosi, Chiara; Barra, Giovanni; Berisio, Rita; Gemma, Sandra; Cusi, Maria Grazia; Campiani, Giuseppe | |
| Exploring the druggability of the UEV domain of human TSG101 in search for broad-spectrum antivirals | 1-gen-2025 | Montero, Fernando; Parra-López, Marisa; Rodríguez-Martínez, Alejandro; Murciano-Calles, Javier; Buzon, Pedro; Han, Ziying; Lin, L-Y; Ramos, Maria C; Ruiz-Sanz, Javier; Martinez, Jose C; Radi, Marco; Moog, Christiane; Diederich, Sandra; Harty, Ronald N; Pérez-Sánchez, Horacio; Vicente, Francisca; Castillo, Francisco; Luque, Irene | |
| Effects of CCL20/CCR6 modulators in a T cell adoptive transfer model of colitis | 1-gen-2025 | Allodi, M.; Flammini, L.; Giorgio, C.; Martina, M. G.; Barbieri, F.; Ballabeni, V.; Barocelli, E.; Radi, M.; Bertoni, S. | |
| Harnessing prebiotic formamide chemistry: a novel platform for antiviral exploration | 1-gen-2025 | Martina, Maria Grazia; Vagaggini, Chiara; Dreassi, Elena; De Angelis, Marta; Nencioni, Lucia; Dragoni, Filippo; Giammarino, Federica; Boccuto, Adele; Zazzi, Maurizio; Vicenti, Ilaria; Radi, Marco | |
| Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses | 1-gen-2025 | Barbieri, Francesca; Martina, Maria Grazia; Pesce, Emanuela; Bianchi, Elena; Cabella, Noemi; Crespan, Emmanuele; Rossi, Sara; Gemma, Sandra; Campiani, Giuseppe; Milite, Ciro; Pepe, Giacomo; Campiglia, Pietro; Sbardella, Gianluca; Maga, Giovanni; Cagno, Valeria; Pedemonte, Nicoletta; Radi, Marco | |
| CHEMISTRY-DRIVEN OPTIMIZATION OF PURINE-BASED ANTIVIRALS FOR THE IDENTIFICATION OF NEW BROAD-SPECTRUM AGENTS | 1-gen-2025 | Valenti, Martina Eleonora; Martina, Maria Grazia; Vincetti, Paolo; Vicenti, Ilaria; Crespan, Emmanuele; Nencioni, Lucia; Kaptein, Suzanne J. F.; Neyts, Johan; Vanderlinden, Evelien; Schols, Dominique; De Forni, Davide; Lori, Franco; Zazzi, Maurizio; Maga, Giovanni; Radi, Marco | |
| DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X | 1-gen-2025 | Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco | |
| DEVELOPMENT OF NOVEL BROAD-SPECTRUM ANTIVIRALS TARGETING THE HUMAN HELICASE DDX3X | 1-gen-2025 | Valenti, Martina Eleonora; Martina, Maria Grazia; Falchi, Federico; Bavagnoli, Laura; Pallotta, Michela; Crespan, Emmanuele; Maga, Giovanni; Radi, Marco | |
| “Investigating PCSK9 inhibition as potential strategy in Alzheimer’s disease” | 1-gen-2025 | Ugolotti, M.; Papotti, B.; Adorni, M. P.; Giannessi, L.; Lupo, M. G.; Ferri, N.; Radi, M.; Bernini, F.; Zimetti, F. | |
| Development of Novel PCSK9 Inhibitors as Potential Broad-Spectrum Antivirals | 1-gen-2025 | Savian, Chiara; Giannessi, Lisa; Martina, Maria Grazia; Ugolotti, Martina; Papotti, Bianca; Palumbo, Marcella; Giovanna Lupo, Maria; Mattina, Beatrice; Padula, Cristina; Nicoli, Sara; Ferri, Nicola; De Forni, Davide; Lori, Franco; Cagno, Valeria; Zimetti, Francesca; Radi, Marco | |
| A sustainable one-pot three step approach for the synthesis of 3,5-disubstituted 1,2,4-triazines as versatile pharmacological tools. | 1-gen-2024 | Rubini, D.; Martina, M. G.; Incerti, M.; Barbieri, F.; Radi, M. | |
| Discovery of small molecule inhibitors of the Tsg101-PTAP interaction as potential host-targeted broad-spectrum antivirals. | 1-gen-2024 | Rubini, Daniele; Martina, Maria Grazia; Valenti, Martina Eleonora; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Harty, Ronald N.; Parra-López, Marisa; Luque, Irene; Radi, Marco | |
| Targeting the ESCRT machinery: a promising strategy for the development of novel Broad-Spectrum Antivirals (BSAs). | 1-gen-2024 | Rubini, Daniele; Martina, Maria Grazia; Valenti, Martina Eleonora; Rodríguez-Martínez, Alejandro; Pérez-Sánchez, Horacio; Harty, Ronald N.; Parra-López, Marisa; Diederich, Sandra; Luque, Irene; Radi, Marco | |
| Identification of 4-amino-2-Pyridones as new potent PCSK9 inhibitors: From phenotypic hit discovery to in vivo tolerability | 1-gen-2024 | Giannessi, L; Lupo, Mg; Rossi, I; Martina, Mg; Vilella, A; Bodria, M; Giuliani, D; Zimetti, F; Zanotti, I; Potì, F; Bernini, F; Ferri, N; Radi, M |
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